Carbamates and crop protection agents containing them

ABSTRACT

Carbamates of the formula I ##STR1## wherein B is a saturated or unsaturated heterocyclic group, and the other substituents are defined in the specification, and having crop protection properties.

This application is a division of application Ser. No. 08/256,628, filed on Jul. 29, 1994, now U.S. Pat. No. 5,824,705, which is a 371 of international Application No. PCT/EP93/00104, filed Jan. 18, 1993.

The present invention relates to carbamates and crop protection agents, in particular for controlling fungi, insects, nematodes and spider mites.

It is known that aniline derivatives, for example isopropyl N-phenylcarbamate or the corresponding 3-chlorophenyl ester (GB 574 995) or methyl N-3,4-dichlorophenylcarbamate (BE 612 550) can be used as crop protection agents. However, their fungicidal action is unsatisfactory.

It has now been found, surprisingly, that carbamates of the formula I ##STR2## where the substituents have the following meanings: Z is methoxy, NH₂, NHCH₃, N(CH₃)₂, CH₃, C₂ H₅, CF₃ or CCl₃,

X and Y independently of one another are each hydrogen,

F, Cl, Br, CF₃₁, CN, NO₂, alkoxy, alkenyloxy, alkynyloxy, alkyl, alkenyl or alkynyl or X and Y may be condensed together to form an unsubstituted or substituted aromatic or heteroaromatic, alicyclic or heterocyclic, partially or completely hydrogenated ring,

R¹ is unsubstituted or substituted alkyl, alkenyl, cyclopropyl, cyclopropylmethyl, cyclobutyl, --CH₂ --CN, --CH₂ OCH₃, --CO₂ CH₃ or --S--R⁵, O-alkyl, O-alkenyl, O-alkynyl, O-cycloalkyl, O-cycloalkenyl or O--CO₂ -alkyl,

A is --O--, --S--, --CR² ═CR³ --, CHR² --O--, --CHR² --S--, --CHR² --O--N═C(R⁴)--, --CR² ═N--O--, --O--N═C(R⁴)--, --C.tbd.C--, --CHR² --CHR³ --, --CHR² --O--, --CO--O--CHR² -- or a single bond,

B can be unsubstituted or substituted and is alkyl, alkenyl, alkynyl, cycloalkyl, cycloalkenyl, cycloalkynyl, aryl, hetaryl, heterocyclyl, hydrogen, unsubstituted or substituted alkylaryl, unsubstituted or substituted alkylhetaryl, unsubstituted or substituted alkylcycloalkyl or unsubstituted or substituted alkylcycloalkenyl,

R² and R³ independently of one another are each hydrogen, alkyl, alkenyl, alkynyl or cycloalkyl,

R⁴ is hydrogen, CN, alkyl, alkenyl, alkynyl, alkoxy or cycloalkyl,

R⁵ is alkyl, cyclopropyl, cyclopropylmethyl or cyclobutyl, and their plant-tolerated acid addition products and base addition products have a good fungicidal, acaricidal, insecticidal and nematocidal action.

Acids for addition products are, for example, mineral acids, such as hydrochloric acid, hydrobromic acid, phosphoric acid, sulfuric acid or nitric acid, or carboxylic acids, such as formic acid, acetic acid, oxalic acid, malonic acid, lactic acid, malic acid, succinic acid, tartaric acid, citric acid, salicylic acid, p-toluenesulfonic acid or dodecylbenzenesulfonic acid, as well as proton-acidic compounds generally, for example saccharin.

Bases for base addition products are, for example, potassium hydroxide, sodium hydroxide, potassium carbonate, sodium carbonate and ammonium hydroxide.

The novel compounds of the formula I may be obtained in the preparation as mixtures of stereoisomers (E/Z isomers, diastereomers, enantiomers), which can be separated into the individual components in a conventional manner, for example by crystallization or chromatography. Both the individual isomers and mixtures thereof may be used as fungicides, acaricides, nematocides or insecticides, and form the subject of the present invention.

The abovementioned alkyl radicals may be substituted and are of 1 to 6 carbon atoms.

The abovementioned alkenyl and alkynyl radicals may be substituted and are of 2 to 6 carbon atoms.

The abovementioned cycloalkyl radicals are of 3 to 10 carbon atoms and are unsubstituted or substituted, for example by 1 to 4 identical or different substituents R⁶.

The abovementioned aryl radicals are of 6, 10 or 14 carbon atoms and are unsubstituted or substituted, for example by 1 to 4 identical or different substituents R⁶.

The abovementioned hetaryl radicals have 5 to 14 ring atoms, including from 1 to 4 hetero atoms selected from the group consisting of N, O and S, are unsaturated and are unsubstituted or substituted, for example by 1 to 4 identical or different substituents R⁶.

The abovementioned heterocyclyl radicals have 5 to 14 carbon atoms, including 1 to 4 hetero atoms selected from the group consisting of N, O and S, are saturated or partially unsaturated and are unsubstituted or substituted, for example by 1 to 4 identical or different substitutents R⁶.

The abovementioned cycloalkenyl radicals are of 5 to 14 carbon atoms and are unsubstituted or substituted, for example by 1 to 4 identical or different substituents R⁶.

Two adjacent substituents R⁶, together with the carbon atoms of which they are substituents, may form a carbocyclic hydrogenated, partially unsaturated or aromatic ring having 3 to 14 carbon atoms or a heterocyclic hydrogenated, partially unsaturated or heteroaromatic ring having 3 to 14 carbon atoms, including 1 to 4 hetero atoms selected from the group consisting of N, O and S.

R⁶ may be unsubstituted or substituted, for example by 1 to 4 identical or different substituents R⁷, and R⁶ is, for example, hydrogen, halogen, cyano, nitro, haloalkyl, alkyl, haloalkoxy, alkenyl, alkynyl, cyclolkyl, aryl, hetaryl, heterocyclyl, cycloalkenyl, alkoxy, alkenyloxy, alkynyloxy, cycloalkoxy, aryloxy, hetaryloxy, heterocyclyloxy, cycloalkenyloxy, alkoximino, alkenyloximino, alkynyloximino, cycloalkoxyimino, cycloalkenyloximino, aryloximino, hetaryloximino, heterocyclyloximino, alkoxycarbonyl, alkenyloxycarbonyl, alkynyloxycarbonyl, cycloalkyloxycarbonyl, aryloxycarbonyl, hetaryloxycarbonyl, heterocyclyloxycarbonyl, cycloalkenyloxycarbonyl, alkylaminocarbonyl, dialkylaminocarbonyl, alkenylaminocarbonyl, dialkenylaminocarbonyl, alkylthio, alkenylthio, alkynylthio, cycloalkylthio, arylthio, hetarylthio, heterocyclylthio, cycloalkenylthio, alkylamino, alkenylamino, alkynylamino, cycloalkylamino, arylamino, hetarylamino, heterocyclylamino, cycloalkenylamino, alkylcarbonyl, alkenylcarbonyl, alkynylcarbonyl, cycloalkylcarbonyl, arylcarbonyl, hetarylcarbonyl, heterocyclylcarbonyl, cycloalkenylcarbonyl, alkylsulfoxyl, alkenylsulfoxyl, alkynylsulfoxyl, cycloalkylsulfoxyl, arylsulfoxyl, hetarylsulfoxyl, heterocyclylsulfoxyl, cycloalkenylsulfoxyl, alkylsulfonyl, alkenylsulfonyl, alkynylsulfonyl, cycloalkylsulfonyl, arylsulfonyl, hetarylsulfonyl, heterocyclylsulfonyl, cycloalkenylsulfonyl, alkylsulfinyl, alkenylsulfinyl, alkynylsulfinyl, cycloalkylsulfinyl, arylsulfinyl, hetarylsulfinyl, heterocyclylsulfinyl or cycloalkenylsulfinyl.

R⁷ is any substituent and is, for example, hydrogen, halogen, cyano, nitro, haloalkyl, alkyl, haloalkoxy, alkenyl, alkynyl, cycloalkyl, aryl, hetaryl, heterocyclyl, cycloalkenyl, alkoxy, alkenyloxy, alkynyloxy, cycloalkoxy, aryloxy, hetaryloxy, heterocyclyloxy, cycloalkenyloxy, alkoximino, alkenyloximino, alkynyloximino, cycloalkoximino, cycloalkenyloximino, aryloximino, hetaryloximino, heterocyclyloximino, alkoxycarbonyl, alkenyloxycarbonyl, alkynyloxycarbonyl, cycloalkyloxycarbonyl, aryloxycarbonyl, hetaryloxycarbonyl, heterocyclyloxycarbonyl, cycloalkenyloxycarbonyl, alkylaminocarbonyl, dialkylaminocarbonyl, alkenylaminocarbonyl, dialkenylaminocarbonyl, alkylthio, alkenylthio, alkynylthio, cycloalkylthio, arylthio, hetarylthio, heterocyclylthio, cycloalkenylthio, alkylamino, alkenylamino, alkynylamino, cycloalkylamino, arylamino, hetarylamino, heterocyclylamino, cycloalkenylamino, alkylcarbonyl, alkenylcarbonyl, alkynylcarbonyl, cycloalkylcarbonyl, arylcarbonyl, hetarylcarbonyl, heterocyclylcarbonyl, cycloalkenylcarbonyl, alkylsulfoxyl; alkenylsulfoxyl, alkynylsulfoxyl, cycloalkylsulfoxyl, arylsulfoxyl, hetarylsulfoxyl, heterocyclylsulfoxyl, cycloalkenylsulfoxyl, alkylsulfonyl, alkenylsulfonyl, alkynylsulfonyl, cycloalkylsulfonyl, arylsulfonyl, hetarylsulfonyl, heterocyclylsulfonyl, cycloalkenylsulfonyl, alkylsulfinyl, alkenylsulfinyl, alkynylsulfinyl, cycloalkylsulfinyl, arylsulfinyl, hetarylsulfinyl, heterocyclylsulfinyl or cycloalkenylsulfinyl.

The abovementioned alkyl radicals may be substituted, are preferably of 1 to 6 carbon atoms and are, in particular, methyl, ethyl, propyl, such as n-propyl or isopropyl, butyl, such as n-butyl, isobutyl, tert-butyl or sec-butyl, pentyl or hexyl.

The abovementioned alkenyl radicals may be substituted, are preferably of 2 to 6 carbon atoms and are, in particular, ethenyl, propenyl, such as prop-1-enyl, prop-2-enyl or prop-1-en-2-yl, butenyl, such as but-1-enyl, but-2-enyl, but-3-enyl, but-1-en-3-yl, but-2-en-2-yl, but-1-en-2-yl, 2-methyl-1-propenyl or 2-methyl-2-propenyl, pentenyl or hexenyl.

The abovementioned alkynyl radicals may be substituted, are preferably of 2 to 6 carbon atoms and are, in particular, ethynyl, propynyl, such as prop-1-ynyl or prop-3-ynyl, butynyl, such as but-1-ynyl, but-2-ynyl, but-3-ynyl or 1-methylprop-2-ynyl, pentynyl or hexynyl.

The abovementioned halogens are fluorine, chlorine, bromine or iodine.

The abovementioned cycloalkyl radicals are preferably cyclopropyl, cyclobutyl, cyclopentyl, cyclohexyl, cycloheptyl, cyclooctyl, cyclononyl, cyclodecyl, bornanyl, norbornanyl, dicyclohexyl, bicyclo[3.3.0]octyl, bicyclo[3.2.1]octyl, bicyclo[2.2.2]octyl or bicyclo[3.3.1]nonyl.

The abovementioned cycloalkenyl radicals are preferably cyclopropenyl, cyclobutenyl, cyclopentenyl, cyclohexenyl, cycloheptenyl, cyclooctenyl, cyclononenyl, cyclodecenyl, bornenyl, norbornenyl, bicyclo[3.3.0]-octenyl, bicyclo[3.2.1]octenyl, bicyclo[2.2.2]octenyl or bicyclo[3.3.1]nonenyl.

The abovementioned haloalkyl radicals are preferably C₁ -C₄ -haloalkyl, in particular C₁ - or C₂ -haloalkyl, such as chloromethyl, dichloromethyl, trichloromethyl, fluoromethyl, difluoromethyl, trifluoromethyl, chlorofluoromethyl, dichlorofluoromethyl, chlorodifluoromethyl, 1-fluoroethyl, 2-fluoroethyl, 2,2-difluoroethyl, 2,2,2-trifluoroethyl, 2-chloro-2-fluoroethyl, 2-chloro-2,2-difluoroethyl, 2,2-dichloro-2-fluoroethyl, 2,2,2-trichloroethyl or pentafluoroethyl.

The abovementioned haloalkoxy radicals are preferably C₁ -C₄ -haloalkoxy, in particular C₁ - or C₂ -haloalkoxy, such as chloromethoxy, dichloromethoxy, trichloromethoxy, fluoromethoxy, difluoromethoxy, trifluoromethoxy, chlorofluoromethoxy, dichlorofluoromethoxy, chlorodifluoromethoxy, 1-fluoroethoxy, 2-fluoroethoxy, 2,2-difluoroethoxy, 2,2,2-trifluoroethoxy, 2-chloro-2-fluoroethoxy, 2-chloro-2,2-difluoroethoxy, 2,2-dichloro-2-fluoroethoxy, 2,2,2-trichloroethoxy or pentafluoroethoxy.

The abovementioned aryl radicals are preferably phenyl, 1-naphthyl, 2-naphtyl, 1-anthracenyl, 2-anthracenyl or 9-anthracenyl.

The abovementioned hetaryl radicals are preferably furyl, such as 2-furyl or 3-furyl, thienyl, such as 2-thienyl or 3-thienyl, pyrrolyl, such as 1-pyrrolyl, 2-pyrrolyl or 3-pyrrolyl, isoxazolyl, such as 3-isoxazolyl, 4-isoxazolyl or 5-isoxazolyl, isothiazolyl, such as 3-isothiazolyl, 4-isothiazolyl or 5-isothiazolyl, pyrazolyl, such as 1-pyrazolyl, 3-pyrazolyl, 4-pyrazolyl or 5-pyrazolyl, oxazolyl, such as 2-oxazolyl, 4-oxazolyl or 5-oxazolyl, thiazolyl, such as 2-thiazolyl, 4-thiazolyl or 5-thiazolyl, imidazolyl, such as 1-imidazolyl, 2-imidazolyl, 4-imidazolyl or 5-imidazolyl, 1,2,3-thiadiazolyl, 1,2,4-thiadiazolyl, 1,2,5-thiadiazolyl, 1,3,4-thiadiazolyl, tetrazolyl, 1,2,3,4-thiatriazolyl, 1,2,3,4-oxatriazolyl, pyridyl, such as 2-pyridyl or 4-pyridyl, pyridazinyl, such as 3-pyridazinyl or 4-pyridazinyl, pyrimidinyl, such as 2-pyrimidinyl, 4-pyrimidinyl or 5-pyrimidinyl, pyrazinyl, such as 2-pyrazinyl or 3-pyrazinyl, 1,2,4-triazinyl, 1,3,5-triazinyl or 1,2,4,5-tetrazinyl.

Adjacent substituents of the hetero atoms may be condensed to form an aromatic or heteroaromatic ring, so that hetaryl also comprises fused ring systems, eg. benzofuranyl, isobenzofuranyl, 1-benzothienyl, 2-benzothienyl, indolyl, isoindolyl, benzisoxazolyl, benzoxazolyl, benzisothiazolyl, benzothiazolyl, such as 2-benzothiazolyl, 4-benzothiazolyl, 5-benzothiazolyl, 6-benzothiazolyl or 7-benzothiazolyl, indazolyl, benzimidazolyl, benzofurazanyl, dibenzofuranyl, dibenzothienyl, acridinyl, phenanthridinyl, carbazolyl, quinolyl, isoquinolyl, phthalazinyl, quinazolinyl, quinoxalinyl, cinnolinyl, 1,5-naphthyridinyl, 1,6-naphthyridinyl, 1,7-naphthyridinyl, 1,8-naphthyridinyl, pteridinyl, pyrrolopyridinyl, pyrrolopyridazinyl, pyrrolopyrimidinyl, pyrrolopyrazinyl, pyrrolotriazinyl, furopyridyl, furopyridazinyl, furopyrimidinyl, furopyrazinyl, furotriazinyl, thienopyridyl, thienopyridazinyl, thienopyrimidinyl, thienopyrazinyl, thienotriazinyl, imidazopyridazinyl, imidazopyrimidinyl, imidazopyrazinyl, pyrazolopyridyl, pyrazolopyridazinyl, pyrazolopyrimidinyl, pyrazopyrazinyl, isoxazolopyrazinyl, oxazolopyridyl, oxazolopyridazinyl, oxazolopyrimidinyl, oxazolopyrazinyl, thiazolopyridyl, thiazolopyridazinyl, isothiazolopyrazinyl, triazolopyridyl, triazolopyridazinyl, triazolopyrimidinyl or triazolopyrazinyl.

The abovementioned heterocycyl radicals are preferably 2-tetrahydrofuranyl, oxiranyl, 3-tetrahydrofuranyl, 2-tetrahydrothienyl, 3-tetrahydrothienyl, 2-pyrrolidinyl, 3-pyrrolidinyl, 3-isoxazolidinyl, 4-isoxazolidinyl, 5-isoxazolidinyl, 3-isothiazolidinyl, 4-isothiazolidinyl, 5-isothiazolidinyl, 3-pyrazolidinyl, 4-pyrazolidinyl, 5-pyrazolidinyl, 2-oxazolidinyl, 4-oxazolidinyl, 5-oxazolidinyl, 2-thiazolidinyl, 4-thiazolidinyl, 5-thiazolidinyl, 2-imidazolidinyl, 4-imidazolidinyl, 1,2,4-oxadiazolidin-3-yl, 1,2,4-oxadiazolidin-5-yl, 1,2,4-thiadiazolidin-3-yl, 1,2,4-thiadiazolidin-5-yl, 1,2,5-triazolidin-3-yl, 1,3,4-oxadiazolidin-2-yl, 1,3,4-thiadiazolidin-2-yl, 1,3,4-triazolidin-2-yl, 2,3-dihydrofur-2-yl, 2,3-dihydrofur-3-yl, 2,5-dihydrofur-2-yl, 2,5-dihydrofur-2-yl, 2,3-dihydrofur-3-yl, 2,3-dihydrothieno-2-yl, 2,3-dihydrothien-3-yl, 2,5-dihydrothien-2-yl, 2,4-pyrrolin-2-yl, 2,3-pyrrolin-3-yl, 2,5-pyrrolin-2-yl, 2,5-pyrrolin-3-yl, 2,3-isoxazolidin-3-yl, 3,4-isoxazolin-3-yl, 4,5-isoxazolin-2-yl, 2,3-isoxazolin-4-yl, 3,4-isoxazolin-3-yl, 4,5-isoxazolin-4-yl, 2,3-isoxazolin-5-yl, 3,4-isoxazolin-5-yl, 4,5-isoxazolin-5-yl, 2,3-isothiazolin-3-yl, 3,4-isothiazolin-3-yl, 4,5-isothiazolin-3-yl, 2,3-isothiazolin-4-yl, 3,4-isothiazolin-4-yl, 4,5-isothiazolin-4-yl, 2,3-isothiazolin-5-yl, 3,4-isothiazolin-5-yl, 4,5-isothiazolin-5-yl, 2,3-dihydropyrazol-1-yl, 2,3-dihydropyrazol-2-yl, 2,3-dihydropyrazol-3-yl, 2,3-dihydropyrazol-4-yl, 2,3-dihydropyrazol-5-yl, 3,4-dihydropyrazol-1-yl, 3,4-dihydropyrazol-2-yl, 3,4-dihydropyrazol-4-yl, 3,4-dihydropyrazol-5-yl, 4,5-dihydropyrazol-1-yl, 4,5-dihydropyrazol-3-yl, 4,5-dihydropyrazol-4-yl, 4,5-dihydropyrazol-5-yl, 3,4-dihydrooxazol-2-yl, 2,3-dihydrooxazol-3-yl, 2,3-dihydrooxazol-4-yl, 2,3-dihydrooxazol-5-yl, 3,4-dihydrooxazol-2-yl, 3,4-dihydrooxazol-3-yl, 3,4-dihydrooxazol-4-yl, 3,4-dihydrooxazol-5-yl, 3,4-dihydrooxazol-2-yl, 3,4-dihydrooxazol-3-yl, 3,4-dihydrooxazol-4-yl, 2-piperidinyl, 3-piperidinyl, 4-piperidinyl, 3-tetrahydropyridazinyl, 4-tetrahydropyridazinyl, 2-tetrahydropyrimidinyl, 4-tetrahydropyrimidinyl, 5-tetrahydropyrimidinyl, 2-tetrahydropyrazinyl, 1,3,5-tetrahydrotriazin-2-yl, 1,2,4-tetrahydrotriazin-3-yl, 1,3-dihydrooxazin-2-yl, 1,3-dithian-2-yl, oxazol-2-in-2-yl, 2-tetrahydropyranyl, 1,3-dioxolan-2-yl, thiazol-2-in-2-yl, 3,4,5,6-tetrahydropyridin-2-yl, 4H-1,3-thiazin-2-yl, 4H-3,1-benzothiazin-2-yl, 1,1-dioxo-2,3,4,5-tetrahydrothien-2-yl, 2H-1,4-benzothiazin-3-yl, 2H-1,4-benzoxazin-3-yl, 1,3-dihydrooxazin-2-yl, 1,3-dithian-2-yl, N-morpholinyl or dihydroquinazolinyl.

The invention furthermore relates to carbamates of the formula I ##STR3## where the substituents have the following meanings: Z is methoxy, NH₂, NHCH₃ or CH₃,

X and Y independently of one another are each hydrogen,

F, Cl, Br, CF₃, CN, NO₂, alkoxy, alkenyloxy, alkynyloxy, alkyl, alkenyl or alkynyl or X and Y may be condensed together to form a phenyl ring,

R¹ is hydrogen, alkyl, alkenyl alkynyl cyclopropyl, cyclopropylmethyl, cyclobutyl, --CH₂ --CN, --CH₂ --O--CH₃, --CO₂ CH₃ or --S--R⁵,

A is --O--, --CR² ═CR³ --, --C.tbd.C--, --CHR² --O--, --CHR² --S--, --CHR² --O--N═C(R⁴)--, --CR² ═N--O-- or --O--N═C(R⁴)--,

a) B is substituted phenyl when A is --CR² .tbd.CR³ --, --C═C--, --CHR² --O--, --CHR² --S--, --CHR² --O--N═C(R⁴)--, --CR² ═N--O-- or --O--N═C(R⁴),

b) or B is unsubstituted or substituted cyclolalkyl, unsubstituted or substituted cycloalkenyl, unsubstituted or substituted heterocyclyl, unsubstituted or substituted hetaryl, unsubstituted or substituted naphthyl, unsubstituted or substituted arylalkyl, unsubstituted or substituted hetarylalkyl, unsubstituted or substituted cycloalkylalkyl, unsubstituted or substituted cycloalkenylalkyl or unsubstituted or substituted anthracenyl,

R² and R³ independently of one another are each hydrogen, alkyl, alkenyl, alkynyl or cycloalkyl,

R⁴ is CN, alkyl, alkenyl, alkynyl or cycloalkyl and

R⁵ is alkyl, cyclopropyl, cyclopropylmethyl or cyclobutyl, and their plant-tolerated acid addition products and base addition products.

The invention furthermore relates to carbamates of the formula II ##STR4## where X, Y, R¹ and B have the meanings stated in claim 2.

The invention furthermore relates to carbamates of the formula III ##STR5## where X, Y, R¹ and B have the meanings stated in claim 2.

The invention furthermore relates to carbamates of the formula I as claimed in claim 2, where A is --CH═CH-- and X, Y, R¹ and B have the meanings stated in claim 2.

The invention furthermore relates to carbamates of the formula VII ##STR6## where the substituents have the following meanings: X and Y independently of one another are each hydrogen,

F, Cl, Br, CF₃, CN, NO₂₁ alkoxy, alkenyloxy, alkynyloxy, alkyl, alkenyl or alkynyl or X and Y may be condensed together to form an unsubstituted or substituted aromatic or heteroaromatic, alicyclic or heterocyclic, partially or completely hydrogenated ring,

R¹ can be unsubstituted or substituted and is alkyl, alkenyl, alkynyl, cycloalkyl, cycloalkenyl or --CO₂ -alkyl,

A is --O--, --S--, --CR² ═CR³ --, CHR² --O--, --CHR² --S--, --CHR² --O--N═C(R⁴)--, --CR² ═N--O--, --O--N═C(R⁴)--, --C.tbd.C--, --CHR² --CHR³ --, --CHR² --O--CO--, --O--CHR² -- or a single bond,

B can be unsubstituted or substituted and is alkyl, alkenyl, alkynyl, cycloalkyl, cycloalkenyl, cycloalkynyl, aryl, hetaryl, heterocyclyl or hydrogen,

R² and R³ independently of one another are each hydrogen, alkyl, alkenyl, alkynyl or cycloalkyl and R⁴ is hydrogen, cyano, alkyl, alkenyl, alkynyl, cycloalkyl or alkoxy, and their plant-tolerated acid addition products and base addition products.

The invention furthermore relates to carbamates of the formula VIII ##STR7## where A, B and R¹ have the meanings stated in claim 9.

The invention furthermore relates to carbamates of the formula IX ##STR8## where R¹ and B have the meanings stated in claim 1.

The invention furthermore relates to carbamates of the formula X ##STR9## where R¹ and B have the meanings stated in claim 1.

The novel compounds can be prepared, for example, by the following processes:

The nitrobenzenes 1 obtainable by standard processes are reduced to the anilines 2, for example with hydrogen or hydrogen transfer agents, such as ammonium formate, in the presence of suitable catalysts, such as Pd, Pt or Ni, with complex reducing agents, eg. Collman's reagent (Na₂ Fe(CO)₄) or by other methods known from the literature (J. March, Advanced Organic Chemistry, 3rd Edition, 1985, page 1103 et seq.). The anilines 2 are reacted under alkaline conditions with methyl chloroformate to give the carbamates 3. The reaction of the carbamates 3 under alkaline conditions with the corresponding alkylating agents, acylating agents or R⁵ --S--S(═O)₂ --R⁵ gives the derivatives 4 (Scheme 1). ##STR10##

The nitrobenzenes 5 can be converted into the carbamates 6 similarly to Scheme 1. The halogen derivatives 7 (Z═Cl or Br) are obtainable by acidic cleavage of the methyl ether of 6 (Scheme 2). ##STR11##

Alternatively, the halogen derivatives 7 (Z═Cl or Br) are obtainable from the derivatives 9 by free radical halogenation. The carbamates 9 are in turn prepared from the corresponding starting materials 8, similarly to Scheme 1 (Scheme 3). ##STR12##

The halogen derivatives 7 (Z═Cl or Br) can be converted into the active ingredients 10 under alkaline conditions. Alternatively, the compounds 7 are converted into the phosphorus compounds 11a and 11b by reaction with P(C₆ H₅)₃ or P(O-Alkyl)₃, or into the carbonyl compounds 12 by oxidation (for example with N-methylmorpholine N-oxide) (Scheme 4). ##STR13##

The corresponding stilbenes 13 are obtainable from the phosphonium salts 11a or phosphonates 11b or carbonyl compounds 12 by a wittig reaction (Scheme 5). ##STR14##

Partial reduction of the nitroaromatics 21 (for example with zinc (similarly to Bamberger et al., Ann. Chem. 316 (1901), 278) or with hydrogen in the presence of suitable catalysts such as platinum (similarly to European Patent 85,890)) gives the hydroxylamines 22, which can be reacted under alkaline conditions with an acylating agent (eg. propionyl chloride) or a carbamoylating agent (eg. methyl isocyanate) to give the compound 23 and then with an electrophile, for example with an alkylating agent, to give the active ingredients 24 (scheme 11). ##STR15##

In addition, the hydroxylamine 25 can be acylated or aminoacylated (for example with methyl isocyanate) (similarly to Bamberger et al., Ann. Chem. 316 (1901), 278; European Patent 85,890) to give the compound 26, which can then be alkylated or alkoxyacylated (for example with chloroformates) to give the hydroxylamine derivative 27. The free radical halogenation of 27, for example with N-bromosuccinamide, bromine, chlorine or SO₂ Cl₂ in the presence of free radical initiator, eg. azobisisobutyronitrile, or with exposure to UV light, then gives the halide 28 (Hal═Cl or Br; Scheme 12). ##STR16##

The halides 28 can then be converted into the compounds 29 with the corresponding nucelphiles (Scheme 13). ##STR17##

In addition, the halides 28 can be converted by free radical reaction to the dihalide 30 and then converted with H₂ O/MeOH in the presence of AgNO₃ into the carbonyl compound 31 or reacted directly with N-methylmorpholine N-oxide to give the carbonyl compound 11. Furthermore, the phosphonates, phosphonium salts or phosphine oxides 32 (P is the particular organophosphorus radical) are obtainable from the halides 8 (Scheme 14). ##STR18##

The carbonyl compounds 31 can then be reacted with the corresponding hydroxylamines to give the oximes 33 or can be subjected to a Wittig reaction to give the olefins 34, The olefins 34 are also obtainable by a Wittig reaction starting from the phosphonates, phosphonium salts or phosphine oxides 32 (Scheme 15). ##STR19##

The saturated compounds 35 can be prepared from the olefins 34 by reduction or, where R² and R³ are each H, the acetylenes 36 can be prepared from said olefins by halogen addition (Hal═Cl, Br or I) and subsequent two-fold elimination of hydrogen halide (Scheme 16). ##STR20##

Alternatively, the ureas 39 can be synthesized by acylation of the hydroxylamines 22 to the compounds 37, subsequent alkylation or acylation to the compounds 38 and substitution of the nucleofugic leaving group V (V is, for example, OCH₃₁, OCCl₃, CCl₃, O -phenyl or O-p-nitrophenyl) by NH₃, H₂ N--CH₃ or HN(CH₃)₂ (Scheme 17). ##STR21##

Alternatively, ureas of the formula 39 can also be obtained by alkylating ureas of the formula 41, which in turn are obtainable from 17 by reacting 17 with the corresponding amines, or directly from 22 by amino-carbonylation (for example with dimethylcarbamoyl chloride or methyl isocyanate) (cf. for example Houben-Weyl, volume E16a, page 208).

Furthermore, ureas of the formula 39 can also be obtained from the N-aryl-O-alkylhydroxylamines of the formula 42 in a similar manner by amino-carbonylation.

The compounds of the formula 42 are in turn obtainable by methods known from the literature, from hydroxylamines of the formula 2 (cf. for example Houben-Weyl, volume E16a, pages 271 and 282-289).

In addition, the hydroxylamines 22 are obtainable from the anilines 43 by formation of the imines 44, oxidation of the compounds 44 with the m-chloroperbenzoic acid and reaction of the oxaziridines 45 with hydroxylamine (Scheme 18; similarly to G. Grundke et al., Synthesis 1987, 1115). ##STR22##

The Examples which follow illustrate the preparation of the novel compounds.

EXAMPLES Example 1

Methyl N-ethyl-N-(2-(2'-methylphenoxymethyl)-phenyl)-carbamate (Table 7, No. 2)

a) Methyl N-(o-methylphenyl)-carbamate

50 g (0.53 mol) of methyl chloroformate are added dropwise to 53 g (0.5 mol) of o-toluidene in 500 ml of methylene chloride. During this procedure, the reaction solution heats up to the boiling point and a colorless solid is precipitated.

Stirring is carried out for one hour, after which 200 ml of 10% strength sodium hydroxide solution are added dropwise, the colorless solid going into solution. The organic phase is dried over MgSO₄ and evaporated down under reduced pressure. The remaining solid is stirred with n-hexane and filtered off under suction. 84 g (0.5 mol, quantitative yield) of the title compound are obtained as a colorless solid. mp.=61-62° C.

¹ H-NMR (DMSO-d₆ ; δ (ppm)): 8.85 (s, 1H, NH); 7.35 (d, broad, 1H, aromatic); 7.1 (m, 3H, aromatic); 3.6 (s, 3H, OCH₃); 2.2 (s, 3H, CH₃)

b) Methyl N-ethyl-N-(o-methylphenyl)-carbamate

5.1 g (0.2 mol) of sodium hydride are added a little at a time to 30 g (0.18 mol) of methyl N-(o-methylphenyl)-carbamate (Example 1a) in 200 ml of dimethylformamide. After the evolution of gas has ceased, 30 g (0.2 mol) of ethyl iodide are added drop-wise, the reaction mixture being lightly cooled in a water bath. A white solid is precipitated. After about 4 hours, the reaction mixture is diluted with water and the aqueous phase is extracted three times with ether. The organic phase is dried over MgSO₄ and evaporated down. The residue is distilled. 32.5 g (0.17 mol=93%) of the title compound are obtained as a colorless oil. bp.⁰.5 =74° C.

¹ H-NMR (CDCl₃ ; δ (ppm): 7.2 (m, 3H, aromatic); 7.1 (m, 1H, aromatic); 3.8 (m, 1H, N--CH_(A)); 3.6 (s, 3H, OCH₃); 3.5 (m, 1H, N--CH_(B)); 2.2 (s, 3H, CH₃); 1.1 (t, 3H, CH₃)

c) Methyl N-ethyl-N-(o-bromomethylphenyl)-carbamate

A mixture of 30 g (0.155 mol) of methyl N-ethyl-N-(o-methylphenyl)-carbamate (Example 1b), 33 g (0.185 mol) of N-bromosuccinimide and 0.1 g of azoisobutyronitrile in 300 ml of carbon tetrachloride is exposed to a 300 W UV lamp for 6 hours. During this procedure, the contents of the flask heat up to about 70° C. Thereafter, the reaction mixture is washed four times with water, dried and evaporated down. The residue obtained comprises 41 g of a brown oil which contains the title compound in about 50% purity and is used without further purification in the next reaction.

¹ H-NMR (CDCl₃ ; δ (ppm)): 7.2 (m, 4H, aromatic); 4.45 (s, 2H, CH₂ --Br); 3.8 (m, 1H, N--CH_(A)); 3.6 (s, 3H, OCH₃); 3.5 (m, 1H, N--CH_(B)); 1.15 (t, 3H, J=8 Hz, CH₃)

d) Methyl N-ethyl-N-(2-(2'-methylphenoxymethyl)-phenyl)-carbamate (Table 7, No. 2)

2.4 g (17 mmol) of sodium hydride are added a little at a time to 8.6 g (80 mmol) of o-cresol in 100 ml of dimethylformamide. Stirring is carried out for 30 minutes at room temperature (20° C.), after which 20.5 g of methyl N-ethyl-N-(o-bromomethylphenyl)-carbamate (Example 1c, about 50% purity, about 37 mmol) are added. Stirring is carried out overnight at room temperature, after which the reaction mixture is diluted with water and the aqueous phase is extracted three times with ether. The combined ether phases are dried over MgSO₄ and evaporated down. The residue is distilled in a kugelrohr (bulb tube) apparatus. 10 g of a yellow oil are obtained at 220° C. and 0.2 mbar, and the oil is then purified by chromatography with cyclohexane/ethyl acetate mixtures over silica gel and then over alumina. The product thus obtained is purified again by kugelrohr distillation. 3.6 g (12 mmol=32%) of the title compound are obtained as a colorless oil.

¹ H-NMR (CDCl₃ ; δ (ppm)): 7.6 (m, 1H, aromatic); 7.35 (m, 2H, aromatic); 7.15 (m, 3H, aromatic); 6.85 (m, 2H, aromatic); 5.0 (dd, broad, 2H, O--CH₂); 3.8 (m, 1H, N--CH_(A)); 3.6 (s, 3H, O--CH₃); 3.5 (m, 1H, N--CH_(B)); 2.3 (s, 3H, CH₃); 1.15 (t, 3H, J=8 Hz, CH₃)

Example 2

Methyl N-[2-(2'-methylphenoxymethyl)-phenyl]-N-methyl-thiocarbamate (Table 7, No. 89)

a) 2-(2'-Methylphenoxymethyl)-nitrobenzene

75 g (0.347 mol) of 2-nitrobenzyl bromide, 37 g (0.342 mol) of o-cresol and 56 g (0.405 mol) of potassium carbonate in 500 ml of dimethylformamide are stirred for 5 hours at room temperature. The reaction mixture is then diluted with water and the aqueous phase is extracted three times with ether. The ether phase is dried and evaporated down. The crystalline residue is stirred with methanol and filtered off under suction. 73 g (0.300 mol=88%) of the title compound are obtained as a colorless solid. mp.=83° C.

¹ H-NMR (CDCl₃ ; δ (ppm)): 8.15 (d, 1H, J=8 Hz, aromatic); 7.95 (d, 1H, J=8 Hz, aromatic); 7.7 (t, 1H, J=8 Hz, aromatic); 7.45 (t, 1H, J=8 Hz, aromatic); 7.15 (m, 2H, aromatic); 6.9 (m, 2H, aromatic); 5.45 (s, 2H, O--CH₂); 2.35 (s, 3H, CH₃)

b) 2-(2'-Methylphenoxymethyl)-aniline

75 g (0.308 mol) of 2-(2'-methylphenoxymethyl)-nitrobenzene (Example 2a) and 10 g of 5% strength Pt/C (platinum adsorbed onto active carbon) in 50 ml of methanol are stirred vigorously for two hours under an H₂ atmosphere. Thereafter, a further 2 g of 5% strength Pt/C are added and stirring is continued overnight. The catalyst is then filtered off under suction and is replaced with 10 g of fresh catalyst. Stirring is continued overnight, the mixture is filtered under suction and the filtrate is evaporated down under reduced pressure. The residue is purified by column chromatography using hexane/ethyl acetate mixtures. 61 g (0.286 mol=93%) of the title compound are obtained as a colorless solid. mp.=56° C.

¹ H-NMR (CDCl₃ ; δ (ppm)): 7.2 (m, 4H, aromatic); 6.95 (d, 1H, J=8 Hz, aromatic); 6.9 (t, 1H, J=6 Hz, aromatic); 6.7 (m, 2H, aromatic); 5.0 (s, 2H, O--CH₂); 4.05 (s, broad, 2H, NH₂); 2.2 (s, 3H, CH₃)

c) Methyl N-[2-(2'-methylphenoxymethyl)-phenyl]-carbamate (Table 7, No. 3)

6 g (63 mmol) of methyl chloroformate are added dropwise to 10 g (47 mmol) of 2-(2'-methylphenoxymethyl)-aniline in 500 of methylene chloride at 20-30° C. Stirring is carried out for 3 hours at room temperature, a white solid being precipitated, and the reaction mixture is then stirred with 20 ml of 10% strength sodium hydroxide solution. The organic phase is filtered off under suction over silica gel, the filtrate is evaporated down and the remaining residue is stirred thoroughly with methanol and filtered under suction. 10.5 g (39 mmol=82%) of the title compound are obtained as a colorless solid. mp.=111° C.

¹ H-NMR (CDCl₃ ; δ (ppm)): 8.0 (d, broad, 1H, aromatic); 7.7 (s, broad, 1H, aromatic); 7.7 (s, broad, 1H, NH); 6.8-7.5 (m, 6H, aromatic); 5.0 (s, 2H, O--CH₂); 3.75 (s, 3H, O--CH₃); 2.25 (s, 3H, CH₃)

d) Methyl N-[2-(2'-methylphenoxymethyl)-phenyl]-N-methylthiocarbamate (Table 7, No. 89)

0.5 g (20.8 mmol) of sodium hydride is added a little at a time to 4.9 g (17.3 mmol) of methyl N-[2-(2'-methylphenoxymethyl)]-phenylcarbamate (Example 2c) in 80 ml of toluene. After the end of gas evolution, 2.4 g (19 mmol) of methyl methanethiosulfonate are added and stirring is carried out overnight at room temperature. Thereafter, the reaction mixture is extracted with water, dried over MgSO₄ and evaporated down under reduced pressure. The residue is purified by column chromatography with hexane/ethyl acetate mixtures over silica gel. 3 g (9.1 mmol=53%) of the title compound are obtained as a yellow oil.

¹ H-NMR (CDCl₃ ; δ (ppm)): 7.65 (d, broad, 1H, aromatic); 7.35 (m, 2H, aromatic); 7.15 (m, 3H, aromatic); 6.85 (m, 2H, aromatic); 5.0 (m, 2H, O--CH₂); 3.75 (s, 3H, O--CR₃); 2.55 (s, 3H, S--CH₃); 2.3 (s, 3H, CH₃)

Example 3

Methyl N-allyl-N-[2-(3"-bromophenylmethyliminoxymethyl)-phenyl]-carbamate (Table 7, No. 91)

a) o-Methoxymethylnitrobenzene

125 g of 30% strength sodium methylate solution (0.69 mol) in methanol are added dropwise to 130 g (0.6 mol) of o-nitrobenzyl bromide in 200 ml of methanol. During this procedure, the reaction mixture heats up to about 50° C. Stirring is continued for a further 3 hours, the reaction mixture being cooled to room temperature, after which ice water is added to the reaction vessel and the reaction mixture is neutralized by adding dilute hydrochloric acid. The aqueous phase is extracted with three times with ether, and the organic phase is dried over MgSO₄ and evaporated down. 101 g (0.6 mol, quantitative yield) of the title compound are obtained as a residue in the form of a brownish oil.

¹ H-NMR (CDCl₃ ; δ (ppm)): 8.1 (d, broad, 1H, aromatic); 7.8 (d, broad, 1H, aromatic); 7.65 (t, broad, 1H, aromatic); 7.45 (t, broad, 1H, aromatic); 4.85 (s, 2H, O--CH₂); 3.5 (s, 3H, OCH₃)

b) Methyl N-(2-methoxymethylphenyl)-carbamate

528 g of 21.8% strength Na₂ [Fe(CO)₄ ] solution (0.6 mol; 1 kg of the solution contains 633 g of water, 218 g of Na₂ [Fe(CO)₄ ], 108 g of Na₂ CO₃ and 41 g of NaOH) are added dropwise to 101 g (0.6 mol) of o-methoxymethylnitrobenzene (Example 3a) in 1 l of methanol at 20-30° C. Stirring is carried out for 1 hour at room temperature, after which the reaction mixture is diluted with ether. A brown oil separates out in the reaction vessel. The total reaction mixture is poured onto a silica gel column and is eluted with ether. Thereafter, the ether phase is evaporated, the residue is taken up in methylene chloride and the solution is dried over MgSO₄. It is filtered under suction over silica gel and the solvent is then evaporated off under reduced pressure. The residue is purified by column chromatography with hexane and methylene chloride. 83.8 g of o-methoxymethylaniline are obtained as a brown oil, which is directly reacted further.

The resulting crude product is dissolved in 700 ml of methylene chloride, 62.4 g (0.66 mol) of methyl chloroformate are added and 52.2 g (0.66 mol) of pyridine are then added dropwise. Stirring is carried out over-night at room temperature and the reaction mixture is then extracted with dilute hydrochloric acid and water. The organic phase is dried over MgSO₄ and evaporated down. The residue is purified by column chromatography with hexane/ethyl acetate mixtures. 89.4 g (0.41 mol=69%, based on 2-methoxymethylnitrobenzene) of the title compound are obtained as a yellow oil in a purity of about 90%.

¹ H-NMR (CDCl₃ ; δ (ppm)): 8.0 (m, 2H, 1×aromatic, NH); 7.35 (t, broad, 1H, aromatic); 7.15 (d, broad, 1H, aromatic); 7.0 (t, broad, 1H, aromatic); 4.5 (s, 2H, OCH₂); 3.8 (s, broad, 3H, OCH₃); 3.4 (s, broad, 3H, OCH₃)

c) Methyl N-(2-bromomethylphenyl)-carbamate

38.6 g (150 mmol) of boron tribromide are added dropwise to 10 g (51 mmol) of methyl N-(2-methoxymethylphenyl)-carbamate (Example 2b) in 100 ml of methylene chloride. Stirring is carried out for 2 hours, after which the vigorously stirred reaction mixture is added dropwise to a solution of 11.8 g (0.17 mol) of NaHCO₃ in water. The organic phase is separated off and the aqueous phase is extracted once with methylene chloride and once with ethyl acetate. The combined organic phases are dried over MgSO₄ and evaporated down. 9.5 g (39 mmol=76%) of the title compound are obtained as a colorless solid. mp.=132° C.

¹ H-NMR (CDCl₃ ; δ (ppm)): 7.85 (d, broad, 1H, aromatic); 7.3 (m, 2H, aromatic); 7.1 (t, broad, 1H, aromatic); 6.9 (s, broad, 1H, NH); 4.5 (s, 2H, CH₂ --Br); 3.8 (s, 3H, OCH₃)

d) Methyl N-[2-(3"-bromophenylmethyliminoxymethyl)-phenyl]-carbamate (Table 7, No. 88)

0.95 g (39 mmol) of sodium hydride is added a little at a time to 7 g (33 mmol) of m-bromoacetophenone oxime in 100 ml of dimethylformamide. When the evolution of gas has ended, 8 g (33 mmol) of methyl N-(2-bromo-methylphenyl)-carbamate (Example 3c), dissolved in 10 ml of dimethylformamide, are added dropwise. Stirring is carried out for 3 hours at room temperature, the reaction mixture is diluted with water and the aqueous phase is extracted three times with ether. The organic phase is washed three times with water, dried and evaporated down. The residue crystallizes and is stirred thoroughly with methanol. 5.1 g (13.5 mmol=41%) of the title compound are obtained as a colorless solid. mp.=124-125° C.

¹ H-NMR (CDCl₃ ; δ (ppm)): 8.6 (s, broad, 1H, NH); 7.8-8.1 (m, 2H, aromatic); 7-7.6 (m, 6H, aromatic); 5.2 (s, 2H, O--CH₂); 3.8 (s, 3H, O--CH₃); 2.2 (s, 3H, CH₃)

e) Methyl N-allyl-N-[2-(3"-bromophenylmethyliminoxy-methyl)-phenyl]-carbamate (Table 7, No. 91)

0.1 g (4.1 mmol) of sodium hydride is added a little at a time to 1.3 g (3.5 mmol) of methyl N-[2-(3"-bromophenylmethyliminoxymethyl)-phenyl]-carbamate (Example 3d) in 20 ml of dimethylformamide. After gas evolution has ended, 0.5 g (3.8 mmol) of allyl bromide are added and stirring is carried out overnight at room temperature. Thereafter, the reaction mixture is diluted with water and extracted three times with ether. The combined ether phases are washed three times with water, dried over MgSO₄ and evaporated down. 1.5 g (quantitative yield) of the title compound are obtained as a residue in the form of a yellow oil.

¹ H-NMR (CDCl₃ ; δ (ppm)): 7.8 (s, broad, 1H, aromatic); 7.1-7.6 (m, 7H, aromatic); 6.0 (m, 1H, C--CH═C); 5.1 (m, 4H, O--CH₂ and C═CH₂); 4.4 (m, 1H, N--CH_(A)); 4.0 (m, 1H, N--CH_(B)) 3.6-3.8 (2s, broad, O--CH₃); 2.2 (s, 3H, CH₃)

The compounds described in the Tables below can be prepared in a similar manner.

                  TABLE 1                                                          ______________________________________                                         1  STR23##                                                                       I: R.sup.1 = H II: R.sup.1 = CH.sub.3 III: R.sup.1 = Allyl IV: R.sup.1         = Propargyl V: R.sup.1 = S--CH.sub.3 VI: R.sup.1 = CH.sub.2 --CN VII:          R.sup.1 = CH.sub.2 --O--CH.sub.3 VIII: R.sup.1 = CO--CH.sub.3                   -  No.         X.sub.m                                                      ______________________________________                                         1         H                                                                      2 2-F                                                                          3 3-F                                                                          4 4-F                                                                          5 2,4-F.sub.2                                                                  6 2,4,6-F.sub.3                                                                7 2,3,4,5,6-F.sub.5                                                            8 2,3-F.sub.2                                                                  9 2-Cl                                                                         10 3-Cl                                                                        11 4-Cl                                                                        12 2,3-Cl.sub.2                                                                13 2,4-Cl.sub.2                                                                14 2,5-Cl.sub.2                                                                15 2,6-Cl.sub.2                                                                16 3,4-Cl.sub.2                                                                17 3,5-Cl.sub.2                                                                18 2,3,4-Cl.sub.3                                                              19 2,3,5-Cl.sub.3                                                              20 2,3,6-Cl.sub.3                                                              21 2,4,5-Cl.sub.3                                                              22 2,4,6-Cl.sub.3                                                              23 3,4,5-Cl.sub.3                                                              24 2,3,4,6-Cl.sub.4                                                            25 2,3,5,6-Cl.sub.4                                                            26 2,3,4,5,6-Cl.sub.5                                                          27 2-Br                                                                        28 3-Br                                                                        29 4-Br                                                                        30 2,4-Br.sub.2                                                                31 2,5-Br.sub.2                                                                32 2,6-Br.sub.2                                                                33 2,4,6-Br.sub.3                                                              34 2,3,4,5,6-Br.sub.5                                                          35 2-I                                                                         36 3-I                                                                         37 4-I                                                                         38 2,4-I.sub.2                                                                 39 2-Cl, 3-F                                                                   40 2-Cl, 4-F                                                                   41 2-Cl, 5-F                                                                   42 2-Cl, 6-F                                                                   43 2-Cl, 3-Br                                                                  44 2-Cl, 4-Br                                                                  45 2-Cl, 5-Br                                                                  46 2-Cl, 6-Br                                                                  47 2-Br, 3-Cl                                                                  48 2-Br, 4-Cl                                                                  49 2-Br, 5-Cl                                                                  50 2-Br, 3-F                                                                   51 2-Br, 4-F                                                                   52 2-Br, 5-F                                                                   53 2-Br, 6-F                                                                   54 2-F, 3-Cl                                                                   55 2-F, 4-Cl                                                                   56 2-F, 5-Cl                                                                   57 3-Cl, 4-F                                                                   58 3-Cl, 5-F                                                                   59 3-Cl, 4-Br                                                                  60 3-Cl, 5-Br                                                                  61 3-F, 4-Cl                                                                   62 3-F, 4-Br                                                                   63 3-Br, 4-Cl                                                                  64 3-Br, 4-F                                                                   65 2,6-Cl.sub.2, 4-Br                                                          66 2-CH.sub.3                                                                  67 3-CH.sub.3                                                                  68 4-CH.sub.3                                                                  69 2,3-(CH.sub.3).sub.2                                                        70 2,4-(CH.sub.3).sub.2                                                        71 2,5-(CH.sub.3).sub.2                                                        72 2,6-(CH.sub.3).sub.2                                                        73 3,4-(CH.sub.3).sub.2                                                        74 3,5-(CH.sub.3).sub.2                                                        75 2,3,5-(CH.sub.3).sub.3                                                      76 2,3,4-(CH.sub.3).sub.3                                                      77 2,3,6-(CH.sub.3).sub.3                                                      78 2,4,5-(CH.sub.3).sub.3                                                      79 2,4,6-(CH.sub.3).sub.3                                                      80 3,4,5-(CH.sub.3).sub.3                                                      81 2,3,4,6-(CH.sub.3).sub.4                                                    82 2,3,5,6-(CH.sub.3).sub.4                                                    83 2,3,4,5,6-(CH.sub.3).sub.5                                                  84 2-C.sub.2 H.sub.5                                                           85 3-C.sub.2 H.sub.5                                                           86 4-C.sub.2 H.sub.5                                                           87 2,4-(C.sub.2 H.sub.5).sub.2                                                 88 2,6-(C.sub.2 H.sub.5).sub.2                                                 89 3,5-(C.sub.2 H.sub.5).sub.2                                                 90 2,4,6-(C.sub.2 H.sub.5).sub.3                                               91 2-n-C.sub.3 H.sub.7                                                         92 3-n-C.sub.3 H.sub.7                                                         93 4-n-C.sub.3 H.sub.7                                                         94 2-i-C.sub.3 H.sub.7                                                         95 3-i-C.sub.3 H.sub.7                                                         96 4-i-C.sub.3 H.sub.7                                                         97 2,4-(i-C.sub.3 H.sub.7).sub.2                                               98 2,6-(i-C.sub.3 H.sub.7).sub.2                                               99 3,5-(i-C.sub.3 H.sub.7).sub.2                                               100 2,4,6-(i-C.sub.3 H.sub.7)3                                                 101 2-s-C.sub.4 H.sub.9                                                        102 3-s-C.sub.4 H.sub.9                                                        103 4-s-C.sub.4 H.sub.9                                                        104 2-t-C.sub.4 H.sub.9                                                        105 3-t-C.sub.4 H.sub.9                                                        106 4-t-C.sub.4 H.sub.9                                                        107 2,3-(t-C.sub.4 H.sub.9).sub.2                                              108 2,4-(t-C.sub.4 H.sub.9).sub.2                                              109 2,5-(t-C.sub.4 H.sub.9).sub.2                                              110 2,6-(t-C.sub.4 H.sub.9).sub.2                                              111 3,4-(t-C.sub.4 H.sub.9).sub.2                                              112 2,4,6-(t-C.sub.4 H.sub.9)3                                                 113 4-n-C.sub.9 H.sub.19                                                       114 4-n-C.sub.12 H.sub.25                                                      115 4-n-C.sub.15 H.sub.31                                                      116 4-(1,1,3,3-Tetramethylbutyl)                                               117 4-(2,4,4-Trimethylpropyl)                                                  118 2-t-C.sub.4 H.sub.9, 4-CH.sub.3                                            119 2-t-C.sub.4 H.sub.9, 5-CH.sub.3                                            120 2,6-(t-C.sub.4 H.sub.9).sub.2, 4-CH.sub.3                                  121 2-CH.sub.3, 4-t-C.sub.4 H.sub.9                                            122 2-CH.sub.3, 6-t-C.sub.4 H.sub.9                                            123 2-CH.sub.3, 4-i-C.sub.3 H.sub.7                                            124 2-CH.sub.3, 5-i-C.sub.3 H.sub.7                                            125 3-CH.sub.3, 4-i-C.sub.3 H.sub.7                                            126 2-i-C.sub.3 H.sub.7, 5-CH.sub.3                                            127 2,4-(t-C.sub.4 H.sub.9).sub.2, 6-i-C.sub.3 H.sub.7                         128 2-Allyl                                                                    129 3-Allyl                                                                    130 4-Allyl                                                                    131 2-Allyl, 6-CH.sub.3                                                        132 2-cyclo-C.sub.6 H.sub.11                                                   133 3-cyclo-C.sub.6 H.sub.11                                                   134 4-cyclo-C.sub.6 H.sub.11                                                   135 2,4-(cyclo-C.sub.6 H.sub.11).sub.2, 6-CH.sub.3                             136 2-CH.sub.3, 4-cyclo-C.sub.6 H.sub.11                                       137 2-CH.sub.2 --C.sub.6 H.sub.5                                               138 3-CH.sub.2 --C.sub.6 H.sub.5                                               139 4-CH.sub.2 --C.sub.6 H.sub.5                                               140 2-CH.sub.2 --C.sub.6 H.sub.5, 4-CH.sub.3                                   141 2-CH.sub.3, 4-CH.sub.2 --C.sub.6 H.sub.5                                   142 2-C.sub.6 H.sub.5                                                          143 3-C.sub.6 H.sub.5                                                          144 4-C.sub.6 H.sub.5                                                          145 4-(2-i-C.sub.3 H.sub.7 --C.sub.6 H.sub.4)                                  146 4-C.sub.6 H.sub.5, 2,6-(CH.sub.3).sub.2                                    147 2-Cl, 4-C.sub.6 H.sub.5                                                    148 2-Br, 4-C.sub.6 H.sub.5                                                    149 2-C.sub.6 H.sub.5, 4-Cl                                                    150 2-C.sub.6 H.sub.5, 4-Br                                                    151 2-CH.sub.2 C.sub.6 H.sub.5, 4-Cl                                           152 2-CH.sub.2 C.sub.6 H.sub.5, 4-Br                                           153 2-Cl, 4-CH.sub.2 C.sub.6 H.sub.5                                           154 2-Br, 4-CH.sub.2 C.sub.6 H.sub.5                                           155 2-cyclo-C.sub.6 H.sub.11, 4-Cl                                             156 2-cyclo-C.sub.6 H.sub.11, 4-Br                                             157 2-Cl, 4-cyclo-C.sub.6 H.sub.11                                             158 2-Br, 4-cyclo-C.sub.6 H.sub.11                                             159 2-OCH.sub.3                                                                160 3-OCH.sub.3                                                                161 4-OCH.sub.3                                                                162 2-OC.sub.2 H.sub.5                                                         163 3-O--C.sub.2 H.sub.5                                                       164 4-O--C.sub.2 H.sub.5                                                       165 2-O-n-C.sub.3 H.sub.7                                                      166 3-O-n-C.sub.3 H.sub.7                                                      167 4-O-n-C.sub.3 H.sub.7                                                      168 2-O-i-C.sub.3 H.sub.7                                                      169 3-O-i-C.sub.3 H.sub.7                                                      170 4-O-i-C.sub.3 H.sub.7                                                      171 2-O-n-C.sub.6 H.sub.13                                                     172 3-O-n-C.sub.6 H.sub.13                                                     173 4-O-n-C.sub.6 H.sub.13                                                     174 2-O-n-C.sub.8 H.sub.17                                                     175 3-O-n-C.sub.8 H.sub.17                                                     176 4-O-n-C.sub.8 H.sub.17                                                     177 2-O--CH.sub.2 C.sub.6 H.sub.5                                              178 3-O--CH.sub.2 C.sub.6 H.sub.5                                              179 4-O--CH.sub.2 C.sub.6 H.sub.5                                              180 2-O--(CH.sub.2).sub.3 C.sub.6 H.sub.5                                      181 3-O--(CH.sub.2).sub.3 C.sub.6 H.sub.5                                      182 4-O--(CH.sub.2).sub.3 C.sub.6 H.sub.5                                      183 2,4-(OCH.sub.3).sub.2                                                      184 2-CF.sub.3                                                                 185 3-CF.sub.3                                                                 186 4-CF.sub.3                                                                 187 2-OCF.sub.3                                                                188 3-OCF.sub.3                                                                189 4-OCF.sub.3                                                                190 3-OCH.sub.2 CHF.sub.2                                                      191 2-NO.sub.2                                                                 192 3-NO.sub.2                                                                 193 4-NO.sub.2                                                                 194 2-CN                                                                       195 3-CN                                                                       196 4-CN                                                                       197 2-CH.sub.3, 3-Cl                                                           198 2-CH.sub.3, 4-Cl                                                           199 2-CH.sub.3, 5-Cl                                                           200 2-CH.sub.3, 6-Cl                                                           201 2-CH.sub.3, 3-F                                                            202 2-CH.sub.3, 4-F                                                            203 2-CH.sub.3, 5-F                                                            204 2-CH.sub.3, 6-F                                                            205 2-CH.sub.3, 3-Br                                                           206 2-CH.sub.3, 4-Br                                                           207 2-CH.sub.3, 5-Br                                                           208 2-CH.sub.3, 6-Br                                                           209 2-Cl, 3-CH.sub.3                                                           210 2-Cl, 4-CH.sub.3                                                           211 2-Cl, 5-CH.sub.3                                                           212 2-F, 3-CH.sub.3                                                            213 2-F, 4-CH.sub.3                                                            214 2-F, 5-CH.sub.3                                                            215 2-Br, 3-CH.sub.3                                                           216 2-Br, 4-CH.sub.3                                                           217 2-Br, 5-CH.sub.3                                                           218 3-CH.sub.3, 4-Cl                                                           219 3-CH.sub.3, 5-Cl                                                           220 3-CH.sub.3, 4-F                                                            221 3-CH.sub.3, 5-F                                                            222 3-CH.sub.3, 4-Br                                                           223 3-CH.sub.3, 5-Br                                                           224 3-F, 4-CH.sub.3                                                            225 3-Cl, 4-CH.sub.3                                                           226 3-Br, 4-CH.sub.3                                                           227 2-Cl, 4,5-(CH.sub.3).sub.2                                                 228 2-Br, 4,5-(CH.sub.3).sub.2                                                 229 2-Cl, 3,5-(CH.sub.3).sub.2                                                 230 2-Br, 3,5-(CH.sub.3).sub.2                                                 231 2,6-Cl.sub.2, 4-CH.sub.3                                                   232 2,6-F.sub.2, 4-CH.sub.3                                                    233 2,6-Br.sub.2, 4-CH.sub.3                                                   234 2,4-Br.sub.2, 6-CH.sub.3                                                   235 2,4-F.sub.2, 6-CH.sub.3                                                    236 2,4-Br.sub.2, 6-CH.sub.3                                                   237 2,6-(CH.sub.3).sub.2, 4-F                                                  238 2,6-(CH.sub.3).sub.2, 4-Cl                                                 239 2,6-(CH.sub.3).sub.2, 4-Br                                                 240 3,5-(CH.sub.3).sub.2, 4-F                                                  241 3,5-(CH.sub.3).sub.2, 4-Cl                                                 242 3,5-(CH.sub.3).sub.2, 4-Br                                                 243 2,3,6-(CH.sub.3).sub.3, 4-F                                                244 2,3,6-(CH.sub.3).sub.3, 4-Cl                                               245 2,3,6-(CH.sub.3).sub.3, 4-Br                                               246 2,4-(CH.sub.3).sub.2, 6-F                                                  247 2,4-(CH.sub.3).sub.2, 6-Cl                                                 248 2,4-(CH.sub.3).sub.2, 6-Br                                                 249 2-i-C.sub.3 H.sub.7, 4-Cl, 5-CH.sub.3                                      250 2-Cl, 4-NO.sub.2                                                           251 2-NO.sub.2, 4-Cl                                                           252 2-OCH.sub.3, 5-NO.sub.2                                                    253 2,4-Cl.sub.2, 5-NO.sub.2                                                   254 2,4-Cl.sub.2, 6-NO.sub.2                                                   255 2,6-Cl.sub.2, 4-NO.sub.2                                                   256 2,6-Br.sub.2, 4-NO.sub.2                                                   257 2,6-I.sub.2, 4-NO.sub.2                                                    258 2-CH.sub.3, 5-i-C.sub.3 H.sub.7, 4-Cl                                      259 2-CO.sub.2 CH.sub.3                                                        260 3-CO.sub.2 CH.sub.3                                                        261 4-CO.sub.2 CH.sub.3                                                        262 2-CO.sub.2 (C.sub.2 H.sub.5)                                               263 3-CO.sub.2 (C.sub.2 H.sub.5)                                               264 4-CO.sub.2 (C.sub.2 H.sub.5)                                               265 2-CO.sub.2 (n-C.sub.3 H.sub.7)                                             266 3-CO.sub.2 (n-C.sub.3 H.sub.7)                                             267 4-CO.sub.2 (n-C.sub.3 H.sub.7)                                             268 2-CO.sub.2 (i-C.sub.3 H.sub.7)                                             269 3-CO.sub.2 (i-C.sub.3 H.sub.7)                                             270 4-CO2(i-C.sub.3 H.sub.7)                                                   271 2-CO.sub.2 (n-C.sub.6 H.sub.13)                                            272 3-CO.sub.2 (n-C.sub.6 H.sub.13)                                            273 4-CO.sub.2 (n-C.sub.6 H.sub.13)                                            274 2-CH.sub.2 --OCH.sub.3                                                     275 3-CH.sub.2 --OCH.sub.3                                                     276 4-CH.sub.2 --OCH.sub.3                                                     277 2-CH.sub.2 O(C.sub.2 H.sub.5)                                              278 3-CH.sub.2 O(C.sub.2 H.sub.5)                                              279 4-CH.sub.2 O(C.sub.2 H.sub.5)                                              280 2-CH.sub.2 O(n-C.sub.2 H.sub.7)                                            281 3-CH.sub.2 O(n-C.sub.3 H.sub.7)                                            282 4-CH.sub.2 O(n-C.sub.3 H.sub.7)                                            283 2-CH.sub.2 O(i-C.sub.3 H.sub.7)                                            284 3-CH.sub.2 O(i-C.sub.3 H.sub.7)                                            285 4-CH.sub.2 O(i-C.sub.3 H.sub.7)                                            286 2-CHO                                                                      287 3-CHO                                                                      288 4-CHO                                                                      289 2-CO--CH.sub.3                                                             290 3-CO--CH.sub.3                                                             291 4-CO--CH.sub.3                                                             292 2-CO--CH.sub.2 --CH.sub.3                                                  293 3-CO--CH.sub.2 --CH.sub.3                                                  294 4-CO--CH.sub.2 --CH.sub.3                                                  295 2-CO--CH.sub.2 --CH.sub.2 --CH.sub.3                                       296 3-CO--CH.sub.2 --CH.sub.2 --CH.sub.3                                       297 4-CO--CH.sub.2 --CH.sub.2 --CH.sub.3                                       298 2-CO--CH(CH.sub.3)--CH.sub.3                                               299 3-CO--CH(CH.sub.3)--CH.sub.3                                               300 4-CO--CH(CH.sub.3)--CH.sub.3                                               301 2-Me-4-CHO                                                                 302 2-Me-4-CH.sub.3 --CO                                                       303 2-Me-4-CH.sub.3 --CH.sub.2 --CO                                            304 2-Me-4-CH.sub.3 --CH.sub.2 --CH.sub.2 --CO                                 305 2-Me-4-CH.sub.3 --CH(CH.sub.3)--CO                                         306 2,5-Me.sub.2 -4-CHO                                                        307 2,5-Me.sub.2 -4-CH.sub.3 --CO                                              308 2,5-Me.sub.2 -4-CH.sub.3 --CH.sub.2 --CO                                   309 2,5-Me.sub.2 -4-CH.sub.3 --CH.sub.2 --CH.sub.2 --CO                        310 2,5-Me.sub.2 -4-CH.sub.3 --CH (CH.sub.3)--CO                               311 2-Cl-4-CHO                                                                 312 2-Cl-4-CH.sub.3 --CO                                                       313 2-Cl-4-CH.sub.3 --CH.sub.2 --CO                                            314 2-Cl-4-CH.sub.3 --CH(CH.sub.3)--CO                                         315 2,5-Cl.sub.2 -4-CHO                                                        316 2,5-Cl.sub.2 -4-CH.sub.3 --CO                                              317 2,5-Cl.sub.2 -4-CH.sub.3 --CH.sub.2 --CO                                   318 2,5-Cl.sub.2 -4-CH.sub.3 --CH.sub.2 --CH.sub.2 --CO                        319 2,5-Cl.sub.2 -4-CH.sub.3 --CH(CH.sub.3)--CO                                320 2-C(═NOCH.sub.3)--CH.sub.3                                             321 3-C(═NOCH.sub.3)--CH.sub.3                                             322 4-C(═NOCH.sub.3)--CH.sub.3                                             323 2-C(═NOC.sub.2 H.sub.5)--CH.sub.3                                      324 3-C(═NOC.sub.2 H.sub.5)--CH.sub.3                                      325 4-C(═NOC.sub.2 H.sub.5)--CH.sub.3                                      326 2-C(═NO-n-C.sub.3 H.sub.7)--CH.sub.3                                   327 3-C(═NO-n-C.sub.3 H.sub.7)--CH.sub.3                                   328 4-C(═NO-n-C.sub.3 H.sub.7)--CH.sub.3                                   329 2-C(═NO-i-C.sub.3 H.sub.7)--CH.sub.3                                   330 3-C(═NO-i-C.sub.3 H.sub.7)--CH.sub.3                                   331 4-C(═NO-i-C.sub.3 H.sub.7)--CH.sub.3                                   332 2-C(═NO-Allyl)-CH.sub.3                                                333 3-C(═NO-Allyl)-CH.sub.3                                                334 4-C(═NO-Allyl)-CH.sub.3                                                335 2-C(═NO-trans-Chloroallyl)-CH.sub.3                                    336 3-C(═NO-trans-Chloroallyl)-CH.sub.3                                    337 4-C(═NO-trans-Chloroallyl)--CH.sub.3                                   338 2-C(═NO-Propargyl)--CH.sub.3                                           339 3-C(═NO-Propargyl)--CH.sub.3                                           340 4-C(═NO-Propargyl)--CH.sub.3                                           341 2-C(═NO-n-C.sub.4 H.sub.9)--CH.sub.3                                   342 3-C(═NO-n-C.sub.4 H.sub.9)--CH.sub.3                                   343 4-C(═NO-n-C.sub.4 H.sub.9)--CH.sub.3                                   344 2-C(═NO--CH.sub.2 --C.sub.6 H.sub.5)--CH.sub.3                         345 3-C(═NO--CH.sub.2 --C.sub.6 H.sub.5)--CH.sub.3                         346 4-C(═NO--CH.sub.2 --C.sub.6 H.sub.5)--CH.sub.3                         347 2-CH.sub.3 -4-CH═NOCH.sub.3                                            348 2-CH.sub.3 -4-CH═NOC.sub.2 H.sub.5                                     349 2-CH.sub.3 -4-CH═NO-n-C.sub.3 H.sub.7                                  350 2-CH.sub.3 -4-CH═NO-i-C.sub.3 H.sub.7                                  351 2-CH.sub.3 -4-CH═NO-Allyl                                              352 2-CH.sub.3 -4-CH═NO-(trans-Chloroallyl)                                353 2-CH.sub.3 -4-CH═NO-Propargyl                                          354 2-CH.sub.3 -4-CH═NO-n-C.sub.4 H.sub.9                                  355 2-CH.sub.3 -4-CH═NO--CH.sub.2 --C.sub.6 H.sub.5                        356 2-CH.sub.3 -4-(CH.sub.3 --C═NOCH.sub.3)                                357 2-CH.sub.3 -4-(CH.sub.3 --C═NOC.sub.2 H.sub.5)                         358 2-CH.sub.3 -4-(CH.sub.3 --C═NO-n-C.sub.3 H.sub.7)                      359 2-CH.sub.3 -4-(CH.sub.3 --C═NO-i-C.sub.3 H.sub.7)                      360 2-CH.sub.3 -4-(CH.sub.3 --C═NO-Allyl)                                  361 2-CH.sub.3 -4-(CH.sub.3 --C═NO-trans-Chloroallyl)                      362 2-CH.sub.3 -4-(CH.sub.3 --C═NO-Propargyl)                              363 2-CH.sub.3 -4-(CH.sub.3 --C═NO-n-C.sub.4 H.sub.9)                      364 2-CH.sub.3 -4-(CH.sub.3 --C═NO-CH.sub.2 --C.sub.6 H.sub.5)                      365 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C═NO--CH.sub.3)                       366 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C═NO--C.sub.2                        H.sub.5)                                                               367 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C═NO-n-C.sub.3 H.sub.7                         368 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C═NO-i-C.sub.3                       H.sub.7                                                                369 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C═NO-Allyl)                           370 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C═NO-trans-Chloroallyl)                        371 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C═NO-Propargyl)                       372 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C═NO-n-C.sub.4                       H.sub.9)                                                               373 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C═NO--CH.sub.2 --C.sub.6                      H.sub.5)                                                               374 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C═NOCH.sub.3)                      375 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C═NOC.sub.2 H.sub.5)                        376 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C═NO-n-C.sub.3                    H.sub.7)                                                               377 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C═NO-i-C.sub.3 H.sub.7)                     378 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C═NO-Allyl)                        379 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C═NO-trans-Chloroal               lyl)                                                                   380 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C═NO-Proparyl)                     381 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C═NO-n-C.sub.4 H.sub.9)                     382 2,5-(CH.sub.3)-2-4-(CH.sub.3 --C═NO--CH.sub.2 --C.sub.6                H.sub.5)                                                              383 2-C.sub.6 H.sub.5                                                          384 3-C.sub.6 H.sub.5                                                          385 4-C.sub.6 H.sub.5                                                          386 2-(2'-F--C.sub.6 H.sub.4)                                                  387 2-(3'-F--C.sub.6 H.sub.4)                                                  388 2-(4'-F--C.sub.6 H.sub.4)                                                  389 3-(2'-F--C.sub.6 H.sub.4)                                                  390 3-(3'-F--C.sub.6 H.sub.4)                                                  391 3-(4'-F--C.sub.6 H.sub.4)                                                  392 4-(2'-F--C.sub.6 H.sub.4)                                                  393 4-(3'-F--C.sub.6 H.sub.4)                                                  394 4-(4'-F--C.sub.6 H.sub.4)                                                  395 2-(2'-Cl-C.sub.6 H.sub.4)                                                  396 2-(3'-Cl-C.sub.6 H.sub.4)                                                  397 2-(4'-Cl-C.sub.6 H.sub.4)                                                  398 3-(2'-Cl-C.sub.6 H.sub.4)                                                  399 3-(3'-Cl-C.sub.6 H.sub.4)                                                  400 3-(4'-Cl-C.sub.6 H.sub.4)                                                  401 4-(2'-Cl-C.sub.6 H.sub.4)                                                  402 4-(3'-Cl-C.sub.6 H.sub.4)                                                  403 4-(4'-Cl-C.sub.6 H.sub.4)                                                  405 2-(2'-CH.sub.3 --C.sub.6 H.sub.4)                                          406 2-(3'-CH.sub.3 --C.sub.6 H.sub.4)                                          407 2-(4'-CH.sub.3 --C.sub.6 H.sub.4)                                          408 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)                                          409 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)                                          410 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)                                          411 4-(2'-CH.sub.3 --C.sub.6 H.sub.4)                                          412 4-(3'-CH.sub.3 --C.sub.6 H.sub.4)                                          413 4-(4'-CH.sub.3 --C.sub.6 H.sub.4)                                          414 2-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                      415 2-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                      416 2-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                      417 3-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                      418 3-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                      419 3-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                      420 4-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                      421 4-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                      422 4-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                      423 2-(2'-(CH.sub.3 --C(═NOAllyl))-C.sub.6 H.sub.4)                        424 2-(3'-(CH.sub.3 --C(═NOAllyl))-C.sub.6 H.sub.4)                        425 2-(4'-(CH.sub.3 --C(═NOAllyl))-C.sub.6 H.sub.4)                        426 3-(2'-(CH.sub.3 --C(═NOAllyl))-C.sub.6 H.sub.4)                        427 3-(3'-(CH.sub.3 --C(═NOAllyl))-C.sub.6 H.sub.4)                        428 3-(4'-(CH.sub.3 --C(═NOAllyl))-C.sub.6 H.sub.4)                        429 4-(2'-(CH.sub.3 --C(═NOAllyl))-C.sub.6 H.sub.4)                        430 4-(3'-(CH.sub.3 --C(═NOAllyl))-C.sub.6 H.sub.4)                        431 4-(4'-(CH.sub.3 --C(═NOAllyl))-C.sub.6 H.sub.4)                        432 2-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                                 433 2-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                                 434 2-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                                 435 3-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                                 436 3-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                                 437 3-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                                 438 4-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                                 439 4-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                                 440 4-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                                 441 2-(2'-CH.sub.3 O--C.sub.6 H.sub.4)                                         442 2-(3'-CH.sub.3 O--C.sub.6 H.sub.4)                                         443 2-(4'-CH.sub.3 O--C.sub.6 H.sub.4)                                         444 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)                                         445 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)                                         446 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)                                         447 4-(2'-CH.sub.3 O--C.sub.6 H.sub.4)                                         448 4-(3'-CH.sub.3 O--C.sub.6 H.sub.4)                                         449 4-(4'-CH.sub.3 O--C.sub.6 H.sub.4)                                         450 2-(2'-O.sub.2 N-C.sub.6 H.sub.4)                                           451 2-(3'-O.sub.2 N-C.sub.6 H.sub.4)                                           452 2-(4'-O.sub.2 N-C.sub.6 H.sub.4)                                           453 3-(2'-O.sub.2 N-C.sub.6 H.sub.4)                                           454 3-(3'-O.sub.2 N-C.sub.6 H.sub.4)                                           455 3-(4'-O.sub.2 N-C.sub.6 H.sub.4)                                           456 4-(2'-O.sub.2 N-C.sub.6 H.sub.4)                                           457 4-(3'-O.sub.2 N-C.sub.6 H.sub.4)                                           458 4-(4'-O.sub.2 N-C.sub.6 H.sub.4)                                           459 2-(2'-NC--C.sub.6 H.sub.4)                                                 460 2-(3'-NC--C.sub.6 H.sub.4)                                                 461 2-(4'-NC--C.sub.6 H.sub.4)                                                 462 3-(2'-NC--C.sub.6 H.sub.4)                                                 463 3-(3'-NC--C.sub.6 H.sub.4)                                                 464 3-(4'-NC--C.sub.6 H.sub.4)                                                 465 4-(2'-NC--C.sub.6 H.sub.4)                                                 466 4-(3'-NC--C.sub.6 H.sub.4)                                                 467 4-(4'-NC--C.sub.6 H.sub.4)                                                 468 2-(2'-CF.sub.3 --C.sub.6 H.sub.4)                                          469 2-(3'-CF.sub.3 --C.sub.6 H.sub.4)                                          470 2-(4'-CF.sub.3 --C.sub.6 H.sub.4)                                          471 3-(2'-CF.sub.3 --C.sub.6 H.sub.4)                                          472 3-(3'-CF.sub.3 --C.sub.6 H.sub.4)                                          473 3-(4'-CF.sub.3 --C.sub.6 H.sub.4)                                          474 4-(2'-CF.sub.3 --C.sub.6 H.sub.4)                                          475 4-(3'-CF.sub.3 --C.sub.6 H.sub.4)                                          476 4-(4'-CF.sub.3 --C.sub.6 H.sub.4)                                          477 2-O--C.sub.6 H.sub.5                                                       475 3-O--C.sub.6 H.sub.5                                                       476 4-O--C.sub.6 H.sub.5                                                       478 2-O-(2'-F--C.sub.6 H.sub.4)                                                479 2-O-(3'-F--C.sub.6 H.sub.4)                                                480 2-O-(4'-F--C.sub.6 H.sub.4)                                                481 3-O-(2'-F--C.sub.6 H.sub.4)                                                482 3-O-(3'-F--C.sub.6 H.sub.4)                                                483 3-O-(4'-F--C.sub.6 H.sub.4)                                                484 4-O-(2'-F--C.sub.6 H.sub.4)                                                485 4-O-(3'-F--C.sub.6 H.sub.4)                                                486 4-O-(4'-F--C.sub.6 H.sub.4)                                                487 2-O-(2'-Cl--C.sub.6 H.sub.4)                                               488 2-O-(3'-Cl--C.sub.6 H.sub.4)                                               489 2-O-(4'-Cl--C.sub.6 H.sub.4)                                               490 3-O-(2'-Cl--C.sub.6 H.sub.4)                                               491 3-O-(3'-Cl--C.sub.6 H.sub.4)                                               492 3-O-(4'-Cl--C.sub.6 H.sub.4)                                               493 3-O-(4'-Cl--C.sub.6 H.sub.4)                                               494 4-O-(2'-Cl--C.sub.6 H.sub.4)                                               495 4-O-(3'-Cl--C.sub.6 H.sub.4)                                               496 4-O-(4'-Cl--C.sub.6 H.sub.4)                                               497 2-O-(2'-CH.sub.3 --C.sub.6 H.sub.4)                                        498 2-O-(3'-CH.sub.3 --C.sub.6 H.sub.4)                                        499 2-O-(4'-CH.sub.3 --C.sub.6 H.sub.4)                                        500 3-O-(2'-CH.sub.3 --C.sub.6 H.sub.4)                                        501 3-O-(3'-CH.sub.3 --C.sub.6 H.sub.4)                                        502 3-o-(4'-CH.sub.3 --C.sub.6 H.sub.4)                                        503 4-O-(2'-CH.sub.3 --C.sub.6 H.sub.4)                                        504 4-O-(3'-CH.sub.3 --C.sub.6 H.sub.4)                                        505 4-O-(4'-CH.sub.3 --C.sub.6 H.sub.4)                                        506 2-O-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                    507 2-O-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                    508 2-O-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                    509 3-O-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                    510 3-O-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                    511 3-O-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                    512 4-O-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                    513 4-O-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                    514 4-O-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                    515 2-O-(2'-(CH.sub.3 --C(═NOAllyl))-C.sub.6 H.sub.4)                      516 2-O-(3'-(CH.sub.3 --C(═NOAllyl))-C.sub.6 H.sub.4)                      517 2-O-(4'-(CH.sub.3 --C(═NOAllyl))-C.sub.6 H.sub.4)                      518 3-O-(2'-(CH.sub.3 --C(═NOAllyl))-C.sub.6 H.sub.4)                      519 3-O-(3'-(CH.sub.3 --C(═NOAllyl))-C.sub.6 H.sub.4)                      520 3-O-(4'-(CH.sub.3 --C(═NOAllyl))-C.sub.6 H.sub.4)                      521 4-O-(2'-(CH.sub.3 --C(═NOAllyl))-C.sub.6 H.sub.4)                      522 4-O-(3'-(CH.sub.3 --C(═NOAllyl))-C.sub.6 H.sub.4)                      523 4-O-(4'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                     524 2-O-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                               525 2-O-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                               526 2-O-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                               527 3-O-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                               528 3-O-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                               529 3-O-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                               530 4-O-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                               531 4-O-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                               532 4-O-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                               533 2-O-(2'-CH.sub.3 O--C.sub.6 H.sub.4)                                       534 2-O-(3'-CH.sub.3 O--C.sub.6 H.sub.4)                                       535 2-O-(4'-CH.sub.3 O--C.sub.6 H.sub.4)                                       536 3-O-(2'-CH.sub.3 O--C.sub.6 H.sub.4)                                       537 3-O-(3'-CH.sub.3 O--C.sub.6 H.sub.4)                                       538 3-O-(4'-CH.sub.3 O--C.sub.6 H.sub.4)                                       539 4-O-(2'-CH.sub.3 O--C.sub.6 H.sub.4)                                       540 4-O-(3'-CH.sub.3 O--C.sub.6 H.sub.4)                                       541 4-O-(4'-CH.sub.3 O--C.sub.6 H.sub.4)                                       542 2-O-(2'-O.sub.2 N-C.sub.6 H.sub.4)                                         543 2-O-(3'-O.sub.2 N-C.sub.6 H.sub.4)                                         544 2-O-(4'-O.sub.2 N-C.sub.6 H.sub.4)                                         545 3-O-(2'-O.sub.2 N-C.sub.6 H.sub.4)                                         546 3-O-(3'-O.sub.2 N-C.sub.6 H.sub.4)                                         547 3-O-(4'-O.sub.2 N-C.sub.6 H.sub.4)                                         548 4-O-(2'-O.sub.2 N-C.sub.6 H.sub.4)                                         549 4-O-(3'-O.sub.2 N-C.sub.6 H.sub.4)                                         550 4-O-(4'-O.sub.2 N-C.sub.6 H.sub.4)                                         551 2-O-(2'-NC--C.sub.6 H.sub.4)                                               552 2-O-(3'-NC--C.sub.6 H.sub.4)                                               553 2-O-(4'-NC--C.sub.6 H.sub.4)                                               554 3-O-(2'-NC--C.sub.6 H.sub.4)                                               555 3-O-(3'-NC--C.sub.6 H.sub.4)                                               556 3-O-(4'-NC--C.sub.6 H.sub.4)                                               557 4-O-(2'-NC--C.sub.6 H.sub.4)                                               558 4-O-(3'-NC--C.sub.6 H.sub.4)                                               559 4-O-(4'-NC--C.sub.6 H.sub.4)                                               560 2-O-(2'-CF.sub.3 --C.sub.6 H.sub.4)                                        561 2-O-(3'-CF.sub.3 --C.sub.6 H.sub.4)                                        562 2-O-(4'-CF.sub.3 --C.sub.6 H.sub.4)                                        563 3-O-(2'-CF.sub.3 --C.sub.6 H.sub.4)                                        564 3-O-(3'-CF.sub.3 --C.sub.6 H.sub.4)                                        565 3-O-(4'-CF.sub.3 --C.sub.6 H.sub.4)                                        566 4-O-(2'-CF.sub.3 --C.sub.6 H.sub.4)                                        567 4-O-(3'-CF.sub.3 --C.sub.6 H.sub.4)                                        568 4-O-(4'-CF.sub.3 --C.sub.6 H.sub.4)                                        569 2-Pyridinyl-2'                                                             570 2-Pyridinyl-3'                                                             571 2-Pyridinyl-4'                                                             572 3-Pyridinyl-2'                                                             573 3-Pyridinyl-3'                                                             574 3-Pyridinyl-4'                                                             575 4-Pyridinyl-2'                                                             576 4-Pyridinyl-3'                                                             577 4-Pyridinyl-4'                                                             578 2-Pyrimidinyl-2'                                                           579 2-Pyrimidinyl-3'                                                           580 2-Pyrimidinyl-4'                                                           581 3-Pyrimidinyl-2'                                                           582 3-Pyrimidinyl-3'                                                           583 3-Pyrimidinyl-4'                                                           584 4-Pyrimidinyl-2'                                                           585 4-Pyrimidinyl-3'                                                           586 4-Pyrimidinyl-4'                                                           587 2-Pyrazolyl-1'                                                             588 2-Pyrazolyl-3'                                                             589 2-Pyrazolyl-4'                                                             590 3-Pyrazolyl-1'                                                             591 3-Pyrazolyl-3'                                                             592 3-Pyrazolyl-4'                                                             593 4-Pyrazolyl-1'                                                             594 4-Pyrazolyl-3'                                                             595 4-Pyrazolyl-4'                                                             596 2-Isoxazolyl-3'                                                            597 2-Isoxazolyl-4'                                                            598 2-Isoxazolyl-5'                                                            599 3-Isoxazolyl-3'                                                            600 3-Isoxazolyl-4'                                                            601 3-Isoxazolyl-5'                                                            602 4-Isoxazolyl-3'                                                            603 4-Isoxazolyl-4'                                                            604 4-Isoxazolyl-5'                                                            605 2-Isothiazolyl-3'                                                          606 2-Isothiazolyl-4'                                                          607 2-Isothiazolyl-5'                                                          608 3-Isothiazolyl-3'                                                          609 3-Isothiazolyl-4'                                                          610 3-Isothiazolyl-5'                                                          611 4-Isothiazolyl-3'                                                          612 4-Isothiazolyl-4'                                                          613 4-Isothiazolyl-5'                                                          614 2-Imidazolyl-1'                                                            615 2-Imidazolyl-2'                                                            616 2-Imidazolyl-4'                                                            617 3-Imidazolyl-1'                                                            618 3-Imidazolyl-2'                                                            619 3-Imidazolyl-4'                                                            620 4-Imidazolyl-1'                                                            621 4-Imidazolyl-2'                                                            622 4-Imidazolyl-4'                                                            623 2-Oxazolyl-2'                                                              624 2-Oxazolyl-4'                                                              625 2-Oxazolyl-5'                                                              626 3-Oxazolyl-2'                                                              627 3-Oxazolyl-4'                                                              628 3-Oxazolyl-5'                                                              629 4-Oxazolyl-2'                                                              630 4-Oxazolyl-4'                                                              631 4-Oxazolyl-5'                                                              632 2-Thiazolyl-2'                                                             633 2-Thiazolyl-4'                                                             634 2-Thiazolyl-5'                                                             635 3-Thiazolyl-2'                                                             636 3-Thiazolyl-4'                                                             637 3-Thiazolyl-5'                                                             638 4-Thiazolyl-2'                                                             639 4-Thiazolyl-4'                                                             640 4-Thiazolyl-5'                                                             641 2-CH.sub.3 -4-(CH.sub.3 --C═N--O--CH.sub.2 --CH.sub.2 --OCH.sub.               3)                                                                     642 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C═N--O--CH.sub.2 --CH.sub.2                   --OCH.sub.3)                                                           643 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C═N--O--CH.sub.2 --CH.sub.2                --OCH.sub.3)                                                           644 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C═N--OCH.sub.3)                     645 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C═N--OC.sub.2 H.sub.5)                       646 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C═N--O-n-C.sub.3                   H.sub.7)                                                               647 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C═N--O-i-C.sub.3 H.sub.7)                    648 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C═N--O-Allyl)                       649 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C═N--O-trans-Chloroa               llyl)                                                                  650 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C═N--O-Propargyl)                   651 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C═N--O-n-C.sub.4 H.sub.9)                    652 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C═N--O--CH.sub.2                   --C.sub.6 H.sub.5)                                                     653 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C═N--OCH.sub.3)                     654 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C═N--OC.sub.2 H.sub.5)                       655 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C═N--O-n-C.sub.3                   H.sub.7)                                                               656 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C═N--O-i-C.sub.3 H.sub.7)                    657 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C═N--O-Allyl)                       658 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C═N--O-trans-Chloroa               llyl)                                                                  659 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C═N--O-Propargyl)                   660 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C═N--O-n-(C.sub.4 H.sub.9)                   661 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C═N--C--CH.sub.2                   --C.sub.6 H.sub.5)                                                     662 2-O-n-C.sub.4 H.sub.9                                                      663 2-O-i-C.sub.4 H.sub.9                                                      664 2-O-s-C.sub.4 H.sub.9                                                      665 2-O-t-C.sub.4 H.sub.9                                                      666 2-Neopentyloxy                                                             667 3-O-n-C.sub.4 H.sub.9                                                      668 3-O-i-C.sub.4 H.sub.9                                                      669 3-O-s-C.sub.4 H.sub.9                                                      670 3-O-t-C.sub.4 H.sub.9                                                      671 3-Neopentyloxy                                                             672 4-O-n-C.sub.4 H.sub.9                                                      673 4-C-i-C.sub.4 H.sub.9                                                      674 4-C-s-C.sub.4 H.sub.9                                                      675 4-C-t-C.sub.4 H.sub.9                                                      676 4-Neopentyloxy                                                             677 3-CH.sub.3 -4-OCH.sub.3                                                    678 3-CH.sub.3 -4-CO.sub.2 H.sub.5                                             679 3-CH.sub.3 -4-O-n-C.sub.3 H.sub.7                                          680 3-CH.sub.3 -4-O-n-C.sub.4 H.sub.9                                          681 3-CH.sub.3 -4-O-i-C.sub.4 H.sub.9                                          682 3-CH.sub.3 -4-O-s-C.sub.4 H.sub.9                                          683 3-CH.sub.3 -4-t-C.sub.4 H.sub.9                                            684 3-CH.sub.3 -4-Neopentyloxy                                                 685 2-CH.sub.3 -3-OCH.sub.3                                                    686 2-CH.sub.3 -4-OCH.sub.3                                                    687 2-CH.sub.3 -5-OCH.sub.3                                                    688 2-CH.sub.3 -6-OCH.sub.3                                                    689 3-CH.sub.3 -4-OCH.sub.3                                                    690 3-CH.sub.3 -5-OCH.sub.3                                                    691 3-CH.sub.3 -6-OCH.sub.3                                                    692 4-CH.sub.3 -5-O--CH.sub.3                                                  693 4-CH.sub.3 -6-O--CH.sub.3                                                  694 4-CH.sub.3 -6-OCH.sub.3                                                    695 2-CH.sub.3 -3-O-i-C.sub.3 H.sub.7                                          696 2-CH.sub.3 -4-O-i-C.sub.3 H.sub.7                                          697 2-CH.sub.3 -5-O-i-C.sub.3 H.sub.7                                          698 2-CH.sub.3 -6-O-i-C.sub.3 H.sub.7                                          699 3-CH.sub.3 -4-O-i-C.sub.3 H.sub.7                                          700 3-CH.sub.3 -5-O-i-C.sub.3 H.sub.7                                          701 3-CH.sub.3 -6-O-i-C.sub.3 H.sub.7                                          702 4-CH.sub.3 -5-O-i-C.sub.3 H.sub.7                                          703 4-CH.sub.3 -6-O-i-C.sub.3 H.sub.7                                          704 5-CH.sub.3 -6-O-i-C.sub.3 H.sub.7                                          705 2-Cl-3-OCH.sub.3                                                           706 2-Cl-4-OCH.sub.3                                                           707 2-Cl-5-OCH.sub.3                                                           708 2-Cl-6-OCH.sub.3                                                           709 3-Cl-4-OCH.sub.3                                                           710 3-Cl-5-OCH.sub.3                                                           711 3-Cl-6-OCH.sub.3                                                           712 4-Cl-5-OCH.sub.3                                                           713 4-Cl-6-OCH.sub.3                                                           714 5-Cl-6-OCH.sub.3                                                         ______________________________________                                    

                  TABLE 2                                                          ______________________________________                                         1  STR24##                                                                        -        I: R.sup.1 = H                                                       II: R.sup.1 = CH.sub.3                                                         III: R.sup.1 = Allyl                                                           IV: R.sup.1 = Propargyl                                                        V: R.sup.1 = S--CH.sub.3                                                       VI: R.sup.1 = CH.sub.2 --CN                                                    VII: R.sup.1 = CH.sub.2 --O--CH.sub.3                                          VIII: R.sup.1 = CO--OCH.sub.3                                                   -                                                                           No.       B                                                                    ______________________________________                                         1         Pyrrolyl-3                                                             2 N-CH.sub.3 -Pyrrolyl-3                                                       3 N-C.sub.6 H.sub.5 -Pyrrolyl-3                                                4 N-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrrolyl-3                                 5 N-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrrolyl-3                                 6 N-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrrolyl-3                                 7 N-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrrolyl-3                                8 N-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrrolyl-3                                9 N-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrrolyl-3                                10 N-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrrolyl-3                                11 N-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrrolyl-3                                12 N-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrrolyl-3                                13 N-(4'-CN-C.sub.6 H.sub.4)-Pyrrolyl-3                                        14 N-(3'-CN-C.sub.6 H.sub.4)-Pyrrolyl-3                                        15 N-(2'-CN-C.sub.6 H.sub.4)-Pyrrolyl-3                                        16 N-(4'-Cl-C.sub.6 H.sub.4)-Pyrrolyl-3                                        17 N-(3'-Cl-C.sub.6 H.sub.4)-Pyrrolyl-3                                        18 N-(2'-Cl-C.sub.6 H.sub.4)-Pyrrolyl-3                                        19 Pyrrolyl-2                                                                  20 N-CH.sub.3 -Pyrrolyl-2                                                      21 N-C.sub.6 H.sub.5 -Pyrrolyl-2                                               22 N-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrrolyl-2                                23 N-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrrolyl-2                                24 N-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrrolyl-2                                25 N-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrrolyl-2                               26 N-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrrolyl-2                               27 N-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrrolyl-2                               28 N-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrrolyl-2                                29 N-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrrolyl-2                                30 N-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrrolyl-2                                31 N-(4'-CN-C.sub.6 H.sub.4)-Pyrrolyl-2                                        32 N-(3'-CN-C.sub.6 H.sub.4)-Pyrrolyl-2                                        33 N-(2'-CN-C.sub.6 H.sub.4)-Pyrrolyl-2                                        34 N-(4'-Cl-C.sub.6 H.sub.4)-Pyrrolyl-2                                        35 N-(3'-Cl-C.sub.6 H.sub.4)-Pyrrolyl-2                                        36 N-(2'-Cl-C.sub.6 H.sub.4)-Pyrrolyl-2                                        37 Furyl-2                                                                     38 5-CH.sub.3 -Furyl-2                                                         39 5-C.sub.6 H.sub.5 -Furyl-2                                                  40 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Furyl-2                                   41 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Furyl-2                                   42 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Furyl-2                                   43 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Furyl-2                                  44 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Furyl-2                                  45 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Furyl-2                                  46 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Furyl-2                                   47 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Furyl-2                                   48 5-(2'-NO.sub.2 O--.sub.6 H.sub.4)-Furyl-2                                   49 5-(4'-CN--C.sub.6 H.sub.4)-Furyl-2                                          50 5-(3'-CN--C.sub.6 H.sub.4)-Furyl-2                                          51 5-(2'-CN--C.sub.6 H.sub.4)-Furyl-2                                          52 5-(4'-Cl--C.sub.6 H.sub.4)-Furyl-2                                          53 5-(3'-Cl--C.sub.6 H.sub.4)-Furyl-2                                          54 5-(2'-Cl--C.sub.6 H.sub.4)-Furyl-2                                          55 4-CH.sub.3 -Furyl-2                                                         56 4-C.sub.6 H.sub.5 -Furyl-2                                                  57 4-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Furyl-2                                   58 4-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Furyl-2                                   59 4-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Furyl-2                                   60 4-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Furyl-2                                  61 4-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Furyl-2                                  62 4-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Furyl-2                                  63 4-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Furyl-2                                   64 4-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Furyl-2                                   65 4-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Furyl-2                                   66 4-(4'-CN--C.sub.6 H.sub.4)-Furyl-2                                          67 4-(3'-CN--C.sub.6 H.sub.4)-Furyl-2                                          68 4-(2'-CN--C.sub.6 H.sub.4)-Furyl-2                                          69 4-(4'-Cl--C.sub.6 H.sub.4)-Furyl-2                                          70 4-(3'-Cl--C.sub.6 H.sub.4)-Furyl-2                                          71 4-(2'-Cl--C.sub.6 H.sub.4)-Furyl-2                                          72 Thienyl-2                                                                   73 5-CH.sub.3 -Thienyl-2                                                       74 5-C.sub.6 H.sub.5 -Thienyl-2                                                75 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-2                                 76 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-2                                 77 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-2                                 78 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-2                                79 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-2                                80 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-2                                81 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-2                                 82 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-2                                 83 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-2                                 84 5-(4'-CN--C.sub.6 H.sub.4)-Thienyl-2                                        85 5-(3'-CN--C.sub.6 H.sub.4)-Thienyl-2                                        86 5-(2'-CN--C.sub.6 H.sub.4)-Thienyl-2                                        87 5-(4'-Cl--C.sub.6 H.sub.4)-Thienyl-2                                        88 5-(3'-Cl--C.sub.6 H.sub.4)-Thienyl-2                                        89 5-(2'-Cl--C.sub.6 H.sub.4)-Thienyl-2                                        90 4-CH.sub.3 -Thienyl-2                                                       91 4-C.sub.6 H.sub.5 -Thienyl-2                                                92 4-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-2                                 93 4-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-2                                 94 4-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-2                                 95 4-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-2                                96 4-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-2                                97 4-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-2                                98 4-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-2                                 99 4-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-2                                 100 4-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-2                                101 4-(4'-CN--C.sub.6 H.sub.4)-Thienyl-2                                       102 4-(3'-CN--C.sub.6 H.sub.4)-Thienyl-2                                       103 4-(2'-CN--C.sub.6 H.sub.4)-Thienyl-2                                       104 4-(4'-Cl--C.sub.6 H.sub.4)-Thienyl-2                                       105 4-(3'-Cl--C.sub.6 H.sub.4)-Thienyl-2                                       106 4-(2'-Cl--C.sub.6 H.sub.4)-Thienyl-2                                       107 Thienyl-3                                                                  108 5-CH.sub.3 -Thienyl-3                                                      109 5-C.sub.6 H.sub.5 -Thienyl-3                                               110 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-3                                111 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-3                                112 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-3                                113 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-3                               114 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-3                               115 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-3                               116 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-3                                117 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-3                                118 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-3                                119 5-(4'-CN--C.sub.6 H.sub.4)-Thienyl-3                                       120 5-(3'-CN--C.sub.6 H.sub.4)-Thienyl-3                                       121 5-(2'-CN--C.sub.6 H.sub.4)-Thienyl-3                                       122 5-(4'-Cl--C.sub.6 H.sub.4)-Thienyl-3                                       123 5-(3'-Cl--C.sub.6 H.sub.4)-Thienyl-3                                       124 5-(2'-Cl--C.sub.6 H.sub.4)-Thienyl-3                                       125 Pyrazolyl-4                                                                126 N-CH.sub.3 -Pyrazolyl-4                                                    127 N-C.sub.6 H.sub.5 -Pyrazolyl-4                                             128 N-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrazolyl-4                              129 N-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrazolyl-4                              130 N-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrazolyl-4                              131 N-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrazolyl-4                             132 N-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrazolyl-4                             133 N-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrazolyl-4                             134 N-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrazolyl-4                              135 N-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrazolyl-4                              136 N-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrazolyl-4                              137 N-(4'-CN--C.sub.6 H.sub.4)-Pyrazolyl-4                                     138 N-(3'-CN--C.sub.6 H.sub.4)-Pyrazolyl-4                                     139 N-(2'-CN--C.sub.6 H.sub.4)-Pyrazolyl-4                                     140 N-(4'-Cl--C.sub.6 H.sub.4)-Pyrazolyl-4                                     141 N-(3'-Cl--C.sub.6 H.sub.4)-Pyrazolyl-4                                     142 N-(2'-Cl--C.sub.6 H.sub.4)-Pyrazolyl-4                                     143 3-CH.sub.3 --N-Methylpyrazolyl-4                                           144 3-C.sub.6 H.sub.5 --N-Methylpyrazolyl-4                                    145 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)-N-Methylpyrazolyl-4                      146 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)-N-Methylpyrazolyl-4                      147 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)-N-Methylpyrazolyl-4                      148 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-N-Methylpyrazolyl-4                     149 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-N-Methylpyrazolyl-4                     150 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-N-Methylpyrazolyl-4                     151 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)-N-Methylpyrazolyl-4                      152 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)-N-Methylpyrazolyl-4                      153 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)-N-Methylpyrazolyl-4                      154 3-(4'-CN--C.sub.6 H.sub.4)-N-Methylpyrazolyl-4                             155 3-(3'-CN--C.sub.6 H.sub.4)-N-Methylpyrazolyl-4                             156 3-(2'-CN--C.sub.6 H.sub.4)-N-Methylpyrazolyl-4                             157 3-(4'-Cl--C.sub.6 H.sub.4)-N-Methylpyrazolyl-4                             158 3-(3'-Cl--C.sub.6 H.sub.4)-N-Methylpyrazolyl-4                             159 3-(2'-Cl--C.sub.6 H.sub.4)-N-Methylpyrazolyl-4                             160 Isoxazolyl-5                                                               161 3-CH.sub.3 -Isoxazolyl-5                                                   162 3-C.sub.6 H.sub.5 -Isoxazolyl-5                                            163 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Isoxazolyl-5                             164 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Isoxazolyl-5                             165 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Isoxazolyl-5                             166 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Isoxazolyl-5                            167 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Isoxazolyl-5                            168 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Isoxazolyl-5                            169 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Isoxazolyl-5                             170 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Isoxazolyl-5                             171 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Isoxazolyl-5                             172 3-(4'-CN--C.sub.6 H.sub.4)-Isoxazolyl-5                                    173 3-(3'-CN--C.sub.6 H.sub.4)-Isoxazolyl-5                                    174 3-(2'-CN--C.sub.6 H.sub.4)-Isoxazolyl-5                                    175 3-(4'-Cl--C.sub.6 H.sub.4)-Isoxazolyl-5                                    176 3-(3'-Cl--C.sub.6 H.sub.4)-Isoxazolyl-5                                    177 3-(2'-Cl--C.sub.6 H.sub.4)-Isoxazolyl-5                                    178 4-Chloroisoxazolyl-5                                                       179 3-CH.sub.3 -4-Chloroisoxazolyl-5                                           180 3-C.sub.6 H.sub.5 -4-Chloroisoxazolyl-5                                    181 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                     182 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                     183 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                     184 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                    185 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                    186 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                    187 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                     188 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                     189 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                     190 3-(4'-CN--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                            191 3-(3'-CN--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                            192 3-(2'-CN--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                            193 3-(4'-Cl--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                            194 3-(3'-Cl--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                            195 3-(2'-Cl--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                            196 Isoxazolyl-3                                                               197 5-CH.sub.3 -Isoxazolyl-3                                                   198 5-C.sub.6 H.sub.5 -Isoxazolyl-3                                            199 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Isoxazolyl-3                             200 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Isoxazolyl-3                             201 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Isoxazolyl-3                             202 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Isoxazolyl-3                            203 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Isoxazolyl-3                            204 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Isoxazolyl-3                            205 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Isoxazolyl-3                             206 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Isoxazolyl-3                             207 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Isoxazolyl-3                             208 5-(4'-CN--C.sub.6 H.sub.4)-Isoxazolyl-3                                    209 5-(3'-CN--C.sub.6 H.sub.4)-Isoxazolyl-3                                    210 5-(2'-CN--C.sub.6 H.sub.4)-Isoxazolyl-3                                    211 5-(4'-Cl--C.sub.6 H.sub.4)-Isoxazolyl-3                                    212 5-(3'-Cl--C.sub.6 H.sub.4)-Isoxazolyl-3                                    213 5-(2'-Cl--C.sub.6 H.sub.4)-Isoxazolyl-3                                    214 Isothiazolyl-5                                                             215 3-CH.sub.3 -Isothiazolyl-5                                                 216 3-C.sub.6 H.sub.5 -Isothiazolyl-5                                          217 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Isothiazolyl-5                           218 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Isothiazolyl-5                           219 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Isothiazolyl-5                           220 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4 )-Isothiazolyl-5                         221 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Isothiazolyl-5                          222 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Isothiazolyl-5                          223 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Isothiazolyl-5                           224 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Isothiazolyl-5                           225 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Isothiazolyl-5                           226 3-(4'-CN--C.sub.6 H.sub.4)-Isothiazolyl-5                                  227 3-(3'-CN--C.sub.6 H.sub.4)-Isothiazolyl-5                                  228 3-(2'-CN--C.sub.6 H.sub.4)-Isothiazolyl-5                                  229 3-(4'-Cl--C.sub.6 H.sub.4)-Isothiazolyl-5                                  230 3-(3'-Cl--C.sub.6 H.sub.4)-Isothiazolyl-5                                  231 3-(2'-Cl--C.sub.6 H.sub.4)-Isothiazolyl-5                                  232 Oxazolyl-4                                                                 233 3-CH.sub.3 -Oxazolyl-4                                                     234 3-C.sub.6 H.sub.5 -Oxazolyl-4                                              235 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Oxazolyl-4                               236 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Oxazolyl-4                               237 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Oxazolyl-4                               238 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Oxazolyl-4                              239 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Oxazolyl-4                              240 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Oxazolyl-4                              241 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Oxazolyl-4                               242 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Oxazolyl-4                               243 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Oxazolyl-4                               244 3-(4'-CN--C.sub.6 H.sub.4)-Oxazolyl-4                                      245 3-(3'-CN--C.sub.6 H.sub.4)-Oxazolyl-4                                      246 3-(2'-CN--C.sub.6 H.sub.4)-Oxazolyl-4                                      247 3-(4'-Cl--C.sub.6 H.sub.4)-Oxazolyl-4                                      248 3-(3'-Cl--C.sub.6 H.sub.4)-Oxazolyl-4                                      249 3-(2'-Cl--C.sub.6 H.sub.4)-Oxazolyl-4                                      250 Thiazolyl-4                                                                251 2-CH.sub.3 -Thiazolyl-4                                                    252 2-C.sub.6 H.sub.5 -Thiazolyl-4                                             253 2-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Thiazolyl-4                              254 2-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Thiazolyl-4                              255 2-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Thiazolyl-4                              256 2-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Thiazolyl-4                             267 2-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Thiazolyl-4                             258 2-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Thiazolyl-4                             259 2-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Thiazolyl-4                              260 2-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Thiazolyl-4                              261 2-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Thiazolyl-4                              262 2-(4'-CN--C.sub.6 H.sub.4)-Thiazolyl-4                                     263 2-(3'-CN--C.sub.6 H.sub.4)-Thiazolyl-4                                     264 2-(2'-CN--C.sub.6 H.sub.4)-Thiazolyl-4                                     265 2-(4'-Cl--C.sub.6 H.sub.4)-Thiazolyl-4                                     266 2-(3'-Cl--C.sub.6 H.sub.4)-Thiazolyl-4                                     267 2-(2'-Cl--C.sub.6 H.sub.4)-Thiazolyl-4                                     268 N--CH.sub.3 -1,2,4-Triazolyl-5                                             269 3-CH.sub.3 --N--CH.sub.3 -1,2,4-Triazolyl-5                                270 3-C.sub.6 H.sub.5 --N--CH.sub.3 -1,2,4-Triazolyl-5                         271 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)-N--CH.sub.3 -1,2,4-Triazolyl-5                    272 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)-N--CH.sub.3 -1,2,4-Triazo               lyl-5                                                                  273 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)-N--CH.sub.3 -1,2,4-Triazolyl-5                    274 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-N--CH.sub.3 -1,2,4-Triaz               olyl-5                                                                 275 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-N--CH.sub.3 -1,2,4-Triazolyl-5                   276 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-N--CH.sub.3 -1,2,4-Triaz               olyl-5                                                                 277 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)-N--CH.sub.3 -1,2,4-Triazolyl-5                    278 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)-N--CH.sub.3 -1,2,4-Triazo               lyl-5                                                                  279 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)-N--CH.sub.3 -1,2,4-Triazolyl-5                    280 3-(4'-CN--C.sub.6 H.sub.4)-N--CH.sub.3 -1,2,4-Triazolyl-5                  281 3-(3'-CN--C.sub.6 H.sub.4)-N--CH.sub.3 -1,2,4-Triazolyl-5                  282 3-(2'-CN--C.sub.6 H.sub.4)-N--CH.sub.3 -1,2,4-Triazolyl-5                  283 3-(4'-Cl--C.sub.6 H.sub.4)-N--CH.sub.3 -1,2,4-Triazolyl-5                  284 3-(3'-Cl--C.sub.6 H.sub.4)-N--CH.sub.3 -1,2,4-Triazolyl-5                  285 3-(2'-Cl--C.sub.6 H.sub.4)-N--CH.sub.3 -1,2,4-Triazolyl-5                  286 1,3,4-Oxadiazolyl-2                                               287 5-CH.sub.3 -1,3,4-Oxadiazolyl-2                                            288 5-C.sub.6 H.sub.5 -1,3,4-Oxadiazolyl-2                                     289 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                      290 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                      291 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                      292 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                     293 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                     294 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                     295 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                      296 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                      297 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                      298 5-(4'-CN--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                             299 5-(3'-CN--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                             300 5-(2'-CN--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                             301 5-(4'-Cl--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                             302 5-(3'-Cl--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                             303 5-(2'-Cl--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                             304 1,2,4-Oxadiazolyl-3                                                        305 5-CH.sub.3 -1,2,4-Oxadiazolyl-3                                            306 5-C.sub.6 H.sub.5 -1,2 4-Oxadiazolyl-3                                     307 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                      308 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                      309 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                      310 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                     311 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                     312 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                     313 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                      314 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                      315 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                      316 5-(4'-CN--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                             317 5-(3'-CN--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                             318 5-(2'-CN--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                             319 5-(4'-Cl--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                             320 5-(3'-Cl--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                             321 5-(2'-Cl--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                             322 1,2,4-Oxadiazolyl-5                                                        323 3-CH.sub.3 -1,2,4-Oxadiazolyl-5                                            324 3-C.sub.6 H.sub.5 -1,2,4-Oxadiazolyl-5                                     325 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                      326 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                      327 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                      328 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                     329 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                     330 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                     331 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                      332 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                      333 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                      334 3-(4'-CN--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                             335 3-(3'-CN--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                             336 3-(2'-CN--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                             337 3-(4'-Cl--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                             338 3-(3'-Cl--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                             339 3-(2'-Cl--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                             340 1,2,4-Thiadiazolyl-3                                                       341 5-CH.sub.3 -1,2,4-Thiadiazolyl-3                                           342 5-C.sub.6 H.sub.5 -1,2,4-Thiadiazolyl-3                                    343 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                     344 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                     345 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                     346 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                    347 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                    348 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                    349 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                     350 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                     351 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                     352 5-(4'-CN--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                            353 5-(3'-CN--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                            354 5-(2'-CN--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                            355 5-(4'-Cl--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                            356 5-(3'-Cl--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                            357 5-(2'-Cl--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                            358 1,3,4-Thiadiazolyl-2                                                       359 5-CH.sub.3 -1,3,4-Thiadiazolyl-2                                           360 5-C.sub.6 H.sub.5 -1,3,4-Thiadiazolyl-2                                    361 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                     362 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                     363 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                     364 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                    365 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                    366 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                    367 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                     368 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                     369 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                     370 5-(4'-CN--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                            371 5-(3'-CN--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                            372 5-(2'-CN--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                            373 5-(4'-Cl--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                            374 5-(3'-Cl--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                            375 5-(2'-Cl--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                            376 Pyridinyl-2                                                                377 Pyridinyl-4                                                                378 Pyridazinyl-3                                                              379 Pyridazinyl-4                                                              380 Pyridazinyl-2                                                              381 Pyrimidinyl-4                                                              382 Pyrimidinyl-5                                                              383 Pyrimidinyl-2                                                              384 1-Naphthyl                                                                 385 2-Naphthyl                                                               ______________________________________                                    

                  TABLE 3                                                          ______________________________________                                         1  STR25##                                                                        -        I: R.sup.1 = H                                                       II: R.sup.1 = CH.sub.3                                                         III: R.sup.1 = Allyl                                                           IV: R.sup.1 = Propargyl                                                        V: R.sup.1 = S--CH.sub.3                                                       VI: R.sup.1 = CH.sub.2 --CN                                                    VII: R.sup.1 = CH.sub.2 --O--CH.sub.3                                          VIII: R.sup.1 = CO--OCH.sub.3                                                No.     X.sub.m                                                                ______________________________________                                          1      H                                                                         2 2-F                                                                          3 3-F                                                                          4 4-F                                                                          5 2,4-F.sub.2                                                                  6 2,4,6-F.sub.3                                                                7 2,3,4,5,6-F.sub.5                                                            8 2,3-F.sub.2                                                                  9 2-Cl                                                                         10 3-Cl                                                                        11 4-Cl                                                                        12 2,3-Cl.sub.2                                                                13 2,4-Cl.sub.2                                                                14 2,5-Cl.sub.2                                                                15 2,6-Cl.sub.2                                                                16 3,4-Cl.sub.2                                                                17 3,5-Cl.sub.2                                                                18 2,3,4-Cl.sub.3                                                              19 2,3,5-Cl.sub.3                                                              20 2,3,6-Cl.sub.3                                                              21 2,4,5-Cl.sub.3                                                              22 2,4,6-Cl.sub.3                                                              23 3,4,5-Cl.sub.3                                                              24 2,3,4,6-Cl.sub.4                                                            25 2,3,5,6-Cl.sub.4                                                            26 2,3,4,5,6-Cl.sub.5                                                          27 2-Br                                                                        28 3-Br                                                                        29 4-Br                                                                        30 2,4-Br.sub.2                                                                31 2,5-Br.sub.2                                                                32 2,6-Br.sub.2                                                                33 2,4,6-Br.sub.3                                                              34 2,3,4,5,6-Br.sub.5                                                          35 2-I                                                                         36 3-I                                                                         37 4-I                                                                         38 2,4-I.sub.2                                                                 39 2-Cl, 3-F                                                                   40 2-Cl, 4-F                                                                   41 2-Cl, 5-F                                                                   42 2-Cl, 6-F                                                                   43 2-Cl, 3-Br                                                                  44 2-Cl, 4-Br                                                                  45 2-Cl, 5-Br                                                                  46 2-Cl, 6-Br                                                                  47 2-Br, 3-Cl                                                                  48 2-Br, 4-Cl                                                                  49 2-Br, 5-Cl                                                                  50 2-Br, 3-F                                                                   51 2-Br, 4-F                                                                   52 2-Br, 5-F                                                                   53 2-Br, 6-F                                                                   54 2-F, 3-Cl                                                                   55 2-F, 4-Cl                                                                   56 2-F, 5-Cl                                                                   57 3-Cl, 4-F                                                                   58 3-Cl, 5-F                                                                   59 3-Cl, 4-Br                                                                  60 3-Cl, 5-Br                                                                  61 3-F, 4-Cl                                                                   62 3-F, 4-Br                                                                   63 3-Br, 4-Cl                                                                  64 3-Br, 4-F                                                                   65 2,6-Cl.sub.2, 4-Br                                                          66 2-CH.sub.3                                                                  67 3-CH.sub.3                                                                  68 4-CH.sub.3                                                                  69 2,3-(CH.sub.3).sub.2                                                        70 2,4-(CH.sub.3).sub.2                                                        71 2,5-(CH.sub.3).sub.2                                                        72 2,6-(CH.sub.3).sub.2                                                        73 3,4-(CH.sub.3).sub.2                                                        74 3,5-(CH.sub.3).sub.2                                                        75 2,3,5-(CH.sub.3).sub.3                                                      76 2,3,4-(CH.sub.3).sub.3                                                      77 2,3,6-(CH.sub.3).sub.3                                                      78 2,4,5-(CH.sub.3).sub.3                                                      79 2,4,6-(CH.sub.3).sub.3                                                      80 3,4,5-(CH.sub.3).sub.3                                                      81 2,3,4,6-(CH.sub.3).sub.4                                                    82 2,3,5,6-(CH.sub.3).sub.4                                                    83 2,3,4,5,6-(CH.sub.3).sub.5                                                  84 2-C.sub.2 H.sub.5                                                           85 3-C.sub.2 H.sub.5                                                           86 4-C.sub.2 H.sub.5                                                           87 2,4-(C.sub.2 H.sub.5).sub.2                                                 88 2,6-(C.sub.2 H.sub.5).sub.2                                                 89 3,5-(C.sub.2 H.sub.5).sub.2                                                 90 2,4,6-(C.sub.2 H.sub.5).sub.3                                               91 2-n-C.sub.3 H.sub.7                                                         92 3-n-C.sub.3 H.sub.7                                                         93 4-n-C.sub.3 H.sub.7                                                         94 2-i-C.sub.3 H.sub.7                                                         95 3-i-C.sub.3 H.sub.7                                                         96 4-i-C.sub.3 H.sub.7                                                         97 2,4-(i-C.sub.3 H.sub.7).sub.2                                               98 2,6-(i-C.sub.3 H.sub.7).sub.2                                               99 3,5-(i-C.sub.3 H.sub.7).sub.2                                              100 2,4,6-(i-C.sub.3 H.sub.7).sub.3                                            101 2-s-C.sub.4 H.sub.9                                                        102 3-s-C.sub.4 H.sub.9                                                        103 4-s-C.sub.4 H.sub.9                                                        104 2-t-C.sub.4 H.sub.9                                                        105 3-t-C.sub.4 H.sub.9                                                        106 4-t-C.sub.4 H.sub.9                                                        107 2,3-(t-C.sub.4 H.sub.9).sub.2                                              108 2,4-(t-C.sub.4 H.sub.9).sub.2                                              109 2,5-(t-C.sub.4 H.sub.9).sub.2                                              110 2,6-(t-C.sub.4 H.sub.9).sub.2                                              111 3,4-(t-C.sub.4 H.sub.9).sub.2                                              112 2,4,6-(t-C.sub.4 H.sub.9).sub.3                                            113 4-n-C.sub.9 H.sub.19                                                       114 4-n-C.sub.12 H.sub.25                                                      115 4-n-C.sub.15 H.sub.31                                                      116 4-(1,1,3,3-Tetramethylbutyl)                                               117 4-(2,4,4-Trimethylpropyl)                                                  118 2-t-C.sub.4 H.sub.9, 4-CH.sub.3                                            119 2-t-C.sub.4 H.sub.9, 5-CH.sub.3                                            120 2,6-(t-C.sub.4 H.sub.9).sub.2, 4-CH.sub.3                                  121 2-CH.sub.3, 4-t-C.sub.4 H.sub.9                                            122 2-CH.sub.3, 6-t-C.sub.4 H.sub.9                                            123 2-CH.sub.3, 4-i-C.sub.3 H.sub.7                                            124 2-CH.sub.3, 5-i-C.sub.3 H.sub.7                                            125 3-CH.sub.3, 4-i-C.sub.3 H.sub.7                                            126 2-i-C.sub.3 H.sub.7, 5-CH.sub.3                                            127 2,4-(t-C.sub.4 H.sub.9).sub.2, 6-i-C.sub.3 H.sub.7                         128 2-Allyl                                                                    129 3-Allyl                                                                    130 4-Allyl                                                                    131 2-Allyl, 6-CH.sub.3                                                        132 2-cyclo-C.sub.6 H.sub.11                                                   133 3-cyclo-C.sub.6 H.sub.11                                                   134 4-cyclo-C.sub.6 H.sub.11                                                   135 2,4-(cyclo-C.sub.6 H.sub.11).sub.2, 6-CH.sub.3                             136 2-CH.sub.3, 4-cyclo-C.sub.6 H.sub.11                                       137 2-CH.sub.2 --C.sub.6 H.sub.5                                               138 3-CH.sub.2 --C.sub.6 H.sub.5                                               139 4-CH.sub.2 --C.sub.6 H.sub.5                                               140 2-CH.sub.2 --C.sub.6 H.sub.5, 4-CH.sub.3                                   141 2-CH.sub.3, 4-CH.sub.2 --C.sub.6 H.sub.5                                   142 2-C.sub.6 H.sub.5                                                          143 3-C.sub.6 H.sub.5                                                          144 4-C.sub.6 H.sub.5                                                          145 4-(2-i-C.sub.3 H.sub.7 --C.sub.6 H.sub.4)                                  146 4-C.sub.6 H.sub.5, 2,6-(CH.sub.3).sub.2                                    147 2-Cl, 4-C.sub.6 H.sub.5                                                    148 2-Br, 4-C.sub.6 H.sub.5                                                    149 2-C.sub.6 H.sub.5, 4-Cl                                                    150 2-C.sub.6 H.sub.5, 4-Br                                                    151 2-CH.sub.2 C.sub.6 H.sub.5, 4-Cl                                           152 2-CH.sub.2 C.sub.6 H.sub.5, 4-Br                                           153 2-Cl, 4-CH.sub.2 C.sub.6 H.sub.5                                           154 2-Br, 4-CH.sub.2 C.sub.6 H.sub.5                                           155 2-cyclo-C.sub.6 H.sub.11, 4-Cl                                             156 2-cyclo-C.sub.6 H.sub.11, 4-Br                                             157 2-Cl, 4-cyclo-C.sub.6 H.sub.11                                             158 2-Br, 4-cyclo-C.sub.6 H.sub.11                                             159 2-OCH.sub.3                                                                160 3-OCH.sub.3                                                                161 4-OCH.sub.3                                                                162 2-OC.sub.2 H.sub.5                                                         163 3-O--C.sub.2 H.sub.5                                                       164 4-O--C.sub.2 H.sub.5                                                       165 2-O-n-C.sub.3 H.sub.7                                                      166 3-O-n-C.sub.3 H.sub.7                                                      167 4-O-n-C.sub.3 H.sub.7                                                      168 2-O-i-C.sub.3 H.sub.7                                                      169 3-O-i-C.sub.3 H.sub.7                                                      170 4-O-i-C.sub.3 H.sub.7                                                      171 2-O-n-C.sub.6 H.sub.13                                                     172 3-O-n-C.sub.6 H.sub.13                                                     173 4-O-n-C.sub.6 H.sub.13                                                     174 2-O-n-C.sub.8 H.sub.17                                                     175 3-O-n-C.sub.8 H.sub.17                                                     176 4-O-n-C.sub.8 H.sub.17                                                     177 2-O--CH.sub.2 C.sub.6 H.sub.5                                              178 3-O--CH.sub.2 C.sub.6 H.sub.5                                              179 4-O--CH.sub.2 C.sub.6 H.sub.5                                              180 2-O--(CH.sub.2).sub.3 C.sub.6 H.sub.5                                      181 3-O--(CH.sub.2).sub.3 C.sub.6 H.sub.5                                      182 4-O--(CH.sub.2).sub.3 C.sub.6 H.sub.5                                      183 2,4-(OCH.sub.3).sub.2                                                      184 2-CF.sub.3                                                                 185 3-CF.sub.3                                                                 186 4-CF.sub.3                                                                 187 2-OCF.sub.3                                                                188 3-OCF.sub.3                                                                189 4-OCF.sub.3                                                                190 3-OCH.sub.2 CHF.sub.2                                                      191 2-NO.sub.2                                                                 192 3-NO.sub.2                                                                 193 4-NO.sub.2                                                                 194 2-CN                                                                       195 3-CN                                                                       196 4-CN                                                                       197 2-CH.sub.3, 3-Cl                                                           198 2-CH.sub.3, 4-Cl                                                           199 2-CH.sub.3, 5-Cl                                                           200 2-CH.sub.3, 6-Cl                                                           201 2-CH.sub.3, 3-F                                                            202 2-CH.sub.3, 4-F                                                            203 2-CH.sub.3, 5-F                                                            204 2-CH.sub.3, 6-F                                                            205 2-CH.sub.3, 3-Br                                                           206 2-CH.sub.3, 4-Br                                                           207 2-CH.sub.3, 5-Br                                                           208 2-CH.sub.3, 6-Br                                                           209 2-Cl, 3-CH.sub.3                                                           210 2-Cl, 4-CH.sub.3                                                           211 2-Cl, 5-CH.sub.3                                                           212 2-F, 3-CH.sub.3                                                            213 2-F, 4-CH.sub.3                                                            214 2-F, 5-CH.sub.3                                                            215 2-Br, 3-CH.sub.3                                                           216 2-Br, 4-CH.sub.3                                                           217 2-Br, 5-CH.sub.3                                                           218 3-CH.sub.3, 4-Cl                                                           219 3-CH.sub.3, 5-Cl                                                           220 3-CH.sub.3, 4-F                                                            221 3-CH.sub.3, 5-F                                                            222 3-CH.sub.3, 4-Br                                                           223 3-CH.sub.3, 5-Br                                                           224 3-F, 4-CH.sub.3                                                            225 3-Cl, 4-CH.sub.3                                                           226 3-Br, 4-CH.sub.3                                                           227 2-Cl, 4,5-(CH.sub.3).sub.2                                                 228 2-Br, 4,5-(CH.sub.3).sub.2                                                 229 2-Cl, 3,5-(CH.sub.3).sub.2                                                 230 2-Br, 3,5-(CH.sub.3).sub.2                                                 231 2,6-Cl.sub.2, 4-CH.sub.3                                                   232 2,6-F.sub.2, 4-CH.sub.3                                                    233 2,6-Br.sub.2, 4-CH.sub.3                                                   234 2,4-Br.sub.2, 6-CH.sub.3                                                   235 2,4-F.sub.2, 6-CH.sub.3                                                    236 2,4-Br.sub.2, 6-CH.sub.3                                                   237 2,6-(CH.sub.3).sub.2, 4-F                                                  238 2,6-(CH.sub.3).sub.2, 4-Cl                                                 239 2,6-(CH.sub.3).sub.2, 4-Br                                                 240 3,5-(CH.sub.3).sub.2, 4-F                                                  241 3,5-(CH.sub.3).sub.2, 4-Cl                                                 242 3,5-(CH.sub.3).sub.2, 4-Br                                                 243 2,3,6-(CH.sub.3).sub.3, 4-F                                                244 2,3,6-(CH.sub.3).sub.3, 4-Cl                                               245 2,3,6-(CH.sub.3).sub.3, 4-Br                                               246 2,4-(CH.sub.3).sub.2, 6-F                                                  247 2,4-(CH.sub.3).sub.2, 6-Cl                                                 248 2,4-(CH.sub.3).sub.2, 6-Br                                                 249 2-i-C.sub.3 H.sub.7, 4-Cl, 5-CH.sub.3                                      250 2-Cl, 4-NO.sub.2                                                           251 2-NO.sub.2, 4-Cl                                                           252 2-OCH.sub.3, 5-NO.sub.2                                                    253 2,4-Cl.sub.2, 5-NO.sub.2                                                   254 2,4-Cl.sub.2, 6-NO2                                                        255 2,6-Cl.sub.2, 4-NO.sub.2                                                   256 2,6-Br.sub.2, 4-NO.sub.2                                                   257 2,6-I.sub.2, 4-NO.sub.2                                                    258 2-CH.sub.3, 5-i-C.sub.3 H.sub.7, 4-Cl                                      259 2-CO.sub.2 CH.sub.3                                                        260 3-CO.sub.2 CH.sub.3                                                        261 4-CO.sub.2 CH.sub.3                                                        262 2-CO.sub.2 (C.sub.2 H.sub.5)                                               263 3-CO.sub.2 (C.sub.2 H.sub.5)                                               264 4-CO.sub.2 (C.sub.2 H.sub.5)                                               265 2-CO.sub.2 (n-C.sub.3 H.sub.7)                                             266 3-CO.sub.2 (n-C.sub.3 H.sub.7)                                             267 4-CO.sub.2 (n-C.sub.3 H.sub.7)                                             268 2-CO.sub.2 (i-C.sub.3 H.sub.7)                                             269 3-CO.sub.2 (i-C.sub.3 H.sub.7)                                             270 4-CO.sub.2 (i-C.sub.3 H.sub.7)                                             271 2-CO.sub.2 (n-C.sub.6 H.sub.13)                                            272 3-CO.sub.2 (n-C.sub.6 H.sub.13)                                            273 4-CO.sub.2 (n-C.sub.6 H.sub.13)                                            274 2-CH.sub.2 --OCH.sub.3                                                     275 3-CH.sub.2 --OCH.sub.3                                                     276 4-CH.sub.2 --OCH.sub.3                                                     277 2-CH.sub.2 O(C.sub.2 H.sub.5)                                              278 3-CH.sub.2 O(C.sub.2 H.sub.5)                                              279 4-CH.sub.2 O(C.sub.2 H.sub.5)                                              280 2-CH.sub.2 O(n-C.sub.3 H.sub.7)                                            281 3-CH.sub.2 O(n-C.sub.3 H.sub.7)                                            282 4-CH.sub.2 O(n-C.sub.3 H.sub.7)                                            283 2-CH.sub.2 O(i-C.sub.3 H.sub.7)                                            284 3-CH.sub.2 O(i-C.sub.3 H.sub.7)                                            285 4-CH.sub.2 O(i-C.sub.3 H.sub.7)                                            286 2-CHO                                                                      287 3-CHO                                                                      288 4-CHO                                                                      289 2-CO-CH.sub.3                                                              290 3-CO-CH.sub.3                                                              291 4-CO-CH.sub.3                                                              292 2-CO--CH.sub.2 --CH.sub.3                                                  293 3-CO--CH.sub.2 --CH.sub.3                                                  294 4-CO--CH.sub.2 --CH.sub.3                                                  295 2-CO--CH.sub.2 --CH.sub.2 --CH.sub.3                                       296 3-CO--CH.sub.2 --CH.sub.2 --CH.sub.3                                       297 4-CO--CH.sub.2 --CH.sub.2 --CH.sub.3                                       298 2-CO--CH(CH.sub.3)--CH.sub.3                                               299 3-CO--CH(CH.sub.3)--CH.sub.3                                               300 4-CO--CH(CH.sub.3)--CH.sub.3                                               301 2-Me-4-CHO                                                                 302 2-Me-4-CH.sub.3 --CO                                                       303 2-Me-4-CH.sub.3 --CH.sub.2 --CO                                            304 2-Me-4-CH.sub.3 --CH.sub.2 --CH.sub.2 --CO                                 305 2-Me-4-CH.sub.3 --CH (CH.sub.3)--CO                                        306 2,5-Me.sub.2 -4-CHO                                                        307 2,5-Me.sub.2 -4-CH.sub.3 --CO                                              308 2,5-Me.sub.2 -4-CH.sub.3 --CH.sub.2 --CO                                   309 2,5-Me.sub.2 -4-CH.sub.3 --CH.sub.2 --CH.sub.2 --CO                        310 2,5-Me.sub.2 -4-CH.sub.3 --CH(CH.sub.3)--CO                                311 2-Cl-4-CHO                                                                 312 2-Cl-4-CH.sub.3 --CO                                                       313 2-Cl-4-CH.sub.3 --CH.sub.2 --CO                                            314 2-Cl-4-CH.sub.3 --CH(CH.sub.3)--CO                                         315 2,5-Cl.sub.2 -4-CHO                                                        316 2,5-Cl.sub.2 -4-CH.sub.3 --CO                                              317 2,5-Cl.sub.2 -4-CH.sub.3 --CH.sub.2 --CO                                   318 2,5-Cl.sub.2 -4-CH.sub.3 --CH.sub.2 --CH.sub.2 --CO                        319 2,5-Cl.sub.2 -4-CH.sub.3 -- --CH(CH.sub.3)--CO                             320 2-C(═NOCH.sub.3)--CH.sub.3                                             321 3-C(═NOCH.sub.3)--CH.sub.3                                             322 4-C(═NOCH.sub.3)--CH.sub.3                                             323 2-C(═NOC.sub.2 H.sub.5)--CH.sub.3                                      324 3-C(═NOC.sub.2 H.sub.5)--CH.sub.3                                      325 4-C(═NOC.sub.2 H.sub.5)--CH.sub.3                                      326 2-C(═NO-n-C.sub.3 H.sub.7)--CH.sub.3                                   327 3-C(═NO-n-C.sub.3 H.sub.7)--CH.sub.3                                   328 4-C(═NO-n-C.sub.3 H.sub.7)--CH.sub.3                                   329 2-C(═NO-i-C.sub.3 H.sub.7)--CH.sub.3                                   330 3-C(═NO-i-C.sub.3 H.sub.7)--CH.sub.3                                   331 4-C(═NO-i-C.sub.3 H.sub.7)--CH.sub.3                                   332 2-C(═NO-Allyl)-CH.sub.3                                                333 3-C(═NO-Allyl)-CH.sub.3                                                334 4-C(═NO-Allyl)-CH.sub.3                                                335 2-C(═NO-trans-Chloroallyl)-CH.sub.3                                    336 3-C(═NO-trans-Chloroallyl)-CH.sub.3                                    337 4-C(═NO-trans-Chloroallyl)-CH.sub.3                                    338 2-C(═NO-Propargyl)-CH.sub.3                                            339 3-C(═NO-Propargyl)-CH.sub.3                                            340 4-C(═NO-Propargyl)-CH.sub.3                                            341 2-C(═NO-n-C.sub.4 H.sub.9)--CH.sub.3                                   342 3-C(═NO-n-C.sub.4 H.sub.9)--CH.sub.3                                   343 4-C(═NO-n-C.sub.4 H.sub.9)--CH.sub.3                                   344 2-C(═NO--CH.sub.2 --C.sub.6 H.sub.5)--CH.sub.3                         345 3-C(═NO--CH.sub.2 --C.sub.6 H.sub.5)--CH.sub.3                         346 4-C(═NO--CH.sub.2 --C.sub.6 H.sub.5)--CH.sub.3                         347 2-CH.sub.3 -4-CH═NOCH.sub.3                                            348 2-CH.sub.3 -4-CH═NOC.sub.2 H.sub.5                                     349 2-CH.sub.3 -4-CH═NO-n-C.sub.3 H.sub.7                                  350 2-CH.sub.3 -4-CH═NO-i-C.sub.3 H.sub.7                                  351 2-CH.sub.3 -4-CH═NO-Allyl                                              352 2-CH.sub.3 -4-CH═NO-(trans-Chloroallyl)                                353 2-CH.sub.3 -4-CH═NO-Propargyl                                          354 2-CH.sub.3 -4-CH═NO-n-C.sub.4 H.sub.9                                  355 2-CH.sub.3 -4-CH═NO--CH.sub.2 --C.sub.6 H.sub.5                        356 2-CH.sub.3 -4-(CH.sub.3 --C═NOCH.sub.3)                                357 2-CH.sub.3 -4-(CH.sub.3 --C═NOC.sub.2 H.sub.5)                         358 2-CH.sub.3 -4-(CH.sub.3 --C═NO-n-C.sub.3 H.sub.7)                      359 2-CH.sub.3 -4-(CH.sub.3 --C═NO-i-C.sub.3 H.sub.7)                      360 2-CH.sub.3 -4-(CH.sub.3 --C═NO-Allyl)                                  361 2-CH.sub.3 -4-(CH.sub.3 --C═NO-trans-Chloroallyl)                      362 2-CH.sub.3 -4-(CH.sub.3 --C═NO-Propargyl)                              363 2-CH.sub.3 -4-(CH.sub.3 --C═NO-n-C.sub.4 H.sub.9)                      364 2-CH.sub.3 -4-(CH.sub.3 --C═NO--CH.sub.2 --C.sub.6 H.sub.5)                   365 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C═NO--CH.sub.3)                       366 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C═NO--C.sub.2 H.sub.5)                367 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C═NO-n-C.sub.3 H.sub.7)        368 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C═NO-i-C.sub.3 H.sub.7                       369 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C═NO-Allyl)                    370 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C═NO-trans-Chloroallyl)                      371 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C═NO-Propargyl)                       372 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C═NO-n-C.sub.4 H.sub.9)        373 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C═NO--CH.sub.2 --C.sub.6                    H.sub.5)                                                                 374 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C═NOCH.sub.3)                      375 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C═NOC.sub.2 H.sub.5)                      376 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C═NO-n-C.sub.3                    H.sub.7)                                                                 377 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C═NO-i-C.sub.3 H.sub.7)                   378 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C═NO-Allyl)                 379 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C═NO-trans-Chloroallyl)                   380 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C═NO-Proparyl)                     381 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C═NO-n-C.sub.4                    H.sub.9)                                                                 382 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C═NO--CH.sub.2 --C.sub.6                 H.sub.5)                                                                 383 2-C.sub.6 H.sub.5                                                          384 3-C.sub.6 H.sub.5                                                          385 4-C.sub.6 H.sub.5                                                          386 2-(2'-F--C.sub.6 H.sub.4)                                                  387 2-(3'-F--C.sub.6 H.sub.4)                                                  388 2-(4'-F--C.sub.6 H.sub.4)                                                  389 3-(2'-F--C.sub.6 H.sub.4)                                                  390 3-(3'-F--C.sub.6 H.sub.4)                                                  391 3-(4'-F--C.sub.6 H.sub.4)                                                  392 4-(2'-F--C.sub.6 H.sub.4)                                                  393 4-(3'-F--C.sub.6 H.sub.4)                                                  394 4-(4'-F--C.sub.6 H.sub.4)                                                  395 2-(2'-Cl--C.sub.6 H.sub.4)                                                 396 2-(3'-Cl--C.sub.6 H.sub.4)                                                 397 2-(4'-Cl--C.sub.6 H.sub.4)                                                 398 3-(2'-Cl--C.sub.6 H.sub.4)                                                 399 3-(3'-Cl--C.sub.6 H.sub.4)                                                 400 3-(4'-Cl--C.sub.6 H.sub.4)                                                 401 4-(2'-Cl--C.sub.6 H.sub.4)                                                 402 4-(3'-Cl--C.sub.6 H.sub.4)                                                 403 4-(4'-Cl--C.sub.6 H.sub.4)                                                 405 2-(2'-CH.sub.3 --C.sub.6 H.sub.4)                                          406 2-(3'-CH.sub.3 --C.sub.6 H.sub.4)                                          407 2-(4'-CH.sub.3 --C.sub.6 H.sub.4)                                          408 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)                                          409 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)                                          410 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)                                          411 4-(2'-CH.sub.3 --C.sub.6 H.sub.4)                                          412 4-(3'-CH.sub.3 --C.sub.6 H.sub.4)                                          413 4-(4'-CH.sub.3 --C.sub.6 H.sub.4)                                          414 2-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                      415 2-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                      416 2-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                      417 3-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                      418 3-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                      419 3-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                      420 4-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                      421 4-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                      422 4-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                      423 2-(2'-(CH.sub.3 --C(═NOAllyl))-C.sub.6 H.sub.4)                        424 2-(3'-(CH.sub.3 --C(═NOAllyl))-C.sub.6 H.sub.4)                        425 2-(4'-(CH.sub.3 --C(═NOAllyl))-C.sub.6 H.sub.4)                        426 3-(2'-(CH.sub.3 --C(═NOAllyl))-C.sub.6 H.sub.4)                        427 3-(3'-(CH.sub.3 --C(═NOAllyl))-C.sub.6 H.sub.4)                        428 3-(4'-(CH.sub.3 --C(═NOAllyl))-C.sub.6 H.sub.4)                        429 4-(2'-(CH.sub.3 --C(═NOAllyl))-C.sub.6 H.sub.4)                        430 4-(3'-(CH.sub.3 --C(═NOAllyl))-C.sub.6 H.sub.4)                        431 4-(4'-(CH.sub.3 --C(═NOAllyl))-C.sub.6 H.sub.4)                        432 2-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                                 433 2-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                                 434 2-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                                 435 3-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                                 436 3-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                                 437 3-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                                 438 4-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                                 439 4-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                                 440 4-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                                 441 2-(2'-CH.sub.3 O--C.sub.6 H.sub.4)                                         442 2-(3'-CH.sub.3 O--C.sub.6 H.sub.4)                                         443 2-(4'-CH.sub.3 O--C.sub.6 H.sub.4)                                         444 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)                                         445 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)                                         446 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)                                         447 4-(2'-CH.sub.3 O--C.sub.6 H.sub.4)                                         448 4-(3'-CH.sub.3 O--C.sub.6 H.sub.4)                                         449 4-(4'-CH.sub.3 O--C.sub.6 H.sub.4)                                         450 2-(2'-O.sub.2 N--C.sub.6 H.sub.4)                                          451 2-(3'-O.sub.2 N--C.sub.6 H.sub.4)                                          452 2-(4'-O.sub.2 N--C.sub.6 H.sub.4)                                          453 3-(2'-O.sub.2 N--C.sub.6 H.sub.4)                                          454 3-(3'-O.sub.2 N--C.sub.6 H.sub.4)                                          455 3-(4'-O.sub.2 N--C.sub.6 H.sub.4)                                          456 4-(2'-O.sub.2 N--C.sub.6 H.sub.4)                                          457 4-(3'-O.sub.2 N--C.sub.6 H.sub.4)                                          458 4-(4'-O.sub.2 N--C.sub.6 H.sub.4)                                          459 2-(2'-NC--C.sub.6 H.sub.4)                                                 460 2-(3'-NC--C.sub.6 H.sub.4)                                                 461 2-(4'-NC--C.sub.6 H.sub.4)                                                 462 3-(2'-NC--C.sub.6 H.sub.4)                                                 463 3-(3'-NC--C.sub.6 H.sub.4)                                                 464 3-(4'-NC--C.sub.6 H.sub.4)                                                 465 4-(2'-NC--C.sub.6 H.sub.4)                                                 466 4-(3'-NC--C.sub.6 H.sub.4)                                                 467 4-(4'-NC--C.sub.6 H.sub.4)                                                 468 2-(2'-CF.sub.3 --C.sub.6 H.sub.4)                                          469 2-(3'-CF.sub.3 --C.sub.6 H.sub.4)                                          470 2-(4'-CF.sub.3 --C.sub.6 H.sub.4)                                          471 3-(2'-CF.sub.3 --C.sub.6 H.sub.4)                                          472 3-(3'-CF.sub.3 --C.sub.6 H.sub.4)                                          473 3-(4'-CF.sub.3 --C.sub.6 H.sub.4)                                          474 4-(2'-CF.sub.3 --C.sub.6 H.sub.4)                                          475 4-(3'-CF.sub.3 --C.sub.6 H.sub.4)                                          476 4-(4'-CF.sub.3 --C.sub.6 H.sub.4)                                          477 2-O--C.sub.6 H.sub.5                                                       475 3-O--C.sub.6 H.sub.5                                                       476 4-O--C.sub.6 H.sub.5                                                       478 2-O-(2'-F--C.sub.6 H.sub.4)                                                479 2-O-(3'-F--C.sub.6 H.sub.4)                                                480 2-O-(4'-F--C.sub.6 H.sub.4)                                                481 3-O-(2'-F--C.sub.6 H.sub.4)                                                482 3-O-(3'-F--C.sub.6 H.sub.4)                                                483 3-O-(4'-F--C.sub.6 H.sub.4)                                                484 4-O-(2'-F--C.sub.6 H.sub.4)                                                485 4-O-(3'-F--C.sub.6 H.sub.4)                                                486 4-O-(4'-F--C.sub.6 H.sub.4)                                                487 2-O-(2'-Cl--C.sub.6 H.sub.4)                                               488 2-O-(3'-Cl--C.sub.6 H.sub.4)                                               489 2-O-(4'-Cl--C.sub.6 H.sub.4)                                               490 3-O-(2'-Cl--C.sub.6 H.sub.4)                                               491 3-O-(3'-Cl--C.sub.6 H.sub.4)                                               492 3-O-(4'-Cl--C.sub.6 H.sub.4)                                               493 3-O-(4'-Cl--C.sub.6 H.sub.4)                                               494 4-O-(2'-Cl--C.sub.6 H.sub.4)                                               495 4-O-(3'-Cl--C.sub.6 H.sub.4)                                               496 4-O-(4'-Cl--C.sub.6 H.sub.4)                                               497 2-O-(2'-CH.sub.3 --C.sub.6 H.sub.4)                                        498 2-O-(3'-CH.sub.3 --C.sub.6 H.sub.4)                                        499 2-O-(4'-CH.sub.3 --C.sub.6 H.sub.4)                                        500 3-O-(2'-CH.sub.3 --C.sub.6 H.sub.4)                                        501 3-O-(3'-CH.sub.3 --C.sub.6 H.sub.4)                                        502 3-O-(4'-CH.sub.3 --C.sub.6 H.sub.4)                                        503 4-O-(2'-CH.sub.3 --C.sub.6 H.sub.4)                                        504 4-O-(3'-CH.sub.3 --C.sub.6 H.sub.4)                                        505 4-O-(4'-CH.sub.3 --C.sub.6 H.sub.4)                                        506 2-O-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                    507 2-O-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                    508 2-O-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                    509 3-O-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                    510 3-O-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                    511 3-O-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                    512 4-O-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                    513 4-O-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                    514 4-O-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                    515 2-O-(2'-(CH.sub.3 --C(═NOAllyl))-C.sub.6 H.sub.4)                      516 2-O-(3'-(CH.sub.3 --C(═NOAllyl))-C.sub.6 H.sub.4)                      517 2-O-(4'-(CH.sub.3 --C(═NOAllyl))-C.sub.6 H.sub.4)                      518 3-O-(2'-(CH.sub.3 --C(═NOAllyl))-C.sub.6 H.sub.4)                      519 3-O-(3'-(CH.sub.3 --C(═NOAllyl))-C.sub.6 H.sub.4)                      520 3-O-(4'-(CH.sub.3 --C(═NOAllyl))-C.sub.6 H.sub.4)                      521 4-O-(2'-(CH.sub.3 --C(═NOAllyl))-C.sub.6 H.sub.4)                      522 4-O-(3'-(CH.sub.3 --C(═NOAllyl))-C.sub.6 H.sub.4)                      523 4-O-(4'-(CH.sub.3 --C(═NOAllyl))-C.sub.6 H.sub.4)                      524 2-O-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                               525 2-O-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                               526 2-O-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                               527 3-O-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                               528 3-O-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                               529 3-O-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                               530 4-O-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                               531 4-O-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                               532 4-O-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                               533 2-O-(2'-CH.sub.3 O--C.sub.6 H.sub.4)                                       534 2-O-(3'-CH.sub.3 O--C.sub.6 H.sub.4)                                       535 2-O-(4'-CH.sub.3 O--C.sub.6 H.sub.4)                                       536 3-O-(2'-CH.sub.3 O--C.sub.6 H.sub.4)                                       537 3-O-(3'-CH.sub.3 O--C.sub.6 H.sub.4)                                       538 3-O-(4'-CH.sub.3 O--C.sub.6 H.sub.4)                                       539 4-O-(2'-CH.sub.3 O--C.sub.6 H.sub.4)                                       540 4-O-(3'-CH.sub.3 O--C.sub.6 H.sub.4)                                       541 4-O-(4'-CH.sub.3 O--C.sub.6 H.sub.4)                                       542 2-O-(2'-O.sub.2 N--C.sub.6 H.sub.4)                                        543 2-O-(3'-O.sub.2 N--C.sub.6 H.sub.4)                                        544 2-O-(4'-O.sub.2 N--C.sub.6 H.sub.4)                                        545 3-O-(2'-O.sub.2 N--C.sub.6 H.sub.4)                                        546 3-O-(3'-O.sub.2 N--C.sub.6 H.sub.4)                                        547 3-O-(4'-O.sub.2 N--C.sub.6 H.sub.4)                                        548 4-O-(2'-O.sub.2 N--C.sub.6 H.sub.4)                                        549 4-O-(3'-O.sub.2 N--C.sub.6 H.sub.4)                                        550 4-O-(4'-O.sub.2 N--C.sub.6 H.sub.4)                                        551 2-O-(2'-NC--C.sub.6 H.sub.4)                                               552 2-O-(3'-NC--C.sub.6 H.sub.4)                                               553 2-O-(4'-NC--C.sub.6 H.sub.4)                                               554 3-O-(2'-NC--C.sub.6 H.sub.4)                                               555 3-O-(3'-NC--C.sub.6 H.sub.4)                                               556 3-O-(4'-NC--C.sub.6 H.sub.4)                                               557 4-O-(2'-NC--C.sub.6 H.sub.4)                                               558 4-O-(3'-NC--C.sub.6 H.sub.4)                                               559 4-O-(4'-NC--C.sub.6 H.sub.4)                                               560 2-O-(2'-CF.sub.3 --C.sub.6 H.sub.4)                                        561 2-O-(3'-CF.sub.3 --C.sub.6 H.sub.4)                                        562 2-O-(4'-CF.sub.3 --C.sub.6 H.sub.4)                                        563 3-O-(2'-CF.sub.3 --C.sub.6 H.sub.4)                                        564 3-O-(3'-CF.sub.3 --C.sub.6 H.sub.4)                                        565 3-O-(4'-CF.sub.3 --C.sub.6 H.sub.4)                                        566 4-O-(2'-CF.sub.3 --C.sub.6 H.sub.4)                                        567 4-O-(3'-CF.sub.3 --C.sub.6 H.sub.4)                                        568 4-O-(4'-CF.sub.3 --C.sub.6 H.sub.4)                                        569 2-Pyridinyl-2'                                                             570 2-Pyridinyl-3'                                                             571 2-Pyridinyl-4'                                                             572 3-Pyridinyl-2'                                                             573 3-Pyridinyl-3'                                                             574 3-Pyridinyl-4'                                                             575 4-Pyridinyl-2'                                                             576 4-Pyridinyl-3'                                                             577 4-Pyridinyl-4'                                                             578 2-Pyrimidinyl-2'                                                           579 2-Pyrimidinyl-3'                                                           580 2-Pyrimidinyl-4'                                                           581 3-Pyrimidinyl-2'                                                           582 3-Pyrimidinyl-3'                                                           583 3-Pyrimidinyl-4'                                                           584 4-Pyrimidinyl-2'                                                           585 4-Pyrimidinyl-3'                                                           586 4-Pyrimidinyl-4'                                                           587 2-Pyrazolyl-1'                                                             588 2-Pyrazolyl-3'                                                             589 2-Pyrazolyl-4'                                                             590 3-Pyrazolyl-1'                                                             591 3-Pyrazolyl-3'                                                             592 3-Pyrazolyl-4'                                                             593 4-Pyrazolyl-1'                                                             594 4-Pyrazolyl-3'                                                             595 4-Pyrazolyl-4'                                                             596 2-Isoxazolyl-3'                                                            597 2-Isoxazolyl-4'                                                            598 2-Isoxazolyl-5'                                                            599 3-Isoxazolyl-3'                                                            600 3-Isoxazolyl-4'                                                            601 3-Isoxazolyl-5'                                                            602 4-Isoxazolyl-3'                                                            603 4-Isoxazolyl-4'                                                            604 4-Isoxazolyl-5'                                                            605 2-Isothiazolyl-3'                                                          606 2-Isothiazolyl-4'                                                          607 2-Isothiazolyl-5'                                                          608 3-Isothiazolyl-3'                                                          609 3-Isothiazolyl-4'                                                          610 3-Isothiazolyl-5'                                                          611 4-Isothiazolyl-3'                                                          612 4-Isothiazolyl-4'                                                          613 4-Isothiazolyl-5'                                                          614 2-Imidazolyl-1'                                                            615 2-Imidazolyl-2'                                                            616 2-Imidazolyl-4'                                                            617 3-Imidazolyl-1'                                                            618 3-Imidazolyl-2'                                                            619 3-Imidazolyl-4'                                                            620 4-Imidazolyl-1'                                                            621 4-Imidazolyl-2'                                                            622 4-Imidazolyl-4'                                                            623 2-Oxazolyl-2'                                                              624 2-Oxazolyl-4'                                                              625 2-Oxazolyl-5'                                                              626 3-Oxazolyl-2'                                                              627 3-Oxazolyl-4'                                                              628 3-Oxazolyl-5'                                                              629 4-Oxazolyl-2'                                                              630 4-Oxazolyl-4'                                                              631 4-Oxazolyl-5'                                                              632 2-Thiazolyl-2'                                                             633 2-Thiazolyl-4'                                                             634 2-Thiazolyl-5'                                                             635 3-Thiazolyl-2'                                                             636 3-Thiazolyl-4'                                                             637 3-Thiazolyl-5'                                                             638 4-Thiazolyl-2'                                                             639 4-Thiazolyl-4'                                                             640 4-Thiazolyl-5'                                                             641 2-CH.sub.3 -4-(CH.sub.3 --C═N--O--CH.sub.2 --CH.sub.2 --OCH.sub.             3)                                                                       642 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C═N--O--CH.sub.2 --CH.sub.2                 --OCH.sub.3)                                                             643 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C═N--O--CH.sub.2 --CH.sub.2              --OCH.sub.3)                                                             644 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C═N--OCH.sub.3)                     645 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C═N--OC.sub.2 H.sub.5)                     646 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C═N--O-n-C.sub.3                   H.sub.7)                                                                 647 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C═N--O-i-C.sub.3 H.sub.7)                  648 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C═N--O-Allyl)                       649 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C═N--O-trans-Chloroall             yl)                                                                      650 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C═N--O-Propargyl)                   651 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C═N--O-n-C.sub.4 H.sub.9)                  652 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C═N--O--CH.sub.2                   --C.sub.6 H.sub.5)                                                       653 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C═N--OCH.sub.3)                     654 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C═N--OC.sub.2 H.sub.5)                     655 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C═N--O-n-C.sub.3                   H.sub.7)                                                                 656 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C═N--O-i-C.sub.3 H.sub.7)                  657 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C═N--O-Allyl)                       658 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C═N--O-trans-Chloroall             yl)                                                                      659 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C═N--O-Propargyl)                   660 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C═N--O-n-C.sub.4 H.sub.9)                  661 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C═N--O--CH.sub.2                   --C.sub.6 H.sub.5)                                                       662 2-O-n-C.sub.4 H.sub.9                                                      663 2-O-i-C.sub.4 H.sub.9                                                      664 2-O-s-C.sub.4 H.sub.9                                                      665 2-O-t-C.sub.4 H.sub.9                                                      666 2-Neopentyloxy                                                             667 3-O-n-C.sub.4 H.sub.9                                                      668 3-O-i-C.sub.4 H.sub.9                                                      669 3-O-s-C.sub.4 H.sub.9                                                      670 3-O-t-C.sub.4 H.sub.9                                                      671 3-Neopentyloxy                                                             672 4-O-n-C.sub.4 H.sub.9                                                      673 4-O-i-C.sub.4 H.sub.9                                                      674 4-O-s-C.sub.4 H.sub.9                                                      675 4-O-t-C.sub.4 H.sub.9                                                      676 4-Neopentyloxy                                                             677 3-CH.sub.3 -4-OCH.sub.3                                                    678 3-CH.sub.3 -4-OC.sub.2 H.sub.5                                             679 3-CH.sub.3 -4-O-n-C.sub.3 H.sub.7                                          680 3-CH.sub.3 -4-O-n-C.sub.4 H.sub.9                                          681 3-CH.sub.3 -4-O-i-C.sub.4 H.sub.9                                          682 3-CH.sub.3 -4-O-s-C.sub.4 H.sub.9                                          683 3-CH.sub.3 -4-O-t-C.sub.4 H.sub.9                                          684 3-CH.sub.3 -4-Neopentyloxy                                                 685 2-CH.sub.3 -3-OCH.sub.3                                                    686 2-CH.sub.3 -4-OCH.sub.3                                                    687 2-CH.sub.3 -5-OCH.sub.3                                                    688 2-CH.sub.3 -6-OCH.sub.3                                                    689 3-CH.sub.3 -4-OCH.sub.3                                                    690 3-CH.sub.3 -5-OCH.sub.3                                                    691 3-CH.sub.3 -6-OCH.sub.3                                                    692 4-CH.sub.3 -5-O--CH.sub.3                                                  693 4-CH.sub.3 -6-O--CH.sub.3                                                  694 4-CH.sub.3 -6-OCH.sub.3                                                    695 2-CH.sub.3 -3-O-i-C.sub.3 H.sub.7                                          696 2-CH.sub.3 -4-O-i-C.sub.3 H.sub.7                                          697 2-CH.sub.3 -5-O-i-C.sub.3 H.sub.7                                          698 2-CH.sub.3 -6-O-i-C.sub.3 H.sub.7                                          699 3-CH.sub.3 -4-O-i-C.sub.3 H.sub.7                                          700 3-CH.sub.3 -5-O-i-C.sub.3 H.sub.7                                          701 3-CH.sub.3 -6-O-i-C.sub.3 H.sub.7                                          702 4-CH.sub.3 -5-O-i-C.sub.3 H.sub.7                                          703 4-CH.sub.3 -6-O-i-C.sub.3 H.sub.7                                          704 5-CH.sub.3 -6-O-i-C.sub.3 H.sub.7                                          705 2-Cl-3-OCH.sub.3                                                           706 2-Cl-4-OCH.sub.3                                                           707 2-Cl-5-OCH.sub.3                                                           708 2-Cl-6-OCH.sub.3                                                           709 3-Cl-4-OCH.sub.3                                                           710 3-Cl-5-OCH.sub.3                                                           711 3-Cl-6-OCH.sub.3                                                           712 4-Cl-5-OCH.sub.3                                                           713 4-Cl-6-OCH.sub.3                                                           714 5-Cl-6-OCH.sub.3                                                         ______________________________________                                    

                  TABLE 4                                                          ______________________________________                                         1  STR26##                                                                       I: R.sup.1 = H                                                                 II: R.sup.1 = CH.sub.3                                                         III: R.sup.1 = Allyl                                                           IV: R.sup.1 = Propargyl                                                        V: R.sup.1 = S--CH.sub.3                                                       VI: R.sup.1 = CH.sub.2 --CN                                                    VII: R.sup.1 = CH.sub.2 --O--CH.sub.3                                          VIII: R.sup.1 = CO--OCH.sub.3                                                  No.        B                                                                 ______________________________________                                          1       Pyrrolyl-3                                                               2 N-CH.sub.3 -Pyrrolyl-3                                                       3 N-C.sub.6 H.sub.5 -Pyrrolyl-3                                                4 N-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrrolyl-3                                 5 N-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrrolyl-3                                 6 N-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrrolyl-3                                 7 N-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrrolyl-3                                8 N-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrrolyl-3                                9 N-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrrolyl-3                                10 N-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrrolyl-3                                11 N-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrrolyl-3                                12 N-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrrolyl-3                                13 N-(4'-CN--C.sub.6 H.sub.4)-Pyrrolyl-3                                       14 N-(3'-CN--C.sub.6 H.sub.4)-Pyrrolyl-3                                       15 N-(2'-CN--C.sub.6 H.sub.4)-Pyrrolyl-3                                       16 N-(4'-Cl--C.sub.6 H.sub.4)-Pyrrolyl-3                                       17 N-(3'-Cl--C.sub.6 H.sub.4)-Pyrrolyl-3                                       18 N-(2'-Cl--C.sub.6 H.sub.4)-Pyrrolyl-3                                       19 Pyrrolyl-2                                                                  20 N--CH.sub.3 -Pyrrolyl-2                                                     21 N--C.sub.6 H.sub.5 -Pyrrolyl-2                                              22 N-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrrolyl-2                                23 N-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrrolyl-2                                24 N-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrrolyl-2                                25 N-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrrolyl-2                               26 N-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrrolyl-2                               27 N-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrrolyl-2                               28 N-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrrolyl-2                                29 N-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrrolyl-2                                30 N-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrrolyl-2                                31 N-(4'-CN--C.sub.6 H.sub.4)-Pyrrolyl-2                                       32 N-(3'-CN--C.sub.6 H.sub.4)-Pyrrolyl-2                                       33 N-(2'-CN--C.sub.6 H.sub.4)-Pyrrolyl-2                                       34 N-(4'-Cl--C.sub.6 H.sub.4)-Pyrrolyl-2                                       35 N-(3'-Cl--C.sub.6 H.sub.4)-Pyrrolyl-2                                       36 N-(2'-Cl--C.sub.6 H.sub.4)-Pyrrolyl-2                                       37 Furyl-2                                                                     38 5-CH.sub.3 -Furyl-2                                                         39 5-C.sub.6 H.sub.5 -Furyl-2                                                  40 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Furyl-2                                   41 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Furyl-2                                   42 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Furyl-2                                   43 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Furyl-2                                  44 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Furyl-2                                  45 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Furyl-2                                  46 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Furyl-2                                   47 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Furyl-2                                   48 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Furyl-2                                   49 5-(4'-CN--C.sub.6 H.sub.4)-Furyl-2                                          50 5-(3'-CN--C.sub.6 H.sub.4)-Furyl-2                                          51 5-(2'-CN--C.sub.6 H.sub.4)-Furyl-2                                          52 5-(4'-Cl--C.sub.6 H.sub.4)-Furyl-2                                          53 5-(3'-Cl--C.sub.6 H.sub.4)-Furyl-2                                          54 5-(2'-Cl--C.sub.6 H.sub.4)-Furyl-2                                          55 4-CH.sub.3 -Furyl-2                                                         56 4-C.sub.6 H.sub.5 -Furyl-2                                                  57 4-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Furyl-2                                   58 4-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Furyl-2                                   59 4-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Furyl-2                                   60 4-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Furyl-2                                  61 4-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Furyl-2                                  62 4-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Furyl-2                                  63 4-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Furyl-2                                   64 4-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Furyl-2                                   65 4-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Furyl-2                                   66 4-(4'-CN--C.sub.6 H.sub.4)-Furyl-2                                          67 4-(3'-CN--C.sub.6 H.sub.4)-Furyl-2                                          68 4-(2'-CN--C.sub.6 H.sub.4)-Furyl-2                                          69 4-(4'-Cl--C.sub.6 H.sub.4)-Furyl-2                                          70 4-(3'-Cl--C.sub.6 H.sub.4)-Furyl-2                                          71 4-(2'-Cl--C.sub.6 H.sub.4)-Furyl-2                                          72 Thienyl-2                                                                   73 5-CH.sub.3 -Thienyl-2                                                       74 5-C.sub.6 H.sub.5 -Thienyl-2                                                75 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-2                                 76 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-2                                 77 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-2                                 78 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-2                                79 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-2                                80 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-2                                81 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-2                                 82 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-2                                 83 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-2                                 84 5-(4'-CN--C.sub.6 H.sub.4)-Thienyl-2                                        85 5-(3'-CN--C.sub.6 H.sub.4)-Thienyl-2                                        86 5-(2'-CN--C.sub.6 H.sub.4)-Thienyl-2                                        87 5-(4'-Cl--C.sub.6 H.sub.4)-Thienyl-2                                        88 5-(3'-Cl--C.sub.6 H.sub.4)-Thienyl-2                                        89 5-(2'-Cl--C.sub.6 H.sub.4)-Thienyl-2                                        90 4-CH.sub.3 -Thienyl-2                                                       91 4-C.sub.6 H.sub.5 -Thienyl-2                                                92 4-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-2                                 93 4-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-2                                 94 4-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-2                                 95 4-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-2                                96 4-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-2                                97 4-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-2                                98 4-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-2                                 99 4-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-2                                100 4-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-2                                101 4-(4'-CN--C.sub.6 H.sub.4)-Thienyl-2                                       102 4-(3'-CN--C.sub.6 H.sub.4)-Thienyl-2                                       103 4-(2'-CN--C.sub.6 H.sub.4)-Thienyl-2                                       104 4-(4'-Cl--C.sub.6 H.sub.4)-Thienyl-2                                       105 4-(3'-Cl--C.sub.6 H.sub.4)-Thienyl-2                                       106 4-(2'-Cl--C.sub.6 H.sub.4)-Thienyl-2                                       107 Thienyl-3                                                                  108 5-CH.sub.3 -Thienyl-3                                                      109 5-C.sub.6 H.sub.5 -Thienyl-3                                               110 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-3                                111 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-3                                112 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-3                                113 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-3                               114 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-3                               115 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-3                               116 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-3                                117 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-3                                118 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-3                                119 5-(4'-CN--C.sub.6 H.sub.4)-Thienyl-3                                       120 5-(3'-CN--C.sub.6 H.sub.4)-Thienyl-3                                       121 5-(2'-CN--C.sub.6 H.sub.4)-Thienyl-3                                       122 5-(4'-Cl--C.sub.6 H.sub.4)-Thienyl-3                                       123 5-(3'-Cl--C.sub.6 H.sub.4)-Thienyl-3                                       124 5-(2'-Cl--C.sub.6 H.sub.4)-Thienyl-3                                       125 Pyrazolyl-4                                                                126 N-CH.sub.3 -Pyrazolyl-4                                                    127 N-C.sub.6 H.sub.5 -Pyrazolyl-4                                             128 N-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrazolyl-4                              129 N-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrazolyl-4                              130 N-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrazolyl-4                              131 N-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrazolyl-4                             132 N-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrazolyl-4                             133 N-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrazolyl-4                             134 N-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrazolyl-4                              135 N-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrazolyl-4                              136 N-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrazolyl-4                              137 N-(4'-CN--C.sub.6 H.sub.4)-Pyrazolyl-4                                     138 N-(3'-CN--C.sub.6 H.sub.4)-Pyrazolyl-4                                     139 N-(2'-CN--C.sub.6 H.sub.4)-Pyrazolyl-4                                     140 N-(4'-Cl--C.sub.6 H.sub.4)-Pyrazolyl-4                                     141 N-(3'-Cl--C.sub.6 H.sub.4)-Pyrazolyl-4                                     142 N-(2'-Cl--C.sub.6 H.sub.4)-Pyrazolyl-4                                     143 3-CH.sub.3 -N-Methylpyrazolyl-4                                            144 3-C.sub.6 H.sub.5 -N-Methylpyrazolyl-4                                     145 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)-N-Methylpyrazolyl-4                      146 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)-N-Methylpyrazolyl-4                      147 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)-N-Methylpyrazolyl-4                      148 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-N-Methylpyrazolyl-4                     149 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-N-Methylpyrazolyl-4                     150 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-N-Methylpyrazolyl-4                     151 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)-N-Methylpyrazolyl-4                      152 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)-N-Methylpyrazolyl-4                      153 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)-N-Methylpyrazolyl-4                      154 3-(4'-CN--C.sub.6 H.sub.4)-N-Methylpyrazolyl-4                             155 3-(3'-CN--C.sub.6 H.sub.4)-N-Methylpyrazolyl-4                             156 3-(2'-CN--C.sub.6 H.sub.4)-N-Methylpyrazolyl-4                             157 3-(4'-Cl--C.sub.6 H.sub.4)-N-Methylpyrazolyl-4                             158 3-(3'-Cl--C.sub.6 H.sub.4)-N-Methylpyrazolyl-4                             159 3-(2'-Cl--C.sub.6 H.sub.4)-N-Methylpyrazolyl-4                             160 Isoxazolyl-5                                                               161 3-CH.sub.3 -Isoxazolyl-5                                                   162 3-C.sub.6 H.sub.5 -Isoxazolyl-5                                            163 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Isoxazolyl-5                             164 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Isoxazolyl-5                             165 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Isoxazolyl-5                             166 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Isoxazolyl-5                            167 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Isoxazolyl-5                            168 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Isoxazolyl-5                            169 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Isoxazolyl-5                             170 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Isoxazolyl-5                             171 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Isoxazolyl-5                             172 3-(4'-CN--C.sub.6 H.sub.4)-Isoxazolyl-5                                    173 3-(3'-CN--C.sub.6 H.sub.4)-Isoxazolyl-5                                    174 3-(2'-CN--C.sub.6 H.sub.4)-Isoxazolyl-5                                    175 3-(4'-Cl--C.sub.6 H.sub.4)-Isoxazolyl-5                                    176 3-(3'-Cl--C.sub.6 H.sub.4)-Isoxazolyl-5                                    177 3-(2'-Cl--C.sub.6 H.sub.4)-Isoxazolyl-5                                    178 4-Chloroisoxazolyl-5                                                       179 3-CH.sub.3 -4-Chloroisoxazolyl-5                                           180 3-C.sub.6 H.sub.5 -4-Chloroisoxazolyl-5                                    181 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                     182 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                     183 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                     184 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                    185 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                    186 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                    187 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                     188 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                     189 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                     190 3-(4'-CN--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                            191 3-(3'-CN--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                            192 3-(2'-CN--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                            193 3-(4'-Cl--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                            194 3-(3'-Cl--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                            195 3-(2'-Cl--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                            196 Isoxazolyl-3                                                               197 5-CH.sub.3 -Isoxazolyl-3                                                   198 5-C.sub.6 H.sub.5 -Isoxazolyl-3                                            199 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Isoxazolyl-3                             200 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Isoxazolyl-3                             201 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Isoxazolyl-3                             202 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Isoxazolyl-3                            203 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Isoxazolyl-3                            204 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Isoxazolyl-3                            205 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Isoxazolyl-3                             206 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Isoxazolyl-3                             207 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Isoxazolyl-3                             208 5-(4'-CN--C.sub.6 H.sub.4)-Isoxazolyl-3                                    209 5-(3'-CN--C.sub.6 H.sub.4)-Isoxazolyl-3                                    210 5-(2'-CN--C.sub.6 H.sub.4)-Isoxazolyl-3                                    211 5-(4'-Cl--C.sub.6 H.sub.4)-Isoxazolyl-3                                    212 5-(3'-Cl--C.sub.6 H.sub.4)-Isoxazolyl-3                                    213 5-(2'-Cl--C.sub.6 H.sub.4)-Isoxazolyl-3                                    214 Isothiazolyl-5                                                             215 3-CH.sub.3 -Isothiazolyl-5                                                 216 3-C.sub.6 H.sub.5 -Isothiazolyl-5                                          217 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Isothiazolyl-5                           218 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Isothiazolyl-5                           219 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Isothiazolyl-5                           220 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Isothiazolyl-5                          221 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Isothiazolyl-5                          222 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Isothiazolyl-5                          223 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Isothiazolyl-5                           224 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Isothiazolyl-5                           225 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Isothiazolyl-5                           226 3-(4'-CN--C.sub.6 H.sub.4)-Isothiazolyl-5                                  227 3-(3'-CN--C.sub.6 H.sub.4)-Isothiazolyl-5                                  228 3-(2'-CN--C.sub.6 H.sub.4)-Isothiazolyl-5                                  229 3-(4'-Cl--C.sub.6 H.sub.4)-Isothiazolyl-5                                  230 3-(3'-Cl--C.sub.6 H.sub.4)-Isothiazolyl-5                                  231 3-(2'-Cl--C.sub.6 H.sub.4)-Isothiazolyl-5                                  232 Oxazolyl-4                                                                 233 2-CH.sub.3 -Oxazolyl-4                                                     234 2-C.sub.6 H.sub.5 -Oxazolyl-4                                              235 2-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Oxazolyl-4                               236 2-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Oxazolyl-4                               237 2-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Oxazolyl-4                               238 2-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Oxazolyl-4                              239 2-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Oxazolyl-4                              240 2-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Oxazolyl-4                              241 2-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Oxazolyl-4                               242 2-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Oxazolyl-4                               243 2-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Oxazolyl-4                               244 2-(4'-CN--C.sub.6 H.sub.4)-Oxazolyl-4                                      245 2-(3'-CN--C.sub.6 H.sub.4)-Oxazolyl-4                                      246 2-(2'-CN--C.sub.6 H.sub.4)-Oxazolyl-4                                      247 2-(4'-Cl--C.sub.6 H.sub.4)-Oxazolyl-4                                      248 2-(3'-Cl--C.sub.6 H.sub.4)-Oxazolyl-4                                      249 2-(2'-Cl--C.sub.6 H.sub.4)-Oxazolyl-4                                      250 Thiazolyl-4                                                                251 2-CH.sub.3 -Thiazolyl-4                                                    252 2-C.sub.6 H.sub.5 -Thiazolyl-4                                             253 2-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Thiazolyl-4                              254 2-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Thiazolyl-4                              255 2-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Thiazolyl-4                              256 2-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Thiazolyl-4                             267 2-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Thiazolyl-4                             258 2-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Thiazolyl-4                             259 2-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Thiazolyl-4                              260 2-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Thiazolyl-4                              261 2-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Thiazolyl-4                              262 2-(4'-CN--C.sub.6 H.sub.4)-Thiazolyl-4                                     263 2-(3'-CN--C.sub.6 H.sub.4)-Thiazolyl-4                                     264 2-(2'-CN--C.sub.6 H.sub.4)-Thiazolyl-4                                     265 2-(4'-Cl--C.sub.6 H.sub.4)-Thiazolyl-4                                     266 2-(3'-Cl--C.sub.6 H.sub.4)-Thiazolyl-4                                     267 2-(2'-Cl--C.sub.6 H.sub.4)-Thiazolyl-4                                     268 N--CH.sub.3 -1,2,4-Triazolyl-5                                             269 3-CH.sub.3 --N--CH.sub.3 -1,2,4-Triazolyl-5                                270 3-C.sub.6 H.sub.5 -N--CH.sub.3 -1,2,4-Triazolyl-5                          271 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5                  272 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazo              lyl-5                                                                   273 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5                  274 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triaz              olyl-5                                                                  275 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5                 276 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triaz              olyl-5                                                                  277 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5                  278 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazo              lyl-5                                                                   279 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5                  280 3-(4'-CN--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5                 281 3-(3'-CN--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5                 282 3-(2'-CN--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5                 283 3-(4'-Cl--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5                 284 3-(3'-Cl--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5                 285 3-(2'-Cl--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5                 286 1,3,4-Oxadiazolyl-2                                                287 5-CH.sub.3 -1,3,4-Oxadiazolyl-2                                            288 5-C.sub.6 H.sub.5 -1,3,4-Oxadiazolyl-2                                     289 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                      290 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                      291 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                      292 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                     293 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                     294 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                     295 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                      296 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                      297 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                      298 5-(4'-CN--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                             299 5-(3'-CN--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                             300 5-(2'-CN--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                             301 5-(4'-Cl--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                             302 5-(3'-Cl--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                             303 5-(2'-Cl--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                             304 1,2,4-Oxadiazolyl-3                                                        305 5-CH.sub.3 -1,2,4-Oxadiazolyl-3                                            306 5-C.sub.6 H.sub.5 -1,2,4-Oxadiazolyl-3                                     307 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                      308 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                      309 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                      310 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                     311 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                     312 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                     313 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                      314 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                      315 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                      316 5-(4'-CN--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                             317 5-(3'-CN--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                             318 5-(2'-CN--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                             319 5-(4'-Cl--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                             320 5-(3'-Cl--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                             321 5-(2'-Cl--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                             322 1,2,4-Oxadiazolyl-5                                                        323 3-CH.sub.3 -1,2,4-Oxadiazolyl-5                                            324 3-C.sub.6 H.sub.5 -1,2,4-Oxadiazolyl-5                                     325 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                      326 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                      327 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                      328 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                     329 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                     330 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-dxadiazolyl-5                     331 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                      332 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                      333 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                      334 3-(4'-CN--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                             335 3-(3'-CN--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                             336 3-(2'-CN--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                             337 3-(4'-Cl--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                             338 3-(3'-Cl--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                             339 3-(2'-Cl--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                             340 1,2,4-Thiadiazolyl-3                                                       341 5-CH.sub.3 -1,2,4-Thiadiazolyl-3                                           342 5-C.sub.6 H.sub.5 -1,2,4-Thiadiazolyl-3                                    343 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                     344 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                     345 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                     346 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                    347 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                    348 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                    349 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                     350 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                     351 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                     352 5-(4'-CN--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                            353 5-(3'-CN--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                            354 5-(2'-CN--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                            355 5-(4'-Cl--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                            356 5-(3'-Cl--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                            357 5-(2'-Cl--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                            358 1,3,4-Thiadiazolyl-2                                                       359 5-CH.sub.3 -1,3,4-Thiadiazolyl-2                                           360 5-C.sub.6 H.sub.5 -1,3,4-Thiadiazolyl-2                                    361 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                     362 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                     363 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                     364 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                    365 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                    366 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                    367 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                     368 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                     369 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                     370 5-(4'-CN--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                            371 5-(3'-CN--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                            372 5-(2'-CN--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                            373 5-(4'-Cl--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                            374 5-(3'-Cl--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                            375 5-(2'-Cl--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                            376 Pyridinyl-2                                                                377 Pyridinyl-4                                                                378 Pyridazinyl-3                                                              379 Pyridazinyl-4                                                              380 Pyridazinyl-2                                                              381 Pyrimidinyl-4                                                              382 Pyrimidinyl-5                                                              383 Pyrimidinyl-2                                                              384 1-Naphthyl                                                                 385 2-Naphthyl                                                               ______________________________________                                    

                  TABLE 5                                                          ______________________________________                                         1  STR27##                                                                       I: R.sup.1 = H II: R.sup.1 = CH.sub.3 III: R.sup.1 = Allyl IV: R.sup.1       = Propargyl V: R.sup.1 = S--CH.sub.3 VI: R.sup.1 = CH.sub.2 --CN VII:          R.sup.1 = CH.sub.2 --O--CH.sub.3 VIII: R.sup.1 = CO--OCH.sub.3                   No.          X.sub.m                                                         ______________________________________                                         1          H                                                                     2 2-F                                                                          3 3-F                                                                          4 4-F                                                                          5 2,4-F.sub.2                                                                  6 2,4,6-F.sub.3                                                                7 2,3,4,5,6-F.sub.5                                                            8 2,3-F.sub.2                                                                  9 2-Cl                                                                         10 3-Cl                                                                        11 4-Cl                                                                        12 2,3-Cl.sub.2                                                                13 2,4-Cl.sub.2                                                                14 2,5-Cl.sub.2                                                                15 2,6-Cl.sub.2                                                                16 3,4-Cl.sub.2                                                                17 3,5-Cl.sub.2                                                                18 2,3,4-Cl.sub.3                                                              19 2,3,5-Cl.sub.3                                                              20 2,3,6-Cl.sub.3                                                              21 2,4,5-Cl.sub.3                                                              22 2,4,6-Cl.sub.3                                                              23 3,4,5-Cl.sub.3                                                              24 2,3,4,6-Cl.sub.4                                                            25 2,3,5,6-Cl.sub.4                                                            26 2,3,4,5,6-Cl.sub.5                                                          27 2-Br                                                                        28 3-Br                                                                        29 4-Br                                                                        30 2,4-Br.sub.2                                                                31 2,5-Br.sub.2                                                                32 2,6-Br.sub.2                                                                33 2,4,6-Br.sub.3                                                              34 2,3,4,5,6-Br.sub.5                                                          35 2-I                                                                         36 3-I                                                                         37 4-I                                                                         38 2,4-I.sub.2                                                                 39 2-Cl, 3-F                                                                   40 2-Cl, 4-F                                                                   41 2-Cl, 5-F                                                                   42 2-Cl, 6-F                                                                   43 2-Cl, 3-Br                                                                  44 2-Cl, 4-Br                                                                  45 2-Cl, 5-Br                                                                  46 2-Cl, 6-Br                                                                  47 2-Br, 3-Cl                                                                  48 2-Br, 4-Cl                                                                  49 2-Br, 5-Cl                                                                  50 2-Br, 3-F                                                                   51 2-Br, 4-F                                                                   52 2-Br, 5-F                                                                   53 2-Br, 6-F                                                                   54 2-F, 3-Cl                                                                   55 2-F, 4-Cl                                                                   56 2-F, 5-Cl                                                                   57 3-Cl, 4-F                                                                   58 3-Cl, 5-F                                                                   59 3-Cl, 4-Br                                                                  60 3-Cl, 5-Br                                                                  61 3-F, 4-Cl                                                                   62 3-F, 4-Br                                                                   63 3-Br, 4-Cl                                                                  64 3-Br, 4-F                                                                   65 2,6-Cl.sub.2, 4-Br                                                          66 2-CH.sub.3                                                                  67 3-CH.sub.3                                                                  68 4-CH.sub.3                                                                  69 2,3-(CH.sub.3).sub.2                                                        70 2,4-(CH.sub.3).sub.2                                                        71 2,5-(CH.sub.3).sub.2                                                        72 2,6-(CH.sub.3).sub.2                                                        73 3,4-(CH.sub.3).sub.2                                                        74 3,5-(CH.sub.3).sub.2                                                        75 2,3,5-(CH.sub.3).sub.3                                                      76 2,3,4-(CH.sub.3).sub.3                                                      77 2,3,6-(CH.sub.3).sub.3                                                      78 2,4,5-(CH.sub.3).sub.3                                                      79 2,4,6-(CH.sub.3).sub.3                                                      80 3,4,5-(CH.sub.3).sub.3                                                      81 2,3,4,6-(CH.sub.3).sub.4                                                    82 2,3,5,6-(CH.sub.3).sub.4                                                    83 2,3,4,5,6-(CH.sub.3).sub.5                                                  84 2-C.sub.2 H.sub.5                                                           85 3-C.sub.2 H.sub.5                                                           86 4-C.sub.2 H.sub.5                                                           87 2,4-(C.sub.2 H.sub.5).sub.2                                                 88 2,6-(C.sub.2 H.sub.5).sub.2                                                 89 3,5-(C.sub.2 H.sub.5).sub.2                                                 90 2,4,6-(C.sub.2 H.sub.5).sub.3                                               91 2-n-C.sub.3 H.sub.7                                                         92 3-n-C.sub.3 H.sub.7                                                         93 4-n-C.sub.3 H.sub.7                                                         94 2-i-C.sub.3 H.sub.7                                                         95 3-i-C.sub.3 H.sub.7                                                         96 4-i-C.sub.3 H.sub.7                                                         97 2,4-(i-C.sub.3 H.sub.7).sub.2                                               98 2,6-(i-C.sub.3 H.sub.7).sub.2                                               99 3,5-(i-C.sub.3 H.sub.7).sub.2                                               100 2,4,6-(i-C.sub.3 H.sub.7).sub.3                                            101 2-s-C.sub.4 H.sub.9                                                        102 3-s-C.sub.4 H.sub.9                                                        103 4-s-C.sub.4 H.sub.9                                                        104 2-t-C.sub.4 H.sub.9                                                        105 3-t-C.sub.4 H.sub.9                                                        106 4-t-C.sub.4 H.sub.9                                                        107 2,3-(t-C.sub.4 H.sub.9).sub.2                                              108 2,4-(t-C.sub.4 H.sub.9).sub.2                                              109 2,5-(t-C.sub.4 H.sub.9).sub.2                                              110 2,6-(t-C.sub.4 H.sub.9).sub.2                                              111 3,4-(t-C.sub.4 H.sub.9).sub.2                                              112 2,4,6-(t-C.sub.4 H.sub.9).sub.3                                            113 4-n-C.sub.9 H.sub.19                                                       114 4-n-C.sub.12 H.sub.25                                                      115 4-n-C.sub.15 H.sub.31                                                      116 4-(1,1,3,3-Tetramethylbutyl)                                               117 4-(2,4,4-Trimethylpropyl)                                                  118 2-t-C.sub.4 H.sub.9, 4-CH.sub.3                                            119 2-t-C.sub.4 H.sub.9, 5-CH.sub.3                                            120 2,6-(t-C.sub.4 H.sub.9).sub.2, 4-CH.sub.3                                  121 2-CH.sub.3, 4-t-C.sub.4 H.sub.9                                            122 2-CH.sub.3, 6-t-C.sub.4 H.sub.9                                            123 2-CH.sub.3, 4-i-C.sub.3 H.sub.7                                            124 2-CH.sub.3, 5-i-C.sub.3 H.sub.7                                            125 3-CH.sub.3, 4-i-C.sub.3 H.sub.7                                            126 2-i-C.sub.3 H.sub.7, 5-CH.sub.3                                            127 2,4-(t-C.sub.4 H.sub.9).sub.2, 6-i-C.sub.3 H.sub.7                         128 2-Allyl                                                                    129 3-Allyl                                                                    130 4-Allyl                                                                    131 2-Allyl, 6-CH.sub.3                                                        132 2-cyclo-C.sub.6 H.sub.11                                                   133 3-cyclo-C.sub.6 H.sub.11                                                   134 4-cyclo-C.sub.6 H.sub.11                                                   135 2,4-(cyclo-C.sub.6 H.sub.11).sub.2, 6-CH.sub.3                             136 2-CH.sub.3, 4-cyclo-C.sub.6 H.sub.11                                       137 2-CH.sub.2 --C.sub.6 H.sub.5                                               138 3-CH.sub.2 --C.sub.6 H.sub.5                                               139 4-CH.sub.2 --C.sub.6 H.sub.5                                               140 2-CH.sub.2 --C.sub.6 H.sub.5, 4-CH.sub.3                                   141 2-CH.sub.3, 4-CH.sub.2 --C.sub.6 H.sub.5                                   142 2-C.sub.6 H.sub.5                                                          143 3-C.sub.6 H.sub.5                                                          144 4-C.sub.6 H.sub.5                                                          145 4-(2-i-C.sub.3 H.sub.7 --C.sub.6 H.sub.4)                                  146 4-C.sub.6 H.sub.5, 2,6-(CH.sub.3).sub.2                                    147 2-Cl, 4-C.sub.6 H.sub.5                                                    148 2-Br, 4-C.sub.6 H.sub.5                                                    149 2-C.sub.6 H.sub.5, 4-Cl                                                    150 2-C.sub.6 H.sub.5, 4-Br                                                    151 2-CH.sub.2 C.sub.6 H.sub.5, 4-Cl                                           152 2-CH.sub.2 C.sub.6 H.sub.5, 4-Br                                           153 2-Cl, 4-CH.sub.2 C.sub.6 H.sub.5                                           154 2-Br, 4-CH.sub.2 C.sub.6 H.sub.5                                           155 2-cyclo-C.sub.6 H.sub.11, 4-Cl                                             156 2-cyclo-C.sub.6 H.sub.11, 4-Br                                             157 2-Cl, 4-cyclo-C.sub.6 H.sub.11                                             158 2-Br, 4-cyclo-C.sub.6 H.sub.11                                             159 2-OCH.sub.3                                                                160 3-OCH.sub.3                                                                161 4-OCH.sub.3                                                                162 2-OC.sub.2 H.sub.5                                                         163 3-O--C.sub.2 H.sub.5                                                       164 4-O--C.sub.2 H.sub.5                                                       165 2-O-n-C.sub.3 H.sub.7                                                      166 3-O-n-C.sub.3 H.sub.7                                                      167 4-O-n-C.sub.3 H.sub.7                                                      168 2-O-i-C.sub.3 H.sub.7                                                      169 3-O-i-C.sub.3 H.sub.7                                                      170 4-O-i-C.sub.3 H.sub.7                                                      171 2-O-n-C.sub.6 H.sub.13                                                     172 3-O-n-C.sub.6 H.sub.13                                                     173 4-O-n-C.sub.6 H.sub.13                                                     174 2-O-n-C.sub.8 H.sub.17                                                     175 3-O-n-C.sub.8 H.sub.17                                                     176 4-O-n-C.sub.8 H.sub.17                                                     177 2-O--CH.sub.2 C.sub.6 H.sub.5                                              178 3-O--CH.sub.2 C.sub.6 H.sub.5                                              179 4-O--CH.sub.2 C.sub.6 H.sub.5                                              180 2-O--(CH.sub.2).sub.3 C.sub.6 H.sub.5                                      181 3-O--(CH.sub.2).sub.3 C.sub.6 H.sub.5                                      182 4-O--(CH.sub.2).sub.3 C.sub.6 H.sub.5                                      183 2,4-(OCH.sub.3).sub.2                                                      184 2-CF.sub.3                                                                 185 3-CF.sub.3                                                                 186 4-CF.sub.3                                                                 187 2-OCF.sub.3                                                                188 3-OCF.sub.3                                                                189 4-OCF.sub.3                                                                190 3-OCH.sub.2 CHF.sub.2                                                      191 2-NO.sub.2                                                                 192 3-NO.sub.2                                                                 193 4-NO.sub.2                                                                 194 2-CN                                                                       195 3-CN                                                                       196 4-CN                                                                       197 2-CH.sub.3, 3-Cl                                                           198 2-CH.sub.3, 4-Cl                                                           199 2-CH.sub.3, 5-Cl                                                           200 2-CH.sub.3, 6-Cl                                                           201 2-CH.sub.3, 3-F                                                            202 2-CH.sub.3, 4-F                                                            203 2-CH.sub.3, 5-F                                                            204 2-CH.sub.3, 6-F                                                            205 2-CH.sub.3, 3-Br                                                           206 2-CH.sub.3, 4-Br                                                           207 2-CH.sub.3, 5-Br                                                           208 2-CH.sub.3, 6-Br                                                           209 2-Cl, 3-CH.sub.3                                                           210 2-Cl, 4-CH.sub.3                                                           211 2-Cl, 5-CH.sub.3                                                           212 2-F, 3-CH.sub.3                                                            213 2-F, 4-CH.sub.3                                                            214 2-F, 5-CH.sub.3                                                            215 2-Br, 3-CH.sub.3                                                           216 2-Br, 4-CH.sub.3                                                           217 2-Br, 5-CH.sub.3                                                           218 3-CH.sub.3, 4-Cl                                                           219 3-CH.sub.3, 5-Cl                                                           220 3-CH.sub.3, 4-F                                                            221 3-CH.sub.3, 5-F                                                            222 3-CH.sub.3, 4-Br                                                           223 3-CH.sub.3, 5-Br                                                           224 3-F, 4-CH.sub.3                                                            225 3-Cl, 4-CH.sub.3                                                           226 3-Br, 4-CH.sub.3                                                           227 2-Cl, 4,5-(CH.sub.3).sub.2                                                 228 2-Br, 4,5-(CH.sub.3).sub.2                                                 229 2-Cl, 3,5-(CH.sub.3).sub.2                                                 230 2-Br, 3,5-(CH.sub.3).sub.2                                                 231 2,6-Cl.sub.2, 4-CH.sub.3                                                   232 2,6-F.sub.2, 4-CH.sub.3                                                    233 2,6-Br.sub.2, 4-CH.sub.3                                                   234 2,4-Br.sub.2, 6-CH.sub.3                                                   235 2,4-F.sub.2, 6-CH.sub.3                                                    236 2,4-Br.sub.2, 6-CH.sub.3                                                   237 2,6-(CH.sub.3).sub.2, 4-F                                                  238 2,6-(CH.sub.3).sub.2, 4-Cl                                                 239 2,6-(CH.sub.3).sub.2, 4-Br                                                 240 3,5-(CH.sub.3).sub.2, 4-F                                                  241 3,5-(CH.sub.3).sub.2, 4-Cl                                                 242 3,5-(CH.sub.3).sub.2, 4-Br                                                 243 2,3,6-(CH.sub.3).sub.3, 4-F                                                244 2,3,6-(CH.sub.3).sub.3, 4-Cl                                               245 2,3,6-(CH.sub.3).sub.3, 4-Br                                               246 2,4-(CH.sub.3).sub.2, 6-F                                                  247 2,4-(CH.sub.3).sub.2, 6-Cl                                                 248 2,4-(CH.sub.3).sub.2, 6-Br                                                 249 2-i-C.sub.3 H.sub.7, 4-Cl, 5-CH.sub.3                                      250 2-Cl, 4-NO.sub.2                                                           251 2-NO.sub.2, 4-Cl                                                           252 2-OCH.sub.3, 5-NO.sub.2                                                    253 2,4-Cl.sub.2, 5-NO.sub.2                                                   254 2,4-Cl.sub.2, 6-NO.sub.2                                                   255 2,6-Cl.sub.2, 4-NO.sub.2                                                   256 2,6-Br.sub.2, 4-NO.sub.2                                                   257 2,6-I.sub.2, 4-NO.sub.2                                                    258 2-CH.sub.3, 5-i-C.sub.3 H.sub.7, 4-Cl                                      259 2-CO.sub.2 CH.sub.3                                                        260 3-CO.sub.2 CH.sub.3                                                        261 4-CO.sub.2 CH.sub.3                                                        262 2-CO.sub.2 (C.sub.2 H.sub.5)                                               263 3-CO.sub.2 (C.sub.2 H.sub.5)                                               264 4-CO.sub.2 (C.sub.2 H.sub.5)                                               265 2-CO.sub.2 (n-C.sub.3 H.sub.7)                                             266 3-CO.sub.2 (n-C.sub.3 H.sub.7)                                             267 4-CO.sub.2 (n-C.sub.3 H.sub.7)                                             268 2-CO.sub.2 (i-C.sub.3 H.sub.7)                                             269 3-CO.sub.2 (i-C.sub.3 H.sub.7)                                             270 4-CO2(i-C.sub.3 H.sub.7)                                                   271 2-CO.sub.2 (n-C.sub.6 H.sub.13)                                            272 3-CO.sub.2 (n-C.sub.6 H.sub.13)                                            273 4-CO.sub.2 (n-C.sub.6 H.sub.13)                                            274 2-CH.sub.2 --CCH.sub.3                                                     275 3-CH.sub.2 --OCH.sub.3                                                     276 4-CH.sub.2 --OCH.sub.3                                                     277 2-CH.sub.2 O(C.sub.2 H.sub.5)                                              278 3-CH.sub.2 O(C.sub.2 H.sub.5)                                              279 4-CH.sub.2 O(C.sub.2 H.sub.5)                                              280 2-CH.sub.2 O(n-C.sub.3 H.sub.7)                                            281 3-CH.sub.2 O(n-C.sub.3 H.sub.7)                                            282 4-CH.sub.2 O(n-C.sub.3 H.sub.7)                                            283 2-CH.sub.2 O(i-C.sub.3 H.sub.7)                                            284 3-CH.sub.2 O(i-C.sub.3 H.sub.7)                                            285 4-CH.sub.2 O(i-C.sub.3 H.sub.7)                                            286 2-CHO                                                                      287 3-CHO                                                                      288 4-CHO                                                                      289 2-CO--CH.sub.3                                                             290 3-CO--CH.sub.3                                                             291 4-CO--CH.sub.3                                                             292 2-CO--CH.sub.2 --CH.sub.3                                                  293 3-CO--CH.sub.2 --CH.sub.3                                                  294 4-CO--CH.sub.2 --CH.sub.3                                                  295 2-CO--CH.sub.2 --CH.sub.2 --CH.sub.3                                       296 3-CO--CH.sub.2 --CH.sub.2 --CH.sub.3                                       297 4-CO--CH.sub.2 --CH.sub.2 --CH.sub.3                                       298 2-CO--CH(CH.sub.3)-CH.sub.3                                                299 3-CO--CH(CH.sub.3)-CH.sub.3                                                300 4-CO--CH(CH.sub.3)-CH.sub.3                                                301 2-Me-4-CHO                                                                 302 2-Me-4-CH.sub.3 --CO                                                       303 2-Me-4-CH.sub.3 --CH.sub.2 --CO                                            304 2-Me-4-CH.sub.3 --CH.sub.2 --CH.sub.2 --CO                                 305 2-Me-4-CH.sub.3 --CH(CH.sub.3)-CO                                          306 2,5-Me.sub.2 -4-CHO                                                        307 2,5-Me.sub.2 -4-CH.sub.3 --CO                                              308 2,5-Me.sub.2 -4-CH.sub.3 --CH.sub.2 --CO                                   309 2,5-Me.sub.2 -4-CH.sub.3 --CH.sub.2 --CH.sub.2 --CO                        310 2,5-Me.sub.2 -4-CH.sub.3 --CH(CH.sub.3)-CO                                 311 2-Cl-4-CHO                                                                 312 2-Cl-4-CH.sub.3 --CO                                                       313 2-Cl-4-CH.sub.3 --CH.sub.2 --CO                                            314 2-Cl-4-CH.sub.3 --CH(CH.sub.3)-CO                                          315 2,5-Cl.sub.2 -4-CHO                                                        316 2,5-Cl.sub.2 -4-CH.sub.3 --CO                                              317 2,5-Cl.sub.2 -4-CH.sub.3 --CH.sub.2 --CO                                   318 2,5-Cl.sub.2 -4-CH.sub.3 --CH.sub.2 --CH.sub.2 --CO                        319 2,5-Cl.sub.2 -4-CH.sub.3 ----CH(CH.sub.3)-CO                               320 2-C(═NOCH.sub.3)-CH.sub.3                                              321 3-C(═NOCH.sub.3)-CH.sub.3                                              322 4-C(═NOCH.sub.3)-CH.sub.3                                              323 2-C(═NOC.sub.2 H.sub.5)-CH.sub.3                                       324 3-C(═NOC.sub.2 H.sub.5)-CH.sub.3                                       325 4-C(═NOC.sub.2 H.sub.5)-CH.sub.3                                       326 2-C(═NO-n-C.sub.3 H.sub.7)-CH.sub.3                                    327 3-C(═NO-n-C.sub.3 H.sub.7)-CH.sub.3                                    328 4-C(═NO-n-C.sub.3 H.sub.7)-CH.sub.3                                    329 2-C(═NO-i-C.sub.3 H.sub.7)-CH.sub.3                                    330 3-C(═NO-i-C.sub.3 H.sub.7)-CH.sub.3                                    331 4-C(═NO-i-C.sub.3 H.sub.7)-CH.sub.3                                    332 2-C(═NO-Allyl)-CH.sub.3                                                333 3-C(═NO-Allyl)-CH.sub.3                                                334 4-C(═NO-Allyl)-CH.sub.3                                                335 2-C(═NO-trans-Chloroallyl)-CH.sub.3                                    336 3-C(═NO-trans-Chloroallyl)-CH.sub.3                                    337 4-C(═NO-trans-Chloroallyl)-CH.sub.3                                    338 2-C(═NO-Propargyl)-CH.sub.3                                            339 3-C(═NO-Proparoyl)-CH.sub.3                                            340 4-C(═NO-Propargyl)-CH.sub.3                                            341 2-C(═NO-n-C.sub.4 H.sub.9)-CH.sub.3                                    342 3-C(═NO-n-C.sub.4 H.sub.9)-CH.sub.3                                    343 4-C(═NO-n-C.sub.4 H.sub.9)-CH.sub.3                                    344 2-C(═NO--CH.sub.2 --C.sub.6 H.sub.5)-CH.sub.3                          345 3-C(═NO--CH.sub.2 --C.sub.6 H.sub.5)-CH.sub.3                          346 4-C(═NO--CH.sub.2 --C.sub.6 H.sub.5)-CH.sub.3                          347 2-CH.sub.3 -4-CH═NOCH.sub.3                                            348 2-CH.sub.3 -4-CH═NOC.sub.2 H.sub.5                                     349 2-CH.sub.3 -4-CH═NO-n-C.sub.3 H.sub.7                                  350 2-CH.sub.3 -4-CH═NO-i-C.sub.3 H.sub.7                                  351 2-CH.sub.3 -4-CH═NO-Allyl                                              352 2-CH.sub.3 -4-CH═NO-(trans-Chloroallyl)                                353 2-CH.sub.3 -4-CH═NO-Propargyl                                          354 2-CH.sub.3 -4-CH═NO-n-C.sub.4 H.sub.9                                  355 2-CH.sub.3 -4-CH═NO--CH.sub.2 --C.sub.6 H.sub.5                        356 2-CH.sub.3 -4-(CH.sub.3 --C═NOCH.sub.3)                                357 2-CH.sub.3 -4-(CH.sub.3 --C═NOC.sub.2 H.sub.5)                         358 2-CH.sub.3 -4-(CH.sub.3 --C═NO-n-C.sub.3 H.sub.7)                      359 2-CH.sub.3 -4-(CH.sub.3 --C═NO-i-C.sub.3 H.sub.7)                      360 2-CH.sub.3 -4-(CH.sub.3 --C═NO-Allyl)                                  361 2-CH.sub.3 -4-(CH.sub.3 --C═NO-trans-Chloroallyl)                      362 2-CH.sub.3 -4-(CH.sub.3 --C═NO-Propargyl)                              363 2-CH.sub.3 -4-(CH.sub.3 --C═NO-n-C.sub.4 H.sub.9)                      364 2-CH.sub.3 -4-(CH.sub.3 --C═NO--CH.sub.2 --C.sub.6 H.sub.5)                      365 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C═NO--CH.sub.3)                       366 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C═NO--C.sub.2                        H.sub.5)                                                              367 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C═NO-n-C.sub.3 H.sub.7)                         368 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C═NO-i-C.sub.3                       H.sub.7                                                               369 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C═NO-Allyl)                           370 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C═NO-trans-Chloroal-                   lyl)                                                                          371 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C═NO-Propargyl)                       372 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C═NO-n-C.sub.4 H.sub.9)                         373 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C═NO--CH.sub.2                       --C.sub.6 H.sub.5)                                                    374 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C═NOCH.sub.3)                      375 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C═NOC.sub.2 H.sub.5)                         376 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C═NO-n-C.sub.3                    H.sub.7)                                                              377 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C═NO-i-C.sub.3 H.sub.7)                      378 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C═NO-Allyl)                        379 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C═NO-trans-Chloro-        allyl)                                                                        380 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C═NO-Proparyl)                     381 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C═NO-n-C.sub.4 H.sub.9)                      382 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C═NO--CH.sub.2                    --C.sub.6 H.sub.5)                                                    383 2-C.sub.6 H.sub.5                                                          384 3-C.sub.6 H.sub.5                                                          385 4-C.sub.6 H.sub.5                                                          386 2-(2'-F--C.sub.6 H.sub.4)                                                  387 2-(3'-F--C.sub.6 H.sub.4)                                                  388 2-(4'-F--C.sub.6 H.sub.4)                                                  389 3-(2'-F--C.sub.6 H.sub.4)                                                  390 3-(3'-F--C.sub.6 H.sub.4)                                                  391 3-(4'-F--C.sub.6 H.sub.4)                                                  392 4-(2'-F--C.sub.6 H.sub.4)                                                  393 4-(3'-F--C.sub.6 H.sub.4)                                                  394 4-(4'-F--C.sub.6 H.sub.4)                                                  395 2-(2'-Cl--C.sub.6 H.sub.4)                                                 396 2-(3'-Cl--C.sub.6 H.sub.4)                                                 397 2-(4'-Cl--C.sub.6 H.sub.4)                                                 398 3-(2'-Cl--C.sub.6 H.sub.4)                                                 399 3-(3'-Cl--C.sub.6 H.sub.4)                                                 400 3-(4'-Cl--C.sub.6 H.sub.4)                                                 401 4-(2'-Cl--C.sub.6 H.sub.4)                                                 402 4-(3'-Cl--C.sub.6 H.sub.4)                                                 403 4-(4'-Cl--C.sub.6 H.sub.4)                                                 405 2-(2'-CH.sub.3 --C.sub.6 H.sub.4)                                          406 2-(3'-CH.sub.3 --C.sub.6 H.sub.4)                                          407 2-(4'-CH.sub.3 --C.sub.6 H.sub.4)                                          408 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)                                          409 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)                                          410 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)                                          411 4-(2'-CH.sub.3 --C.sub.6 H.sub.4)                                          412 4-(3'-CH.sub.3 --C.sub.6 H.sub.4)                                          413 4-(4'-CH.sub.3 --C.sub.6 H.sub.4)                                          414 2-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                      415 2-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                      416 2-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                      417 3-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                      418 3-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                      419 3-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                      420 4-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                      421 4-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                      422 4-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                      423 2-(2'-(CH.sub.3 --C(═NOAllyl))-C.sub.6 H.sub.4)                        424 2-(3'-(CH.sub.3 --C(═NOAllyl))-C.sub.6 H.sub.4)                        425 2-(4'-(CH.sub.3 --C(═NOAllyl))-C.sub.6 H.sub.4)                        426 3-(2'-(CH.sub.3 --C(═NOAllyl))-C.sub.6 H.sub.4)                        427 3-(3'-(CH.sub.3 --C(═NOAllyl))-C.sub.6 H.sub.4)                        428 3-(4'-(CH.sub.3 --C(═NOAllyl))-C.sub.6 H.sub.4)                        429 4-(2'-(CH.sub.3 --C(═NOAllyl))-C.sub.6 H.sub.4)                        430 4-(3'-(CH.sub.3 --C(═NOAllyl))-C.sub.6 H.sub.4)                        431 4-(4'-(CH.sub.3 --C(═NOAllyl))-C.sub.6 H.sub.4)                        432 2-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                                 433 2-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                                 434 2-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                                 435 3-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                                 436 3-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                                 437 3-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                                 438 4-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                                 439 4-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                                 440 4-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                                 441 2-(2'-CH.sub.3 O--C.sub.6 H.sub.4)                                         442 2-(3'-CH.sub.3 O--C.sub.6 H.sub.4)                                         443 2-(4'-CH.sub.3 O--C.sub.6 H.sub.4)                                         444 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)                                         445 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)                                         446 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)                                         447 4-(2'-CH.sub.3 O--C.sub.6 H.sub.4)                                         448 4-(3'-CH.sub.3 O--C.sub.6 H.sub.4)                                         449 4-(4'-CH.sub.3 O--C.sub.6 H.sub.4)                                         450 2-(2'-O.sub.2 N--C.sub.6 H.sub.4)                                          451 2-(3'-O.sub.2 N--C.sub.6 H.sub.4)                                          452 2-(4'-O.sub.2 N--C.sub.6 H.sub.4)                                          453 3-(2'-O.sub.2 N--C.sub.6 H.sub.4)                                          454 3-(3'-O.sub.2 N--C.sub.6 H.sub.4)                                          455 3-(4'-O.sub.2 N--C.sub.6 H.sub.4)                                          456 4-(2'-O.sub.2 N--C.sub.6 H.sub.4)                                          457 4-(3'-O.sub.2 N--C.sub.6 H.sub.4)                                          458 4-(4'-O.sub.2 N--C.sub.6 H.sub.4)                                          459 2-(2'-NC--C.sub.6 H.sub.4)                                                 460 2-(3'-NC--C.sub.6 H.sub.4)                                                 461 2-(4'-NC--C.sub.6 H.sub.4)                                                 462 3-(2'-NC--C.sub.6 H.sub.4)                                                 463 3-(3'-NC--C.sub.6 H.sub.4)                                                 464 3-(4'-NC--C.sub.6 H.sub.4)                                                 465 4-(2'-NC--C.sub.6 H.sub.4)                                                 466 4-(3'-NC--C.sub.6 H.sub.4)                                                 467 4-(4'-NC--C.sub.6 H.sub.4)                                                 468 2-(2'-CF.sub.3 --C.sub.6 H.sub.4)                                          469 2-(3'-CF.sub.3 --C.sub.6 H.sub.4)                                          470 2-(4'-CF.sub.3 --C.sub.6 H.sub.4)                                          471 3-(2'-CF.sub.3 --C.sub.6 H.sub.4)                                          472 3-(3'-CF.sub.3 --C.sub.6 H.sub.4)                                          473 3-(4'-CF.sub.3 --C.sub.6 H.sub.4)                                          474 4-(2'-CF.sub.3 --C.sub.6 H.sub.4)                                          475 4-(3'-CF.sub.3 --C.sub.6 H.sub.4)                                          476 4-(4'-CF.sub.3 --C.sub.6 H.sub.4)                                          477 2-O--C.sub.6 H.sub.5                                                       475 3-O--C.sub.6 H.sub.5                                                       476 4-O--C.sub.6 H.sub.5                                                       478 2-O-(2'-F--C.sub.6 H.sub.4)                                                479 2-O-(3'-F--C.sub.6 H.sub.4)                                                480 2-O-(4'-F--C.sub.6 H.sub.4)                                                481 3-O-(2'-F--C.sub.6 H.sub.4)                                                482 3-O-(3'-F--C.sub.6 H.sub.4)                                                483 3-O-(4'-F--C.sub.6 H.sub.4)                                                484 4-O-(2'-F--C.sub.6 H.sub.4)                                                485 4-O-(3'-F--C.sub.6 H.sub.4)                                                486 4-O-(4'-F--C.sub.6 H.sub.4)                                                487 2-O-(2'-Cl--C.sub.6 H.sub.4)                                               488 2-O-(3'-Cl--C.sub.6 H.sub.4)                                               489 2-O-(4'-Cl--C.sub.6 H.sub.4)                                               490 3-O-(2'-Cl--C.sub.6 H.sub.4)                                               491 3-O-(3'-Cl--C.sub.6 H.sub.4)                                               492 3-O-(4'-Cl--C.sub.6 H.sub.4)                                               493 3-O-(4'-Cl--C.sub.6 H.sub.4)                                               494 4-O-(2'-Cl--C.sub.6 H.sub.4)                                               495 4-O-(3'-Cl--C.sub.6 H.sub.4)                                               496 4-O-(4'-Cl--C.sub.6 H.sub.4)                                               497 2-O-(2'-CH.sub.3 --C.sub.6 H.sub.4)                                        498 2-O-(3'-CH.sub.3 --C.sub.6 H.sub.4)                                        499 2-O-(4'-CH.sub.3 --C.sub.6 H.sub.4)                                        500 3-O-(2'-CH.sub.3 --C.sub.6 H.sub.4)                                        501 3-O-(3'-CH.sub.3 --C.sub.6 H.sub.4)                                        502 3-O-(4'-CH.sub.3 --C.sub.6 H.sub.4)                                        503 4-O-(2'-CH.sub.3 --C.sub.6 H.sub.4)                                        504 4-O-(3'-CH.sub.3 --C.sub.6 H.sub.4)                                        505 4-O-(4'-CH.sub.3 --C.sub.6 H.sub.4)                                        506 2-O-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                    507 2-O-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                    508 2-O-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                    509 3-O-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                    510 3-O-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                    511 3-O-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                    512 4-O-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                    513 4-O-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                    514 4-O-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                    515 2-O-(2'-(CH.sub.3 --C(═NOAllyl))-C.sub.6 H.sub.4)                      516 2-O-(3'-(CH.sub.3 --C(═NOAllyl))-C.sub.6 H.sub.4)                      517 2-O-(4'-(CH.sub.3 --C(═NOAllyl))-C.sub.6 H.sub.4)                      518 3-O-(2'-(CH.sub.3 --C(═NOAllyl))-C.sub.6 H.sub.4)                      519 3-O-(3'-(CH.sub.3 --C(═NOAllyl))-C.sub.6 H.sub.4)                      520 3-O-(4'-(CH.sub.3 --C(═NcAllyl))-C.sub.6 H.sub.4)                      521 4-O-(2'-(CH.sub.3 --C(═NOAllyl))-C.sub.6 H.sub.4)                      522 4-O-(3'-(CH.sub.3 --C(═NOAllyl))-C.sub.6 H.sub.4)                      523 4-O-(4'-(CH.sub.3 --C(═NOAllyl))-C.sub.6 H.sub.4)                      524 2-O-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                               525 2-O-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                               526 2-O-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                               527 3-O-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                               528 3-O-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                               529 3-O-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                               530 4-O-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                               531 4-O-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                               532 4-O-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                               533 2-O-(2'-CH.sub.3 O--C.sub.6 H.sub.4)                                       534 2-O-(3'-CH.sub.3 O--C.sub.6 H.sub.4)                                       535 2-O-(4'-CH.sub.3 O--C.sub.6 H.sub.4)                                       536 3-O-(2'-CH.sub.3 O--C.sub.6 H.sub.4)                                       537 3-O-(3'-CH.sub.3 O--C.sub.6 H.sub.4)                                       538 3-O-(4'-CH.sub.3 O--C.sub.6 H.sub.4)                                       539 4-O-(2'-CH.sub.3 O--C.sub.6 H.sub.4)                                       540 4-O-(3'-CH.sub.3 O--C.sub.6 H.sub.4)                                       541 4-O-(4'-CH.sub.3 O--C.sub.6 H.sub.4)                                       542 2-O-(2'-O.sub.2 N--C.sub.6 H.sub.4)                                        543 2-O-(3'-O.sub.2 N--C.sub.6 H.sub.4)                                        544 2-O-(4'-O.sub.2 N--C.sub.6 H.sub.4)                                        545 3-O-(2'-O.sub.2 N--C.sub.6 H.sub.4)                                        546 3-O-(3'-O.sub.2 N--C.sub.6 H.sub.4)                                        547 3-O-(4'-O.sub.2 N--C.sub.6 H.sub.4)                                        548 4-O-(2'-O.sub.2 N--C.sub.6 H.sub.4)                                        549 4-O-(3'-O.sub.2 N--C.sub.6 H.sub.4)                                        550 4-O-(4'-O.sub.2 N--C.sub.6 H.sub.4)                                        551 2-O-(2'-NC--C.sub.6 H.sub.4)                                               552 2-O-(3'-NC--C.sub.6 H.sub.4)                                               553 2-O-(4'-NC--C.sub.6 H.sub.4)                                               554 3-O-(2'-NC--C.sub.6 H.sub.4)                                               555 3-O-(3'-NC--C.sub.6 H.sub.4)                                               556 3-O-(4'-NC--C.sub.6 H.sub.4)                                               557 4-O-(2'-NC--C.sub.6 H.sub.4)                                               558 4-O-(3'-NC--C.sub.6 H.sub.4)                                               559 4-O-(4'-NC--C.sub.6 H.sub.4)                                               560 2-O-(2'-CF.sub.3 --C.sub.6 H.sub.5)                                        561 2-O-(3'-CF.sub.3 --C.sub.6 H.sub.5)                                        562 2-O-(4'-CF.sub.3 --C.sub.6 H.sub.5)                                        563 3-O-(2'-CF.sub.3 --C.sub.6 H.sub.5)                                        564 3-O-(3'-CF.sub.3 --C.sub.6 H.sub.5)                                        565 3-O-(4'-CF.sub.3 --C.sub.6 H.sub.5)                                        566 4-O-(2'-CF.sub.3 --C.sub.6 H.sub.5)                                        567 4-O-(3'-CF.sub.3 --C.sub.6 H.sub.5)                                        568 4-O-(4'-CF.sub.3 --C.sub.6 H.sub.5)                                        569 2-Pyridinyl-2'                                                             570 2-Pyridinyl-3'                                                             571 2-Pyridinyl-4'                                                             572 3-Pyridinyl-2'                                                             573 3-Pyridinyl-3'                                                             574 3-Pyridinyl-4'                                                             575 4-Pyridinyl-2'                                                             576 4-Pyridinyl-3'                                                             577 4-Pyridinyl-4'                                                             578 2-Pyrimidinyl-2'                                                           579 2-Pyrimidinyl-3'                                                           580 2-Pyrimidinyl-4'                                                           581 3-Pyrimidinyl-2'                                                           582 3-Pyrimidinyl-3'                                                           583 3-Pyrimidinyl-4'                                                           584 4-Pyrimidinyl-2'                                                           585 4-Pyrimidinyl-3'                                                           586 4-Pyrimidinyl-4'                                                           587 2-Pyrazolyl-1'                                                             588 2-Pyrazolyl-3'                                                             589 2-Pyrazolyl-4'                                                             590 3-Pyrazolyl-1'                                                             591 3-Pyrazolyl-3'                                                             592 3-Pyrazolyl-4'                                                             593 4-Pyrazolyl-1'                                                             594 4-Pyrazolyl-3'                                                             595 4-Pyrazolyl-4'                                                             596 2-Isoxazolyl-3'                                                            597 2-Isoxazolyl-4'                                                            598 2-Isoxazolyl-5'                                                            599 3-Isoxazolyl-3'                                                            600 3-Isoxazolyl-4'                                                            601 3-Isoxazolyl-5'                                                            602 4-Isoxazolyl-3'                                                            603 4-Isoxazolyl-4'                                                            604 4-Isoxazolyl-5'                                                            605 2-Isothiazolyl-3'                                                          606 2-Isothiazolyl-4'                                                          607 2-Isothiazolyl-5'                                                          608 3-Isothiazolyl-3'                                                          609 3-Isothiazolyl-4'                                                          610 3-Isothiazolyl-5'                                                          611 4-Isothiazolyl-3'                                                          612 4-Isothiazolyl-4'                                                          613 4-Isothiazolyl-5'                                                          614 2-Imidazolyl-1'                                                            615 2-Imidazolyl-2'                                                            616 2-Imidazolyl-4'                                                            617 3-Imidazolyl-1'                                                            618 3-Imidazolyl-2'                                                            619 3-Imidazolyl-4'                                                            620 4-Imidazolyl-1'                                                            621 4-Imidazolyl-2'                                                            622 4-Imidazolyl-4'                                                            623 2-Oxazolyl-2'                                                              624 2-Oxazolyl-4'                                                              625 2-Oxazolyl-5'                                                              626 3-Oxazolyl-2'                                                              627 3-Oxazolyl-4'                                                              628 3-Oxazolyl-5'                                                              629 4-Oxazolyl-2'                                                              630 4-Oxazolyl-4'                                                              631 4-Oxazolyl-5'                                                              632 2-Thiazolyl-2'                                                             633 2-Thiazolyl-4'                                                             634 2-Thiazolyl-5'                                                             635 3-Thiazolyl-2'                                                             636 3-Thiazolyl-4'                                                             637 3-Thiazolyl-5'                                                             638 4-Thiazolyl-2'                                                             639 4-Thiazolyl-4'                                                             640 4-Thiazolyl-5'                                                           ______________________________________                                    

                  TABLE 6                                                          ______________________________________                                         1  STR28##                                                                        -        I: R.sup.1 = H                                                       II: R.sup.1 = CH.sub.3                                                         III: R.sup.1 = Allyl                                                           IV: R.sup.1 = Propargyl                                                        V: R.sup.1 = S--CH.sub.3                                                       VI: R.sup.1 = CH.sub.2 --CN                                                    VII: R.sup.1 = CH.sub.2 --O--CH.sub.3                                          VIII: R.sup.1 = CO--OCH.sub.3                                                No        B                                                                    ______________________________________                                          1        Pyrrolyl-3                                                              2 N-CH.sub.3 -Pyrrolyl-3                                                       3 N-C.sub.6 H.sub.5 -Pyrrolyl-3                                                4 N-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrrolyl-3                                 5 N-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrrolyl-3                                 6 N-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrrolyl-3                                 7 N-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrrolyl-3                                8 N-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrrolyl-3                                9 N-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrrolyl-3                                10 N-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrrolyl-3                                11 N-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrrolyl-3                                12 N-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrrolyl-3                                13 N-(4'-CN--C.sub.6 H.sub.4)-Pyrrolyl-3                                       14 N-(3'-CN--C.sub.6 H.sub.4)-Pyrrolyl-3                                       15 N-(2'-CN--C.sub.6 H.sub.4)-Pyrrolyl-3                                       16 N-(4'-Cl--C.sub.6 H.sub.4)-Pyrrolyl-3                                       17 N-(3'-Cl--C.sub.6 H.sub.4)-Pyrrolyl-3                                       18 N-(2'-Cl--C.sub.6 H.sub.4)-Pyrrolyl-3                                       19 Pyrrolyl-2                                                                  20 N-CH.sub.3 -Pyrrolyl-2                                                      21 N-C.sub.6 H.sub.5 -Pyrrolyl-2                                               22 N-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrrolyl-2                                23 N-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrrolyl-2                                24 N-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrrolyl-2                                25 N-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrrolyl-2                               26 N-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrrolyl-2                               27 N-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrrolyl-2                               28 N-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrrolyl-2                                29 N-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrrolyl-2                                30 N-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrrolyl-2                                31 N-(4'-CN--C.sub.6 H.sub.4)-Pyrrolyl-2                                       32 N-(3'-CN--C.sub.6 H.sub.4)-Pyrrolyl-2                                       33 N-(2'-CN--C.sub.6 H.sub.4)-Pyrrolyl-2                                       34 N-(4'-Cl--C.sub.6 H.sub.4)-Pyrrolyl-2                                       35 N-(3'-Cl--C.sub.6 H.sub.4)-Pyrrolyl-2                                       36 N-(2'-Cl--C.sub.6 H.sub.4)-Pyrrolyl-2                                       37 Furyl-2                                                                     38 5-CH.sub.3 -Furyl-2                                                         39 5-C.sub.6 H.sub.5 -Furyl-2                                                  40 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Furyl-2                                   41 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Furyl-2                                   42 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Furyl-2                                   43 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Furyl-2                                  44 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Furyl-2                                  45 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Furyl-2                                  46 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Furyl-2                                   47 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Furyl-2                                   48 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Furyl-2                                   49 5-(4'-CN--C.sub.6 H.sub.4)-Furyl-2                                          50 5-(3'-CN--C.sub.6 H.sub.4)-Furyl-2                                          51 5-(2'-CN--C.sub.6 H.sub.4)-Furyl-2                                          52 5-(4'-Cl--C.sub.6 H.sub.4)-Furyl-2                                          53 5-(3'-Cl--C.sub.6 H.sub.4)-Furyl-2                                          54 5-(2'-Cl--C.sub.6 H.sub.4)-Furyl-2                                          55 4-CH.sub.3 -Furyl-2                                                         56 4-C.sub.6 H.sub.5 -Furyl-2                                                  57 4-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Furyl-2                                   58 4-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Furyl-2                                   59 4-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Furyl-2                                   60 4-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Furyl-2                                  61 4-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Furyl-2                                  62 4-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Furyl-2                                  63 4-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Furyl-2                                   64 4-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Furyl-2                                   65 4-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Furyl-2                                   66 4-(4'-CN--C.sub.6 H.sub.4)-Furyl-2                                          67 4-(3'-CN--C.sub.6 H.sub.4)-Furyl-2                                          68 4-(2'-CN--C.sub.6 H.sub.4) Furyl-2                                          69 4-(4'-Cl--C.sub.6 H.sub.4)-Furyl-2                                          70 4-(3'-Cl--C.sub.6 H.sub.4)-Furyl-2                                          71 4-(2'-Cl--C.sub.6 H.sub.4)-Furyl-2                                          72 Thienyl-2                                                                   73 5-CH.sub.3 -Thienyl-2                                                       74 5-C.sub.6 H.sub.5 -Thienyl-2                                                75 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-2                                 76 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-2                                 77 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-2                                 78 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-2                                79 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-2                                80 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-2                                81 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-2                                 82 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-2                                 83 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-2                                 84 5-(4'-CN--C.sub.6 H.sub.4)-Thienyl-2                                        85 5-(3'-CN--C.sub.6 H.sub.4)-Thienyl-2                                        86 5-(2'-CN--C.sub.6 H.sub.4)-Thienyl-2                                        87 5-(4'-Cl--C.sub.6 H.sub.4)-Thienyl-2                                        88 5-(3'-Cl--C.sub.6 H.sub.4)-Thienyl-2                                        89 5-(2'-Cl--C.sub.6 H.sub.4)-Thienyl-2                                        90 4-CH.sub.3 -Thienyl-2                                                       91 4-C.sub.6 H.sub.5 -Thienyl-2                                                92 4-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-2                                 93 4-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-2                                 94 4-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-2                                 95 4-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-2                                96 4-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-2                                97 4-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-2                                98 4-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-2                                 99 4-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-2                                100 4-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-2                                101 4-(4'-CN--C.sub.6 H.sub.4)-Thienyl-2                                       102 4-(3'-CN--C.sub.6 H.sub.4)-Thienyl-2                                       103 4-(2'-CN--C.sub.6 H.sub.4)-Thienyl-2                                       104 4-(4'-Cl--C.sub.6 H.sub.4)-Thienyl-2                                       105 4-(3'-Cl--C.sub.6 H.sub.4)-Thienyl-2                                       106 4-(2'-Cl--C.sub.6 H.sub.4)-Thienyl-2                                       107 Thienyl-3                                                                  108 5-CH.sub.3 -Thienyl-3                                                      109 5-C.sub.6 H.sub.5 -Thienyl-3                                               110 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-3                                111 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-3                                112 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-3                                113 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-3                               114 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-3                               115 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-3                               116 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-3                                117 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-3                                118 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-3                                119 5-(4'-CN--C.sub.6 H.sub.4)-Thienyl-3                                       120 5-(3'-CN--C.sub.6 H.sub.4)-Thienyl-3                                       121 5-(2'-CN--C.sub.6 H.sub.4)-Thienyl-3                                       122 5-(4'-Cl--C.sub.6 H.sub.4)-Thienyl-3                                       123 5-(3'-Cl--C.sub.6 H.sub.4)-Thienyl-3                                       124 5-(2'-Cl--C.sub.6 H.sub.4)-Thienyl-3                                       125 Pyrazolyl-4                                                                126 N-CH.sub.3 -Pyrazolyl-4                                                    127 N-C.sub.6 H.sub.5 -Pyrazolyl-4                                             128 N-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrazolyl-4                              129 N-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrazolyl-4                              130 N-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrazolyl-4                              131 N-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrazolyl-4                             132 N-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrazolyl-4                             133 N-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrazolyl-4                             134 N-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrazolyl-4                              135 N-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrazolyl-4                              136 N-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrazolyl-4                              137 N-(4'-CN--C.sub.6 H.sub.4)-Pyrazolyl-4                                     138 N-(3'-CN--C.sub.6 H.sub.4)-Pyrazolyl-4                                     139 N-(2'-CN--C.sub.6 H.sub.4)-Pyrazolyl-4                                     140 N-(4'-Cl--C.sub.6 H.sub.4)-Pyrazolyl-4                                     141 N-(3'-Cl--C.sub.6 H.sub.4)-Pyrazolyl-4                                     142 N-(2'-Cl--C.sub.6 H.sub.4)-Pyrazolyl-4                                     143 3-CH.sub.3 --N-Methylpyrazolyl-4                                           144 3-C.sub.6 H.sub.5 --N-Methylpyrazolyl-4                                    145 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)--N-Methylpyrazolyl-4                     146 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)--N-Methylpyrazolyl-4                     147 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)--N-Methylpyrazolyl-4                     148 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)--N-Methylpyrazolyl-4                    149 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)--N-Methylpyrazolyl-4                    150 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)--N-Methylpyrazolyl-4                    151 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)--N-Methylpyrazolyl-4                     152 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)--N-Methylpyrazolyl-4                     153 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)--N-Methylpyrazolyl-4                     154 3-(4'-CN--C.sub.6 H.sub.4)--N-Methylpyrrazolyl-4                           155 3-(3'-CN--C.sub.6 H.sub.4)--N-Methylpyrazolyl-4                            156 3-(2'-CN--C.sub.6 H.sub.4)--N-Methylpyrazolyl-4                            157 3-(4'-Cl--C.sub.6 H.sub.4)--N-Methylpyrazolyl-4                            158 3-(3'-Cl--C.sub.6 H.sub.4)--N-Methylpyrazolyl-4                            159 3-(2'-Cl--C.sub.6 H.sub.4)--N-Methylpyrazolyl-4                            160 Isoxazolyl-5                                                               161 3-CH.sub.3 -Isoxazolyl-5                                                   162 3-C.sub.6 H.sub.5 -Isoxazolyl-5                                            163 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Isoxazolyl-5                             164 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Isoxazolyl-5                             165 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Isoxazolyl-5                             166 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Isoxazolyl-5                            167 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Isoxazolyl-5                            168 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Isoxazolyl-5                            169 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Isoxazolyl-5                             170 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Isoxazolyl-5                             171 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Isoxazolyl-5                             172 3-(4'-CN--C.sub.6 H.sub.4)-Isoxazolyl-5                                    173 3-(3'-CN--C.sub.6 H.sub.4)-Isoxazolyl-5                                    174 3-(2'-CN--C.sub.6 H.sub.4)-Isoxazolyl-5                                    175 3-(4'-Cl--C.sub.6 H.sub.4)-Isoxazolyl-5                                    176 3-(3'-Cl--C.sub.6 H.sub.4)-Isoxazolyl-5                                    177 3-(2'-Cl--C.sub.6 H.sub.4)-Isoxazolyl-5                                    178 4-Chloroisoxazolyl-5                                                       179 3-CH.sub.3 -4-Chloroisoxazolyl-5                                           180 3-C.sub.6 H.sub.5 -4-Chloroisoxazolyl-5                                    181 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                     182 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                     183 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                     184 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                    185 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                    186 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                    187 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                     188 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                     189 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                     190 3-(4'-CN--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                            191 3-(3'-CN--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                            192 3-(2'-CN--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                            193 3-(4'-Cl--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                            194 3-(3'-Cl--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                            195 3-(2'-Cl--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                            196 Isoxazolyl-3                                                               197 5-CH.sub.3 -Isoxazolyl-3                                                   198 5-C.sub.6 H.sub.5 -Isoxazolyl-3                                            199 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Isoxazolyl-3                             200 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Isoxazolyl-3                             201 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Isoxazolyl-3                             202 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Isoxazolyl-3                            203 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Isoxazolyl-3                            204 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Isoxazolyl-3                            205 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Isoxazolyl-3                             206 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Isoxazolyl-3                             207 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Isoxazolyl-3                             208 5-(4'-CN--C.sub.6 H.sub.4)-Isoxazolyl-3                                    209 5-(3'-CN--C.sub.6 H.sub.4)-Isoxazolyl-3                                    210 5-(2'-CN--C.sub.6 H.sub.4)-Isoxazolyl-3                                    211 5-(4'-Cl--C.sub.6 H.sub.4)-Isoxazolyl-3                                    212 5-(3'-Cl--C.sub.6 H.sub.4)-Isoxazolyl-3                                    213 5-(2'-Cl--C.sub.6 H.sub.4)-Isoxazolyl-3                                    214 Isothiazolyl-5                                                             215 3-CH.sub.3 -Isothiazolyl-5                                                 216 3-C.sub.6 H.sub.5 -Isothiazolyl-5                                          217 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Isothiazolyl-5                           218 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Isothiazolyl-5                           219 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Isothiazolyl-5                           220 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Isothiazolyl-5                          221 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Isothiazolyl-5                          222 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Isothiazolyl-5                          223 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Isothiazolyl-5                           224 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Isothiazolyl-5                           225 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Isothiazolyl-5                           226 3-(4'-CN--C.sub.6 H.sub.4)-Isothiazolyl-5                                  227 3-(3'-CN--C.sub.6 H.sub.4)-Isothiazolyl-5                                  228 3-(2'-CN--C.sub.6 H.sub.4)-Isothiazolyl-5                                  229 3-(4'-Cl--C.sub.6 H.sub.4)-Isothiazolyl-5                                  230 3-(3'-Cl--C.sub.6 H.sub.4)-Isothiazolyl-5                                  231 3-(2'-Cl--C.sub.6 H.sub.4)-Isothiazolyl-5                                  232 Oxazolyl-4                                                                 233 2-CH.sub.3 -Oxazolyl-4                                                     234 2-C.sub.6 H.sub.5 -Oxazolyl-4                                              235 2-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Oxazolyl-4                               236 2-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Oxazolyl-4                               237 2-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Oxazolyl-4                               238 2-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Oxazolyl-4                              239 2-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Oxazolyl-4                              240 2-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Oxazolyl-4                              241 2-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Oxazolyl-4                               242 2-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Oxazolyl-4                               243 2-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Oxazolyl-4                               244 2-(4'-CN--C.sub.6 H.sub.4)-Oxazolyl-4                                      245 2-(3'-CN--C.sub.6 H.sub.4)-Oxazolyl-4                                      246 2-(2'-CN--C.sub.6 H.sub.4)-Oxazolyl-4                                      247 2-(4'-Cl--C.sub.6 H.sub.4)-Oxazolyl-4                                      248 2-(3'-Cl--C.sub.6 H.sub.4)-Oxazolyl-4                                      249 2-(2'-Cl--C.sub.6 H.sub.4)-Oxazolyl-4                                      250 Thiazolyl-4                                                                251 2-CH.sub.3 -Thiazolyl-4                                                    252 2-C.sub.6 H.sub.5 -Thiazolyl-4                                             253 2-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Thiazolyl-4                              254 2-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Thiazolyl-4                              255 2-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Thiazolyl-4                              256 2-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Thiazolyl-4                             267 2-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Thiazolyl-4                             258 2-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Thiazolyl-4                             259 2-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Thiazolyl-4                              260 2-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Thiazolyl-4                              261 2-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Thiazolyl-4                              262 2-(4'-CN--C.sub.6 H.sub.4)-Thiazolyl-4                                     263 2-(3'-CN--C.sub.6 H.sub.4)-Thiazolyl-4                                     264 2-(2'-CN--C.sub.6 H.sub.4)-Thiazolyl-4                                     265 2-(4'-Cl--C.sub.6 H.sub.4)-Thiazolyl-4                                     266 2-(3'-Cl--C.sub.6 H.sub.4)-Thiazolyl-4                                     267 2-(2'-Cl--C.sub.6 H.sub.4)-Thiazolyl-4                                     268 N-CH.sub.3 -1,2,4-Triazolyl-5                                              269 3-CH.sub.3 --N--CH.sub.3 -1,2,4-Triazolyl-5                                270 3-C.sub.6 H.sub.5 --N--CH.sub.3 -1,2,4-Triazolyl-5                         271 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5                   272 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triaz               olyl-5                                                                 273 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5                   274 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Tria               zolyl-5                                                                275 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5                  276 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Tria               zolyl-5                                                                277 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5                   278 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triaz               olyl-5                                                                 279 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5                   280 3-(4'-CN--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5        281 3-(3'-CN--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5                 282 3-(2'-CN--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5                 283 3-(4'-Cl--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5                 284 3-(3'-Cl--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5                 285 3-(2'-Cl--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5                 286 1,3,4-Oxadiazolyl-2                                                        287 5-CH.sub.3 -1,3,4-Oxadiazolyl-2                                            288 5-C.sub.6 H.sub.5 -1,3,4-Oxadiazolyl-2                                     289 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                      290 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                      291 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                      292 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                     293 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                     294 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                     295 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                      296 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                      297 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                      298 5-(4'-CN--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                             299 5-(3'-CN--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                             300 5-(2'-CN--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                             301 5-(4'-Cl--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                             302 5-(3'-Cl--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                             303 5-(2'-Cl--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                             304 1,2,4-Oxadiazolyl-3                                                        305 5-CH.sub.3 -1,2,4-Oxadiazolyl-3                                            306 5-C.sub.6 H.sub.5 -1,2,4-Oxadiazolyl-3                                     307 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                      308 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                      309 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                      310 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                     311 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                     312 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                     313 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                      314 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                      315 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                      316 5-(4'-CN--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                             317 5-(3'-CN--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                             318 5-(2'-CN--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                             319 5-(4'-Cl--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                             320 5-(3'-Cl--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                             321 5-(2'-Cl--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                             322 1,2,4-Oxadiazolyl-5                                                        323 3-CH.sub.3 -1,2,4-Oxadiazolyl-5                                            324 3-C.sub.6 H.sub.5 -1,2,4-Oxadiazolyl-5                                     325 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                      326 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                      327 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                      328 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Oxadazolyl-5                      329 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                     330 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                     331 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                      332 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                      333 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                      334 3-(4'-CN--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                             335 3-(3'-CN--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                             336 3-(2'-CN--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                             337 3-(4'-Cl--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                             338 3-(3'-Cl--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                             339 3-(2'-Cl--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                             340 1,2,4-Thiadiazolyl-3                                                       341 5-CH.sub.3 -1,2,4-Thiadiazolyl-3                                           342 5-C.sub.6 H.sub.5 -1,2,4-Thiadiazolyl-3                                    343 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                     344 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                     345 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                     346 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                    347 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                    348 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                    349 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                     350 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                     351 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                     352 5-(4'-CN--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                            353 5-(3'-CN--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                            354 5-(2'-CN--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                            355 5-(4'-Cl--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                            356 5-(3'-Cl--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                            357 5-(2'-Cl--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                            358 1,3,4-Thiadiazolyl-2                                                       359 5-CH.sub.3 -1,3,4-Thiadiazolyl-2                                           360 5-C.sub.6 H.sub.5 -1,3,4-Thiadiazolyl-2                                    361 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                     362 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                     363 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                     364 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                    365 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                    366 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                    367 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                     368 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                     369 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                     370 5-(4'-CN--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                            371 5-(3'-CN--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                            372 5-(2'-CN--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                            373 5-(4'-Cl--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                            374 5-(3'-Cl--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                            375 5-(2'-Cl--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                            376 Pyridinyl-2                                                                377 Pyridinyl-4                                                                378 Pyridazinyl-3                                                              379 Pyridazinyl-4                                                              380 Pyridazinyl-2                                                              381 Pyrimidinyl-4                                                              382 Pyrimidinyl-5                                                              383 Pyrimidinyl-2                                                            ______________________________________                                    

                                      TABLE 7                                      __________________________________________________________________________     Selected physical data of some compounds                                       No.                                                                               Compound                          mp/° C.                                                                     IR/cm.sup.-1                          __________________________________________________________________________        1                                                                                                                    1  -- 1707, 1484, 1457, 1447,                                                  1303, 1277                               -  2                                                                                                                 2  -- 1708, 1495, 1457, 1449,                                                  1304, 1241                               -  3                                                                                                                 3  111  ##                               -  4                                                                                                                 4  73 32##                               -  5                                                                                                                 5  54 33##                               -  6                                                                                                                 6  -- 1706, 1496, 1456, 1447,                                                  1294, 1243                               -  7                                                                                                                 7  73 35##                               -  8                                                                                                                 8  57 36##                               -  9                                                                                                                 9  86 37##                               - 10                                                                                                                 0  -- 1709, 1599, 1497, 1453,                                                  1346, 1241                               - 11                                                                                                                 1  -- 1708, 1599, 1497, 1455,                                                  1447, 1397, 1238                         - 12                                                                                                                 2  -- 1740, 1593, 1527, 1489,                                                  1456, 1252, 1225                         - 13                                                                                                                 3  -- 1710, 1603, 1584, 1490,                                                  1451, 1364, 1254                         - 14                                                                                                                 4  -- 1709, 1490, 1456, 1447,                                                  1379, 1300, 1258                         - 15                                                                                                                 5  -- 1712, 1490, 1456, 1447,                                                  1378, 1298, 1259                         - 16                                                                                                                 6  88 44##                               - 17                                                                                                                 7  -- 1710, 1511, 1451, 1364,                                                  1302, 1238                               - 18                                                                                                                 8  -- 1709, 1511, 1456, 1447,                                                  1379, 1301, 1236                         - 19                                                                                                                 9  -- 1712, 1511, 1447, 1378,                                                  1298, 1233                               - 20                                                                                                                 0  -- 1738, 1723, 1582, 1522,                                                  1452, 1223                               - 21                                                                                                                 1  -- 1711, 1492, 1480, 1447,                                                  1362, 1303, 1192, 1159                   (2 isomers approx. 4:3)                                                        - 22                                                                                                                 2  -- 1708, 1491, 1479, 1446,                                                  1376, 1300, 1277, 1150                   (2 isomers approx. 4:3)                                                        - 23                                                                                                                 3  -- 1712, 1511, 1447, 1378,                                                  1298, 1233                               (2 isomers approx. 4:3)                                                        - 24                                                                                                                 4  -- 1736, 1582, 1523, 1453,                                                  1221                                     (2 isomrs approx. 4:3)                                                         - 25                                                                                                                 5  -- 1706, 1495, 1485, 1363,                                                  1303, 1193, 1160                         (2 isomers approx. 4:3)                                                        - 26                                                                                                                 6  -- 1706, 1484, 1447, 1377,                                                  1301, 1280, 1150                         (2 isomers approx. 4:3)                                                        - 27                                                                                                                 7  -- 1710, 1495, 1483, 1446,                                                  1376, 1299, 1233                         (2 isomers approx. 4:3)                                                        - 28                                                                                                                 8  92 56##                               (2 isomers approx. 4:1)                                                        - 29                                                                                                                 9  -- 1709, 1489, 1447, 1362,                                                  1303, 1192, 1159                         (2 isomers approx. 4:1)                                                        - 30                                                                                                                 0  -- 1706, 1484, 1447, 1377,                                                  1301, 1280, 1150                         (2 isomers approx. 4:1)                                                        - 31                                                                                                                 1  -- 1711, 1488, 1446, 1375,                                                  1299, 1232                               (2 isomers approx. 4:1)                                                        - 32                                                                                                                 2  132  ##                               - 33                                                                                                                 3  -- 1709, 1495, 1486, 1451,                                                  1366, 1161, 1008                         - 34                                                                                                                 4  -- 1708, 1487, 1455, 1447,                                                  1379, 1300, 1009                         - 35                                                                                                                 5  -- 1711, 1488, 1447, 1378,                                                  1297, 1232, 1023, 1008                   - 36                                                                                                                 6  -- 1696, 1532, 1515, 1453,                                                  1267, 1245, 1069                         - 37                                                                                                                 7  -- 1712, 1486, 1447, 1361,                                                  1303, 1191, 1160                         - 38                                                                                                                 8  -- 1708, 1485, 1446, 1376,                                                  1300, 1274                               - 39                                                                                                                 9  -- 1709, 1484, 1446, 1374,                                                  1297, 1277, 1232                         - 40                                                                                                                 0  -- 1712, 1495, 1457, 1447,                                                  1378, 1298, 1237                         - 41                                                                                                                 1  110  ##                               - 42                                                                                                                 2  -- 1739, 1593, 1528, 1511,                                                  1457, 1226, 1035                         - 43                                                                                                                 3  102  ##                               - 44                                                                                                                 4  -- 1708, 1513, 1457, 1447,                                                  1378, 1302, 1246, 1035                   - 45                                                                                                                 5  102  ##                               - 46                                                                                                                 6  74 74##                               - 47                                                                                                                 7  -- 1709, 1606, 1512, 1364,                                                  1245, 1228, 1171, 1162, 1033,                                                  1005                                     - 48                                                                                                                 8  59 76##                               - 49                                                                                                                 9  -- 1709, 1447, 1364, 1261,                                                  1157, 1034, 1007                         - 50                                                                                                                 0  -- 1709, 1576, 1446, 1379,                                                  1300, 1260, 1239, 1156, 1037                                                     - 51                                                                         1  89 79##                               - 52                                                                                                                 2  -- 1740, 1593, 1575, 1527,                                                  1457, 1316, 1300, 1224, 1067,                                                  1029                                     - 53                                                                                                                 3  81 81##                               - 54                                                                                                                 4  -- 1711, 1574, 1447, 1365,                                                  1322, 1303, 1213, 1160, 1033,                                                  1008                                     - 55                                                                                                                 5  -- 1709, 1574, 1446, 1378,                                                  1321, 1301, 1284, 1213, 1034                                                     - 56                                                                         6  -- 1711, 1505, 1451, 1365,                                                  1304, 1245, 1160, 1143, 1035,                                                  1007                                     - 57                                                                                                                 7  63 85##                               - 58                                                                                                                 8  -- 1710, 1487, 1450, 1364,                                                  1301, 1246, 1160, 1030, 1006                                                     - 59                                                                         9  -- 1708, 1487, 1449, 1378,                                                  1300, 1247, 1030, 1009                   - 60                                                                                                                 0  -- 1743, 1593, 1528, 1502,                                                  1457, 1301, 1255, 1190, 1066,                                                  1006                                     - 61                                                                                                                 1  77 89##                               - 62                                                                                                                 2  -- 1712, 1503, 1453, 1363,                                                  1303, 1259, 1244, 1160, 1136,                                                  1006                                     - 63                                                                                                                 3  -- 1711, 1503, 1457, 1447,                                                  1380, 1301, 1258, 1239, 1136,                                                  1015                                     - 64                                                                                                                 4  92 1743, 1593, 1528, 1502,                                                  1457, 1301, 1255, 1190, 1066,                                                  1006                                     - 65                                                                                                                 5  90 93##                               - 66                                                                                                                 6  70 94##                               - 67                                                                                                                 7  75 95##                               - 68                                                                                                                 8  108  ##                               - 69                                                                                                                 9  93 97##                               - 70                                                                                                                 0  74 98##                               - 71                                                                                                                 1  -- 1712, 1504, 1450, 1363,                                                  1303, 1255, 1222, 1159, 1134                                                     - 72                                                                         2  -- 1712, 1510, 1498, 1450,                                                  1365, 1327, 1246, 1150, 1035,                                                  1005                                     - 73                                                                                                                 3  60 101##                              - 74                                                                                                                 4  -- 1711, 1509, 1497, 1451,                                                  1363, 1302, 1264, 1193, 1156,                                                  1129                                     - 75                                                                                                                 5  -- 1710, 1496, 1475, 1149,                                                  1365, 1301, 1263, 1195, 1159                                                     - 76                                                                         6  66 104##                              - 77                                                                                                                 7  86 105##                              - 78                                                                                                                 8  91 106##                              - 79                                                                                                                 9  100  7##                              - 80                                                                                                                 0  -- 1710, 1593, 1497, 1452,                                                  1364, 1323, 1297, 1193, 1165,                                                  1153                                     - 81                                                                                                                 1  -- 1715, 1510, 1447, 1367,                                                  1324, 1299, 1243, 1149, 1027,                                                  996                                      - 82                                                                                                                 2  -- 1710, 1509, 1456, 1446,                                                  1377, 1326, 1300, 1241, 1149,                                                  1306                                     - 83                                                                                                                 3  -- 1723, 1509, 1453, 1437,                                                  1316, 1292, 1241, 1149, 1064,                                                  1036                                     - 84                                                                                                                 4  -- 1738, 1611, 1581, 1539,                                                  1446, 1312, 1301, 1231, 1201,                                                  1067                                     - 85                                                                                                                 5  -- 1713, 1504, 1447, 1375,                                                  1313, 1300, 1233, 1143, 1027                                                     - 86                                                                         6  -- 1711, 1486, 1447, 1376,                                                  1300, 1281, 1150, 1034, 1013                                                     - 87                                                                         7  -- 1714, 1487, 1447, 1376,                                                  1300, 1231, 1023, 999                    - 88                                                                                                                 8  -- 1733, 1594, 1533, 1457,                                                  1396, 1231, 1013, 984                    - 89                                                                                                                 9  -- 1721, 1495, 1453, 1437,                                                  1313, 1290, 1239, 1123                   - 90                                                                                                                 0  -- 1709, 1453, 1366, 1303,                                                  1228, 1160, 1014                         - 91                                                                                                                 1  -- 1708, 1455, 1447, 1378,                                                  1299, 1282, 1015, 996                    - 92                                                                                                                 2  -- 1710, 1447, 1378, 1296,                                                  1232, 1045, 1023, 995                    - 93                                                                                                                 3  108  1##                              - 94                                                                                                                 4  -- 1717, 1495, 1457, 1444,                                                  1376, 1298, 1241, 1228, 1193                                                     - 95                                                                         5  -- 1739, 1614, 1603, 1542,                                                  1450, 1262, 129, 1179                    - 96                                                                                                                 6  170  4##                              - 97                                                                                                                 7  180  5##                              - 98                                                                                                                 8  173  6##                              - 99                                                                                                                 9  150  7##                              - 100                                                                                                                0  129  8##                              - 101                                                                                                                1  112  9##                              - 102                                                                                                                2  116  0##                              - 103                                                                                                                3  127  1##                              - 104                                                                                                                4  108  2##                              - 105                                                                                                                5  -- 1710, 1486, 1447, 1363,                                                  1307, 1193, 1159, 1031, 1006,                                                  919                                      - 106                                                                                                                6  -- 1706, 1484, 1447, 1376,                                                  1302, 1279, 1150, 1031, 1011,                                                  923                                      - 107                                                                                                                7  -- 1711, 1484, 1446, 1376,                                                  1298, 1232, 1144, 1024, 995, 922         - 108                                                                                                                8  147  6##                              - 109                                                                                                                9   1716, 1455, 1445, 1376,                                                    1297, 1279, 1097, 1069, 1017,                                                  1008                                     - 110                                                                                                                0   1718, 1487, 1447, 1394,                                                    1374, 1306, 1232, 1025, 1008                                                     - 111                                                                        1  109  9##                              - 112                                                                                                                2   1706, 1487, 1450, 1387,                                                    1304, 1276, 1155, 1022, 1009,                                                  769                                      - 113                                                                                                                3   1706, 1487, 1453, 1383,                                                    1312, 1301, 1274, 1155, 1033,                                                  1008                                     - 114                                                                                                                4  115  2##                              - 115                                                                                                                5  167  3##                              - 116                                                                                                                6   1729, 1575, 1565, 1545,                                                    1523, 1445, 1434, 1224, 1060                                                     - 117                                                                        7  110  5##                              - 118                                                                                                                8  77 146##                              - 119                                                                                                                9   1712, 1494, 1447, 1378,                                                    1298, 1232, 1045, 1024, 818, 771         - 120                                                                                                                0  115  8##                              - 121                                                                                                                1   1717, 1455, 1445, 1376,                                                    1298, 1278, 1097, 1068, 1016,                                                  999                                      - 122                                                                                                                2  81 150##                              - 123                                                                                                                3   1712, 1493, 1447, 1378,                                                    1297, 1232, 1047, 1024, 998, 772         - 124                                                                                                                4  107  2##                              - 125                                                                                                                5   1717, 1455, 1445, 1376,                                                    1298, 1279, 1096, 1068, 1017,                                                  999                                      - 126                                                                                                                6  128  4##                              - 127                                                                                                                7   1712, 1492, 1447, 1378,                                                    1298, 1232, 1096, 1044, 1023                                                     - 128                                                                        8  119  6##                              - 129                                                                                                                9   1717, 1492, 1455, 1445,                                                    1376, 1298, 1096, 1068, 1012,                                                  1000                                     - 130                                                                                                                0  133  8##                              - 131                                                                                                                1   1712, 1511, 1494, 1447,                                                    1378, 1298, 1232, 1045, 1024,                                                  837                                      - 132                                                                                                                2  113  0##                              - 133                                                                                                                3   1716, 1511, 1455, 1445,                                                    1376, 1298, 1228, 1097, 1068,                                                  999                                      - 134                                                                                                                4   1737, 1592, 1529, 1509,                                                    1489, 1455, 1303, 1231, 1067,                                                  1014                                     - 135                                                                                                                5   1712, 1586, 1507, 1489,                                                    1454, 1378, 1297, 1239, 1023                                                     - 136                                                                        6  148  4##                              - 137                                                                                                                7   1716, 1587, 1507, 1490,                                                    1455, 1375, 1298, 1240, 1068                                                     - 138                                                                        8  90 166##                              - 139                                                                                                                9   1719, 1495, 1464, 1446,                                                    1375, 1295, 1239, 1104, 1075,                                                  1014                                     - 140                                                                                                                0   1715, 1495, 1463, 1448,                                                    1376, 1298, 1239                         - 141                                                                                                                1  134  9##                              - 142                                                                                                                2   1744, 1583, 1522, 1503,                                                    1458, 1442, 1223, 1304, 1035,                                                  1004                                     - 143                                                                                                                3   1720, 1465, 1446, 1372,                                                    1296, 1280, 1243, 1144, 1035,                                                  1014                                     - 144                                                                                                                4   1716, 1505, 1465, 1448,                                                    1374, 1298, 1279, 1241, 1141,                                                  999                                      - 145                                                                                                                5  109  3##                              - 146                                                                                                                6  158  4##                              - 147                                                                                                                7   1718, 1463, 1445, 1376,                                                    1294, 1104, 1073, 1024, 1010                                                     - 148                                                                        8   1714, 1462, 1447, 1377,                                                    1297, 1238, 1025, 1009                   - 149                                                                                                                9  140 77##                           __________________________________________________________________________

Example 4

Methyl N-(2-methylphenyl)-N-methoxy-carbamate (Table 14, No. 1)

(a Methyl N-(2-methylphenyl)-N-hydroxy-carbamate

At 25-30° C., 14.0 g (0.148 mol) of methyl Chloroocarbonate is added dropwise to 16.4 g of N-(2-methylphenyl)-hydroxylamine (crude product, obtained according to Bamberger et al., Ann. Chem. 316 (1901), 278) and 12.9 g (0.163 mol) of pyridine in 100 ml of methylene Chloroide. The mixture is stirred overnight at room temperature (20° C.) and is then extracted with dilute hydroChloroic acid and water. The organic phase is dried over MgSO₄ and evaporated down. The residue is purified by column chromatography with mixtures of hexane and ethyl acetate. There is obtained 7 g (39mmol) of the title compound as a yellow oil.

¹ H-NMR (CDCl₃ ; δ in ppm): 8.6 (s, broad, OH); 7.3 (m, 4H, phenyl); 3.75 (s, 3H, OCH₃); 2.3 (s, 3H, CH₃)

b) Methyl N-(2-methylphenyl)-N-methoxy-carbamate (Table 14, No. 1)

At 20-30° C., 1.1 g (44.1 mmol) of sodium hydride is added in portions to 6.6 g (36.5 mmol) of the hydroxyl compound from Example 1a in 50 ml of dimethylformamide. Upon conclusion of gas evolution 5.7 g (40.1 mmol) of methyl iodide is added and the mixture is stirred over-night at room temperature. The reaction mixture is then diluted with water and the aqueous phase is extracted three times with methyl-t-butyl ether. The combined organic phases are dried over MgSO₄ and evaporated down. The residue is purified by column chromatography with mixtures of hexane and ethyl acetate. There is obtained 5.2 g (27 mmol=73%) of the title compound as a yellow oil.

¹ H-NMR (CDCl₃ ; δ in ppm): 7.25 (m, 4H, phenyl); 3.8; 3.75 (s, 3H, OCH₃ ; 3.75 (s, 3H, OCH₃); 2.3 (s, 3H, CH₃)

Example 5

Methyl N-(2-bromomethylphenyl)-N-methoxy-carbamate (Table 14, No. 2)

2.5 g (12.8 mmol) of the N-methoxycarbamate from Example 4b, 2.5 g (14.1 mmol) of N-bromosuccinimide and a spatula-tip (1 g) of azoisobutyrodinitrile in 20 ml of carbon tetraChloraide were irradiated with a 300 W UV lamp; the reaction mixture heated up to 30-40° C. After three hours the reaction mixture is extracted twice with water. The organic phase is dried over MgSO₄ and evaporated down. The residue is purified by column chromatography with mixtures of hexane and ethyl acetate. There is obtained 1.4 g (5.1 mmol=40%) of the title compound as a yellow oil.

¹ H-NMR (CDCl₃ ; δ in ppm): 7.5 (m, 1H, phenyl); 7.35 (m, 3H, phenyl); 4.55 (s, 2H, CH₂ --Br); 3.8 (2s, 6H, 2× OCH₃)

Example 6

Methyl N-[2-(2'-methylphenoxymethyl)-phenyl]-N-methoxy-carbamate (Table 14, No. 3)

1.2 g (4.4 mmol) of the methyl bromide from Example 5, 0.45 g (4.2 mmol) o-cresol and 0.7 g (4.8 mmol) of K₂ CO₃ in 30 ml of dimethylformamide are stirred overnight at room temperature. The reaction mixture is then diluted with water and the aqueous phase is extracted three times with methyl-t-butyl ether. The combined organic phases are dried over MgSO₄ and evaporated down. The residue is purified by column chromatography with mixtures of hexane and ethyl acetate. There is obtained 1.2 g of the title compound containing o-cresol as impurity. The mixture is heated in a furnace at about 1 mbar for about 1 hour at 125° C. The residue obtained is 0.9 g (3 mmol=68%) of the title compound as a yellow oil.

¹ H-NMR (CDCl₃ ; δ in ppm): 7.7 (m, 1H, phenyl); 7.4 (m, 3H, phenyl); 7.15 (m, 2H, phenyl); 6.9 (t, broad, 2H, phenyl); 5.15 (s, 2H, O--CH₂); 3.8 (s, 3H, OCH₃), 3.75 (s, 3H, OCH₃); 2.3 (s, 3H, CH₃)

                  TABLE 8                                                          ______________________________________                                         1  STR178##                                                                                 I: R.sup.1 = CH.sub.3                                               II: R.sup.1 = CH.sub.2 --CH.sub.3                                               -                                                                           No.     Xm                                                                     ______________________________________                                          1      H                                                                         2 2-F                                                                          3 3-F                                                                          4 4-F                                                                          5 2,4-F.sub.2                                                                  6 2,4,6-F.sub.3                                                                7 2,3,4,5,6-F.sub.5                                                            8 2,3-F.sub.2                                                                  9 2-Cl                                                                         10 3-Cl                                                                        11 4-Cl                                                                        12 2,3-Cl.sub.2                                                                13 2,4-Cl.sub.2                                                                14 2,5-Cl.sub.2                                                                15 2,6-Cl.sub.2                                                                16 3,4-Cl.sub.2                                                                17 3,5-Cl.sub.2                                                                18 2,3,4-Cl.sub.3                                                              19 2,3,5-Cl.sub.3                                                              20 2,3,6-Cl.sub.3                                                              21 2,4,5-Cl.sub.3                                                              22 2,4,6-Cl.sub.3                                                              23 3,4,5-Cl.sub.3                                                              24 2,3,4,6-Cl.sub.4                                                            25 2,3,5,6-Cl.sub.4                                                            26 2,3,4,5,6-Cl.sub.5                                                          27 2-Br                                                                        28 3-Br                                                                        29 4-Br                                                                        30 2,4-Br.sub.2                                                                31 2,5-Br.sub.2                                                                32 2,6-Br.sub.2                                                                33 2,4,6-Br.sub.3                                                              34 2,3,4,5,6-Br.sub.5                                                          35 2-I                                                                         36 3-I                                                                         37 4-I                                                                         38 2,4-I.sub.2                                                                 39 2-Cl, 3-F                                                                   40 2-Cl, 4-F                                                                   41 2-Cl, 5-F                                                                   42 2-Cl, 6-F                                                                   43 2-Cl, 3-Br                                                                  44 2-Cl, 4-Br                                                                  45 2-Cl, 5-Br                                                                  46 2-Cl, 6-Br                                                                  47 2-Br, 3-Cl                                                                  48 2-Br, 4-Cl                                                                  49 2-Br, 5-Cl                                                                  50 2-Br, 3-F                                                                   51 2-Br, 4-F                                                                   52 2-Br, 5-F                                                                   53 2-Br, 6-F                                                                   54 2-F, 3-Cl                                                                   55 2-F, 4-Cl                                                                   56 2-F, 5-Cl                                                                   57 3-Cl, 4-F                                                                   58 3-Cl, 5-F                                                                   59 3-Cl, 4-Br                                                                  60 3-Cl, 5-Br                                                                  61 3-F, 4-Cl                                                                   62 3-F, 4-Br                                                                   63 3-Br, 4-Cl                                                                  64 3-Br, 4-F                                                                   65 2,6-Cl.sub.2, 4-Br                                                          66 2-CH.sub.3                                                                  67 3-CH.sub.3                                                                  68 4-CH.sub.3                                                                  69 2,3-(CH.sub.3).sub.2                                                        70 2,4-(CH.sub.3).sub.2                                                        71 2,5-(CH.sub.3).sub.2                                                        72 2,6-(CH.sub.3).sub.2                                                        73 3,4-(CH.sub.3).sub.2                                                        74 3,5-(CH.sub.3).sub.2                                                        75 2,3,5-(CH.sub.3).sub.3                                                      76 2,3,4-(CH.sub.3).sub.3                                                      77 2,3,6-(CH.sub.3).sub.3                                                      78 2,4,5-(CH.sub.3).sub.3                                                      79 2,4,6-(CH.sub.3).sub.3                                                      80 3,4,5-(CH.sub.3).sub.3                                                      81 2,3,4,6-(CH.sub.3).sub.4                                                    82 2,3,5,6-(CH.sub.3).sub.4                                                    83 2,3,4,5,6-(CH.sub.3).sub.5                                                  84 2-C.sub.2 H.sub.5                                                           85 3-C.sub.2 H.sub.5                                                           86 4-C.sub.2 H.sub.5                                                           87 2,4-(C.sub.2 H.sub.5).sub.2                                                 88 2,6-(C.sub.2 H.sub.5).sub.2                                                 89 3,5-(C.sub.2 H.sub.5).sub.2                                                 90 2,4,6-(C.sub.2 H.sub.5).sub.3                                               91 2-n-C.sub.3 H.sub.7                                                         92 3-n-C.sub.3 H.sub.7                                                         93 4-n-C.sub.3 H.sub.7                                                         94 2-i-C.sub.3 H.sub.7                                                         95 3-i-C.sub.3 H.sub.7                                                         96 4-i-C.sub.3 H.sub.7                                                         97 2,4-(i-C.sub.3 H.sub.7).sub.2                                               98 2,6-(i-C.sub.3 H.sub.7).sub.2                                               99 3,5-(i-C.sub.3 H.sub.7).sub.2                                              100 2,4,6-(i-C.sub.3 H.sub.7).sub.3                                            101 2-s-C.sub.4 H.sub.9                                                        102 3-s-C.sub.4 H.sub.9                                                        103 4-s-C.sub.4 H.sub.9                                                        104 2-t-C.sub.4 H.sub.9                                                        105 3-t-C.sub.4 H.sub.9                                                        106 4-t-C.sub.4 H.sub.9                                                        107 2,3-(t-C.sub.4 H.sub.9).sub.2                                              108 2,4-(t-C.sub.4 H.sub.9).sub.2                                              109 2,5-(t-C.sub.4 H.sub.9).sub.2                                              110 2,6-(t-C.sub.4 H.sub.9).sub.2                                              111 3,4-(t-C.sub.4 H.sub.9).sub.2                                              112 2,4,6-(t-C.sub.4 H.sub.9).sub.3                                            113 4-n-C.sub.9 H.sub.19                                                       114 4-n-C.sub.12 H.sub.25                                                      115 4-n-C.sub.15 H.sub.31                                                      116 4-(1,1,3,3-Tetramethylbutyl)                                               117 4-(2,4,4-Trimethylpropyl)                                                  118 2-t-C.sub.4 H.sub.9, 4-CH.sub.3                                            119 2-t-C.sub.4 H.sub.9, 5-CH.sub.3                                            120 2,6-(t-C.sub.4 H.sub.9).sub.2, 4-CH.sub.3                                  121 2-CH.sub.3, 4-t-C.sub.4 H.sub.9                                            122 2-CH.sub.3, 6-t-C.sub.4 H.sub.9                                            123 2-CH.sub.3, 4-i-C.sub.3 H.sub.7                                            124 2-CH.sub.3, 5-i-C.sub.3 H.sub.7                                            125 3-CH.sub.3, 4-i-C.sub.3 H.sub.7                                            126 2-i-C.sub.3 H.sub.7, 5-CH.sub.3                                            127 2,4-(t-C.sub.4 H.sub.9).sub.2, 6-i-C.sub.3 H.sub.7                         128 2-Allyl                                                                    129 3-Allyl                                                                    130 4-Allyl                                                                    131 2-Allyl, 6-CH.sub.3                                                        132 2-cyclo-C.sub.6 H.sub.11                                                   133 3-cyclo-C.sub.6 H.sub.11                                                   134 4-cyclo-C.sub.6 H.sub.11                                                   135 2,4-(cyclo-C.sub.6 H.sub.11).sub.2, 6-CH.sub.3                             136 2-CH.sub.3, 4-cyclo-C.sub.6 H.sub.11                                       137 2-CH.sub.2 --C.sub.6 H.sub.5                                               138 3-CH.sub.2 --C.sub.6 H.sub.5                                               139 4-CH.sub.2 --C.sub.6 H.sub.5                                               140 2-CH.sub.2 --C.sub.6 H.sub.5, 4-CH.sub.3                                   141 2-CH.sub.3, 4-CH.sub.2 --C.sub.6 H.sub.5                                   142 2-C.sub.6 H.sub.5                                                          143 3-C.sub.6 H.sub.5                                                          144 4-C.sub.6 H.sub.5                                                          145 4-(2-i-C.sub.3 H.sub.7 --C.sub.6 H.sub.4)                                  146 4-C.sub.6 H.sub.5, 2,6-(CH.sub.3).sub.2                                    147 2-Cl, 4-C.sub.6 H.sub.5                                                    148 2-Br, 4-C.sub.6 H.sub.5                                                    149 2-C.sub.6 H.sub.5, 4-Cl                                                    150 2-C.sub.6 H.sub.5, 4-Br                                                    151 2-CH.sub.2 C.sub.6 H.sub.5, 4-Cl                                           152 2-CH.sub.2 C.sub.6 H.sub.5, 4-Br                                           153 2-Cl, 4-CH.sub.2 C.sub.6 H.sub.5                                           154 2-Br, 4-CH.sub.2 C.sub.6 H.sub.5                                           155 2-cyclo-C.sub.6 H.sub.11, 4-Cl                                             156 2-cyclo-C.sub.6 H.sub.11, 4-Br                                             157 2-Cl, 4-cyclo-C.sub.6 H.sub.11                                             158 2-Br, 4-cyclo-C.sub.6 H.sub.11                                             159 2-OCH.sub.3                                                                160 3-OCH.sub.3                                                                161 4-OCH.sub.3                                                                162 2-OC.sub.2 H.sub.5                                                         163 3-O--C.sub.2 H.sub.5                                                       164 4-O--C.sub.2 H.sub.5                                                       165 2-O-n-C.sub.3 H.sub.7                                                      166 3-O-n-C.sub.3 H.sub.7                                                      167 4-O-n-C.sub.3 H.sub.7                                                      168 2-O-i-C.sub.3 H.sub.7                                                      169 3-O-i-C.sub.3 H.sub.7                                                      170 4-O-i-C.sub.3 H.sub.7                                                      171 2-O-n-C.sub.6 H.sub.13                                                     172 3-O-n-C.sub.6 H.sub.13                                                     173 4-O-n-C.sub.6 H.sub.13                                                     174 2-O-n-C.sub.8 H.sub.17                                                     175 3-O-n-C.sub.8 H.sub.17                                                     176 4-O-n-C.sub.8 H.sub.17                                                     177 2-O--CH.sub.2 C.sub.6 H.sub.5                                              178 3-O--CH.sub.2 C.sub.6 H.sub.5                                              179 4-O--CH.sub.2 C.sub.6 H.sub.5                                              180 2-O--(CH.sub.2).sub.3 C.sub.6 H.sub.5                                      181 3-O--(CH.sub.2).sub.3 C.sub.6 H.sub.5                                      182 4-O--(CH.sub.2).sub.3 C.sub.6 H.sub.5                                      183 2,4-(OCH.sub.3).sub.2                                                      184 2-CF.sub.3                                                                 185 3-CF.sub.3                                                                 186 4-CF.sub.3                                                                 187 2-OCF.sub.3                                                                188 3-OCF.sub.3                                                                189 4-OCF.sub.3                                                                190 3-OCH.sub.2 CHF.sub.2                                                      191 2-NO.sub.2                                                                 192 3-NO.sub.2                                                                 193 4-NO.sub.2                                                                 194 2-CN                                                                       195 3-CN                                                                       196 4-CN                                                                       197 2-CH.sub.3, 3-Cl                                                           198 2-CH.sub.3, 4-Cl                                                           199 2-CH.sub.3, 5-Cl                                                           200 2-CH.sub.3, 6-Cl                                                           201 2-CH.sub.3, 3-F                                                            202 2-CH.sub.3, 4-F                                                            203 2-CH.sub.3, 5-F                                                            204 2-CH.sub.3, 6-F                                                            205 2-CH.sub.3, 3-Br                                                           206 2-CH.sub.3, 4-Br                                                           207 2-CH.sub.3, 5-Br                                                           208 2-CH.sub.3, 6-Br                                                           209 2-Cl, 3-CH.sub.3                                                           210 2-Cl, 4-CH.sub.3                                                           211 2-Cl, 5-CH.sub.3                                                           212 2-F, 3-CH.sub.3                                                            213 2-F, 4-CH.sub.3                                                            214 2-F, 5-CH.sub.3                                                            215 2-Br, 3-CH.sub.3                                                           216 2-Br, 4-CH.sub.3                                                           217 2-Br, 5-CH.sub.3                                                           218 3-CH.sub.3, 4-Cl                                                           219 3-CH.sub.3, 5-Cl                                                           220 3-CH.sub.3, 4-F                                                            221 3-CH.sub.3, 5-F                                                            222 3-CH.sub.3, 4-Br                                                           223 3-CH.sub.3, 5-Br                                                           224 3-F, 4-CH.sub.3                                                            225 3-Cl, 4-CH.sub.3                                                           226 3-Br, 4-CH.sub.3                                                           227 2-Cl, 4,5-(CH.sub.3).sub.2                                                 228 2-Br, 4,5-(CH.sub.3).sub.2                                                 229 2-Cl, 3,5-(CH.sub.3).sub.2                                                 230 2-Br, 3,5-(CH.sub.3).sub.2                                                 231 2,6-Cl.sub.2, 4-CH.sub.3                                                   232 2,6-F.sub.2, 4-CH.sub.3                                                    233 2,6-Br.sub.2, 4-CH.sub.3                                                   234 2,4-Br.sub.2, 6-CH.sub.3                                                   235 2,4-F.sub.2, 6-CH.sub.3                                                    236 2,4-Br.sub.2, 6-CH.sub.3                                                   237 2,6-(CH.sub.3).sub.2, 4-F                                                  238 2,6-(CH.sub.3).sub.2, 4-Cl                                                 239 2,6-(CH.sub.3).sub.2, 4-Br                                                 240 3,5-(CH.sub.3).sub.2, 4-F                                                  241 3,5-(CH.sub.3).sub.2, 4-Cl                                                 242 3,5-(CH.sub.3).sub.2, 4-Br                                                 243 2,3,6-(CH.sub.3).sub.3, 4-F                                                244 2,3,6-(CH.sub.3).sub.3, 4-Cl                                               245 2,3,6-(CH.sub.3).sub.3, 4-Br                                               246 2,4-(CH.sub.3).sub.2, 6-F                                                  247 2,4-(CH.sub.3).sub.2, 6-Cl                                                 248 2,4-(CH.sub.3).sub.2, 6-Br                                                 249 2-i-C.sub.3 H.sub.7, 4-Cl, 5-CH.sub.3                                      250 2-Cl, 4-NO.sub.2                                                           251 2-NO.sub.2, 4-Cl                                                           252 2-OCH.sub.3, 5-NO.sub.2                                                    253 2,4-Cl.sub.2, 5-NO.sub.2                                                   254 2,4-Cl.sub.2, 6-NO.sub.2                                                   255 2,6-Cl.sub.2, 4-NO.sub.2                                                   256 2,6-Br.sub.2, 4-NO.sub.2                                                   257 2,6-I.sub.2, 4-NO.sub.2                                                    258 2-CH.sub.3, 5-i-C.sub.3 H.sub.7, 4-Cl                                      259 2-CO.sub.2 CH.sub.3                                                        260 3-CO.sub.2 CH.sub.3                                                        261 4-CO.sub.2 CH.sub.3                                                        262 2-CO.sub.2 (C.sub.2 H.sub.5)                                               263 3-CO.sub.2 (C.sub.2 H.sub.5)                                               264 4-CO.sub.2 (C.sub.2 H.sub.5)                                               265 2-CO.sub.2 (n-C.sub.3 H.sub.7)                                             266 3-CO.sub.2 (n-C.sub.3 H.sub.7)                                             267 4-CO.sub.2 (n-C.sub.3 H.sub.7)                                             268 2-CO.sub.2 (i-C.sub.3 H.sub.7)                                             269 3-CO.sub.2 (i-C.sub.3 H.sub.7)                                             270 4-CO.sub.2 (i-C.sub.3 H.sub.7)                                             271 2-CO.sub.2 (n-C.sub.6 H.sub.13)                                            272 3-CO.sub.2 (n-C.sub.6 H.sub.13)                                            273 4-CO.sub.2 (n-C.sub.6 H.sub.13)                                            274 2-CH.sub.2 --OCH.sub.3                                                     275 3-CH.sub.2 --OCH.sub.3                                                     276 4-CH.sub.2 --OCH.sub.3                                                     277 2-CH.sub.2 O(C.sub.2 H.sub.5)                                              278 3-CH.sub.2 O(C.sub.2 H.sub.5)                                              279 4-CH.sub.2 O(C.sub.2 H.sub.5)                                              280 2-CH.sub.2 O(n-C.sub.3 H.sub.7)                                            281 3-CH.sub.2 O(n-C.sub.3 H.sub.7)                                            282 4-CH.sub.2 O(n-C.sub.3 H.sub.7)                                            283 2-CH.sub.2 O(i-C.sub.3 H.sub.7)                                            284 3-CH.sub.2 O(i-C.sub.3 H.sub.7)                                            285 4-CH.sub.2 O(i-C.sub.3 H.sub.7)                                            286 2-CHO                                                                      287 3-CHO                                                                      288 4-CHO                                                                      289 2-CO--CH.sub.3                                                             290 3-CO--CH.sub.3                                                             291 4-CO--CH.sub.3                                                             292 2-CO--CH.sub.2 --CH.sub.3                                                  293 3-CO--CH.sub.2 --CH.sub.3                                                  294 4-CO--CH.sub.2 --CH.sub.3                                                  295 2-CO--CH.sub.2 --CH.sub.2 --CH.sub.3                                       296 3-CO--CH.sub.2 --CH.sub.2 --CH.sub.3                                       297 4-CO--CH.sub.2 --CH.sub.2 --CH.sub.3                                       298 2-CO--CH(CH.sub.3)--CH.sub.3                                               299 3-CO--CH(CH.sub.3)--CH.sub.3                                               300 4-CO--CH(CH.sub.3)--CH.sub.3                                               301 2-Me-4-CHO                                                                 302 2-Me-4-CH.sub.3 --CO                                                       303 2-Me-4-CH.sub.3 --CH.sub.2 --CO                                            304 2-Me-4-CH.sub.3 --CH.sub.2 --CH.sub.2 --CO                                 305 2-Me-4-CH.sub.3 --CH(CH.sub.3)--CO                                         306 2,5-Me.sub.2 -4-CHO                                                        307 2, 5-Me.sub.2 -4-CH.sub.3 --CO                                             308 2, 5-Me.sub.2 -4-CH.sub.3 --CH.sub.2 --CO                                  309 2, 5-Me.sub.2 -4-CH.sub.3 --CH.sub.2 --CH.sub.2 --CO                       310 2, 5-Me.sub.2 -4-CH.sub.3 --CH(CH.sub.3)--CO                               311 2-Cl-4-CHO                                                                 312 2-Cl-4-CH.sub.3 --CO                                                       313 2-Cl-4-CH.sub.3 --CH.sub.2 --CO                                            314 2-Cl-4-CH.sub.3 --CH(CH.sub.3)--CO                                         315 2,5-Cl.sub.2 -4-CHO                                                        316 2,5-Cl.sub.2 -4-CH.sub.3 --CO                                              317 2,5-Cl.sub.2 -4-CH.sub.3 --CH.sub.2 --CO                                   318 2,5-Cl.sub.2 -4-CH.sub.3 --CH.sub.2 --CH.sub.2 --CO                        319 2,5-Cl.sub.2 -4-CH.sub.3 --CH(CH.sub.3)--CO                                320 2-C(═NOCH.sub.3)--CH.sub.3                                             321 3-C(═NOCH.sub.3)--CH.sub.3                                             322 4-C(═NOCH.sub.3)--CH.sub.3                                             323 2-C(═NOC.sub.2 H.sub.5)--CH.sub.3                                      324 3-C(═NOC.sub.2 H.sub.5)--CH.sub.3                                      325 4-C(═NOC.sub.2 H.sub.5)--CH.sub.3                                      326 2-C(═NO-n-C.sub.3 H.sub.7)--CH.sub.3                                   327 3-C(═NO-n-C.sub.3 H.sub.7)--CH.sub.3                                   328 4-C(═NO-n-C.sub.3 H.sub.7)--CH.sub.3                                   329 2-C(═NO-i-C.sub.3 H.sub.7)--CH.sub.3                                   330 3-C(═NO-i-C.sub.3 H.sub.7)--CH.sub.3                                   331 4-C(═NO-i-C.sub.3 H.sub.7)--CH.sub.3                                   332 2-C(═NO-Allyl)--CH.sub.3                                               333 3-C(═NO-Allyl)--CH.sub.3                                               334 4-C(═NO-Allyl)--CH.sub.3                                               335 2-C(═NO-trans-Chloroallyl)--CH.sub.3                                   336 3-C(═NO-trans-Chloroallyl)--CH.sub.3                                   337 4-C(═NO-trans-Chloroallyl)--CH.sub.3                                   338 2-C(═NO-Propargyl)--CH.sub.3                                           339 3-C(═NO-Propargyl)--CH.sub.3                                           340 4-C(═NO-Propargyl)--CH.sub.3                                           341 2-C(═NO-n-C.sub.4 H.sub.9)--CH.sub.3                                   342 3-C(═NO-n-C.sub.4 H.sub.9)--CH.sub.3                                   343 4-C(═NO-n-C.sub.4 H.sub.9)--CH.sub.3                                   344 2-C(═NO--CH.sub.2 --C.sub.6 H.sub.5)--CH.sub.3                         345 3-C(═NO--CH.sub.2 --C.sub.6 H.sub.5)--CH.sub.3                         346 4-C(═NO--CH.sub.2 --C.sub.6 H.sub.5)--CH.sub.3                         347 2-CH.sub.3 -4-CH═NOCH.sub.3                                            348 2-CH.sub.3 -4-CH═NOC.sub.2 H.sub.5                                     349 2-CH.sub.3 -4-CH═NO-n-C.sub.3 H.sub.7                                  350 2-CH.sub.3 -4-CH═NO-i-C.sub.3 H.sub.7                                  351 2-CH.sub.3 -4-CH═NO-Allyl                                              352 2-CH.sub.3 -4-CH═NO-(trans-Chloroallyl)                                353 2-CH.sub.3 -4-CH═NO-Propargyl                                          354 2-CH.sub.3 -4-CH═NO-n-C.sub.4 H.sub.9                                  355 2-CH.sub.3 -4-CH═NO-CH.sub.2 --C.sub.6 H.sub.5                         356 2-CH.sub.3 -4-(CH.sub.3 --C═NOCH.sub.3)                                357 2-CH.sub.3 -4-(CH.sub.3 --C═NOC.sub.2 H.sub.5)                         358 2-CH.sub.3 -4-(CH.sub.3 --C═NO-n-C.sub.3 H.sub.7)                      359 2-CH.sub.3 -4-(CH.sub.3 --C═NO-i-C.sub.3 H.sub.7)                      360 2-CH.sub.3 -4-(CH.sub.3 --C═NO-Allyl)                                  361 2-CH.sub.3 -4-(CH.sub.3 --C═NO-trans-Chloroallyl)                      362 2-CH.sub.3 -4-(CH.sub.3 --C═NO-Propargyl)                              363 2-CH.sub.3 -4-(CH.sub.3 --C═NO-n-C.sub.4 H.sub.9)                      364 2-CH.sub.3 -4-(CH.sub.3 --C═NO--CH.sub.2 --C.sub.6 H.sub.5)                   365 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C═NO--CH.sub.3)                       366 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C═NO--C.sub.2 H.sub.5)                367 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C═NO-n-C.sub.3 H.sub.7)        368 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C═NO-i-C.sub.3 H.sub.7                       369 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C═NO-Allyl)                    370 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C═NO-trans-Chloroallyl)                      371 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C═NO-Propargyl)                       372 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C═NO-n-C.sub.4 H.sub.9)        373 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C═NO--CH.sub.2 --C.sub.6                    H.sub.5)                                                                 374 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C═NOCH.sub.3)                      375 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C═NOC.sub.2 H.sub.5)                      376 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C═NO-n-C.sub.3                    H.sub.7)                                                                 377 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C═NO-i-C.sub.3 H.sub.7)                   378 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C═NO-Allyl)                 379 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C═NO-trans-Chloroallyl)                   380 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C═NO-Proparyl)                     381 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C═NO-n-C.sub.4                    H.sub.9)                                                                 382 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C═NO--CH.sub.2 --C.sub.6                 H.sub.5)                                                                 383 2-C.sub.6 H.sub.5                                                          384 3-C.sub.6 H.sub.5                                                          385 4-C.sub.6 H.sub.5                                                          386 2-(2'-F--C.sub.6 H.sub.4)                                                  387 2-(3'-F--C.sub.6 H.sub.4)                                                  388 2-(4'-F--C.sub.6 H.sub.4)                                                  389 3-(2'-F--C.sub.6 H.sub.4)                                                  390 3-(3'-F--C.sub.6 H.sub.4)                                                  391 3-(4'-F--C.sub.6 H.sub.4)                                                  392 4-(2'-F--C.sub.6 H.sub.4)                                                  393 4-(3'-F--C.sub.6 H.sub.4)                                                  394 4-(4'-F--C.sub.6 H.sub.4)                                                  395 2-(2'-Cl--C.sub.6 H.sub.4)                                                 396 2-(3'-Cl--C.sub.6 H.sub.4)                                                 397 2-(4'-Cl--C.sub.6 H.sub.4)                                                 398 3-(2'-Cl--C.sub.6 H.sub.4)                                                 399 3-(3'-Cl--C.sub.6 H.sub.4)                                                 400 3-(4'-Cl--C.sub.6 H.sub.4)                                                 401 4-(2'-Cl--C.sub.6 H.sub.4)                                                 402 4-(3'-Cl--C.sub.6 H.sub.4)                                                 403 4-(4'-Cl--C.sub.6 H.sub.4)                                                 405 2-(2'-CH.sub.3 --C.sub.6 H.sub.4)                                          406 2-(3'-CH.sub.3 --C.sub.6 H.sub.4)                                          407 2-(4'-CH.sub.3 --C.sub.6 H.sub.4)                                          408 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)                                          409 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)                                          410 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)                                          411 4-(2'-CH.sub.3 --C.sub.6 H.sub.4)                                          412 4-(3'-CH.sub.3 --C.sub.6 H.sub.4)                                          413 4-(4'-CH.sub.3 --C.sub.6 H.sub.4)                                          414 2-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                      415 2-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                      416 2-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                      417 3-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                      418 3-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                      419 3-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                      420 4-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                      421 4-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                      422 4-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                      423 2-(2'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                       424 2-(3'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                       425 2-(4'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                       426 3-(2'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                       427 3-(3'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                       428 3-(4'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                       429 4-(2'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                       430 4-(3'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                       431 4-(4'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                       432 2-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                                 433 2-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                                 434 2-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                                 435 3-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                                 436 3-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                                 437 3-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                                 438 4-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                                 439 4-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                                 440 4-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                                 441 2-(2'-CH.sub.3 O--C.sub.6 H.sub.4)                                         442 2-(3'-CH.sub.3 O--C.sub.6 H.sub.4)                                         443 2-(4'-CH.sub.3 O--C.sub.6 H.sub.4)                                         444 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)                                         445 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)                                         446 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)                                         447 4-(2'-CH.sub.3 O--C.sub.6 H.sub.4)                                         448 4-(3'-CH.sub.3 O--C.sub.6 H.sub.4)                                         449 4-(4'-CH.sub.3 O--C.sub.6 H.sub.4)                                         450 2-(2'-O.sub.2 N--C.sub.6 H.sub.4)                                          451 2-(3'-O.sub.2 N--C.sub.6 H.sub.4)                                          452 2-(4'-O.sub.2 N--C.sub.6 H.sub.4)                                          453 3-(2'-O.sub.2 N--C.sub.6 H.sub.4)                                          454 3-(3'-O.sub.2 N--C.sub.6 H.sub.4)                                          455 3-(4'-O.sub.2 N--C.sub.6 H.sub.4)                                          456 4-(2'-O.sub.2 N--C.sub.6 H.sub.4)                                          457 4-(3'-O.sub.2 N--C.sub.6 H.sub.4)                                          458 4-(4'-O.sub.2 N--C.sub.6 H.sub.4)                                          459 2-(2'-NC--C.sub.6 H.sub.4)                                                 460 2-(3'-NC--C.sub.6 H.sub.4)                                                 461 2-(4'-NC--C.sub.6 H.sub.4)                                                 462 3-(2'-NC--C.sub.6 H.sub.4)                                                 463 3-(3'-NC--C.sub.6 H.sub.4)                                                 464 3-(4'-NC--C.sub.6 H.sub.4)                                                 465 4-(2'-NC--C.sub.6 H.sub.4)                                                 466 4-(3'-NC--C.sub.6 H.sub.4)                                                 467 4-(4'-NC--C.sub.6 H.sub.4)                                                 468 2-(2'-CF.sub.3 --C.sub.6 H.sub.4)                                          469 2-(3'-CF.sub.3 --C.sub.6 H.sub.4)                                          470 2-(4'-CF.sub.3 --C.sub.6 H.sub.4)                                          471 3-(2'-CF.sub.3 --C.sub.6 H.sub.4)                                          472 3-(3'-CF.sub.3 --C.sub.6 H.sub.4)                                          473 3-(4'-CF.sub.3 --C.sub.6 H.sub.4)                                          474 4-(2'-CF.sub.3 --C.sub.6 H.sub.4)                                          475 4-(3'-CF.sub.3 --C.sub.6 H.sub.4)                                          476 4-(4'-CF.sub.3 --C.sub.6 H.sub.4)                                          477 2-O--C.sub.6 H.sub.5                                                       475 3-O--C.sub.6 H.sub.5                                                       476 4-O--C.sub.6 H.sub.5                                                       478 2-O--(2'-F--C.sub.6 H.sub.4)                                               479 2-O--(3'-F--C.sub.6 H.sub.4)                                               480 2-O--(4'-F--C.sub.6 H.sub.4)                                               481 3-O--(2'-F--C.sub.6 H.sub.4)                                               482 3-O--(3'-F--C.sub.6 H.sub.4)                                               483 3-O--(4'-F--C.sub.6 H.sub.4)                                               484 4-O--(2'-F--C.sub.6 H.sub.4)                                               485 4-O--(3'-F--C.sub.6 H.sub.4)                                               486 4-O--(4'-F--C.sub.6 H.sub.4)                                               487 2-O--(2'-Cl--C.sub.6 H.sub.4)                                              488 2-O--(3'-Cl--C.sub.6 H.sub.4)                                              489 2-O--(4'-Cl--C.sub.6 H.sub.4)                                              490 3-O--(2'-Cl--C.sub.6 H.sub.4)                                              491 3-O--(3'-Cl--C.sub.6 H.sub.4)                                              492 3-O--(4'-Cl--C.sub.6 H.sub.4)                                              493 3-O--(4'-Cl--C.sub.6 H.sub.4)                                              494 4-O--(2'-Cl--C.sub.6 H.sub.4)                                              495 4-O--(3'-Cl--C.sub.6 H.sub.4)                                              496 4-O--(4'-Cl--C.sub.6 H.sub.4)                                              497 2-O--(2'-CH.sub.3 --C.sub.6 H.sub.4)                                       498 2-O--(3'-CH.sub.3 --C.sub.6 H.sub.4)                                       499 2-O--(4'-CH.sub.3 --C.sub.6 H.sub.4)                                       500 3-O--(2'-CH.sub.3 --C.sub.6 H.sub.4)                                       501 3-O--(3'-CH.sub.3 --C.sub.6 H.sub.4)                                       502 3-O--(4'-CH.sub.3 --C.sub.6 H.sub.4)                                       503 4-O--(2'-CH.sub.3 --C.sub.6 H.sub.4)                                       504 4-O--(3'-CH.sub.3 --C.sub.6 H.sub.4)                                       505 4-O--(4'-CH.sub.3 --C.sub.6 H.sub.4)                                       506 2-O--(2'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                   507 2-O--(3'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                   508 2-O--(4'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                   509 3-O--(2'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                   510 3-O--(3'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                   511 3-O--(4'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                   512 4-O--(2'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                   513 4-O--(3'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                   514 4-O--(4'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                   515 2-O--(2'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                    516 2-O--(3'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                    517 2-O--(4'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                    518 3-O--(2'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                    519 3-O--(3'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                    520 3-O--(4'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                    521 4-O--(2'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                    522 4-O--(3'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                    523 4-O--(4'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                    524 2-O--(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                              525 2-O--(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                              526 2-O--(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                              527 3-O--(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                              528 3-O--(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                              529 3-O--(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                              530 4-O--(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                              531 4-O--(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                              532 4-O--(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                              533 2-O--(2'-CH.sub.3 O--C.sub.6 H.sub.4)                                      534 2-O--(3'-CH.sub.3 O--C.sub.6 H.sub.4)                                      535 2-O--(4'-CH.sub.3 O--C.sub.6 H.sub.4)                                      536 3-O--(2'-CH.sub.3 O--C.sub.6 H.sub.4)                                      537 3-O--(3'-CH.sub.3 O--C.sub.6 H.sub.4)                                      538 3-O--(4'-CH.sub.3 O--C.sub.6 H.sub.4)                                      539 4-O--(2'-CH.sub.3 O--C.sub.6 H.sub.4)                                      540 4-O--(3'-CH.sub.3 O--C.sub.6 H.sub.4)                                      541 4-O--(4'-CH.sub.3 O--C.sub.6 H.sub.4)                                      542 2-O--(2'-O.sub.2 N--C.sub.6 H.sub.4)                                       543 2-O--(3'-O.sub.2 N--C.sub.6 H.sub.4)                                       544 2-O--(4'-O.sub.2 N--C.sub.6 H.sub.4)                                       545 3-O--(2'-O.sub.2 N--C.sub.6 H.sub.4)                                       546 3-O--(3'-O.sub.2 N--C.sub.6 H.sub.4)                                       547 3-O--(4'-O.sub.2 N--C.sub.6 H.sub.4)                                       548 4-O--(2'-O.sub.2 N--C.sub.6 H.sub.4)                                       549 4-O--(3'-O.sub.2 N--C.sub.6 H.sub.4)                                       550 4-O--(4'-O.sub.2 N--C.sub.6 H.sub.4)                                       551 2-O--(2'-NC--C.sub.6 H.sub.4)                                              552 2-O--(3'-NC--C.sub.6 H.sub.4)                                              553 2-O--(4'-NC--C.sub.6 H.sub.4)                                              554 3-O--(2'-NC--C.sub.6 H.sub.4)                                              555 3-O--(3'-NC--C.sub.6 H.sub.4)                                              556 3-O--(4'-NC--C.sub.6 H.sub.4)                                              557 4-O--(2'-NC--C.sub.6 H.sub.4)                                              558 4-O--(3'-NC--C.sub.6 H.sub.4)                                              559 4-O--(4'-NC--C.sub.6 H.sub.4)                                              560 2-O--(2'-CF.sub.3 --C.sub.6 H.sub.4)                                       561 2-O--(3'-CF.sub.3 --C.sub.6 H.sub.4)                                       562 2-O--(4'-CF.sub.3 --C.sub.6 H.sub.4)                                       563 3-O--(2'-CF.sub.3 --C.sub.6 H.sub.4)                                       564 3-O--(3'-CF.sub.3 --C.sub.6 H.sub.4)                                       565 3-O--(4'-CF.sub.3 --C.sub.6 H.sub.4)                                       566 4-O--(2'-CF.sub.3 --C.sub.6 H.sub.4)                                       567 4-O--(3'-CF.sub.3 --C.sub.6 H.sub.4)                                       568 4-O--(4'-CF.sub.3 --C.sub.6 H.sub.4)                                       569 2-Pyridinyl-2'                                                             570 2-Pyridinyl-3'                                                             571 2-Pyridinyl-4'                                                             572 3-Pyridinyl-2'                                                             573 3-Pyridinyl-3'                                                             574 3-Pyridinyl-4'                                                             575 4-Pyridinyl-2'                                                             576 4-Pyridinyl-3'                                                             577 4-Pyridinyl-4'                                                             578 2-Pyrimidinyl-2'                                                           579 2-Pyrimidinyl-3'                                                           580 2-Pyrimidinyl-4'                                                           581 3-Pyrimidinyl-2'                                                           582 3-Pyrimidinyl-3'                                                           583 3-Pyrimidinyl-4'                                                           584 4-Pyrimidinyl-2'                                                           585 4-Pyrimidinyl-3'                                                           586 4-Pyrimidinyl-4'                                                           587 2-Pyrazolyl-1'                                                             588 2-Pyrazolyl-3'                                                             589 2-Pyrazolyl-4'                                                             590 3-Pyrazolyl-1'                                                             591 3-Pyrazolyl-3'                                                             592 3-Pyrazolyl-4'                                                             593 4-Pyrazolyl-1'                                                             594 4-Pyrazolyl-3'                                                             595 4-Pyrazolyl-4'                                                             596 2-Isoxazolyl-3'                                                            597 2-Isoxazolyl-4'                                                            598 2-Isoxazolyl-5'                                                            599 3-Isoxazolyl-3'                                                            600 3-Isoxazolyl-4'                                                            601 3-Isoxazolyl-5'                                                            602 4-Isoxazolyl-3'                                                            603 4-Isoxazolyl-4'                                                            604 4-Isoxazolyl-5'                                                            605 2-Isothiazolyl-3'                                                          606 2-Isothiazolyl-4'                                                          607 2-Isothiazolyl-5'                                                          608 3-Isothiazolyl-3'                                                          609 3-Isothiazolyl-4'                                                          610 3-Isothiazolyl-5'                                                          611 4-Isothiazolyl-3'                                                          612 4-Isothiazolyl-4'                                                          613 4-Isothiazolyl-5'                                                          614 2-Imidazolyl-1'                                                            615 2-Imidazolyl-2'                                                            616 2-Imidazolyl-4'                                                            617 3-Imidazolyl-1'                                                            618 3-Imidazolyl-2'                                                            619 3-Imidazolyl-4'                                                            620 4-Imidazolyl-1'                                                            621 4-Imidazolyl-2'                                                            622 4-Imidazolyl-4'                                                            623 2-Oxazolyl-2'                                                              624 2-Oxazolyl-4'                                                              625 2-Oxazolyl-5'                                                              626 3-Oxazolyl-2'                                                              627 3-Oxazolyl-4'                                                              628 3-Oxazolyl-5'                                                              629 4-Oxazolyl-2'                                                              630 4-Oxazolyl-4'                                                              631 4-Oxazolyl-5'                                                              632 2-Thiazolyl-2'                                                             633 2-Thiazolyl-4'                                                             634 2-Thiazolyl-5'                                                             635 3-Thiazolyl-2'                                                             636 3-Thiazolyl-4'                                                             637 3-Thiazolyl-5'                                                             638 4-Thiazolyl-2'                                                             639 4-Thiazolyl-4'                                                             640 4-Thiazolyl-5'                                                             641 2-CH.sub.3 -4-(CH.sub.3 --C═N--O--CH.sub.2 --CH.sub.2 --OCH.sub.             3)                                                                       642 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C═N--O--CH.sub.2 --CH.sub.2                 --OCH.sub.3)                                                             643 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C═N--O--CH.sub.2 --CH.sub.2              --OCH.sub.3)                                                             644 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C═N--OCH.sub.3)                     645 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C═N--OC.sub.2 H.sub.5)                     646 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C═N--O-n-C.sub.3                   H.sub.7)                                                                 647 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C═N--O-i-C.sub.3 H.sub.7)                  648 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C═N--O-Allyl)                       649 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C═N--O-trans-Chloroall             yl)                                                                      650 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C═N--O-Propargyl)                   651 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C═N--O-n-C.sub.4 H.sub.9)                  652 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C═N--O--CH.sub.2                   --C.sub.6 H.sub.5)                                                       653 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C═N--OCH.sub.3)                     654 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C═N--OC.sub.2 H.sub.5)                     655 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C═N--O-n-C.sub.3                   H.sub.7)                                                                 656 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C═N--O-i-C.sub.3 H.sub.7)                  657 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C═N--O-Allyl)                       658 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C═N--O-trans-Chloroall             yl)                                                                      659 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C═N--O-Propargyl)                   660 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C═N--O-n-C.sub.4 H.sub.9)                  661 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C═N--O--CH.sub.2                   --C.sub.6 H.sub.5)                                                       662 2-O-n-C.sub.4 H.sub.9                                                      663 2-O-i-C.sub.4 H.sub.9                                                      664 2-O-s-C.sub.4 H.sub.9                                                      665 2-O-t-C.sub.4 H.sub.9                                                      666 2-Neopentyloxy                                                             667 3-O-n-C.sub.4 H.sub.9                                                      668 3-O-i-C.sub.4 H.sub.9                                                      669 3-O-s-C.sub.4 H.sub.9                                                      670 3-O-t-C.sub.4 H.sub.9                                                      671 3-Neopentyloxy                                                             672 4-O-n-C.sub.4 H.sub.9                                                      673 4-O-i-C.sub.4 H.sub.9                                                      674 4-O-s-C.sub.4 H.sub.9                                                      675 4-O-t-C.sub.4 H.sub.9                                                      676 4-Neopentyloxy                                                             677 3-CH.sub.3 -4-OCH.sub.3                                                    678 3-CH.sub.3 -4-OC.sub.2 H.sub.5                                             679 3-CH.sub.3 -4-O-n-C.sub.3 H.sub.7                                          680 3-CH.sub.3 -4-O-n-C.sub.4 H.sub.9                                          681 3-CH.sub.3 -4-O-i-C.sub.4 H.sub.9                                          682 3-CH.sub.3 -4-O-s-C.sub.4 H.sub.9                                          683 3-CH.sub.3 -4-O-t-C.sub.4 H.sub.9                                          684 3-CH.sub.3 -4-Neopentyloxy                                                 685 2-CH.sub.3 -3-OCH.sub.3                                                    686 2-CH.sub.3 -4-OCH.sub.3                                                    687 2-CH.sub.3 -5-OCH.sub.3                                                    688 2-CH.sub.3 -6-OCH.sub.3                                                    689 3-CH.sub.3 -4-OCH.sub.3                                                    690 3-CH.sub.3 -5-OCH.sub.3                                                    691 3-CH.sub.3 -6-OCH.sub.3                                                    692 4-CH.sub.3 -5-O--CH.sub.3                                                  693 4-CH.sub.3 -6-O--CH.sub.3                                                  694 4-CH.sub.3 -6-OCH.sub.3                                                    695 2-CH.sub.3 -3-O-i-C.sub.3 H.sub.7                                          696 2-CH.sub.3 -4-O-i-C.sub.3 H.sub.7                                          697 2-CH.sub.3 -5-O-i-C.sub.3 H.sub.7                                          698 2-CH.sub.3 -6-O-i-C.sub.3 H.sub.7                                          699 3-CH.sub.3 -4-O-i-C.sub.3 H.sub.7                                          700 3-CH.sub.3 -5-O-i-C.sub.3 H.sub.7                                          701 3-CH.sub.3 -6-O-i-C.sub.3 H.sub.7                                          702 4-CH.sub.3 -5-O-i-C.sub.3 H.sub.7                                          703 4-CH.sub.3 -6-O-i-C.sub.3 H.sub.7                                          704 5-CH.sub.3 -6-O-i-C.sub.3 H.sub.7                                          705 2-Cl-3-OCH.sub.3                                                           706 2-Cl-4-OCH.sub.3                                                           707 2-Cl-5-OCH.sub.3                                                           708 2-Cl-6-OCH.sub.3                                                           709 3-Cl-4-OCH.sub.3                                                           710 3-Cl-5-OCH.sub.3                                                           711 3-Cl-6-OCH.sub.3                                                           712 4-Cl-5-OCH.sub.3                                                           713 4-Cl-6-OCH.sub.3                                                           714 5-Cl-6-OCH.sub.3                                                         ______________________________________                                    

                  TABLE 9                                                          ______________________________________                                         2  STR179##                                                                       -         I: R.sup.1 = CH.sub.3                                               II: R.sup.1 = CH.sub.2 --CH.sub.3                                            No.       B                                                                    ______________________________________                                          1        Pyrrolyl-3                                                              2 N--CH.sub.3 -Pyrrolyl-3                                                      3 N--C.sub.6 H.sub.5 -Pyrrolyl-3                                               4 N-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrrolyl-3                                 5 N-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrrolyl-3                                 6 N-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrrolyl-3                                 7 N-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrrolyl-3                                8 N-(3'-CH.sub.3 O--C.sub.6 H.sub.4) Pyrrolyl-3                                9 N-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrrolyl-3                                10 N-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrrolyl-3                                11 N-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrrolyl-3                                12 N-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrrolyl-3                                13 N-(4'-CN--C.sub.6 H.sub.4)-Pyrrolyl-3                                       14 N-(3'-CN--C.sub.6 H.sub.4)-Pyrrolyl-3                                       15 N-(2'-CN--C.sub.6 H.sub.4)-Pyrrolyl-3                                       16 N-(4'-Cl--C.sub.6 H.sub.4)-Pyrrolyl-3                                       17 N-(3'-Cl--C.sub.6 H.sub.4)-Pyrrolyl-3                                       18 N-(2'-Cl--C.sub.6 H.sub.4)-Pyrrolyl-3                                       19 Pyrrolyl-2                                                                  20 N--CH.sub.3 -Pyrrolyl-2                                                     21 N--C.sub.6 H.sub.5 -Pyrrolyl-2                                              22 N-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrrolyl-2                                23 N-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrrolyl-2                                24 N-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrrolyl-2                                25 N-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrrolyl-2                               26 N-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrrolyl-2                               27 N-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrrolyl-2                               28 N-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrrolyl-2                                29 N-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrrolyl-2                                30 N-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrrolyl-2                                31 N-(4'-CN--C.sub.6 H.sub.4)-Pyrrolyl-2                                       32 N-(3'-CN--C.sub.6 H.sub.4)-Pyrrolyl-2                                       33 N-(2'-CN--C.sub.6 H.sub.4)-Pyrrolyl-2                                       34 N-(4'-Cl--C.sub.6 H.sub.4)-Pyrrolyl-2                                       35 N-(3'-Cl--C.sub.6 H.sub.4)-Pyrrolyl-2                                       36 N-(2'-Cl--C.sub.6 H.sub.4)-Pyrrolyl-2                                       37 Furyl-2                                                                     38 5-CH.sub.3 -Furyl-2                                                         39 5-C.sub.6 H.sub.5 -Furyl-2                                                  40 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Furyl-2                                   41 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Furyl-2                                   42 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Furyl-2                                   43 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Furyl-2                                  44 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Furyl-2                                  45 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Furyl-2                                  46 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Furyl-2                                   47 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Furyl-2                                   48 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Furyl-2                                   49 5-(4'-CN--C.sub.6 H.sub.4)-Furyl-2                                          50 5-(3'-CN--C.sub.6 H.sub.4)-Furyl-2                                          51 5-(2'-CN--C.sub.6 H.sub.4)-Furyl-2                                          52 5-(4'-Cl--C.sub.6 H.sub.4)-Furyl-2                                          53 5-(3'-Cl--C.sub.6 H.sub.4)-Furyl-2                                          54 5-(2'-Cl--C.sub.6 H.sub.4)-Furyl-2                                          55 4-CH.sub.3 -Furyl-2                                                         56 4-C.sub.6 H.sub.5 -Furyl-2                                                  57 4-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Furyl-2                                   58 4-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Furyl-2                                   59 4-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Furyl-2                                   60 4-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Furyl-2                                  61 4-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Furyl-2                                  62 4-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Furyl-2                                  63 4-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Furyl-2                                   64 4-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Furyl-2                                   65 4-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Furyl-2                                   66 4-(4'-CN--C.sub.6 H.sub.4)-Furyl-2                                          67 4-(3'-CN--C.sub.6 H.sub.4)-Furyl-2                                          68 4-(2'-CN--C.sub.6 H.sub.4)-Furyl-2                                          69 4-(4'-Cl--C.sub.6 H.sub.4)-Furyl-2                                          70 4-(3'-Cl--C.sub.6 H.sub.4)-Furyl-2                                          71 4-(2'-Cl--C.sub.6 H.sub.4)-Furyl-2                                          72 Thienyl-2                                                                   73 5-CH.sub.3 -Thienyl-2                                                       74 5-C.sub.6 H.sub.5 -Thienyl-2                                                75 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-2                                 76 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-2                                 77 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-2                                 78 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-2                                79 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4) Thienyl-2                                80 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-2                                81 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-2                                 82 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-2                                 83 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-2                                 84 5-(4'-CN--C.sub.6 H.sub.4)-Thienyl-2                                        85 5-(3'-CN--C.sub.6 H.sub.4)-Thienyl-2                                        86 5-(2'-CN--C.sub.6 H.sub.4)-Thienyl-2                                        87 5-(4'-Cl--C.sub.6 H.sub.4)-Thienyl-2                                        88 5-(3'-Cl--C.sub.6 H.sub.4)-Thienyl-2                                        89 5-(2'-Cl--C.sub.6 H.sub.4)-Thienyl-2                                        90 4-CH.sub.3 -Thienyl-2                                                       91 4-C.sub.6 H.sub.5 -Thienyl-2                                                92 4-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-2                                 93 4-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-2                                 94 4-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-2                                 95 4-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-2                                96 4-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-2                                97 4-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-2                                98 4-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-2                                 99 4-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-2                                100 4-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-2                                101 4-(4'-CN--C.sub.6 H.sub.4)-Thienyl-2                                       102 4-(3'-CN--C.sub.6 H.sub.4)-Thienyl-2                                       103 4-(2'-CN--C.sub.6 H.sub.4)-Thienyl-2                                       104 4-(4'-Cl--C.sub.6 H.sub.4)-Thienyl-2                                       105 4-(3'-Cl--C.sub.6 H.sub.4)-Thienyl-2                                       106 4-(2'-Cl--C.sub.6 H.sub.4)-Thienyl-2                                       107 Thienyl-3                                                                  108 5-CH.sub.3 -Thienyl-3                                                      109 5-C.sub.6 H.sub.5 -Thienyl-3                                               110 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-3                                111 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-3                                112 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-3                                113 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-3                               114 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-3                               115 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-3                               116 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-3                                117 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-3                                118 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-3                                119 5-(4'-CN--C.sub.6 H.sub.4)-Thienyl-3                                       120 5-(3'-CN--C.sub.6 H.sub.4)-Thienyl-3                                       121 5-(2'-CN--C.sub.6 H.sub.4)-Thienyl-3                                       122 5-(4'-Cl--C.sub.6 H.sub.4)-Thienyl-3                                       123 5-(3'-Cl--C.sub.6 H.sub.4)-Thienyl-3                                       124 5-(2'-Cl--C.sub.6 H.sub.4)-Thienyl-3                                       125 Pyrazolyl-4                                                                126 N--CH.sub.3 -Pyrazolyl-4                                                   127 N--C.sub.6 H.sub.5 -Pyrazolyl-4                                            128 N-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrazolyl-4                              129 N-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrazolyl-4                              130 N-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrazolyl-4                              131 N-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrazolyl-4                             132 N-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrazoly-4                              133 N-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrazolyl-4                             134 N-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrazolyl-4                              135 N-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrazolyl-4                              136 N-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrazolyl-4                              137 N-(4'-CN--C.sub.6 H.sub.4)-Pyrazolyl-4                                     138 N-(3'-CN--C.sub.6 H.sub.4)-Pyrazolyl-4                                     139 N-(2'-CN--C.sub.6 H.sub.4)-Pyrazolyl-4                                     140 N-(4'-Cl--C.sub.6 H.sub.4)-Pyrazolyl-4                                     141 N-(3'-Cl--C.sub.6 H.sub.4)-Pyrazolyl-4                                     142 N-(2'-Cl--C.sub.6 H.sub.4)-Pyrazolyl-4                                     143 3-CH.sub.3 --N-Methylpyrazolyl-4                                           144 3-C.sub.6 H.sub.5 --N-Methylpyrazolyl-4                                    145 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)--N-Methylpyrazolyl-4                     146 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)--N-Methylpyrazolyl-4                     147 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)--N-Methylpyrazolyl-4                     148 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)--N-Methylpyrazolyl-4                    149 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)--N-Methylpyrazolyl-4                    150 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)--N-Methylpyrazolyl-4                    151 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)--N-Methylpyrazolyl-4                     152 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)--N-Methylpyrazolyl-4                     153 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)--N-Methylpyrazolyl-4                     154 3-(4'-CN--C.sub.6 H.sub.4)--N-Methylpyrazolyl-4                            155 3-(3'-CN--C.sub.6 H.sub.4)--N-Methylpyrazolyl-4                            156 3-(2'-CN--C.sub.6 H.sub.4)--N-Methylpyrazolyl-4                            157 3-(4'-Cl--C.sub.6 H.sub.4)--N-Methylpyrazolyl-4                            158 3-(3'-Cl--C.sub.6 H.sub.4)--N-Methylpyrazolyl-4                            159 3-(2'-Cl--C.sub.6 H.sub.4)--N-Methylpyrazolyl-4                            160 Isoxazolyl-5                                                               161 3-CH.sub.3 -Isoxazolyl-5                                                   162 3-C.sub.6 H.sub.5 -Isoxazolyl-5                                            163 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Isoxazolyl-5                             164 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Isoxazolyl-5                             165 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Isoxazolyl-5                             166 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Isoxazolyl-5                            167 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Isoxazolyl-5                            168 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Isoxazolyl-5                            169 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Isoxazolyl-5                             170 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Isoxazolyl-5                             171 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Isoxazolyl-5                             172 3-(4'-CN--C.sub.6 H.sub.4)-Isoxazolyl-5                                    173 3-(3'-CN--C.sub.6 H.sub.4)-Isoxazolyl-5                                    174 3-(2'-CN--C.sub.6 H.sub.4)-Isoxazolyl-5                                    175 3-(4'-Cl--C.sub.6 H.sub.4)-Isoxazolyl-5                                    176 3-(3'-Cl--C.sub.6 H.sub.4)-Isoxazolyl-5                                    177 3-(2'-Cl--C.sub.6 H.sub.4)-Isoxazolyl-5                                    178 4-Chloroisoxazolyl-5                                                       179 3-CH.sub.3 -4-Chloroisoxazolyl-5                                           180 3-C.sub.6 H.sub.5 -4-Chloroisoxazolyl-5                                    181 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                     182 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                     183 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                     184 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                    185 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                    186 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                    187 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                     188 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                     189 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                     190 3-(4'-CN--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                            191 3-(3'-CN--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                            192 3-(2'-CN--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                            193 3-(4'-Cl--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                            194 3-(3'-Cl--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                            195 3-(2'-Cl--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                            196 Isoxazolyl-3                                                               197 5-CH.sub.3 -Isoxazolyl-3                                                   198 5-C.sub.6 H.sub.5 -Isoxazolyl-3                                            199 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Isoxazolyl-3                             200 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Isoxazolyl-3                             201 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Isoxazolyl-3                             202 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Isoxazolyl-3                            203 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Isoxazolyl-3                            204 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Isoxazolyl-3                            205 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Isoxazolyl-3                             206 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Isoxazolyl-3                             207 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Isoxazolyl-3                             208 5-(4'-CN--C.sub.6 H.sub.4)-Isoxazolyl-3                                    209 5-(3'-CN--C.sub.6 H.sub.4)-Isoxazolyl-3                                    210 5-(2'-CN--C.sub.6 H.sub.4)-Isoxazolyl-3                                    211 5-(4'-Cl--C.sub.6 H.sub.4)-Isoxazolyl-3                                    212 5-(3'-Cl--C.sub.6 H.sub.4)-Isoxazolyl-3                                    213 5-(2'-Cl--C.sub.6 H.sub.4)-Isoxazolyl-3                                    214 Isothiazolyl-5                                                             215 3-CH.sub.3 -Isothiazolyl-5                                                 216 3-C.sub.6 H.sub.5 -Isothiazolyl-5                                          217 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Isothiazolyl-5                           218 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Isothiazolyl-5                           219 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Isothiazolyl-5                           220 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Isothiazolyl-5                          221 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Isothiazolyl-5                          222 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Isothiazolyl-5                          223 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Isothiazolyl-5                           224 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Isothiazolyl-5                           225 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Isothiazolyl-5                           226 3-(4'-CN--C.sub.6 H.sub.4)-Isothiazolyl-5                                  227 3-(3'-CN--C.sub.6 H.sub.4)-Isothiazolyl-5                                  228 3-(2'-CN--C.sub.6 H.sub.4)-Isothiazolyl-5                                  229 3-(4'-Cl--C.sub.6 H.sub.4)-Isothiazolyl-5                                  230 3-(3'-Cl--C.sub.6 H.sub.4)-Isothiazolyl-5                                  231 3-(2'-Cl--C.sub.6 H.sub.4)-Isothiazolyl-5                                  232 Oxazolyl-4                                                                 233 2-CH.sub.3 -Oxazolyl-4                                                     234 2-C.sub.6 H.sub.5 -Oxazolyl-4                                              235 2-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Oxazolyl-A                               236 2-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Oxazolyl-4                               237 2-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Oxazolyl-4                               238 2-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Oxazolyl-4                              239 2-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Oxazolyl-4                              240 2-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Oxazolyl-4                              241 2-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Oxazolyl-4                               242 2-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Oxazolyl-4                               243 2-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Oxazolyl-4                               244 2-(4'-CN--C.sub.6 H.sub.4)-Oxazolyl-4                                      245 2-(3'-CN--C.sub.6 H.sub.4)-Oxazolyl-4                                      246 2-(2'-CN--C.sub.6 H.sub.4)-Oxazolyl-4                                      247 2-(4'-Cl--C.sub.6 H.sub.4)-Oxazolyl-4                                      248 2-(3'-Cl--C.sub.6 H.sub.4)-Oxazolyl-4                                      249 2-(2'-Cl--C.sub.6 H.sub.4)-Oxazolyl-4                                      250 Thiazolyl-4                                                                251 2-CH.sub.3 -Thiazolyl-4                                                    252 2-C.sub.6 H.sub.5 -Thiazolyl-4                                             253 2-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Thiazolyl-4                              254 2-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Thiazolyl-4                              255 2-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Thiazolyl-4                              256 2-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Thiazolyl-4                             267 2-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Thiazolyl-4                             258 2-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Thiazolyl-4                             259 2-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Thiazolyl-4                              260 2-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Thiazolyl-4                              261 2-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Thiazolyl-4                              262 2-(4'-CN--C.sub.6 H.sub.4)-Thiazolyl-4                                     263 2-(3'-CN--C.sub.6 H.sub.4)-Thiazolyl-4                                     264 2-(2'-CN--C.sub.6 H.sub.4)-Thiazolyl-4                                     265 2-(4'-Cl--C.sub.6 H.sub.4)-Thiazolyl-4                                     266 2-(3'-Cl--C.sub.6 H.sub.4)-Thiazolyl-4                                     267 2-(2'-Cl--C.sub.6 H.sub.4)-Thiazolyl-4                                     268 N--CH.sub.3 -1,2,4-Triazolyl-5                                             269 3-CH.sub.3 --N--CH.sub.3 -1,2,4-Triazolyl-5                                270 3-C.sub.6 H.sub.5 --N--CH.sub.3 -1,2,4-Triazolyl-5                         271 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5                   272 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triaz               olyl-5                                                                 273 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5                   274 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Tria               zolyl-5                                                                275 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5                  276 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Tria               zolyl-5                                                                277 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5                   278 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triaz               olyl-5                                                                 279 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5                   280 3-(4'-CN--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5        281 3-(3'-CN--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5                 282 3-(2'-CN--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5                 283 3-(4'-Cl--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5                 284 3-(3'-Cl--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5                 285 3-(2'-Cl--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5                 286 1,3,4-Oxadiazolyl-2                                                        287 5-CH.sub.3 -1,3,4-Oxadiazolyl-2                                            288 5-C.sub.6 H.sub.5 -1,3,4-Oxadiazolyl-2                                     289 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                      290 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                      291 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                      292 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                     293 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                     294 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                     295 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                      296 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                      297 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                      298 5-(4'-CN--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                             299 5-(3'-CN--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                             300 5-(2'-CN--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                             301 5-(4'-Cl--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                             302 5-(3'-Cl--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                             303 5-(2'-Cl--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                             304 1,2,4-Oxadiazolyl-3                                                        305 5-CH.sub.3 -1,2,4-Oxadiazolyl-3                                            306 5-C.sub.6 H.sub.5 -1,2,4-Oxadiazolyl-3                                     307 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                      308 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                      309 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                      310 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                     311 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                     312 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                     313 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                      314 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                      315 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Oxa;diazolyl-3                     316 5-(4'-CN--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                             317 5-(3'-CN--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                             318 5-(2'-CN--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                             319 5-(4'-Cl--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                             320 5-(3'-Cl--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                             321 5-(2'-Cl--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                             322 1,2,4-Oxadiazolyl-5                                                        323 3-CH.sub.3 -1,2,4-Oxadiazolyl-5                                            324 3-C.sub.6 H.sub.5 -1,2,4-Oxadiazolyl-5                                     325 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                      326 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                      327 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                      328 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                     329 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                     330 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                     331 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                      332 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                      333 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                      334 3-(4'-CN--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                             335 3-(3'-CN--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                             336 3-(2'-CN--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                             337 3-(4'-Cl--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                             338 3-(3'-Cl--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                             339 3-(2'-Cl--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                             340 1,2,4-Thiadiazolyl-3                                                       341 5-CH.sub.3 -1,2,4-Thiadiazolyl-3                                           342 5-C.sub.6 H.sub.5 -1,2,4-Thiadiazolyl-3                                    343 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                     344 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                     345 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                     346 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                    347 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                    348 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                    349 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                     350 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                     351 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                     352 5-(4'-CN--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                            353 5-(3'-CN--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                            354 5-(2'-CN--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                            355 5-(4'-Cl--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                            356 5-(3'-Cl--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                            357 5-(2'-Cl--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                            358 1,3,4-Thiadiazolyl-2                                                       359 5-CH.sub.3 -1,3,4-Thiadiazolyl-2                                           360 5-C.sub.6 H.sub.5 -1,3,4-Thiadiazolyl-2                                    36i 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                     362 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                     363 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                     364 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                    365 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                    366 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                    367 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                     368 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                     369 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                     370 5-(4'-CN--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                            371 5-(3'-CN--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                            372 5-(2'-CN--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                            373 5-(4'-Cl--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                            374 5-(3'-Cl--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                            375 5-(2'-Cl--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                            376 Pyridinyl-2                                                                377 Pyridinyl-4                                                                378 Pyridazinyl-3                                                              379 Pyridazinyl-4                                                              380 Pyridazinyl-2                                                              381 Pyrimidinyl-4                                                              382 Pyrimidinyl-5                                                              383 Pyrimidinyl-2                                                              384 Pyridinyl-3                                                                385 1-Naphthyl                                                                 386 2-Naphthyl                                                               ______________________________________                                    

                  TABLE 10                                                         ______________________________________                                         1  STR180##                                                                      I: R.sup.1 = CH.sub.3                                                          II: R.sup.1 = CH.sub.2 --CH.sub.3                                              No.       Xm                                                                 ______________________________________                                         1       H                                                                        2 2-F                                                                          3 3-F                                                                          4 4-F                                                                          5 2,4-F.sub.2                                                                  6 2,4,6-F.sub.3                                                                7 2,3,4,5,6-F.sub.5                                                            8 2,3-F.sub.2                                                                  9 2-Cl                                                                         10 3-Cl                                                                        11 4-C1                                                                        12 2,3-Cl.sub.2                                                                13 2,4-Cl.sub.2                                                                14 2,5-Cl.sub.2                                                                15 2,6-Cl.sub.2                                                                16 3,4-Cl.sub.2                                                                17 3,5-Cl.sub.2                                                                18 2,3,4-Cl.sub.3                                                              19 2,3,5-Cl.sub.3                                                              20 2,3,6-Cl.sub.3                                                              21 2,4,5-Cl.sub.3                                                              22 2,4,6-Cl.sub.3                                                              23 3,4,5-Cl.sub.3                                                              24 2,3,4,6-Cl.sub.4                                                            25 2,3,5,6-Cl.sub.4                                                            26 2,3,4,5,6-Cl.sub.5                                                          27 2-Br                                                                        28 3-Br                                                                        29 4-Br                                                                        30 2,4-Br.sub.2                                                                31 2,5-Br.sub.2                                                                32 2,6-Br.sub.2                                                                33 2,4,6-Br.sub.3                                                              34 2,3,4,5,6-Br.sub.5                                                          35 2-I                                                                         36 3-I                                                                         37 4-I                                                                         38 2,4-I.sub.2                                                                 39 2-Cl, 3-F                                                                   40 2-Cl, 4-F                                                                   41 2-Cl, 5-F                                                                   42 2-Cl, 6-F                                                                   43 2-Cl, 3-Br                                                                  44 2-Cl, 4-Br                                                                  45 2-Cl, 5-Br                                                                  46 2-Cl, 6-Br                                                                  47 2-Br, 3-Cl                                                                  48 2-Br, 4-Cl                                                                  49 2-Br, 5-Cl                                                                  50 2-Br, 3-F                                                                   51 2-Br, 4-F                                                                   52 2-Br, 5-F                                                                   53 2-Br, 6-F                                                                   54 2-F, 3-Cl                                                                   55 2-F, 4-Cl                                                                   56 2-F, 5-Cl                                                                   57 3-Cl, 4-F                                                                   58 3-Cl, 5-F                                                                   59 3-Cl, 4-Br                                                                  60 3-Cl, 5-Br                                                                  61 3-F, 4-Cl                                                                   62 3-F, 4-Br                                                                   63 3-Br, 4-Cl                                                                  64 3-Br, 4-F                                                                   65 2,6-Cl.sub.2, 4-Br                                                          66 2-CH.sub.3                                                                  67 3-CH.sub.3                                                                  68 4-CH.sub.3                                                                  69 2,3-(CH.sub.3).sub.2                                                        70 2,4-(CH.sub.3).sub.2                                                        71 2,5-(CH.sub.3).sub.2                                                        72 2,6-(CH.sub.3).sub.2                                                        73 3,4-(CH.sub.3).sub.2                                                        74 3,5-(CH.sub.3).sub.2                                                        75 2,3,5-(CH.sub.3).sub.3                                                      76 2,3,4-(CH.sub.3).sub.3                                                      77 2,3,6-(CH.sub.3).sub.3                                                      78 2,4,5-(CH.sub.3).sub.3                                                      79 2,4,6-(CH.sub.3).sub.3                                                      80 3,4,5-(CH.sub.3).sub.3                                                      81 2,3,4,6-(CH.sub.3).sub.4                                                    82 2,3,5,6-(CH.sub.3).sub.4                                                    83 2,3,4,5,6-(CH.sub.3).sub.5                                                  84 2-C.sub.2 H.sub.5                                                           85 3-C.sub.2 H.sub.5                                                           86 4-C.sub.2 H.sub.5                                                           87 2,4-(C.sub.2 H.sub.5).sub.2                                                 88 2,6-(C.sub.2 H.sub.5).sub.2                                                 89 3,5-(C.sub.2 H.sub.5).sub.2                                                 90 2,4,6-(C2H5)3                                                               91 2-n-C.sub.3 H.sub.7                                                         92 3-n-C.sub.3 H.sub.7                                                         93 4-n-C.sub.3 H.sub.7                                                         94 2-i-C.sub.3 H.sub.7                                                         95 3-i-C.sub.3 H.sub.7                                                         96 4-i-C.sub.3 H.sub.7                                                         97 2,4-(i-C.sub.3 H.sub.7).sub.2                                               98 2,6-(i-C.sub.3 H.sub.7).sub.2                                               99 3,5-(i-C.sub.3 H.sub.7).sub.2                                               100 2,4,6-(i-C.sub.3 H.sub.7).sub.3                                            101 2-s-C.sub.4 H.sub.9                                                        102 3-s-C.sub.4 H.sub.9                                                        103 4-s-C.sub.4 H.sub.9                                                        104 2-t-C.sub.4 H.sub.9                                                        105 3-t-C.sub.4 H.sub.9                                                        106 4-t-C.sub.4 H.sub.9                                                        107 2,3-(t-C.sub.4 H.sub.9).sub.2                                              108 2,4-(t-C.sub.4 H.sub.9).sub.2                                              109 2,5-(t-C.sub.4 H.sub.9).sub.2                                              110 2,6-(t-C.sub.4 H.sub.9).sub.2                                              111 3,4-(t-C.sub.4 H.sub.9).sub.2                                              112 2,4,6-(t-C.sub.4 H.sub.9).sub.3                                            113 4-n-C.sub.9 H.sub.19                                                       114 4-n-C.sub.12 H.sub.25                                                      115 4-n-C.sub.15 H.sub.31                                                      116 4-(1,1,3,3-Tetramethylbutyl)                                               117 4-(2,4,4-Trimethylpropyl)                                                  118 2-t-C.sub.4 H.sub.9, 4-CH.sub.3                                            119 2-t-C.sub.4 H.sub.9, 5-CH.sub.3                                            120 2,6-(t-C.sub.4 H.sub.9).sub.2, 4-CH.sub.3                                  121 2-CH.sub.3, 4-t-C.sub.4 H.sub.9                                            122 2-CH.sub.3, 6-t-C.sub.4 H.sub.9                                            123 2-CH.sub.3, 4-i-C.sub.3 H.sub.7                                            124 2-CH.sub.3, 5-i-C.sub.3 H.sub.7                                            125 3-CH.sub.3, 4-i-C.sub.3 H.sub.7                                            126 2-i-C.sub.3 H.sub.7, 5-CH.sub.3                                            127 2,4-(t-C.sub.4 H.sub.9).sub.2, 6-i-C.sub.3 H.sub.7                         128 2-Allyl                                                                    129 3-Allyl                                                                    130 4-Allyl                                                                    131 2-Allyl, 6-CH.sub.3                                                        132 2-cyclo-C.sub.6 H.sub.11                                                   133 3-cyclo-C.sub.6 H.sub.11                                                   134 4-cyclo-C.sub.6 H.sub.11                                                   135 2,4-(cyclo-C.sub.6 H.sub.11).sub.2, 6-CH.sub.3                             136 2-CH.sub.3, 4-cyclo-C.sub.6 H.sub.11                                       137 2-CH.sub.2 --C.sub.6 H.sub.5                                               138 3-CH.sub.2 --C.sub.6 H.sub.5                                               139 4-CH.sub.2 --C.sub.6 H.sub.5                                               140 2-CH.sub.2 --C.sub.6 H.sub.5, 4-CH.sub.3                                   141 2-CH.sub.3, 4-CH.sub.2 --C.sub.6 H.sub.5                                   142 2-C.sub.6 H.sub.5                                                          143 3-C.sub.6 H.sub.5                                                          144 4-C.sub.6 H.sub.5                                                          145 4-(2-i-C.sub.3 H.sub.7 --C.sub.6 H.sub.4)                                  146 4-C.sub.6 H.sub.5, 2,6-(CH.sub.3).sub.2                                    147 2-Cl, 4-C.sub.6 H.sub.5                                                    148 2-Br, 4-C.sub.6 H.sub.5                                                    149 2-C.sub.6 H.sub.5, 4-Cl                                                    150 2-C.sub.6 H.sub.5, 4-Br                                                    151 2-CH.sub.2 C.sub.6 H.sub.5, 4-Cl                                           152 2-CH.sub.2 C.sub.6 H.sub.5, 4-Br                                           153 2-Cl, 4-CH.sub.2 C.sub.6 H.sub.5                                           154 2-Br, 4-CH.sub.2 C.sub.6 H.sub.5                                           155 2-cyclo-C.sub.6 H.sub.11, 4-Cl                                             156 2-cyclo-C.sub.6 H.sub.11, 4-Br                                             157 2-Cl, 4-cyclo-C.sub.6 H.sub.11                                             158 2-Br, 4-cyclo-C.sub.6 H.sub.11                                             159 2-OCH.sub.3                                                                160 3-OCH.sub.3                                                                161 4-OCH.sub.3                                                                162 2-OC.sub.2 H.sub.5                                                         163 3-O--C.sub.2 H.sub.5                                                       164 4-O--C.sub.2 H.sub.5                                                       165 2-O-n-C.sub.3 H.sub.7                                                      166 3-O-n-C.sub.3 H.sub.7                                                      167 4-O-n-C.sub.3 H.sub.7                                                      168 2-O-i-C.sub.3 H.sub.7                                                      169 3-O-i-C.sub.3 H.sub.7                                                      170 4-O-i-C.sub.3 H.sub.7                                                      171 2-O-n-C.sub.6 H.sub.13                                                     172 3-O-n-C.sub.6 H.sub.13                                                     173 4-O-n-C.sub.6 H.sub.13                                                     174 2-O-n-C.sub.8 H.sub.17                                                     175 3-O-n-C.sub.8 H.sub.17                                                     176 4-O-n-C.sub.8 H.sub.17                                                     177 2-O-CH.sub.2 C.sub.6 H.sub.5                                               178 3-O-CH.sub.2 C.sub.6 H.sub.5                                               179 4-O-CH.sub.2 C.sub.6 H.sub.5                                               180 2-O-(CH.sub.2).sub.3 C.sub.6 H.sub.5                                       181 3-O-(CH.sub.2).sub.3 C.sub.6 H.sub.5                                       182 4-O-(CH.sub.2).sub.3 C.sub.6 H.sub.5                                       183 2,4-(OCH.sub.3).sub.2                                                      184 2-CF.sub.3                                                                 185 3-CF.sub.3                                                                 186 4-CF.sub.3                                                                 187 2-OCF.sub.3                                                                188 3-OCF.sub.3                                                                189 4-OCF.sub.3                                                                190 3-OCH.sub.2 CHF.sub.2                                                      191 2-NO.sub.2                                                                 192 3-NO.sub.2                                                                 193 4-NO.sub.2                                                                 194 2-CN                                                                       195 3-CN                                                                       196 4-CN                                                                       197 2-CH.sub.3, 3-Cl                                                           198 2-CH.sub.3, 4-Cl                                                           199 2-CH.sub.3, 5-Cl                                                           200 2-CH.sub.3, 6-Cl                                                           201 2-CH.sub.3, 3-F                                                            202 2-CH.sub.3, 4-F                                                            203 2-CH.sub.3, 5-F                                                            204 2-CH.sub.3, 6-F                                                            205 2-CH.sub.3, 3-Br                                                           206 2-CH.sub.3, 4-Br                                                           207 2-CH.sub.3, 5-Br                                                           208 2-CH.sub.3, 6-Br                                                           209 2-Cl, 3-CH.sub.3                                                           210 2-Cl, 4-CH.sub.3                                                           211 2-Cl, 5-CH.sub.3                                                           212 2-F, 3-CH.sub.3                                                            213 2-F, 4-CH.sub.3                                                            214 2-F, 5-CH.sub.3                                                            215 2-Br, 3-CH.sub.3                                                           216 2-Br, 4-CH.sub.3                                                           217 2-Br, 5-CH.sub.3                                                           218 3-CH.sub.3, 4-Cl                                                           219 3-CH.sub.3, 5-Cl                                                           220 3-CH.sub.3, 4-F                                                            221 3-CH.sub.3, 5-F                                                            222 3-CH.sub.3, 4-Br                                                           223 3-CH.sub.3, 5-Br                                                           224 3-F, 4-CH.sub.3                                                            225 3-Cl, 4-CH3                                                                226 3-Br, 4-CH3                                                                227 2-Cl, 4,5-(CH.sub.3).sub.2                                                 228 2-Br, 4,5-(CH.sub.3).sub.2                                                 229 2-Cl, 3,5-(CH.sub.3).sub.2                                                 230 2-Br, 3,5-(CH.sub.3).sub.2                                                 231 2,6-Cl.sub.2, 4-CH.sub.3                                                   232 2,6-F.sub.2, 4-CH.sub.3                                                    233 2,6-Br.sub.2, 4-CH.sub.3                                                   234 2,4-Br.sub.2, 6-CH.sub.3                                                   235 2,4-F.sub.2, 6-CH.sub.3                                                    236 2,4-Br.sub.2, 6-CH.sub.3                                                   237 2,6-(CH.sub.3).sub.2, 4-F                                                  238 2,6-(CH.sub.3).sub.2, 4-Cl                                                 239 2,6-(CH.sub.3).sub.2, 4-Br                                                 240 3,5-(CH.sub.3).sub.2, 4-F                                                  241 3,5-(CH.sub.3).sub.2, 4-Cl                                                 242 3,5-(CH.sub.3).sub.2, 4-Br                                                 243 2,3,6-(CH.sub.3).sub.3, 4-F                                                244 2,3,6-(CH.sub.3).sub.3, 4-Cl                                               245 2,3,6-(CH.sub.3).sub.3, 4-Br                                               246 2,4-(CH.sub.3).sub.2, 6-F                                                  247 2,4-(CH.sub.3).sub.2, 6-Cl                                                 248 2,4-(CH.sub.3).sub.2, 6-Br                                                 249 2-i-C.sub.3 H.sub.7, 4-Cl, 5-CH.sub.3                                      250 2-Cl, 4-NO.sub.2                                                           251 2-NO.sub.2, 4-Cl                                                           252 2-OCH.sub.3, 5-NO.sub.2                                                    253 2,4-Cl.sub.2, 5-NO.sub.2                                                   254 2,4-Cl.sub.2, 6-NO.sub.2                                                   255 2,6-Cl.sub.2, 4-NO.sub.2                                                   256 2,6-Br.sub.2, 4-NO.sub.2                                                   257 2,6-I.sub.2 , 2,4-NO.sub.2                                                 258 2-CH.sub.3, 5-i-C.sub.3 H.sub.7, 4-Cl                                      259 2-CO.sub.2 CH.sub.3                                                        260 3-CO.sub.2 CH.sub.3                                                        261 4-CO.sub.2 CH.sub.3                                                        262 2-CO.sub.2 (C.sub.2 H.sub.5)                                               263 3-CO.sub.2 (C.sub.2 H.sub.5)                                               264 4-CO.sub.2 (C.sub.2 H.sub.5)                                               265 2-CO.sub.2 (n-C.sub.3 H.sub.7)                                             266 3-CO.sub.2 (n-C.sub.3 H.sub.7)                                             267 4-CO.sub.2 (n-C.sub.3 H.sub.7)                                             268 2-CO.sub.2 (i-C.sub.3 H.sub.7)                                             269 3-CO.sub.2 (i-C.sub.3 H.sub.7)                                             270 4-CO.sub.2 (i-C.sub.3 H.sub.7)                                             271 2-CO.sub.2 (n-C.sub.6 H.sub.13)                                            272 3-CO.sub.2 (n-C.sub.6 H.sub.13)                                            273 4-CO.sub.2 (n-C.sub.6 H.sub.13)                                            274 2-CH.sub.2 --OCH.sub.3                                                     275 3-CH.sub.2 --OCH.sub.3                                                     276 4-CH.sub.2 --OCH.sub.3                                                     277 2-CH.sub.2 O(C.sub.2 H.sub.5)                                              278 3-CH.sub.2 O(C.sub.2 H.sub.5)                                              279 4-CH.sub.2 O(C.sub.2 H.sub.5)                                              280 2-CH.sub.2 O(n-C.sub.3 H.sub.7)                                            281 3-CH.sub.2 O(n-C.sub.3 H.sub.7)                                            282 4-CH.sub.2 O(n-C.sub.3 H.sub.7)                                            283 2-CH.sub.2 O(i-C.sub.3 H.sub.7)                                            284 3-CH.sub.2 O(i-C.sub.3 H.sub.7)                                            285 4-CH.sub.2 O(i-C.sub.3 H.sub.7)                                            286 2-CHO                                                                      287 3-CHO                                                                      288 4-CHO                                                                      289 2-CO--CH.sub.3                                                             290 3-CO--CH.sub.3                                                             291 4-CO--CH.sub.3                                                             292 2-CO--CH.sub.2 --CH.sub.3                                                  293 3-CO--CH.sub.2 --CH.sub.3                                                  294 4-CO--CH.sub.2 --CH.sub.3                                                  295 2-CO--CH.sub.2 --CH.sub.2 --CH.sub.3                                       296 3-CO--CH.sub.2 --CH.sub.2 --CH.sub.3                                       297 4-CO--CH.sub.2 --CH.sub.2 --CH.sub.3                                       298 2-CO--CH(CH.sub.3)--CH.sub.3                                               299 3-CO--CH(CH.sub.3)--CH.sub.3                                               300 4-CO--CH(CH.sub.3)--CH.sub.3                                               301 2-Me-4-CHO                                                                 302 2-Me-4-CH.sub.3 --CO                                                       303 2-Me-4-CH.sub.3 --CH.sub.2 --CO                                            304 2-Me-4-CH.sub.3 --CH.sub.2 --CH.sub.2 --CO                                 305 2-Me-4-CH.sub.3 --CH (CH.sub.3)--CO                                        306 2,5-Me.sub.2 -4-CHO                                                        307 2,5-Me.sub.2 -4-CH.sub.3 --CO                                              308 2,5-Me.sub.2 -4-CH.sub.3 --CH.sub.2 --CO                                   309 2,5-Me.sub.2 -4-CH.sub.3 --CH.sub.2 --CH.sub.2 --CO                        310 2,5-Me.sub.2 -4-CH.sub.3 --CH(CH.sub.3)--CO                                311 2-Cl-4-CHO                                                                 312 2-Cl-4-CH.sub.3 --CO                                                       313 2-Cl-4-CH.sub.3 --CH.sub.2 --CO                                            314 2-Cl-4-CH.sub.3 --CH(CH.sub.3)--CO                                         315 2,5-Cl.sub.2 -4-CHO                                                        316 2,5-Cl.sub.2 -4-CH.sub.3 --CO                                              317 2,5-Cl.sub.2 -4-CH.sub.3 --CH.sub.2 --CO                                   318 2,5-Cl.sub.2 -4-CH.sub.3 --CH.sub.2 --CH.sub.2 --CO                        319 2,5-Cl.sub.2 -4-CH.sub.3 --CH (CH.sub.3)--CO                               320 2-C(═NOCH.sub.3)--CH.sub.3                                             321 3-C(═NOCH.sub.3)--CH.sub.3                                             322 4-C(═NOCH.sub.3)--CH.sub.3                                             323 2-C(═NOC.sub.2 H.sub.5)--CH.sub.3                                      324 3-C(═NOC.sub.2 H.sub.5)--CH.sub.3                                      325 4-C(═NOC.sub.2 H.sub.5)--CH.sub.3                                      326 2-C(═NO-n-C.sub.3 H.sub.7)--CH.sub.3                                   327 3-C(═NO-n-C.sub.3 H.sub.7)--CH.sub.3                                   328 4-C(═NO-n-C.sub.3 H.sub.7)--CH.sub.3                                   329 2-C(═NO-i-C.sub.3 H.sub.7)--CH.sub.3                                   330 3-C(═NO-i-C.sub.3 H.sub.7)--CH.sub.3                                   331 4-C(═NO-i-C.sub.3 H.sub.7)--CH.sub.3                                   332 2-C(═NO-Allyl)-CH.sub.3                                                333 3-C(═NO-Allyl)-CH.sub.3                                                334 4-C(═NO-Allyl)-CH.sub.3                                                335 2-C═NO-trans-Chloroallyl)-CH.sub.3                                     336 3-C(═NO-trans-Chloroallyl)-CH.sub.3                                    337 4-C(═NO-trans-Chloroallyl)-CH.sub.3                                    338 2-C(═NO-Propargyl)-CH.sub.3                                            339 3-C(═NO-Propargyl)-CH.sub.3                                            340 4-C(═NO-Propargyl)-CH.sub.3                                            341 2-C(═NO-n-C.sub.4 H.sub.9)--CH.sub.3                                   342 3-C(═NO-n-C.sub.4 H.sub.9)--CH.sub.3                                   343 4-C(═NO-n-C.sub.4 H.sub.9)--CH.sub.3                                   344 2-C(═NO--CH.sup.2 --C.sup.6 H.sup.5)--CH.sub.3                         345 3-C(═NO--CH.sub.2 --C.sub.6 H.sub.5)--CH.sub.3                         346 4-C(═NO--CH.sub.2 --C.sub.6 H.sub.5)--CH.sub.3                         347 2-CH.sub.3 -4-CH═NOCH.sub.3                                            348 2-CH.sub.3 -4-CH═NOC.sub.2 H.sub.5                                     349 2-CH.sub.3 -4-CH═NC-n-C.sub.3 H.sub.7                                  350 2-CH.sub.3 -4-CH═NO-i-C.sub.3 H.sub.7                                  351 2-CH.sub.3 -4-CH═NO-Allyl                                              352 2-CH.sub.3 -4-CH═NO-(trans-Chloroallyl)                                353 2-CH.sub.3 -4-CH═NO-Propargyl                                          354 2-CH.sub.3 -4-CH═NO-n-C.sub.4 H.sub.9                                  355 2-CH.sub.3 -4-CH═NO--CH.sub.2 --C.sub.6 H.sub.5                        356 2-CH.sub.3 -4-(CH.sub.3 --C═NOCH.sub.3)                                357 2-CH.sub.3 -4-(CH.sub.3 --C═NOC.sub.2 H.sub.5)                         358 2-CH.sub.3 -4-(CH.sub.3 --C═NO-n-C.sub.3 H.sub.7)                      359 2-CH.sub.3 -4-(CH.sub.3 --C═NO-i-C.sub.3 H.sub.7)                      360 2-CH.sub.3 -4-(CH.sub.3 --C═NO-Allyl)                                  361 2-CH.sub.3 -4-(CH.sub.3 --C═NO-trans-Chloroallyl)                      362 2-CH.sub.3 -4-(CH.sub.3 --C═NO-Propargyl)                              363 2-CH.sub.3 -4-(CH.sub.3 --C═NO-n-C.sub.4 H.sub.9)                      364 2-CH.sub.3 -4-(CH.sub.3 --C═NO--CH.sub.2 --C.sub.6 H.sub.5)                   365 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C═NO--CH.sub.3)                       366 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C═NO--C.sub.2 H.sub.5)                367 2-CH.sub.3 -4-(C.sub.2 H.sub.5 -C═NO-n-C.sub.3 H.sub.7)                368 2-CH.sub.3 -4-(C.sub.2 H.sub.5 -C═NO-i-C.sub.3 H.sub.7                 369 2-CH.sub.3 -4-(C.sub.2 H.sub.5 -C═NO-Allyl                      370 2-CH.sub.3 -4-(C.sub.2 H.sub.5 -C═NO-trans-Chloroallyl)                       371 2-CH.sub.3 -4-(C.sub.2 H.sub.5 -C═NO-Propagyl)                  372 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C═NO-n-C.sub.4 H.sub.9)                      373 2-CH.sub.3 -4-(C.sub.2 H.sub.5 -C═NO--CH.sub.2 --C.sub.6              H.sub.5)                                                                 374 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C═NOCH.sub.3)                      375 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C═NOC.sub.2 H.sub.5)                      376 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C═NO-n-C.sub.3                    H.sub.7)                                                                 377 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C═NO-i-C.sub.3 H.sub.7)                   378 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C═NO-Allyl)                 379 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C═NO-trans-Chloroal-                       lyl)                                                                   380 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C═NO-Proparyl)                     381 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C═NO-n-C.sub.4 H.sub.9)                   382 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C═NO-CH.sub.2                     --C.sub.6 H.sub.5)                                                       383 2-C.sub.6 H.sub.5                                                          384 3-C6H5                                                                     385 4-C6H5                                                                     386 2-(2'-F--C6H4)                                                             387 2-(3'-F--C.sub.6 H.sub.4)                                                  388 2-(4'-F--C.sub.6 H.sub.4)                                                  389 3-(2'-F--C.sub.6 H.sub.4)                                                  390 3-(3'-F--C.sub.6 H.sub.4)                                                  391 3-(4'-F--C.sub.6 H.sub.4)                                                  392 4-(2'-F--C.sub.6 H.sub.4)                                                  393 4-(3'-F--C.sub.6 H.sub.4)                                                  394 4-(4'-F--C.sub.6 H.sub.4)                                                  395 2-(2'-Cl--C.sub.6 H.sub.4)                                                 396 2-(3'-Cl--C.sub.6 H.sub.4)                                                 397 2-(4'-Cl--C.sub.6 H.sub.4)                                                 398 3-(2'-Cl--C6H4)                                                            399 3-(3'-Cl--C.sub.6 H.sub.4)                                                 400 3-(4'-Cl--C.sub.6 H.sub.4)                                                 401 4-(2'-Cl--C.sub.6 H.sub.4)                                                 402 4-(3'-Cl--C.sub.6 H.sub.4)                                                 403 4-(4'-Cl--C.sub.6 H.sub.4)                                                 405 2-(2'-CH.sub.3 --C.sub.6 H.sub.4)                                          406 2-(3'-CH.sub.3 --C.sub.6 H.sub.4)                                          407 2-(4'-CH.sub.3 --C.sub.6 H.sub.4)                                          408 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)                                          409 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)                                          410 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)                                          411 4-(2'-CH.sub.3 --C.sub.6 H.sub.4)                                          412 4-(3'-CH.sub.3 --C.sub.6 H.sub.4)                                          413 4-(4'-CH.sub.3 --C.sub.6 H.sub.4)                                          414 2-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                      415 2-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                      416 2-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                      417 3-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                      418 3-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                      419 3-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                      420 4-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                      421 4-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                      422 4-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                      423 2-(2'-(CH.sub.3 --C(═NOAllyl))-C.sub.6 H.sub.4)                        424 2-(3'-(CH.sub.3 --C(═NOAllyl))-C.sub.6 H.sub.4)                        425 2-(4'-(CH.sub.3 --C(═NOAllyl))-C.sub.6 H.sub.4)                        426 3-(2'-(CH.sub.3 --C(═NOAllyl))-C.sub.6 H.sub.4)                        427 3-(3'-(CH.sub.3 --C(═NOAllyl))-C.sub.6 H.sub.4)                        428 3-(4'-(CH.sub.3 --C(═NOAllyl))-C.sub.6 H.sub.4)                        429 4-(2'-(CH.sub.3 --C(═NOAllyl))-C.sub.6 H.sub.4)                        430 4-(3'-(CH.sub.3 --C(═NOAllyl))-C.sub.6 H.sub.4)                        431 4-(4'-(CH.sub.3 --C(═NOAllyl))-C.sub.6 H.sub.4)                        432 2-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                                 433 2-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                                 434 2-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                                 435 3-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                                 436 3-(3'-CH3O2C--C6H4)                                                        437 3-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                                 438 4-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                                 439 4-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                                 440 4-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                                 441 2-(2'-CH.sub.3 O--C.sub.6 H.sub.4)                                         442 2-(3'-CH.sub.3 O--C.sub.6 H.sub.4)                                         443 2-(4'-CH.sub.3 O--C.sub.6 H.sub.4)                                         444 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)                                         445 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)                                         446 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)                                         447 4-(2'-CH.sub.3 O--C.sub.6 H.sub.4)                                         448 4-(3'-CH.sub.3 O--C.sub.6 H.sub.4)                                         449 4-(4'-CH.sub.3 O--C.sub.6 H.sub.4)                                         450 2-(2'-O.sub.2 N--C.sub.6 H.sub.4)                                          451 2-(3'-O.sub.2 N--C.sub.6 H.sub.4)                                          452 2-(4'-O.sub.2 N--C.sub.6 H.sub.4)                                          453 3-(2'-O.sub.2 N--C.sub.6 H.sub.4)                                          454 3-(3'-O.sub.2 N--C.sub.6 H.sub.4)                                          455 3-(4'-O.sub.2 N--C.sub.6 H.sub.4)                                          456 4-(2'-O.sub.2 N--C.sub.6 H.sub.4)                                          457 4-(3'-O.sub.2 N--C.sub.6 H.sub.4)                                          458 4-(4'-O.sub.2 N--C.sub.6 H.sub.4)                                          459 2-(2'-NC--C.sub.6 H.sub.4)                                                 460 2-(3'-NC--C.sub.6 H.sub.4)                                                 461 2-(4'-NC--C.sub.6 H.sub.4)                                                 462 3-(2'-NC--C.sub.6 H.sub.4)                                                 463 3-(3'-NC--C.sub.6 H.sub.4)                                                 464 3-(4'-NC--C.sub.6 H.sub.4)                                                 465 4-(2'-NC--C.sub.6 H.sub.4)                                                 466 4-(3'-NC--C.sub.6 H.sub.4)                                                 467 4-(4'-NC--C.sub.6 H.sub.4)                                                 468 2-(2'-CF.sub.3 --C.sub.6 H.sub.4)                                          469 2-(3'-CF.sub.3 --C.sub.6 H.sub.4)                                          470 2-(4'-CF.sub.3 --C.sub.6 H.sub.4)                                          471 3-(2'-CF.sub.3 --C.sub.6 H.sub.4)                                          472 3-(3'-CF.sub.3 --C.sub.6 H.sub.4)                                          473 3-(4'-CF.sub.3 --C.sub.6 H.sub.4)                                          474 4-(2'-CF.sub.3 --C.sub.6 H.sub.4)                                          475 4-(3'-CF.sub.3 --C.sub.6 H.sub.4)                                          476 4-(4'-CF.sub.3 --C.sub.6 H.sub.4)                                          477 2-O--C.sub.6 H.sub.5                                                       475 3-O--C6H5                                                                  476 4-O--C6H5                                                                  478 2-O-(2'-F--C6H4)                                                           479 2-O-(3'-F--C.sub.6 H.sub.4)                                                480 2-O-(4'-F--C.sub.6 H.sub.4)                                                481 3-O-(2'-F--C.sub.6 H.sub.4)                                                482 3-O-(3'-F--C.sub.6 H.sub.4)                                                483 3-O-(4'-F--C.sub.6 H.sub.4)                                                484 4-O-(2'-F--C.sub.6 H.sub.4)                                                485 4-O-(3'-F--C.sub.6 H.sub.4)                                                486 4-O-(4'-F--C.sub.6 H.sub.4)                                                487 2-O-(2'-Cl--C.sub.6 H.sub.4)                                               488 2-O-(3'-Cl--C.sub.6 H.sub.4)                                               489 2-O-(4'-Cl--C.sub.6 H.sub.4)                                               490 3-O-(2'-Cl--C.sub.6 H.sub.4)                                               491 3-O-(3'-Cl--C.sub.6 H.sub.4)                                               492 3-C-(4'-Cl--C.sub.6 H.sub.4)                                               493 3-O-(4'-Cl--C.sub.6 H.sub.4)                                               494 4-O-(2'-Cl--C.sub.6 H.sub.4)                                               495 4-O-(3'-Cl--C.sub.6 H.sub.4)                                               496 4-O-(4'-Cl--C.sub.6 H.sub.4)                                               497 2-O-(2'-CH.sub.3 --C.sub.6 H.sub.4)                                        498 2-O-(3'-CH.sub.3 --C.sub.6 H.sub.4)                                        499 2-O-(4'-CH.sub.3 --C.sub.6 H.sub.4)                                        500 3-O-(2'-CH.sub.3 --C.sub.6 H.sub.4)                                        501 3-O-(3'-CH.sub.3 --C.sub.6 H.sub.4)                                        502 3-O-(4'-CH.sub.3 --C.sub.6 H.sub.4)                                        503 4-O-(2'-CH.sub.3 --C.sub.6 H.sub.4)                                        504 4-O-(3'-CH.sub.3 --C.sub.6 H.sub.4)                                        505 4-O-(4'-CH.sub.3 --C.sub.6 H.sub.4)                                        506 2-O-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                    507 2-O-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                    508 2-O-(4'-CH3--CO--C6H4)                                                     509 3-O-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                    510 3-O-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                    511 3-O-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                    512 4-O-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                    513 4-O-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                    514 4-O-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                    515 2-O-(2'-(CH.sub.3 --C(═NOAllyl))-C.sub.6 H.sub.4)                      516 2-O-(3'-(CH.sub.3 --C(═NOAllyl))-C.sub.6 H.sub.4)                      517 2-O-(4'-(CH.sub.3 --C(═NOAllyl))-C.sub.6 H.sub.4)                      518 3-O-(2'-(CH.sub.3 --C(═NOAllyl))-C.sub.6 H.sub.4)                      519 3-O-(3'-(CH.sub.3 --C(═NOAllyl))-C.sub.6 H.sub.4)                      520 3-O-(4'-(CH.sub.3 --C(═NOAllyl))-C.sub.6 H.sub.4)                      521 4-O-(2'-(CH.sub.3 --C(═NOAllyl))-C.sub.6 H.sub.4)                      522 4-O-(3'-(CH.sub.3 --C(═NOAllyl))-C.sub.6 H.sub.4)                      523 4-O-(4'-(CH.sub.3 --C(═NOAllyl))-C.sub.6 H.sub.4)                      524 2-O-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                               525 2-O-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                               526 2-O-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                               527 3-O-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                               528 3-O-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                               529 3-O-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                               530 4-O-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                               531 4-O-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                               532 4-O-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                               533 2-O-(2'-CH.sub.3 O--C.sub.6 H.sub.4)                                       534 2-O-(3'-CH.sub.3 O--C.sub.6 H.sub.4)                                       535 2-O-(4'-CH.sub.3 O--C.sub.6 H.sub.4)                                       536 3-O-(2'-CH.sub.3 O--C.sub.6 H.sub.4)                                       537 3-O-(3'-CH.sub.3 O--C.sub.6 H.sub.4)                                       538 3-O-(4'-CH.sub.3 O--C.sub.6 H.sub.4)                                       539 4-O-(2'-CH.sub.3 O--C.sub.6 H.sub.4)                                       540 4-O-(3'-CH.sub.3 O--C.sub.6 H.sub.4)                                       541 4-O-(4'-CH.sub.3 O--C.sub.6 H.sub.4)                                       542 2-O-(2'-O.sub.2 N--C.sub.6 H.sub.4)                                        543 2-O-(3'-O.sub.2 N--C.sub.6 H.sub.4)                                        544 2-O-(4'-O.sub.2 N--C.sub.6 H.sub.4)                                        545 3-O-(2'-O.sub.2 N--C.sub.6 H.sub.4)                                        546 3-O-(3'-O.sub.2 N--C.sub.6 H.sub.4)                                        547 3-O-(4'-O.sub.2 N--C.sub.6 H.sub.4)                                        548 4-O-(2'-O.sub.2 N--C.sub.6 H.sub.4)                                        549 4-O-(3'-O.sub.2 N--C.sub.6 H.sub.4)                                        550 4-O-(4'-O.sub.2 N--C.sub.6 H.sub.4)                                        551 2-O-(2'-NC--C.sub.6 H.sub.4)                                               552 2-O-(3'-NC--C.sub.6 H.sub.4)                                               553 2-O-(4'-NC--C.sub.6 H.sub.4)                                               554 3-O-(2'-NC--C.sub.6 H.sub.4)                                               555 3-O-(3'-NC--C.sub.6 H.sub.4)                                               556 3-O-(4'-NC--C.sub.6 H.sub.4)                                               557 4-O-(2'-NC--C.sub.6 H.sub.4)                                               558 4-O-(3'-NC--C.sub.6 H.sub.4)                                               559 4-O-(4'-NC--C.sub.6 H.sub.4)                                               560 2-O-(2'-CF.sub.3 --C.sub.6 H.sub.4)                                        561 2-O-(3'-CF.sub.3 --C.sub.6 H.sub.4)                                        562 2-O-(4'-CF.sub.3 --C.sub.6 H.sub.4)                                        563 3-O-(2'-CF.sub.3 --C.sub.6 H.sub.4)                                        564 3-O-(3'-CF.sub.3 --C.sub.6 H.sub.4)                                        565 3-O-(4'-CF.sub.3 --C.sub.6 H.sub.4)                                        566 4-O-(2'-CF.sub.3 --C.sub.6 H.sub.4)                                        567 4-O-(3'-CF.sub.3 --C.sub.6 H.sub.4)                                        568 4-O-(4'-CF.sub.3 --C.sub.6 H.sub.4)                                        569 2-Pyridinyl-2'                                                             570 2-Pyridinyl-3'                                                             571 2-Pyridinyl-4'                                                             572 3-Pyridinyl-2'                                                             573 3-Pyridinyl-3'                                                             574 3-Pyridinyl-4'                                                             575 4-Pyridinyl-2'                                                             576 4-Pyridinyl-3'                                                             577 4-Pyridinyl-4'                                                             578 2-Pyrimidinyl-2'                                                           579 2-Pyrimidinyl-3'                                                           580 2-Pyrimidinyl-4'                                                           581 3-Pyrimidinyl-2'                                                           582 3-Pyrimidinyl-3'                                                           583 3-Pyrimidinyl-4'                                                           584 4-Pyrimidinyl-2'                                                           585 4-Pyrimidinyl-3'                                                           586 4-Pyrimidinyl-4'                                                           587 2-Pyrazolyl-1'                                                             588 2-Pyrazolyl-3'                                                             589 2-Pyrazolyl-4'                                                             590 3-Pyrazolyl-1'                                                             591 3-Pyrazolyl-3'                                                             592 3-Pyrazolyl-4'                                                             593 4-Pyrazolyl-1'                                                             594 4-Pyrazolyl-3'                                                             595 4-Pyrazolyl-4'                                                             596 2-Isoxazolyl-3'                                                            597 2-Isoxazolyl-4'                                                            598 2-Isoxazolyl-5'                                                            599 3-Isoxazolyl-3'                                                            600 3-Isoxazolyl-4'                                                            601 3-Isoxazolyl-5'                                                            602 4-Isoxazolyl-3'                                                            603 4-Isoxazolyl-4'                                                            604 4-Isoxazolyl-5'                                                            605 2-Isothiazolyl-3'                                                          606 2-Isothiazolyl-4'                                                          607 2-Isothiazolyl-5'                                                          608 3-Isothiazolyl-3'                                                          609 3-Isothiazolyl-4'                                                          610 3-Isothiazolyl-5'                                                          611 4-Isothiazolyl-3'                                                          612 4-Isothiazolyl-4'                                                          613 4-Isothiazolyl-5'                                                          614 2-Imidazolyl-1'                                                            615 2-Imidazolyl-2'                                                            616 2-Imidazolyl-4'                                                            617 3-Imidazolyl-1'                                                            618 3-Imidazolyl-2'                                                            619 3-Imidazolyl-4'                                                            620 4-Imidazolyl-1'                                                            621 4-Imidazolyl-2'                                                            622 4-Imidazolyl-4'                                                            623 2-Oxazolyl-2'                                                              624 2-Oxazolyl-4'                                                              625 2-Oxazolyl-5'                                                              626 3-Oxazolyl-2'                                                              627 3-Oxazolyl-4'                                                              628 3-Oxazolyl-5'                                                              629 4-Oxazolyl-2'                                                              630 4-Oxazolyl-4'                                                              631 4-Oxazolyl-5'                                                              632 2-Thiazolyl-2'                                                             633 2-Thiazolyl-4'                                                             634 2-Thiazolyl-5'                                                             635 3-Thiazolyl-2'                                                             636 3-Thiazolyl-4'                                                             637 3-Thiazolyl-5'                                                             638 4-Thiazolyl-2'                                                             639 4-Thiazolyl-4'                                                             640 4-Thiazolyl-5'                                                             641 2-CH.sub.3 -4-(CH.sub.3 --C═N--O--CH.sub.2 --CH.sub.2 --OCH.sub.             3)                                                                       642 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C═N--O--CH.sub.2 --CH.sub.2                 --OCH.sub.3)                                                             643 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C═N--O--CH.sub.2 --CH.sub.2              --OCH.sub.3)                                                             644 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C═N--OCH.sub.3)                     645 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C═N--OC.sub.2 H.sub.5)                     646 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C═N--O-n-C.sub.3                   H.sub.7)                                                                 647 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C═N--O-i-C.sub.3 H.sub.7)                  648 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C═N--O-Allyl)                       649 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C═N--O-trans-Chloroall             yl)                                                                      650 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C═N--O-Propargyl)                   651 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C═N--O-n-C.sub.4 H.sub.9)                  652 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C═N--O--CH.sub.2                   --C.sub.6 H.sub.5)                                                       653 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C═N--OCH.sub.3)                     654 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C═N--OC.sub.2 H.sub.5)                     655 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C═N--O-n-C.sub.3                   H.sub.7)                                                                 656 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C═N--O-i-C.sub.3 H.sub.7)                  657 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C═N--O-Allyl)                       658 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C═N--O-trans-Chloroall             yl)                                                                      659 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C═N--O-Proparoyl)                   660 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C═N--O-n-C.sub.4 H.sub.9)                  661 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C═N--O--CH.sub.2                   --C.sub.6 H.sub.5)                                                       662 2-O-n-C.sub.4 H.sub.9                                                      663 2-O-i-C.sub.4 H.sub.9                                                      664 2-O-s-C.sub.4 H.sub.9                                                      665 2-O-t-C.sub.4 H.sub.9                                                      666 2-Neopentyloxy                                                             667 3-O-n-C.sub.4 H.sub.9                                                      668 3-O-i-C.sub.4 H.sub.9                                                      669 3-O-s-C.sub.4 H.sub.9                                                      670 3-O-t-C.sub.4 H.sub.9                                                      671 3-Neopentyloxy                                                             672 4-O-n-C.sub.4 H.sub.9                                                      673 4-O-i-C.sub.4 H.sub.9                                                      674 4-O-s-C.sub.4 H.sub.9                                                      675 4-O-t-C.sub.4 H.sub.                                                       676 4-Neopentyloxy                                                             677 3-CH.sub.3 -4-OCH.sub.3                                                    678 3-CH.sub.3 -4-OC.sub.2 H.sub.5                                             679 3-CH.sub.3 -4-O-n-C.sub.3 H.sub.7                                          680 3-COH.sub.3 -4-O-n-C.sub.4 H.sub.9                                         681 3-CH.sub.3 -4-O-i-C.sub.4 H.sub.9                                          682 3-CH.sub.3 -4-O-s-C.sub.4 H.sub.9                                          683 3-CH.sub.3 -4-O-t-C.sub.4 H.sub.9                                          684 3-CH.sub.3 -4-Neopentyloxy                                                 685 2-CH.sub.3 -3-OCH.sub.3                                                    686 2-CH.sub.3 -4-OCH.sub.3                                                    687 2-CH.sub.3 -5-OCH.sub.3                                                    688 2-CH.sub.3 -6-OCH.sub.3                                                    689 3-CH.sub.3 -4-OOH.sub.3                                                    690 3-CH.sub.3 -5-OCH.sub.3                                                    691 3-CH.sub.3 -6-OCH.sub.3                                                    692 4-CH.sub.3 -5-O--CH.sub.3                                                  693 4-CH.sub.3 -6-O--CH.sub.3                                                  694 4-CH.sub.3 -6-OCH.sub.3                                                    695 2-CH.sub.3 -3-O-i-C.sub.3 H.sub.7                                          696 2-CH.sub.3 -4-O-i-C.sub.3 H.sub.7                                          697 2-CH.sub.3 -5-O-i-C.sub.3 H.sub.7                                          698 2-CH.sub.3 -6-O-i-C.sub.3 H.sub.7                                          699 3-CH.sub.3 -4-O-i-C.sub.3 H.sub.7                                          700 3-CH.sub.3 -5-O-i-C.sub.3 H.sub.7                                          701 3-CH.sub.3 -6-O-i-C.sub.3 H.sub.7                                          702 4-CH.sub.3 -5-O-i-C.sub.3 H.sub.7                                          703 4-CH.sub.3 -6-O-i-C.sub.3 H.sub.7                                          704 5-CH.sub.3 -6-C-i-C.sub.3 H.sub.7                                          705 2-Cl-3-OCH.sub.3                                                           706 2-Cl-4-OCH.sub.3                                                           707 2-Cl-5-OCH.sub.3                                                           708 2-Cl-6-OCH.sub.3                                                           709 3-Cl-4-OCH.sub.3                                                           710 3-Cl-5-OCH.sub.3                                                           711 3-Cl-6-OCH.sub.3                                                           712 4-Cl-5-OCH.sub.3                                                           713 4-Cl-6-OCH.sub.3                                                           714 5-Cl-6-OCH.sub.3                                                         ______________________________________                                    

                  TABLE 11                                                         ______________________________________                                         2  STR181##                                                                      I: R.sup.1 = CH.sub.3                                                          II: R.sup.1 = CH.sub.2 --CH.sub.3                                              No.       B                                                                  ______________________________________                                         1       Pyrrolyl-3                                                               2 N--CH.sub.3 -Pyrrolyl-3                                                      3 N--C.sub.6 H.sub.5 -Pyrrolyl-3                                               4 N-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrrolyl-3                                 5 N-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrrolyl-3                                 6 N-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrrolyl-3                                 7 N-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrrolyl-3                                8 N-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrrolyl-3                                9 N-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrrolyl-3                                10 N-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrrolyl-3                                11 N-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrrolyl-3                                12 N-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrrolyl-3                                13 N-(4'-CN--C.sub.6 H.sub.4)-Pyrrolyl-3                                       14 N-(3'-CN--C.sub.6 H.sub.4)-Pyrrolyl-3                                       15 N-(2'-CN--C.sub.6 H.sub.4)-Pyrrolyl-3                                       16 N-(4'-Cl--C.sub.6 H.sub.4)-Pyrrolyl-3                                       17 N-(3'-Cl--C.sub.6 H.sub.4)-Pyrrolyl-3                                       18 N-(2'-Cl--C.sub.6 H.sub.4)-Pyrrolyl-3                                       19 Pyrrolyl-2                                                                  20 N--CH.sub.3 -Pyrrolyl-2                                                     21 N--C.sub.6 H.sub.5 -Pyrrolyl-2                                              22 N-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrrolyl-2                                23 N-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrrolyl-2                                24 N-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrrolyl-2                                25 N-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrrolyl-2                               26 N-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrrolyl-2                               27 N-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrrolyl-2                               28 N-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrrolyl-2                                29 N-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrrolyl-2                                30 N-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrrolyl-2                                31 N-(4'-CN--C.sub.6 H.sub.4)-Pyrrolyl-2                                       32 N-(3'-CN--C.sub.6 H.sub.4)-Pyrrolyl-2                                       33 N-(2'-CN--C.sub.6 H.sub.4)-Pyrrolyl-2                                       34 N-(4'-Cl--C.sub.6 H.sub.4)-Pyrrolyl-2                                       35 N-(3'-Cl--C.sub.6 H.sub.4)-Pyrrolyl-2                                       36 N-(2'-Cl--C.sub.6 H.sub.4)-Pyrrolyl-2                                       37 Furyl-2                                                                     38 5-CH.sub.3 -Furyl-2                                                         39 5-C.sub.6 H.sub.5 -Furyl-2                                                  40 5-(4'-CH.sub.3 --C.sub.6 H.sub.4 -Furyl-2                                   41 5-(3'-CH.sub.3 --C.sub.6 H.sub.4 -Furyl-2                                   42 5-(2'-CH.sub.3 --C.sub.6 H.sub.4 -Furyl-2                                   43 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4 -Furyl-2                                  44 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4 -Furyl-2                                  45 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4 -Furyl-2                                  46 5-(4'-NO.sub.2 --C.sub.6 H.sub.4 -Furyl-2                                   47 5-(3'-NO.sub.2 --C.sub.6 H.sub.4 -Furyl-2                                   48 5-(2'-NO.sub.2 --C.sub.6 H.sub.4 -Furyl-2                                   49 5-(4'-CN--C.sub.6 H.sub.4 -Furyl-2                                          50 5-(3'-CN--C.sub.6 H.sub.4 -Furyl-2                                          51 5-(2'-CN--C.sub.6 H.sub.4 -Furyl-2                                          52 5-(4'-Cl--C.sub.6 H.sub.4 -Furyl-2                                          53 5-(3'-Cl--C.sub.6 H.sub.4 -Furyl-2                                          54 5-(2'-Cl--C.sub.6 H.sub.4 -Furyl-2                                          55 4-CH.sub.3 -Furyl-2                                                         56 4-C.sub.6 H.sub.5 -Furyl-2                                                  57 4-(4'-CH.sub.3 --C.sub.6 H.sub.4 -Furyl-2                                   58 4-(3'-CH.sub.3 --C.sub.6 H.sub.4 -Furyl-2                                   59 4-(2'-CH.sub.3 --C.sub.6 H.sub.4 -Furyl-2                                   60 4-(4'-CH.sub.3 O--C.sub.6 H.sub.4 -Furyl-2                                  61 4-(3'-CH.sub.3 O--C.sub.6 H.sub.4 -Furyl-2                                  62 4-(2'-CH.sub.3 O--C.sub.6 H.sub.4 -Furyl-2                                  63 4-(4'-NO.sub.2 --C.sub.6 H.sub.4 -Furyl-2                                   64 4-(3'-NO.sub.2 --C.sub.6 H.sub.4 -Furyl-2                                   65 4-(2'-NO.sub.2 --C.sub.6 H.sub.4 -Furyl-2                                   66 4-(4'-CN--C.sub.6 H.sub.4 -Furyl-2                                          67 4-(3'-CN--C.sub.6 H.sub.4 -Furyl-2                                          68 4-(2'-CN--C.sub.6 H.sub.4 -Furyl-2                                          69 4-(4'-Cl--C.sub.6 H.sub.4 -Furyl-2                                          70 4-(3'-Cl--C.sub.6 H.sub.4 -Furyl-2                                          71 4-(2'-Cl--C.sub.6 H.sub.4 -Furyl-2                                          72 Thienyl-2                                                                   73 5-CH.sub.3 -Thienyl-2                                                       74 5-C.sub.6 H.sub.5 -Thienyl-2                                                75 5-(4'-CH.sub.3 --C.sub.6 H.sub.4 -Thienyl-2                                 76 5-(3'-CH.sub.3 --C.sub.6 H.sub.4 -Thienyl-2                                 77 5-(2'-CH.sub.3 --C.sub.6 H.sub.4 -Thienyl-2                                 78 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4 -Thienyl-2                                79 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4 -Thienyl-2                                80 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4 -Thienyl-2                                81 5-(4'-NO.sub.2 --C.sub.6 H.sub.4 -Thienyl-2                                 82 5-(3'-NO.sub.2 --C.sub.6 H.sub.4 -Thienyl-2                                 83 5-(2'-NO.sub.2 --C.sub.6 H.sub.4 -Thienyl-2                                 84 5-(4'-CN--C.sub.6 H.sub.4 -Thienyl-2                                        85 5-(3'-CN--C.sub.6 H.sub.4 -Thienyl-2                                        86 5-(2'-CN--C.sub.6 H.sub.4 -Thienyl-2                                        87 5-(4'-Cl--C.sub.6 H.sub.4 -Thienyl-2                                        88 5-(3'-Cl--C.sub.6 H.sub.4 -Thienyl-2                                        89 5-(2'-Cl--C.sub.6 H.sub.4 -Thienyl-2                                        90 4-CH.sub.3 -Thienyl-2                                                       91 4-C.sub.6 H.sub.5 -Thienyl-2                                                92 4-(4'-CH.sub.3 --C.sub.6 H.sub.4 -Thienyl-2                                 93 4-(3'-CH.sub.3 --C.sub.6 H.sub.4 -Thienyl-2                                 94 4-(2'-CH.sub.3 --C.sub.6 H.sub.4 -Thienyl-2                                 95 4-(4'-CH.sub.3 O--C.sub.6 H.sub.4 -Thienyl-2                                96 4-(3'-CH.sub.3 O--C.sub.6 H.sub.4 -Thienyl-2                                97 4-(2'-CH.sub.3 O--C.sub.6 H.sub.4 -Thienyl-2                                98 4-(4'-NO.sub.2 --C.sub.6 H.sub.4 -Thienyl-2                                 99 4-(3'-NO.sub.2 --C.sub.6 H.sub.4 -Thienyl-2                                 100 4-(2'-NO.sub.2 --C.sub.6 H.sub.4 -Thienyl-2                                101 4-(4'-CN--C.sub.6 H.sub.4 -Thienyl-2                                       102 4-(3'-CN--C.sub.6 H.sub.4 -Thienyl-2                                       103 4-(2'-CN--C.sub.6 H.sub.4 -Thienyl-2                                       104 4-(4'-Cl--C.sub.6 H.sub.4 -Thienyl-2                                       105 4-(3'-Cl--C.sub.6 H.sub.4 -Thienyl-2                                       106 4-(2'-Cl--C.sub.6 H.sub.4 -Thienyl-2                                       107 Thienyl-3                                                                  108 5-CH.sub.3 -Thienyl-3                                                      109 5-C.sub.6 H.sub.5 -Thienyl-3                                               110 5-(4'-CH.sub.3 --C.sub.6 H.sub.4 -Thienyl-3                                111 5-(3'-CH.sub.3 --C.sub.6 H.sub.4 -Thienyl-3                                112 5-(2'-CH.sub.3 --C.sub.6 H.sub.4 -Thienyl-3                                113 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4 -Thienyl-3                               114 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4 -Thienyl-3                               115 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4 -Thienyl-3                               116 5-(4'-NO.sub.2 --C.sub.6 H.sub.4 -Thienyl-3                                117 5-(3'-NO.sub.2 --C.sub.6 H.sub.4 -Thienyl-3                                118 5-(2'-NO.sub.2 --C.sub.6 H.sub.4 -Thienyl-3                                119 5-(4'-CN--C.sub.6 H.sub.4 -Thienyl-3                                       120 5-(3'-CN--C.sub.6 H.sub.4 -Thienyl-3                                       121 5-(2'-CN--C.sub.6 H.sub.4 -Thienyl-3                                       122 5-(4'-Cl--C.sub.6 H.sub.4 -Thienyl-3                                       123 5-(3'-Cl--C.sub.6 H.sub.4 -Thienyl-3                                       124 5-(2'-Cl--C.sub.6 H.sub.4 -Thienyl-3                                       125 Pyrazolyl-4                                                                126 N--CH.sub.3 -Pyrazolyl-4                                                   127 N--C.sub.6 H.sub.5 -Pyrazolyl-4                                            128 N-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrazolyl-4                              129 N-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrazolyl-4                              130 N-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrazolyl-4                              131 N-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrazolyl-4                             132 N-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrazolyl-4                             133 N-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrazolyl-4                             134 N-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrazolyl-4                              135 N-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrazolyl-4                              136 N-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrazolyl-4                              137 N-(4'-CN--C.sub.6 H.sub.4)-Pyrazolyl-4                                     138 N-(3'-CN--C.sub.6 H.sub.4)-Pyrazolyl-4                                     139 N-(2'-CN--C.sub.6 H.sub.4)-Pyrazolyl-4                                     140 N-(4'-Cl--C.sub.6 H.sub.4)-Pyrazolyl-4                                     141 N-(3'-Cl--C.sub.6 H.sub.4)-Pyrazolyl-4                                     142 N-(2'-Cl--C.sub.6 H.sub.4)-Pyrazolyl-4                                     143 3-CH.sub.3 --N-Methylpyrazolyl-4                                           144 3-C.sub.6 H.sub.5 --N-Methylpyrazolyl-4                                    145 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)--N-Methylpyrazolyl-4                     146 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)--N-Methylpyrazolyl-4                     147 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)--N-Methylpyrazolyl-4                     148 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)--N-Methylpyrazolyl-4                    149 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)--N-Methylpyrazolyl-4                    150 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)--N-Methylpyrazolyl-4                    151 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)--N-Methylpyrazolyl-4                     152 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)--N-Methylpyrazolyl-4                     153 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)--N-Methylpyrazolyl-4                     154 3-(4'-CN--C.sub.6 H.sub.4)--N-Methylpyrazolyl-4                            155 3-(3'-CN--C.sub.6 H.sub.4)--N-Methylpyrazolyl-4                            156 3-(2'-CN--C.sub.6 H.sub.4)--N-Methylpyrazolyl-4                            157 3-(4'-Cl--C.sub.6 H.sub.4)--N-Methylpyrazolyl-4                            158 3-(3'-Cl--C.sub.6 H.sub.4)--N-Methylpyrazolyl-4                            159 3-(2'-Cl--C.sub.6 H.sub.4)--N-Methylpyrazolyl-4                            160 Isoxazolyl-5                                                               161 3-CH.sub.3 -Isoxazolyl-5                                                   162 3-C.sub.6 H.sub.5 -Isoxazolyl-5                                            163 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Isoxazolyl-5                             164 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Isoxazolyl-5                             165 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Isoxazolyl-5                             166 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Isoxazolyl-5                            167 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Isoxazolyl-5                            168 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Isoxazolyl-5                            169 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Isoxazolyl-5                             170 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Isoxazolyl-5                             171 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Isoxazolyl-5                             172 3-(4'-CN--C.sub.6 H.sub.4)-Isoxazolyl-5                                    173 3-(3'-CN--C.sub.6 H.sub.4)-Isoxazolyl-5                                    174 3-(2'-CN--C.sub.6 H.sub.4)-Isoxazolyl-5                                    175 3-(4'-Cl--C.sub.6 H.sub.4)-Isoxazolyl-5                                    176 3-(3'-Cl--C.sub.6 H.sub.4)-Isoxazolyl-5                                    177 3-(2'-Cl--C.sub.6 H.sub.4)-Isoxazolyl-5                                    178 4-Chloroisoxazolyl-5                                                       179 3-CH.sub.3 -4-Chloroisoxazolyl-5                                           180 3-C.sub.6 H.sub.5 -4-Chloroisoxazolyl-5                                    181 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                     182 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                     183 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                     184 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                    185 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                    186 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                    187 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                     188 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                     189 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                     190 3-(4'-CN--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                            191 3-(3'-CN--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                            192 3-(2'-CN--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                            193 3-(4'-Cl--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                            194 3-(3'-Cl--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                            195 3-(2'-Cl--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                            196 Isoxazolyl-3                                                               197 5-CH.sub.3 -Isoxazolyl-3                                                   198 5-C.sub.6 H.sub.5 -Isoxazolyl-3                                            199 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Isoxazolyl-3                             200 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Isoxazolyl-3                             201 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Isoxazolyl-3                             202 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Isoxazolyl-3                            203 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Isoxazolyl-3                            204 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Isoxazolyl-3                            205 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Isoxazolyl-3                             206 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Isoxazolyl-3                             207 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Isoxazolyl-3                             208 5-(4'-CN--C.sub.6 H.sub.4)-Isoxazolyl-3                                    209 5-(3'-CN--C.sub.6 H.sub.4)-Isoxazolyl-3                                    210 5-(2'-CN--C.sub.6 H.sub.4)-Isoxazolyl-3                                    211 5-(4'-Cl--C.sub.6 H.sub.4)-Isoxazolyl-3                                    212 5-(3'-Cl--C.sub.6 H.sub.4)-Isoxazolyl-3                                    213 5-(2'-Cl--C.sub.6 H.sub.4)-Isoxazolyl-3                                    214 Isothiazolyl-5                                                             215 3-CH.sub.3 -Isothiazolyl-5                                                 216 3-C.sub.6 H.sub.5 -Isothiazolyl-5                                          217 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Isothiazolyl-5                           218 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Isothiazolyl-5                           219 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Isothiazolyl-5                           220 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Isothiazolyl-5                          221 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Isothiazolyl-5                          222 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Isothiazolyl-5                          223 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Isothiazolyl-5                           224 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Isothiazolyl-5                           225 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Isothiazolyl-5                           226 3-(4'-CN--C.sub.6 H.sub.4)-Isothiazolyl-5                                  227 3-(3'-CN--C.sub.6 H.sub.4)-Isothiazolyl-5                                  228 3-(2'-CN--C.sub.6 H.sub.4)-Isothiazolyl-5                                  229 3-(4'-Cl--C.sub.6 H.sub.4)-Isothiazolyl-5                                  230 3-(3'-Cl--C.sub.6 H.sub.4)-Isothiazolyl-5                                  231 3-(2'-Cl--C.sub.6 H.sub.4)-Isothiazolyl-5                                  232 Oxazolyl-4                                                                 233 2-CH.sub.3 -Oxazolyl-4                                                     234 2-C.sub.6 H.sub.5 -Oxazolyl-4                                              235 2-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Oxazolyl-4                               236 2-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Oxazolyl-4                               237 2-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Oxazolyl-4                               238 2-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Oxazolyl-4                              239 2-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Oxazolyl-4                              240 2-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Oxazolyl-4                              241 2-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Oxazolyl-4                               242 2-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Oxazolyl-4                               243 2-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Oxazolyl-4                               244 2-(4'-CN--C.sub.6 H.sub.4)-Oxazolyl-4                                      245 2-(3'-CN--C.sub.6 H.sub.4)-Oxazolyl-4                                      246 2-(2'-CN--C.sub.6 H.sub.4)-Oxazolyl-4                                      247 2-(4'-Cl--C.sub.6 H.sub.4)-Oxazolyl-4                                      248 2-(3'-Cl--C.sub.6 H.sub.4)-Oxazolyl-4                                      249 2-(2'-Cl--C.sub.6 H.sub.4)-Oxazolyl-4                                      250 Thiazolyl-4                                                                251 2-CH.sub.3 -Thiazolyl-4                                                    252 2-C.sub.6 H.sub.5 -Thiazolyl-4                                             253 2-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Thiazolyl-4                              254 2-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Thiazolyl-4                              255 2-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Thiazolyl-4                              256 2-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Thiazolyl-4                             267 2-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Thiazolyl-4                             258 2-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Thiazolyl-4                             259 2-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Thiazolyl-4                              260 2-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Thiazolyl-4                              261 2-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Thiazolyl-4                              262 2-(4'-CN--C.sub.6 H.sub.4)-Thiazolyl-4                                     263 2-(3'-CN--C.sub.6 H.sub.4)-Thiazolyl-4                                     264 2-(2'-CN--C.sub.6 H.sub.4)-Thiazolyl-4                                     265 2-(4'-Cl--C.sub.6 H.sub.4)-Thiazolyl-4                                     266 2-(3'-Cl--C.sub.6 H.sub.4)-Thiazolyl-4                                     267 2-(2'-Cl--C.sub.6 H.sub.4)-Thiazolyl-4                                     268 N--CH.sub.3 -1,2,4-Triazolyl-5                                             269 3-CH.sub.3 --N--CH.sub.3 -1,2,4-Triazolyl-5                                270 3-C.sub.6 H.sub.5 --N--CH.sub.3 -1,2,4-Triazolyl-5                         271 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5                 272 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazol             yl-5                                                                     273 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5                 274 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazo             lyl-5                                                                    275 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5                276 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazo             lyl-5                                                                    277 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5                 278 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazol             yl-5                                                                     279 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5                 280 3-(4'-CN--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5                 281 3-(3'-CN--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5                 282 3-(2'-CN--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5                 283 3-(4'-Cl--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5                 284 3-(3'-Cl--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5                 285 3-(2'-Cl--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5                 286 1,3,4-Oxadiazolyl-2                                                 287 5-CH.sub.3 -1,3,4-Oxadiazolyl-2                                            288 5-C.sub.6 H.sub.5 -1,2,3-Oxadiazolyl-2                                     289 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                      290 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                      291 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                      292 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                     293 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                     294 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                     295 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                      296 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                      297 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                      298 5-(4'-CN--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                             299 5-(3'-CN--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                             300 5-(2'-CN--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                             301 5-(4'-Cl--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                             302 5-(3'-Cl--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                             303 5-(2'-Cl--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                             304 1,2,4-Oxadiazolyl-3                                                        305 5-CH.sub.3 -1,2,4-Oxadiazolyl-3                                            306 5-C.sub.6 H.sub.5 -1,2,4-Oxadiazolyl-3                                     307 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                      308 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                      309 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                      310 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                     311 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                     312 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                     313 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                      314 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                      315 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                      316 5-(4'-CN--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                             317 5-(3'-CN--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                             318 5-(2'-CN--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                             319 5-(4'-Cl--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                             320 5-(3'-Cl--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                             321 5-(2'-Cl--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                             322 1,2,4-Oxadiazolyl-5                                                        323 3-CH.sub.3 -1,2,4-Oxadiazolyl-5                                            324 3-C.sub.6 H.sub.5 -1,2,4-Oxadiazolyl-5                                     325 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                      326 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                      327 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                      328 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                     329 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                     330 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                     331 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                      332 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                      333 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                      334 3-(4'-CN--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                             335 3-(3'-CN--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                             336 3-(2'-CN--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                             337 3-(4'-Cl--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                             338 3-(3'-Cl--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                             339 3-(2'-Cl--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                             340 1,2,4-Thiadiazolyl-3                                                       341 5-CH.sub.3 -1,2,4-Thiadiazolyl-3                                           342 5-C.sub.6 H.sub.5 -1,2,4-Thiadiazolyl-3                                    343 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                     344 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                     345 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                     346 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                    347 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                    348 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                    349 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                     350 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                     351 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                     352 5-(4'-CN--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                            353 5-(3'-CN--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                            354 5-(2'-CN--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                            355 5-(4'-Cl--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                            356 5-(3'-Cl--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                            357 5-(2'-Cl--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                            358 1,3,4-Thiadiazolyl-2                                                       359 5-CH.sub.3 -1,3,4-Thiadiazolyl-2                                           360 5-C.sub.6 H.sub.5 -1,3,4-Thiadiazolyl-2                                    361 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                     362 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                     363 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                     364 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                    365 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                    366 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                    367 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                     368 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                     369 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                     370 5-(4'-CN--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                            371 5-(3'-CN--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                            372 5-(2'-CN--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                            373 5-(4'-Cl--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                            374 5-(3'-Cl--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                            375 5-(2'-Cl--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                            376 Pyridinyl-2                                                                377 Pyridinyl-4                                                                378 Pyridazinyl-3                                                              379 Pyridazinyl-4                                                              380 Pyridazinyl-2                                                              381 Pyrimidinyl-4                                                              382 Pyrimidinyl-5                                                              383 Pyrimidinyl-2                                                              384 Pyridinyl-3                                                                385 1-Naphthyl                                                                 386 2-Naphthyl                                                               ______________________________________                                    

                  TABLE 12                                                         ______________________________________                                         1  STR182##                                                                                 I: R.sup.1 = CH.sub.3                                               II: R.sup.1 = CH.sub.2 --CH.sub.3                                               -                                                                           No.       X.sub.m                                                              ______________________________________                                         1         H                                                                      2 2-F                                                                          3 3-F                                                                          4 4-F                                                                          5 2,4-F.sub.2                                                                  6 2,4,6-F.sub.3                                                                7 2,3,4,5,6-F.sub.5                                                            8 2,3-F.sub.2                                                                  9 2-Cl                                                                         10 3-Cl                                                                        11 4-Cl                                                                        12 2,3-Cl.sub.2                                                                13 2,4-Cl.sub.2                                                                14 2,5-Cl.sub.2                                                                15 2,6-Cl.sub.2                                                                16 3,4-Cl.sub.2                                                                17 3,5-Cl.sub.2                                                                18 2,3,4-Cl.sub.3                                                              19 2,3,5-Cl.sub.3                                                              20 2,3,6-Cl.sub.3                                                              21 2,4,5-Cl.sub.3                                                              22 2,4,6-Cl.sub.3                                                              23 3,4,5-Cl.sub.3                                                              24 2,3,4,6-Cl.sub.4                                                            25 2,3,5,6-Cl.sub.4                                                            26 2,3,4,5,6-Cl.sub.5                                                          27 2-Br                                                                        28 3-Br                                                                        29 4-Br                                                                        30 2,4-Br.sub.2                                                                31 2,5-Br.sub.2                                                                32 2,6-Br.sub.2                                                                33 2,4,6-Br.sub.3                                                              34 2,3,4,5,6-Br.sub.5                                                          35 2-I                                                                         36 3-I                                                                         37 4-I                                                                         38 2,4-I.sub.2                                                                 39 2-Cl, 3-F                                                                   40 2-Cl, 4-F                                                                   41 2-Cl, 5-F                                                                   42 2-Cl, 6-F                                                                   43 2-Cl, 3-Br                                                                  44 2-Cl, 4-Br                                                                  45 2-Cl, 5-Br                                                                  46 2-Cl, 6-Br                                                                  47 2-Br, 3-Cl                                                                  48 2-Br, 4-Cl                                                                  49 2-Br, 5-Cl                                                                  50 2-Br, 3-F                                                                   51 2-Br, 4-F                                                                   52 2-Br, 5-F                                                                   53 2-Br, 6-F                                                                   54 2-F, 3-Cl                                                                   55 2-F, 4-Cl                                                                   56 2-F, 5-Cl                                                                   57 3-Cl, 4-F                                                                   58 3-Cl, 5-F                                                                   59 3-Cl, 4-Br                                                                  60 3-Cl, 5-Br                                                                  61 3-F, 4-Cl                                                                   62 3-F, 4-Br                                                                   63 3-Br, 4-Cl                                                                  64 3-Br, 4-F                                                                   65 2,6-Cl.sub.2, 4-Br                                                          66 2-CH.sub.3                                                                  67 3-CH.sub.3                                                                  68 4-CH.sub.3                                                                  69 2,3-(CH.sub.3).sub.2                                                        70 2,4-(CH.sub.3).sub.2                                                        71 2,5-(CH.sub.3).sub.2                                                        72 2,6-(CH.sub.3).sub.2                                                        73 3,4-(CH.sub.3).sub.2                                                        74 3,5-(CH.sub.3).sub.2                                                        75 2,3,5-(CH.sub.3).sub.3                                                      76 2,3,4-(CH.sub.3).sub.3                                                      77 2,3,6-(CH.sub.3).sub.3                                                      78 2,4,5-(CH.sub.3).sub.3                                                      79 2,4,6-(CH.sub.3).sub.3                                                      80 3,4,5-(CH.sub.3).sub.3                                                      81 2,3,4,6-(CH.sub.3).sub.4                                                    82 2,3,5,6-(CH.sub.3).sub.4                                                    83 2,3,4,5,6-(CH.sub.3).sub.5                                                  84 2-C.sub.2 H.sub.5                                                           85 3-C.sub.2 H.sub.5                                                           86 4-C.sub.2 H.sub.5                                                           87 2,4-(C.sub.2 H.sub.5).sub.2                                                 88 2,6-(C.sub.2 H.sub.5).sub.2                                                 89 3,5-(C.sub.2 H.sub.5).sub.2                                                 90 2,4,6-(C.sub.2 H.sub.5).sub.3                                               91 2-n-C.sub.3 H.sub.7                                                         92 3-n-C.sub.3 H.sub.7                                                         93 4-n-C.sub.3 H.sub.7                                                         94 2-i-C.sub.3 H.sub.7                                                         95 3-i-C.sub.3 H.sub.7                                                         96 4-i-C.sub.3 H.sub.7                                                         97 2,4-(i-C.sub.3 H.sub.7).sub.2                                               98 2,6-(i-C.sub.3 H.sub.7).sub.2                                               99 3,5-(i-C.sub.3 H.sub.7).sub.2                                               100 2,4,6-(i-C.sub.3 H.sub.7).sub.3                                            101 2-s-C.sub.4 H.sub.9                                                        102 3-s-C.sub.4 H.sub.9                                                        103 4-s-C.sub.4 H.sub.9                                                        104 2-t-C.sub.4 H.sub.9                                                        105 3-t-C.sub.4 H.sub.9                                                        106 4-t-C.sub.4 H.sub.9                                                        107 2,3-(t-C.sub.4 H.sub.9).sub.2                                              108 2,4-(t-C.sub.4 H.sub.9).sub.2                                              109 2,5-(t-C.sub.4 H.sub.9).sub.2                                              110 2,6-(t-C.sub.4 H.sub.9).sub.2                                              111 3,4-(t-C.sub.4 H.sub.9).sub.2                                              112 2,4,6-(t-C.sub.4 H.sub.9).sub.3                                            113 4-n-C.sub.9 H.sub.19                                                       114 4-n-C.sub.12 H.sub.25                                                      115 4-n-C.sub.15 H.sub.31                                                      116 4-(1,1,3,3-Tetramethylbutyl)                                               117 4-(2,4,4-Trimethylpropyl)                                                  118 2-t-C.sub.4 H.sub.9, 4-CH.sub.3                                            119 2-t-C.sub.4 H.sub.9, 5-CH.sub.3                                            120 2,6-(t-C.sub.4 H.sub.9).sub.2, 4-CH.sub.3                                  121 2-CH.sub.3, 4-t-C.sub.4 H.sub.9                                            122 2-CH.sub.3, 6-t-C.sub.4 H.sub.9                                            123 2-CH.sub.3, 4-i-C.sub.3 H.sub.7                                            124 2-CH.sub.3, 5-i-C.sub.3 H.sub.7                                            125 3-CH.sub.3, 4-i-C.sub.3 H.sub.7                                            126 2-i-C.sub.3 H.sub.7, 5-CH.sub.3                                            127 2,4-(t-C.sub.4 H.sub.9).sub.2, 6-i-C.sub.3 H.sub.7                         128 2-Allyl                                                                    129 3-Allyl                                                                    130 4-Allyl                                                                    131 2-Allyl, 6-CH.sub.3                                                        132 2-cyclo-C.sub.6 H.sub.11                                                   133 3-cyclo-C.sub.6 H.sub.11                                                   134 4-cyclo-C.sub.6 H.sub.11                                                   135 2,4-(cyclo-C.sub.6 H.sub.11).sub.2, 6-CH.sub.3                             136 2-CH.sub.3, 4-cyclo-C.sub.6 H.sub.11                                       137 2-CH.sub.2 --C.sub.6 H.sub.5                                               138 3-CH.sub.2 --C.sub.6 H.sub.5                                               139 4-CH.sub.2 --C.sub.6 H.sub.5                                               140 2-CH.sub.2 --C.sub.6 H.sub.5, 4-CH.sub.3                                   141 2-CH.sub.3, 4-CH.sub.2 --C.sub.6 H.sub.5                                   142 2-C.sub.6 H.sub.5                                                          143 3-C.sub.6 H.sub.5                                                          144 4-C.sub.6 H.sub.5                                                          145 4-(2-i-C.sub.3 H.sub.7 --C.sub.6 H.sub.4)                                  146 4-C.sub.6 H.sub.5, 2,6-(CH.sub.3).sub.2                                    147 2-Cl, 4-C.sub.6 H.sub.5                                                    148 2-Br, 4-C.sub.6 H.sub.5                                                    149 2-C.sub.6 H.sub.5, 4-Cl                                                    150 2-C.sub.6 H.sub.5, 4-Br                                                    151 2-CH.sub.2 C.sub.6 H.sub.5, 4-Cl                                           152 2-CH.sub.2 C.sub.6 H.sub.5, 4-Br                                           153 2-Cl, 4-CH.sub.2 C.sub.6 H.sub.5                                           154 2-Br, 4-CH.sub.2 C.sub.6 H.sub.5                                           155 2-cyclo-C.sub.6 H.sub.11, 4-Cl                                             156 2-cyclo-C.sub.6 H.sub.11, 4-Br                                             157 2-Cl, 4-cyclo-C.sub.6 H.sub.11                                             158 2-Br, 4-cyclo-C.sub.6 H.sub.11                                             159 2-OCH.sub.3                                                                160 3-OCH.sub.3                                                                161 4-OCH.sub.3                                                                162 2-OC.sub.2 H.sub.5                                                         163 3-O--C.sub.2 H.sub.5                                                       164 4-O--C.sub.2 H.sub.5                                                       165 2-O-n-C.sub.3 H.sub.7                                                      166 3-O-n-C.sub.3 H.sub.7                                                      167 4-O-n-C.sub.3 H.sub.7                                                      168 2-O-i-C.sub.3 H.sub.7                                                      169 3-O-i-C.sub.3 H.sub.7                                                      170 4-O-i-C.sub.3 H.sub.7                                                      171 2-O-n-C.sub.6 H.sub.13                                                     172 3-O-n-C.sub.6 H.sub.13                                                     173 4-O-n-C.sub.6 H.sub.13                                                     174 2-O-n-C.sub.8 H.sub.17                                                     175 3-O-n-C.sub.8 H.sub.17                                                     176 4-O-n-C.sub.8 H.sub.17                                                     177 2-O--CH.sub.2 C.sub.6 H.sub.5                                              178 3-O--CH.sub.2 C.sub.6 H.sub.5                                              179 4-O--CH.sub.2 C.sub.6 H.sub.5                                              180 2-O--(CH.sub.2).sub.3 C.sub.6 H.sub.5                                      181 3-O--(CH.sub.2).sub.3 C.sub.6 H.sub.5                                      182 4-O--(CH.sub.2).sub.3 C.sub.6 H.sub.5                                      183 2,4-(OCH.sub.3).sub.2                                                      184 2-CF.sub.3                                                                 185 3-CF.sub.3                                                                 186 4-CF.sub.3                                                                 187 2-OCF.sub.3                                                                188 3-OCF.sub.3                                                                189 4-OCF.sub.3                                                                190 3-OCH.sub.2 CHF.sub.2                                                      191 2-NO.sub.2                                                                 192 3-NO.sub.2                                                                 193 4-NO.sub.2                                                                 194 2-CN                                                                       195 3-CN                                                                       196 4-CN                                                                       197 2-CH.sub.3, 3-Cl                                                           198 2-CH.sub.3, 4-Cl                                                           199 2-CH.sub.3, 5-Cl                                                           200 2-CH.sub.3, 6-Cl                                                           201 2-CH.sub.3, 3-F                                                            202 2-CH.sub.3, 4-F                                                            203 2-CH.sub.3, 5-F                                                            204 2-CH.sub.3, 6-F                                                            205 2-CH.sub.3, 3-Br                                                           206 2-CH.sub.3, 4-Br                                                           207 2-CH.sub.3, 5-Br                                                           208 2-CH.sub.3, 6-Br                                                           209 2-Cl, 3-CH.sub.3                                                           210 2-Cl, 4-CH.sub.3                                                           211 2-Cl, 5-CH.sub.3                                                           212 2-F, 3-CH.sub.3                                                            213 2-F, 4-CH.sub.3                                                            214 2-F, 5-CH.sub.3                                                            215 2-Br, 3-CH.sub.3                                                           216 2-Br, 4-CH.sub.3                                                           217 2-Br, 5-CH.sub.3                                                           218 3-CH.sub.3, 4-Cl                                                           219 3-CH.sub.3, 5-Cl                                                           220 3-CH.sub.3, 4-F                                                            221 3-CH.sub.3, 5-F                                                            222 3-CH.sub.3, 4-Br                                                           223 3-CH.sub.3, 5-Br                                                           224 3-F, 4-CH.sub.3                                                            225 3-Cl, 4-CH.sub.3                                                           226 3-Br, 4-CH.sub.3                                                           227 2-Cl, 4,5-(CH.sub.3).sub.2                                                 228 2-Br, 4,5-(CH.sub.3).sub.2                                                 229 2-Cl, 3,5-(CH.sub.3).sub.2                                                 230 2-Br, 3,5-(CH.sub.3).sub.2                                                 231 2,6-Cl.sub.2, 4-CH.sub.3                                                   232 2,6-F.sub.2, 4-CH.sub.3                                                    233 2,6-Br.sub.2, 4-CH.sub.3                                                   234 2,4-Br.sub.2, 6-CH.sub.3                                                   235 2,4-F.sub.2, 6-CH.sub.3                                                    236 2,4-Br.sub.2, 6-CH.sub.3                                                   237 2,6-(CH.sub.3).sub.2, 4-F                                                  238 2,6-(CH.sub.3).sub.2, 4-Cl                                                 239 2,6-(CH.sub.3).sub.2, 4-Br                                                 240 3,5-(CH.sub.3).sub.2, 4-F                                                  241 3,5-(CH.sub.3).sub.2, 4-Cl                                                 242 3,5-(CH.sub.3).sub.2, 4-Br                                                 243 2,3,6-(CH.sub.3).sub.3, 4-F                                                244 2,3,6-(CH.sub.3).sub.3, 4-Cl                                               245 2,3,6-(CH.sub.3).sub.3, 4-Br                                               246 2,4-(CH.sub.3).sub.2, 6-F                                                  247 2,4-(CH.sub.3).sub.2, 6-Cl                                                 248 2,4-(CH.sub.3).sub.2, 6-Br                                                 249 2-i-C.sub.3 H.sub.7, 4-Cl, 5-CH.sub.3                                      250 2-Cl, 4-NO.sub.2                                                           251 2-NO.sub.2, 4-Cl                                                           252 2-OCH.sub.3, 5-NO.sub.2                                                    253 2,4-Cl.sub.2, 5-NO.sub.2                                                   254 2,4-Cl.sub.2, 6-NO.sub.2                                                   255 2,6-Cl.sub.2, 4-NO.sub.2                                                   256 2,6-Br.sub.2, 4-NO.sub.2                                                   257 2,6-I.sub.2, 4-NO.sub.2                                                    258 2-CH.sub.3, 5-i-C.sub.3 H.sub.7, 4-Cl                                      259 2-CO.sub.2 CH.sub.3                                                        260 3-CO.sub.2 CH.sub.3                                                        261 4-CO.sub.2 CH.sub.3                                                        262 2-CO.sub.2 (C.sub.2 H.sub.5)                                               263 3-CO.sub.2 (C.sub.2 H.sub.5)                                               264 4-CO.sub.2 (C.sub.2 H.sub.5)                                               265 2-CO.sub.2 (n-C.sub.3 H.sub.7)                                             266 3-CO.sub.2 (n-C.sub.3 H.sub.7)                                             267 4-CO.sub.2 (n-C.sub.3 H.sub.7)                                             268 2-CO.sub.2 (i-C.sub.3 H.sub.7)                                             269 3-CO.sub.2 (i-C.sub.3 H.sub.7)                                             270 4-CO.sub.2 (i-C.sub.3 H.sub.7)                                             271 2-CO.sub.2 (n-C.sub.6 H.sub.13)                                            272 3-CO.sub.2 (n-C.sub.6 H.sub.13)                                            273 4-CO.sub.2 (n-C.sub.6 H.sub.13)                                            274 2-CH.sub.2 --OCH.sub.3                                                     275 3-CH.sub.2 --OCH.sub.3                                                     276 4-CH.sub.2 --OCH.sub.3                                                     277 2-CH.sub.2 O(C.sub.2 H.sub.5)                                              278 3-CH.sub.2 O(C.sub.2 H.sub.5)                                              279 4-CH.sub.2 O(C.sub.2 H.sub.5)                                              280 2-CH.sub.2 O(n-C.sub.3 H.sub.7)                                            281 3-CH.sub.2 O(n-C.sub.3 H.sub.7)                                            282 4-CH.sub.2 O(n-C.sub.3 H.sub.7)                                            283 2-CH.sub.2 O(i-C.sub.3 H.sub.7)                                            284 3-CH.sub.2 O(i-C.sub.3 H.sub.7)                                            285 4-CH.sub.2 O(i-C.sub.3 H.sub.7)                                            286 2-CHO                                                                      287 3-CHO                                                                      288 4-CHO                                                                      289 2-CO--CH.sub.3                                                             290 3-CO--CH.sub.3                                                             291 4-CO--CH.sub.3                                                             292 2-CO--CH.sub.2 --CH.sub.3                                                  293 3-CO--CH.sub.2 --CH.sub.3                                                  294 4-CO--CH.sub.2 --CH.sub.3                                                  295 2-CO--CH.sub.2 --CH.sub.2 --CH.sub.3                                       296 3-CO--CH.sub.2 --CH.sub.2 --CH.sub.3                                       297 4-CO--CH.sub.2 --CH.sub.2 --CH.sub.3                                       298 2-CO--CH(CH.sub.3)--CH.sub.3                                               299 3-CO--CH(CH.sub.3)--CH.sub.3                                               300 4-CO--CH(CH.sub.3)--CH.sub.3                                               301 2-Me-4-CHO                                                                 302 2-Me-4-CH.sub.3 --CO                                                       303 2-Me-4-CH.sub.3 --CH.sub.2 --CO                                            304 2-Me-4-CH.sub.3 --CH.sub.2 --CH.sub.2 --CO                                 305 2-Me-4-CH.sub.3 --CH(CH.sub.3)--CO                                         306 2,5-Me.sub.2 -4-CHO                                                        307 2,5-Me.sub.2 -4-CH.sub.3 --CO                                              308 2,5-Me.sub.2 -4-CH.sub.3 --CH.sub.2 --CO                                   309 2,5-Me.sub.2 -4-CH.sub.3 --CH.sub.2 --CH.sub.2 --CO                        310 2,5-Me.sub.2 -4-CH.sub.3 --CH(CH.sub.3)--CO                                311 2-Cl-4-CHO                                                                 312 2-Cl-4-CH.sub.3 --CO                                                       313 2-Cl-4-CH.sub.3 --CH.sub.2 --CO                                            314 2-Cl-4-CH.sub.3 --CH(CH.sub.3)--CO                                         315 2,5-Cl.sub.2 -4-CHO                                                        316 2,5-Cl.sub.2 -4-CH.sub.3 --CO                                              317 2,5-Cl.sub.2 -4-CH.sub.3 --CH.sub.2 --CO                                   318 2,5-Cl.sub.2 -4-CH.sub.3 --CH.sub.2 --CH.sub.2 --CO                        319 2,5-Cl.sub.2 -4-CH.sub.3 --CH(CH.sub.3)--CO                                320 2-C(═NOCH.sub.3)--CH.sub.3                                             321 3-C(═NOCH.sub.3)--CH.sub.3                                             322 4-C(═NOCH.sub.3)--CH.sub.3                                             323 2-C(═NOC.sub.2 H.sub.5)--CH.sub.3                                      324 3-C(═NOC.sub.2 H.sub.5)--CH.sub.3                                      325 4-C(═NOC.sub.2 H.sub.5)--CH.sub.3                                      326 2-C(═NO-n-C.sub.3 H.sub.7)--CH.sub.3                                   327 3-C(═NO-n-C.sub.3 H.sub.7)--CH.sub.3                                   328 4-C(═NO-n-C.sub.3 H.sub.7)--CH.sub.3                                   329 2-C(═NO-i-C.sub.3 H.sub.7)--CH.sub.3                                   330 3-C(═NO-i-C.sub.3 H.sub.7)--CH.sub.3                                   331 4-C(═NO-i-C.sub.3 H.sub.7)--CH.sub.3                                   332 2-C(═NO-Allyl)--CH.sub.3                                               333 3-C(═NO-Allyl)--CH.sub.3                                               334 4-C(═NO-Allyl)--CH.sub.3                                               335 2-C(═NO-trans-Chloroallyl)--CH.sub.3                                   336 3-C(═NO-trans-Chloroallyl)--CH.sub.3                                   337 4-C(═NO-trans-Chloroallyl)--CH.sub.3                                   338 2-C(═NO-Propargyl)--CH.sub.3                                           339 3-C(═NO-Propargyl)--CH.sub.3                                           340 4-C(═NO-Propargyl)--CH.sub.3                                           341 2-C(═NO-n-C.sub.4 H.sub.9)--CH.sub.3                                   342 3-C(═NO-n-C.sub.4 H.sub.9)--CH.sub.3                                   343 4-C(═NO-n-C.sub.4 H.sub.9)--CH.sub.3                                   344 2-C(═NO--CH.sub.2 --C.sub.6 H.sub.5)--CH.sub.3                         345 3-C(═NO--CH.sub.2 --C.sub.6 H.sub.5)--CH.sub.3                         346 4-C(═NO--CH.sub.2 --C.sub.6 H.sub.5)--CH.sub.3                         347 2-CH.sub.3 -4-CH═NOCH.sub.3                                            348 2-CH.sub.3 -4-CH═NOC.sub.2 H.sub.5                                     349 2-CH.sub.3 -4-CH═NO-n-C.sub.3 H.sub.7                                  350 2-CH.sub.3 -4-CH═NO-i-C.sub.3 H.sub.7                                  351 2-CH.sub.3 -4-CH═NO-Allyl                                              352 2-CH.sub.3 -4-CH═NO-(trans-Chloroallyl)                                353 2-CH.sub.3 -4-CH═NO-Propargyl                                          354 2-CH.sub.3 -4-CH═NO-n-C.sub.4 H.sub.9                                  355 2-CH.sub.3 -4-CH═NO--CH.sub.2 --C.sub.6 H.sub.5                        356 2-CH.sub.3 -4-(CH.sub.3 --C═NOCH.sub.3)                                357 2-CH.sub.3 -4-(CH.sub.3 --C═NOC.sub.2 H.sub.5)                         358 2-CH.sub.3 -4-(CH.sub.3 --C═NO-n-C.sub.3 H.sub.7)                      359 2-CH.sub.3 -4-(CH.sub.3 --C═NO-i-C.sub.3 H.sub.7)                      360 2-CH.sub.3 -4-(CH.sub.3 --C═NO-Allyl)                                  361 2-CH.sub.3 -4-(CH.sub.3 --C═NO-trans-Chloroallyl)                      362 2-CH.sub.3 -4-(CH.sub.3 --C═NO-Propargyl)                              363 2-CH.sub.3 -4-(CH.sub.3 --C═NO-n-C.sub.4 H.sub.9)                      364 2-CH.sub.3 -4-(CH.sub.3 --C═NO--CH.sub.2 --C.sub.6 H.sub.5)                     365 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C═NO--CH.sub.3)                       366 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C═NO--C.sub.2                        H.sub.5)                                                               367 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C═NO-n-C.sub.3 H.sub.7)                        368 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C═NO-i-C.sub.3                       H.sub.7)                                                               369 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C═NO-Allyl)                           370 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C═NO-trans-Chloroallyl)                        371 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C═NO-Propargyl)                       372 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C═NO-n-C.sub.4                       H.sub.9)                                                               373 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C═NO--CH.sub.2 --C.sub.6                      H.sub.5)                                                               374 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C═NOCH.sub.3)                      375 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C═NOC.sub.2 H.sub.5)                        376 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C═NO-n-C.sub.3                    H.sub.7)                                                               377 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C═NO-i-C.sub.3 H.sub.7)                     378 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C═NO-Allyl)                        379 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C═NO-trans-Chloroal               lyl)                                                                   380 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C═NO-Proparyl)                     381 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C═NO-n-C.sub.4 H.sub.9)                     382 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C═NO--CH.sub.2                    --C.sub.6 H.sub.5)                                                     383 2-C.sub.6 H.sub.5                                                          384 3-C.sub.6 H.sub.5                                                          385 4-C.sub.6 H.sub.5                                                          386 2-(2'-F--C.sub.6 H.sub.4)                                                  387 2-(3'-F--C.sub.6 H.sub.4)                                                  388 2-(4'-F--C.sub.6 H.sub.4)                                                  389 3-(2'-F--C.sub.6 H.sub.4)                                                  390 3-(3'-F--C.sub.6 H.sub.4)                                                  391 3-(4'-F--C.sub.6 H.sub.4)                                                  392 4-(2'-F--C.sub.6 H.sub.4)                                                  393 4-(3'-F--C.sub.6 H.sub.4)                                                  394 4-(4'-F--C.sub.6 H.sub.4)                                                  395 2-(2'-Cl--C.sub.6 H.sub.4)                                                 396 2-(3'-Cl--C.sub.6 H.sub.4)                                                 397 2-(4'-Cl--C.sub.6 H.sub.4)                                                 398 3-(2'-Cl--C.sub.6 H.sub.4)                                                 399 3-(3'-Cl--C.sub.6 H.sub.4)                                                 400 3-(4'-Cl--C.sub.6 H.sub.4)                                                 401 4-(2'-Cl--C.sub.6 H.sub.4)                                                 402 4-(3'-Cl--C.sub.6 H.sub.4)                                                 403 4-(4'-Cl--C.sub.6 H.sub.4)                                                 405 2-(2'-CH.sub.3 --C.sub.6 H.sub.4)                                          406 2-(3'-CH.sub.3 --C.sub.6 H.sub.4)                                          407 2-(4'-CH.sub.3 --C.sub.6 H.sub.4)                                          408 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)                                          409 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)                                          410 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)                                          411 4-(2'-CH.sub.3 --C.sub.6 H.sub.4)                                          412 4-(3'-CH.sub.3 --C.sub.6 H.sub.4)                                          413 4-(4'-CH.sub.3 --C.sub.6 H.sub.4)                                          414 2-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                      415 2-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                      416 2-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                      417 3-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                      418 3-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                      419 3-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                      420 4-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                      421 4-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                      422 4-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                      423 2-(2'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                       424 2-(3'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                       425 2-(4'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                       426 3-(2'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                       427 3-(3'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                       428 3-(4'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                       429 4-(2'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                       430 4-(3'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                       431 4-(4'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                       432 2-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                                 433 2-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                                 434 2-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                                 435 3-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                                 436 3-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                                 437 3-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                                 438 4-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                                 439 4-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                                 440 4-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                                 441 2-(2'-CH.sub.3 O--C.sub.6 H.sub.4)                                         442 2-(3'-CH.sub.3 O--C.sub.6 H.sub.4)                                         443 2-(4'-CH.sub.3 O--C.sub.6 H.sub.4)                                         444 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)                                         445 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)                                         446 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)                                         447 4-(2'-CH.sub.3 O--C.sub.6 H.sub.4)                                         448 4-(3'-CH.sub.3 O--C.sub.6 H.sub.4)                                         449 4-(4'-CH.sub.3 O--C.sub.6 H.sub.4)                                         450 2-(2'-O.sub.2 N--C.sub.6 H.sub.4)                                          451 2-(3'-O.sub.2 N--C.sub.6 H.sub.4)                                          452 2-(4'-O.sub.2 N--C.sub.6 H.sub.4)                                          453 3-(2'-O.sub.2 N--C.sub.6 H.sub.4)                                          454 3-(3'-O.sub.2 N--C.sub.6 H.sub.4)                                          455 3-(4'-O.sub.2 N--C.sub.6 H.sub.4)                                          456 4-(2'-O.sub.2 N--C.sub.6 H.sub.4)                                          457 4-(3'-O.sub.2 N--C.sub.6 H.sub.4)                                          458 4-(4'-O.sub.2 N--C.sub.6 H.sub.4)                                          459 2-(2'-NC--C.sub.6 H.sub.4)                                                 460 2-(3'-NC--C.sub.6 H.sub.4)                                                 461 2-(4'-NC--C.sub.6 H.sub.4)                                                 462 3-(2'-NC--C.sub.6 H.sub.4)                                                 463 3-(3'-NC--C.sub.6 H.sub.4)                                                 464 3-(4'-NC--C.sub.6 H.sub.4)                                                 465 4-(2'-NC--C.sub.6 H.sub.4)                                                 466 4-(3'-NC--C.sub.6 H.sub.4)                                                 467 4-(4'-NC--C.sub.6 H.sub.4)                                                 468 2-(2'-CF.sub.3 --C.sub.6 H.sub.4)                                          469 2-(3'-CF.sub.3 --C.sub.6 H.sub.4)                                          470 2-(4'-CF.sub.3 --C.sub.6 H.sub.4)                                          471 3-(2'-CF.sub.3 --C.sub.6 H.sub.4)                                          472 3-(3'-CF.sub.3 --C.sub.6 H.sub.4)                                          473 3-(4'-CF.sub.3 --C.sub.6 H.sub.4)                                          474 4-(2'-CF.sub.3 --C.sub.6 H.sub.4)                                          475 4-(3'-CF.sub.3 --C.sub.6 H.sub.4)                                          476 4-(4'-CF.sub.3 --C.sub.6 H.sub.4)                                          477 2-O--C.sub.6 H.sub.5                                                       475 3-O--C.sub.6 H.sub.5                                                       476 4-O--C.sub.6 H.sub.5                                                       478 2-O-(2'-F--C.sub.6 H.sub.4)                                                479 2-O-(3'-F--C.sub.6 H.sub.4)                                                480 2-O-(4'-F--C.sub.6 H.sub.4)                                                481 3-O-(2'-F--C.sub.6 H.sub.4)                                                482 3-O-(3'-F--C.sub.6 H.sub.4)                                                483 3-O-(4'-F--C.sub.6 H.sub.4)                                                484 4-O-(2'-F--C.sub.6 H.sub.4)                                                485 4-O-(3'-F--C.sub.6 H.sub.4)                                                486 4-O-(4'-F--C.sub.6 H.sub.4)                                                487 2-O-(2'-Cl--C.sub.6 H.sub.4)                                               488 2-O-(3'-Cl--C.sub.6 H.sub.4)                                               489 2-O-(4'-Cl--C.sub.6 H.sub.4)                                               490 3-O-(2'-Cl--C.sub.6 H.sub.4)                                               491 3-O-(3'-Cl--C.sub.6 H.sub.4)                                               492 3-O-(4'-Cl--C.sub.6 H.sub.4)                                               493 3-O-(4'-Cl--C.sub.6 H.sub.4)                                               494 4-O-(2'-Cl--C.sub.6 H.sub.4)                                               495 4-O-(3'-Cl--C.sub.6 H.sub.4)                                               496 4-O-(4'-Cl--C.sub.6 H.sub.4)                                               497 2-O-(2'-CH.sub.3 --C.sub.6 H.sub.4)                                        498 2-O-(3'-CH.sub.3 --C.sub.6 H.sub.4)                                        499 2-O-(4'-CH.sub.3 --C.sub.6 H.sub.4)                                        500 3-O-(2'-CH.sub.3 --C.sub.6 H.sub.4)                                        501 3-O-(3'-CH.sub.3 --C.sub.6 H.sub.4)                                        502 3-O-(4'-CH.sub.3 --C.sub.6 H.sub.4)                                        503 4-O-(2'-CH.sub.3 --C.sub.6 H.sub.4)                                        504 4-O-(3'-CH.sub.3 --C.sub.6 H.sub.4)                                        505 4-O-(4'-CH.sub.3 --C.sub.6 H.sub.4)                                        506 2-O-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                    507 2-O-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                    508 2-O-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                    509 3-O-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                    510 3-O-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                    511 3-O-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                    512 4-O-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                    513 4-O-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                    514 4-O-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                    515 2-O-(2'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                     516 2-O-(3'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                     517 2-O-(4'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                     518 3-O-(2'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                     519 3-O-(3'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                     520 3-O-(4'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                     521 4-O-(2'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                     522 4-O-(3'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                     523 4-O-(4'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                     524 2-O-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                               525 2-O-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                               526 2-O-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                               527 3-O-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                               528 3-O-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                               529 3-O-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                               530 4-O-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                               531 4-O-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                               532 4-O-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                               533 2-O-(2'-CH.sub.3 O--C.sub.6 H.sub.4)                                       534 2-O-(3'-CH.sub.3 O--C.sub.6 H.sub.4)                                       535 2-O-(4'-CH.sub.3 O--C.sub.6 H.sub.4)                                       536 3-O-(2'-CH.sub.3 O--C.sub.6 H.sub.4)                                       537 3-O-(3'-CH.sub.3 O--C.sub.6 H.sub.4)                                       538 3-O-(4'-CH.sub.3 O--C.sub.6 H.sub.4)                                       539 4-O-(2'-CH.sub.3 O--C.sub.6 H.sub.4)                                       540 4-O-(3'-CH.sub.3 O--C.sub.6 H.sub.4)                                       541 4-O-(4'-CH.sub.3 O--C.sub.6 H.sub.4)                                       542 2-O-(2'-O.sub.2 N--C.sub.6 H.sub.4)                                        543 2-O-(3'-O.sub.2 N--C.sub.6 H.sub.4)                                        544 2-O-(4'-O.sub.2 N--C.sub.6 H.sub.4)                                        545 3-O-(2'-O.sub.2 N--C.sub.6 H.sub.4)                                        546 3-O-(3'-O.sub.2 N--C.sub.6 H.sub.4)                                        547 3-O-(4'-O.sub.2 N--C.sub.6 H.sub.4)                                        548 4-O-(2'-O.sub.2 N--C.sub.6 H.sub.4)                                        549 4-O-(3'-O.sub.2 N--C.sub.6 H.sub.4)                                        550 4-O-(4'-O.sub.2 N--C.sub.6 H.sub.4)                                        551 2-O-(2'-NC--C.sub.6 H.sub.4)                                               552 2-O-(3'-NC--C.sub.6 H.sub.4)                                               553 2-O-(4'-NC--C.sub.6 H.sub.4)                                               554 3-O-(2'-NC--C.sub.6 H.sub.4)                                               555 3-O-(3'-NC--C.sub.6 H.sub.4)                                               556 3-O-(4'-NC--C.sub.6 H.sub.4)                                               557 4-O-(2'-NC--C.sub.6 H.sub.4)                                               558 4-O-(3'-NC--C.sub.6 H.sub.4)                                               559 4-O-(4'-NC--C.sub.6 H.sub.4)                                               560 2-O-(2'-CF.sub.3 --C.sub.6 H.sub.4)                                        561 2-O-(3'-CF.sub.3 --C.sub.6 H.sub.4)                                        562 2-O-(4'-CF.sub.3 --C.sub.6 H.sub.4)                                        563 3-O-(2'-CF.sub.3 --C.sub.6 H.sub.4)                                        564 3-O-(3'-CF.sub.3 --C.sub.6 H.sub.4)                                        565 3-O-(4'-CF.sub.3 --C.sub.6 H.sub.4)                                        566 4-O-(2'-CF.sub.3 --C.sub.6 H.sub.4)                                        567 4-O-(3'-CF.sub.3 --C.sub.6 H.sub.4)                                        568 4-O-(4'-CF.sub.3 --C.sub.6 H.sub.4)                                        569 2-Pyridinyl-2'                                                             570 2-Pyridinyl-3'                                                             571 2-Pyridinyl-4'                                                             572 3-Pyridinyl-2'                                                             573 3-Pyridinyl-3'                                                             574 3-Pyridinyl-4'                                                             575 4-Pyridinyl-2'                                                             576 4-Pyridinyl-3'                                                             577 4-Pyridinyl-4'                                                             578 2-Pyrimidinyl-2'                                                           579 2-Pyrimidinyl-3'                                                           580 2-Pyrimidinyl-4'                                                           581 3-Pyrimidinyl-2'                                                           582 3-Pyrimidinyl-3'                                                           583 3-Pyrimidinyl-4'                                                           584 4-Pyrimidinyl-2'                                                           585 4-Pyrimidinyl-3'                                                           586 4-Pyrimidinyl-4'                                                           587 2-Pyrazolyl-1'                                                             588 2-Pyrazolyl-3'                                                             589 2-Pyrazolyl-4'                                                             590 3-Pyrazolyl-1'                                                             591 3-Pyrazolyl-3'                                                             592 3-Pyrazolyl-4'                                                             593 4-Pyrazolyl-1'                                                             594 4-Pyrazolyl-3'                                                             595 4-Pyrazolyl-4'                                                             596 2-Isoxazolyl-3'                                                            597 2-Isoxazolyl-4'                                                            598 2-Isoxazolyl-5'                                                            599 3-Isoxazolyl-3'                                                            600 3-Isoxazolyl-4'                                                            601 3-Isoxazolyl-5'                                                            602 4-Isoxazolyl-3'                                                            603 4-Isoxazolyl-4'                                                            604 4-Isoxazolyl-5'                                                            605 2-Isothiazolyl-3'                                                          606 2-Isothiazolyl-4'                                                          607 2-Isothiazolyl-5'                                                          608 3-Isothiazolyl-3'                                                          609 3-Isothiazolyl-4'                                                          610 3-Isothiazolyl-5'                                                          611 4-Isothiazolyl-3'                                                          612 4-Isothiazolyl-4'                                                          613 4-Isothiazolyl-5'                                                          614 2-Imidazolyl-1'                                                            615 2-Imidazolyl-2'                                                            616 2-Imidazolyl-4'                                                            617 3-Imidazolyl-1'                                                            618 3-Imidazolyl-2'                                                            619 3-Imidazolyl-4'                                                            620 4-Imidazolyl-1'                                                            621 4-Imidazolyl-2'                                                            622 4-Imidazolyl-4'                                                            623 2-Oxazolyl-2'                                                              624 2-Oxazolyl-4'                                                              625 2-Oxazolyl-5'                                                              626 3-Oxazolyl-2'                                                              627 3-Oxazolyl-4'                                                              628 3-Oxazolyl-5'                                                              629 4-Oxazolyl-2'                                                              630 4-Oxazolyl-4'                                                              631 4-Oxazolyl-5'                                                              632 2-Thiazolyl-2'                                                             633 2-Thiazolyl-4'                                                             634 2-Thiazolyl-5'                                                             635 3-Thiazolyl-2'                                                             636 3-Thiazolyl-4'                                                             637 3-Thiazolyl-5'                                                             638 4-Thiazolyl-2'                                                             639 4-Thiazolyl-4'                                                             640 4-Thiazolyl-5'                                                           ______________________________________                                    

                  TABLE 13                                                         ______________________________________                                         3  STR183##                                                                      I: R.sup.1 = CH.sub.3                                                          II: R.sup.1 = CH.sub.2 --CH.sub.3                                              No.       B                                                                  ______________________________________                                         1       Pyrrolyl-3                                                               2 N--CH.sub.3 -Pyrrolyl-3                                                      3 N--C.sub.6 H.sub.5 -Pyrrolyl-3                                               4 N-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrrolyl-3                                 5 N-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrrolyl-3                                 6 N-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrrolyl-3                                 7 N-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrrolyl-3                                8 N-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrrolyl-3                                9 N-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrrolyl-3                                10 N-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrrolyl-3                                11 N-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrrolyl-3                                12 N-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrrolyl-3                                13 N-(4'-CN--C.sub.6 H.sub.4)-Pyrrolyl-3                                       14 N-(3'-CN--C.sub.6 H.sub.4)-Pyrrolyl-3                                       15 N-(2'-CN--C.sub.6 H.sub.4)-Pyrrolyl-3                                       16 N-(4'-Cl--C.sub.6 H.sub.4)-Pyrrolyl-3                                       17 N-(3'-Cl--C.sub.6 H.sub.4)-Pyrrolyl-3                                       18 N-(2'-Cl--C.sub.6 H.sub.4)-Pyrrolyl-3                                       19 Pyrrolyl-2                                                                  20 N--CH.sub.3 -Pyrrolyl-2                                                     21 N--C.sub.6 H.sub.5 -Pyrrolyl-2                                              22 N-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrrolyl-2                                23 N-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrrolyl-2                                24 N-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrrolyl-2                                25 N-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrrolyl-2                               26 N-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrrolyl-2                               27 N-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrrolyl-2                               28 N-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrrolyl-2                                29 N-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrrolyl-2                                30 N-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrrolyl-2                                31 N-(4'-CN--C.sub.6 H.sub.4)-Pyrrolyl-2                                       32 N-(3'-CN--C.sub.6 H.sub.4)-Pyrrolyl-2                                       33 N-(2'-CN--C.sub.6 H.sub.4)-Pyrrolyl-2                                       34 N-(4'-Cl--C.sub.6 H.sub.4)-Pyrrolyl-2                                       35 N-(3'-Cl--C.sub.6 H.sub.4)-Pyrrolyl-2                                       36 N-(2'-Cl--C.sub.6 H.sub.4)-Pyrrolyl-2                                       37 Furyl-2                                                                     38 5-CH.sub.3 -Furyl-2                                                         39 5-C.sub.6 H.sub.5 -Furyl-2                                                  40 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Furyl-2                                   41 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Furyl-2                                   42 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Furyl-2                                   43 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Furyl-2                                  44 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Furyl-2                                  45 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Furyl-2                                  46 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Furyl-2                                   47 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Furyl-2                                   48 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Furyl-2                                   49 5-(4'-CN--C.sub.6 H.sub.4)-Furyl-2                                          50 5-(3'-CN--C.sub.6 H.sub.4)-Furyl-2                                          51 5-(2'-CN--C.sub.6 H.sub.4)-Furyl-2                                          52 5-(4'-Cl--C.sub.6 H.sub.4)-Furyl-2                                          53 5-(3'-Cl--C.sub.6 H.sub.4)-Furyl-2                                          54 5-(2'-Cl--C.sub.6 H.sub.4)-Furyl-2                                          55 4-CH.sub.3 -Furyl-2                                                         56 4-C.sub.6 H.sub.5 -Furyl-2                                                  57 4-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Furyl-2                                   58 4-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Furyl-2                                   59 4-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Furyl-2                                   60 4-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Furyl-2                                  61 4-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Furyl-2                                  62 4-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Furyl-2                                  63 4-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Furyl-2                                   64 4-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Furyl-2                                   65 4-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Furyl-2                                   66 4-(4'-CN--C.sub.6 H.sub.4)-Furyl-2                                          67 4-(3'-CN--C.sub.6 H.sub.4)-Furyl-2                                          68 4-(2'-CN--C.sub.6 H.sub.4)-Furyl-2                                          69 4-(4'-Cl--C.sub.6 H.sub.4)-Furyl-2                                          70 4-(3'-Cl--C.sub.6 H.sub.4)-Furyl-2                                          71 4-(2'-Cl--C.sub.6 H.sub.4)-Furyl-2                                          72 Thienyl-2                                                                   73 5-CH.sub.3 -Thienyl-2                                                       74 5-C.sub.6 H.sub.5 -Thienyl-2                                                75 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-2                                 76 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-2                                 77 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-2                                 78 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-2                                79 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-2                                80 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-2                                81 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-2                                 82 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-2                                 83 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-2                                 84 5-(4'-CN--C.sub.6 H.sub.4)-Thienyl-2                                        85 5-(3'-CN--C.sub.6 H.sub.4)-Thienyl-2                                        86 5-(2'-CN--C.sub.6 H.sub.4)-Thienyl-2                                        87 5-(4'-Cl--C.sub.6 H.sub.4)-Thienyl-2                                        88 5-(3'-Cl--C.sub.6 H.sub.4)-Thienyl-2                                        89 5-(2'-Cl--C.sub.6 H.sub.4)-Thienyl-2                                        90 4-CH.sub.3 -Thienyl-2                                                       91 4-C.sub.6 H.sub.5 -Thienyl-2                                                92 4-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-2                                 93 4-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-2                                 94 4-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-2                                 95 4-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-2                                96 4-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-2                                97 4-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-2                                98 4-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-2                                 99 4-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-2                                 100 4-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-2                                101 4-(4'-CN--C.sub.6 H.sub.4)-Thienyl-2                                       102 4-(3'-CN--C.sub.6 H.sub.4)-Thienyl-2                                       103 4-(2'-CN--C.sub.6 H.sub.4)-Thienyl-2                                       104 4-(4'-Cl--C.sub.6 H.sub.4)-Thienyl-2                                       105 4-(3'-Cl--C.sub.6 H.sub.4)-Thienyl-2                                       106 4-(2'-Cl--C.sub.6 H.sub.4)-Thienyl-2                                       107 Thienyl-3                                                                  108 5-CH.sub.3 -Thienyl-3                                                      109 5-C.sub.6 H.sub.5 -Thienyl-3                                               110 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-3                                111 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-3                                112 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-3                                113 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-3                               114 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-3                               115 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-3                               116 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-3                                117 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-3                                118 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-3                                119 5-(4'-CN--C.sub.6 H.sub.4)-Thienyl-3                                       120 5-(3'-CN--C.sub.6 H.sub.4)-Thienyl-3                                       121 5-(2'-CN--C.sub.6 H.sub.4)-Thienyl-3                                       122 5-(4'-Cl--C.sub.6 H.sub.4)-Thienyl-3                                       123 5-(3'-Cl--C.sub.6 H.sub.4)-Thienyl-3                                       124 5-(2'-Cl--C.sub.6 H.sub.4)-Thienyl-3                                       125 Pyrazolyl-4                                                                126 N--CH.sub.3 -Pyrazolyl-4                                                   127 N--C.sub.6 H.sub.5 -Pyrazolyl-4                                            128 N-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrazolyl-4                              129 N-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrazolyl-4                              130 N-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrazolyl-4                              131 N-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrazolyl-4                             132 N-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrazolyl-4                             133 N-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrazolyl-4                             134 N-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrazolyl-4                              135 N-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrazolyl-4                              136 N-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrazolyl-4                              137 N-(4'-CN--C.sub.6 H.sub.4)-Pyrazolyl-4                                     138 N-(3'-CN--C.sub.6 H.sub.4)-Pyrazolyl-4                                     139 N-(2'-CN--C.sub.6 H.sub.4)-Pyrazolyl-4                                     140 N-(4'-Cl--C.sub.6 H.sub.4)-Pyrazolyl-4                                     141 N-(3'-Cl--C.sub.6 H.sub.4)-Pyrazolyl-4                                     142 N-(2'-Cl--C.sub.6 H.sub.4)-Pyrazolyl-4                                     143 3-CH.sub.3 --N-Methylpyrazolyl-4                                           144 3-C.sub.6 H.sub.5 --N-Methylpyrazolyl-4                                    145 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)--N-Methylpyrazolyl-4                     146 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)--N-Methylpyrazolyl-4                     147 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)--N-Methylpyrazolyl-4                     148 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)--N-Methylpyrazolyl-4                    149 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)--N-Methylpyrazolyl-4                    150 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)--N-Methylpyrazolyl-4                    151 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)--N-Methylpyrazolyl-4                     152 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)--N-Methylpyrazolyl-4                     153 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)--N-Methylpyrazolyl-4                     154 3-(4'-CN--C.sub.6 H.sub.4)--N-Methylpyrazolyl-4                            155 3-(3'-CN--C.sub.6 H.sub.4)--N-Methylpyrazolyl-4                            156 3-(2'-CN--C.sub.6 H.sub.4)--N-Methylpyrazolyl-4                            157 3-(4'-Cl--C.sub.6 H.sub.4)--N-Methylpyrazolyl-4                            158 3-(3'-Cl--C.sub.6 H.sub.4)--N-Methylpyrazolyl-4                            159 3-(2'-Cl--C.sub.6 H.sub.4)--N-Methylpyrazolyl-4                            160 Isoxazolyl-5                                                               161 3-CH.sub.3 -Isoxazolyl-5                                                   162 3-C.sub.6 H.sub.5 -Isoxazolyl-5                                            163 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Isoxazolyl-5                             164 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Isoxazolyl-5                             165 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Isoxazolyl-5                             166 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Isoxazolyl-5                            167 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Isoxazolyl-5                            168 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Isoxazolyl-5                            169 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Isoxazolyl-5                             170 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Isoxazolyl-5                             171 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Isoxazolyl-5                             172 3-(4'-CN--C.sub.6 H.sub.4)-Isoxazolyl-5                                    173 3-(3'-CN--C.sub.6 H.sub.4)-Isoxazolyl-5                                    174 3-(2'-CN--C.sub.6 H.sub.4)-Isoxazolyl-5                                    175 3-(4'-Cl--C.sub.6 H.sub.4)-Isoxazolyl-5                                    176 3-(3'-Cl--C.sub.6 H.sub.4)-Isoxazolyl-5                                    177 3-(2'-Cl--C.sub.6 H.sub.4)-Isoxazolyl-5                                    178 4-Chloroisoxazolyl-5                                                       179 3-CH.sub.3 -4-Chloroisoxazolyl-5                                           180 3-C.sub.6 H.sub.5 -4-Chloroisoxazolyl-5                                    181 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                     182 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                     183 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                     184 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                    185 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                    186 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                    187 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                     188 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                     189 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                     190 3-(4'-CN--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                            191 3-(3'-CN--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                            192 3-(2'-CN--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                            193 3-(4'-Cl--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                            194 3-(3'-Cl--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                            195 3-(2'-Cl--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                            196 Isoxazolyl-3                                                               196 5-CH.sub.3 -Isoxazolyl-3                                                   197 5-C.sub.6 H.sub.5 -Isoxazolyl-3                                            198 5-C.sub.6 H.sub.5 -Isoxazolyl-3                                            199 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Isoxazolyl-3                             200 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Isoxazolyl-3                             201 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Isoxazolyl-3                             202 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Isoxazolyl-3                            203 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Isoxazolyl-3                            204 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Isoxazolyl-3                            205 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Isoxazolyl-3                             206 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Isoxazolyl-3                             207 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Isoxazolyl-3                             208 5-(4'-CN--C.sub.6 H.sub.4)-Isoxazolyl-3                                    209 5-(3'-CN--C.sub.6 H.sub.4)-Isoxazolyl-3                                    210 5-(2'-CN--C.sub.6 H.sub.4)-Isoxazolyl-3                                    211 5-(4'-Cl--C.sub.6 H.sub.4)-Isoxazolyl-3                                    212 5-(3'-Cl--C.sub.6 H.sub.4)-Isoxazolyl-3                                    213 5-(2'-Cl--C.sub.6 H.sub.4)-Isoxazolyl-3                                    214 Isothiazolyl-5                                                             215 3-CH.sub.3 -Isothiazolyl-5                                                 216 3-C.sub.6 H.sub.5 -Isothiazolyl-5                                          217 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Isothiazolyl-5                           218 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Isothiazolyl-5                           219 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Isothiazolyl-5                           220 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Isothiazolyl-5                          221 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Isothiazolyl-5                          222 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Isothiazolyl-5                          223 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Isothiazolyl-5                           224 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Isothiazolyl-5                           225 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Isothiazolyl-5                           226 3-(4'-CN--C.sub.6 H.sub.4)-Isothiazolyl-5                                  227 3-(3'-CN--C.sub.6 H.sub.4)-Isothiazolyl-5                                  228 3-(2'-CN--C.sub.6 H.sub.4)-Isothiazolyl-5                                  229 3-(4'-Cl--C.sub.6 H.sub.4)-Isothiazolyl-5                                  230 3-(3'-Cl--C.sub.6 H.sub.4)-Isothiazolyl-5                                  231 3-(2'-Cl--C.sub.6 H.sub.4)-Isothiazolyl-5                                  232 Oxazolyl-4                                                                 233 2-CH.sub.3 -Oxazolyl-4                                                     234 2-C.sub.6 H.sub.5 -Oxazolyl-4                                              235 2-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Oxazolyl-4                               236 2-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Oxazolyl-4                               237 2-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Oxazolyl-4                               238 2-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Oxazolyl-4                              239 2-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Oxazolyl-4                              240 2-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Oxazolyl-4                              241 2-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Oxazolyl-4                               242 2-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Oxazolyl-4                               243 2-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Oxazolyl-4                               244 2-(4'-CN--C.sub.6 H.sub.4)-Oxazolyl-4                                      245 2-(3'-CN--C.sub.6 H.sub.4)-Oxazolyl-4                                      246 2-(2'-CN--C.sub.6 H.sub.4)-Oxazolyl-4                                      247 2-(4'-Cl--C.sub.6 H.sub.4)-Oxazolyl-4                                      248 2-(3'-Cl--C.sub.6 H.sub.4)-Oxazolyl-4                                      249 2-(2'-Cl--C.sub.6 H.sub.4)-Oxazolyl-4                                      250 Thiazolyl-4                                                                251 2-CH.sub.3 -Thiazolyl-4                                                    252 2-C.sub.6 H.sub.5 -Thiazolyl-4                                             253 2-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Thiazolyl-4                              254 2-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Thiazolyl-4                              255 2-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Thiazolyl-4                              256 2-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Thiazolyl-4                             267 2-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Thiazolyl-4                             258 2-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Thiazolyl-4                             259 2-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Thiazolyl-4                              260 2-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Thiazolyl-4                              261 2-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Thiazolyl-4                              262 2-(4'-CN--C.sub.6 H.sub.4)-Thiazolyl-4                                     263 2-(3'-CN--C.sub.6 H.sub.4)-Thiazolyl-4                                     264 2-(2'-CN--C.sub.6 H.sub.4)-Thiazolyl-4                                     265 2-(4'-Cl--C.sub.6 H.sub.4)-Thiazolyl-4                                     266 2-(3'-Cl--C.sub.6 H.sub.4)-Thiazolyl-4                                     267 2-(2'-Cl--C.sub.6 H.sub.4)-Thiazolyl-4                                     268 N--CH.sub.3 -1,2,4-Triazolyl-5                                             269 3-CH.sub.3 --N--CH.sub.3 -1,2,4-Triazolyl-5                                270 3-C.sub.6 H.sub.5 -N--CH.sub.3 -1,2,4-Triazolyl-5                          271 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5                 272 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazol             yl-5                                                                     273 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5                 274 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazo             lyl-5                                                                    275 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5                276 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazo             lyl-5                                                                    277 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5                 278 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazol             yl-5                                                                     279 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5                 280 3-(4'-CN--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5                 281 3-(3'-CN--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5                 282 3-(2'-CN--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5                 283 3-(4'-Cl--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5                 284 3-(3'-Cl--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5                 285 3-(2'-Cl--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5                 286 1,3,4-Oxadiazolyl-2                                                 287 5-CH.sub.3 -1,3,4-Oxadiazolyl-2                                            288 5-C.sub.6 H.sub.5 -1,3,4-Oxadiazolyl-2                                     289 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                      290 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                      291 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                      292 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                     293 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                     294 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                     295 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                      296 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                      297 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                      298 5-(4'-CN--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                             299 5-(3'-CN--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                             300 5-(2'-CN--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                             301 5-(4'-Cl--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                             302 5-(3'-Cl--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                             303 5-(2'-Cl--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                             304 1,2,4-Oxadiazolyl-3                                                        305 5-CH.sub.3 -1,2,4-Oxadiazolyl-3                                            306 5-C.sub.6 H.sub.5 -1,2,4-Oxadiazolyl-3                                     307 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                      308 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                      309 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                      310 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                     311 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                     312 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                     313 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                      314 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                      315 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                      316 5-(4'-CN--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                             317 5-(3'-CN--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                             318 5-(2'-CN--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                             319 5-(4'-Cl--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                             320 5-(3'-Cl--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                             321 5-(2'-Cl--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                             322 1,2,4-Oxadiazolyl-5                                                        323 3-CH.sub.3 -1,2,4-Oxadiazolyl-5                                            324 3-C.sub.6 H.sub.5 -1,2,4-Oxadiazolyl-5                                     325 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                      326 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                      327 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                      328 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                     329 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                     330 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                     331 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                      332 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                      333 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                      334 3-(4'-CN--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                             335 3-(3'-CN--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                             336 3-(2'-CN--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                             337 3-(4'-Cl--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                             338 3-(3'-Cl--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                             339 3-(2'-Cl--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                             340 1,2,4-Thiadiazolyl-3                                                       341 5-CH.sub.3 -1,2,4-Thiadiazolyl-3                                           342 5-C.sub.6 H.sub.5 -1,2,4-Thiadiazolyl-3                                    343 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                     344 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                     345 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                     346 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                    347 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                    348 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                    349 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                     350 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                     351 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                     352 5-(4'-CN--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                            353 5-(3'-CN--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                            354 5-(2'-CN--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                            355 5-(4'-Cl--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                            356 5-(3'-Cl--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                            357 5-(2'-Cl--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                            358 1,3,4-Thiadiazolyl-2                                                       359 5-CH.sub.3 -1,3,4-Thiadiazolyl-2                                           360 5-C.sub.6 H.sub.5 -1,3,4-Thiadiazolyl-2                                    361 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                     362 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                     363 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                     364 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                    365 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                    366 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                    367 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                     368 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                     369 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                     370 5-(4'-CN--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                            371 5-(3'-CN--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                            372 5-(2'-CN--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                            373 5-(4'-Cl--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                            374 5-(3'-Cl--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                            375 5-(2'-Cl--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                            376 Pyridinyl-2                                                                377 Pyridinyl-4                                                                378 Pyridazinyl-3                                                              379 Pyridazinyl-4                                                              380 Pyridazinyl-2                                                              381 Pyrimidinyl-4                                                              382 Pyrimidinyl-5                                                              383 Pyrimidinyl-2                                                              384 Pyridinyl-3                                                              ______________________________________                                    

                                      TABLE 14                                     __________________________________________________________________________     Selected physical data of some compounds                                       No.                                                                               Compound             .sup.1 H--NMR (ppm)                                    __________________________________________________________________________       1                                                                                                                2  3.8(s, 3H); 3.75(s, 3H)                    - 2                                                                                                             3  3.8(2s, 2×3H)                        - 3                                                                                                             4  3.8(s, 3H); 3.75(s, 3H)                    - 4                                                                                                             5  3.95(q, 2H, I=7.5Hz); 3.8(s, 3H)                                              - 5                                                                          6  4.05(q, 2H, I=7.5 Hz); 3.85(s, 3H)         - 6                                                                                                             7  4.0(q, 2H, I=7.5Hz); 3.8(s, 3H)                                               - 7                                                                          8  3.8(s, 3H); 3.75(s, 3H)                    - 8                                                                                                             9  3.8(s, 3H); 3.75(s, 3H)                    - 9                                                                                                             0  3.85(s, 3H); 3.8(s, 3H)                    - 10                                                                                                            1  4.0(s, 3H); 3.8(s, 3H), 3.75(s,                                             3H)                                           - 11                                                                                                            2  3.8(s, 3H); 3.75(s, 3H)                    - 12                                                                                                            3  3.8(s, 3H); 3.75(s, 3H)                    - 13                                                                                                            4  3.8(s, 3H); 3.75(s, 3H)                    - 14                                                                                                            5  3.8(s, 3H); 3.75(s, 3H)66                  - 15                                                                                                            6  3.8(s, 3H); 3.75(s, 3H)                    - 16                                                                                                            7  4.0(q, 2H, I=7.5Hz); 3.8(s, 3H)                                               - 17                                                                         8  3.8(2s, each 3H)                           - 18                                                                                                            9  3.8(2s, each 3H)                           - 19                                                                                                            0  3.8(s, 3H); 3.75(s, 3H)                    - 20                                                                                                            1  3.8(s, 3H); 3.75(s, 3H)                    - 21                                                                                                            2  3.8(s, 3H); 3.75(s, 3H)                    - 22                                                                                                            3  3.8(s, 3H); 3.75(s, 3H)                    - 23                                                                                                            4  3.8(s, 3H); 3.75(s, 3H)                    - 24                                                                                                            5  3.8(s, 6H)                                 - 25                                                                                                            4  3.75(2s, each 3H)                          - 26                                                                                                            6  3.8(s, 3H); 3.75(s, 3H)                    - 27                                                                                                            7  3.8(s, 3H); 3.75(s, 3H)                    - 28                                                                                                            8  3.8(s, 3H); 3.75(s, 3H)                    - 29                                                                                                            9  3.8(s, 3H); 3.75(s, 3H)                    - 30                                                                                                            8  3.8(s, 6H)                              __________________________________________________________________________

                  TABLE 52                                                         ______________________________________                                         Selected physical data of some compounds                                          -                                                                           2  STR214##                                                                      No.    X.sub.m       mp (° C.)                                                                      .sup.1 H-NMR(ppm) or IR(cm.sup.-1)               ______________________________________                                          1   H                      3.75(2s, each 3H)                                     2 2-CH.sub.3  3.75(2s, each 3H)                                                3 3-CH.sub.3  3.75(2s, each 3H)                                                4 2,4-(CH.sub.3).sub.2  3.75(2s, each 3H)                                      5 4-C.sub.2 H.sub.5  3.75(2s, each 3H)                                         6 4-i-C.sub.3 H.sub.7  3.75(2s, each 3H)                                       7 4-t-C.sub.4 H.sub.9  3.75(2s, each 3H)                                       8 3,4-(CH.sub.3).sub.2  3.75(2s, each 3H)                                      9 3-Cl  3.75(2s, each 3H)                                                     10 3-Br  3.75(2s, each 3H)                                                     11 3-CF.sub.3  3.75(2s, each 3H)                                               12 4-Br  3.75(2s, each 3H)                                                     13 4-F  3.75(2s, each 3H)                                                      14 4-CF.sub.3  3.75(2s, each 3H)                                               15 4-OCH.sub.3  3.8(s, 3H); 3.75(2s,                                              each 3H)                                                                    16 4-CN  3.75(2s, each 3H)                                                     17 3-CH.sub.3 -4-O-i-C.sub.3 H.sub.7  3.75(2s, each 3H)                        18 3,4-Cl.sub.2  3.75(2s, each 3H)                                             19 3-CH.sub.3 -4-OCH.sub.3  3.85(s, 3H); 3.75                                     (2s, each 3H)                                                               20 4-NO.sub.2 112                                                              21 3,5-(CH.sub.3).sub.2  3.75(2s, each 3H)                                     22 3-CH.sub.3 -4-Cl  3.75(2s, each 3H)                                         23 3-Cl-4-CH.sub.3  3.75(2s, each 3H)                                        ______________________________________                                    

                  TABLE 53                                                         ______________________________________                                         Selected physical data of some compounds                                          -                                                                           3  STR215##                                                                       -                        mp    .sup.1 H-NMR(ppm) or                           No. X.sub.m (° C.) IR(cm.sup.-1)                                      ______________________________________                                          1   2-CH.sub.3 -4-C(CH.sub.3)═N--O--C.sub.2 H.sub.5                                                       3.8(s, 3H); 3.75(s,                                 3H)                                                                          2 2-CH.sub.3 -4-C(CH.sub.3)═N--O-  3.8(s, 3H); 3.75(s,                     (trans-CH.sub.2 --CH═CHCl)  3H)                                            3 2,5-(CH.sub.3).sub.2 -4-C(CH.sub.3)═N--  3.95(s, 3H); 3.8(s,                                            OCH.sub.3  3H); 3.75(s, 3H)                     4 2,5-(CH.sub.3).sub.2 -4-C(CH.sub.3)═N--  3.8(s, 3H); 3.75(s,                                            OC.sub.2 H.sub.5  3H)                           5 2,5-(CH.sub.3).sub.2 -4-C(CH.sub.3)═N--O-  3.85(s, 3H); 3.75(s,                                         (trans-CH.sub.2 --CH═CHCl)  3H)                                            6 2-CH.sub.3 -4-C(C.sub.2 H.sub.5)═N                                     --OCH.sub.3  3.95(s, 3H); 3.8(s,                    3H); 3.75 (s, 3H)                                                            7 2-CH.sub.3 -4-C(C.sub.2 H.sub.5)═N--  3.8(s, 3H); 3.75(s,                                               O--C.sub.2 H.sub.5  3H)                         8 2-CH.sub.3 -4-C(C.sub.2 H.sub.5)═N--O-Allyl  3.8(s, 3H); 3.75(s,           3H)                                                                          9 2-CH.sub.3 -4-C(C.sub.2 H.sub.5)═N--O-  3.8(s, 3H); 3.75(s,                                             (trans-CH.sub.2 --CH═CHCl)  3H)                                           10 2,5-(CH.sub.3).sub.2 -4-C(C.sub.2                                          H.sub.5)═N--  3.95(S, 3H); 3.8(s,                                            OCH.sub.3  3H); 3.75(s, 3H)                    11 2,5-(CH.sub.3).sub.2 -4-C(C.sub.2 H.sub.5)═N--  3.8(s, 3H);                                           3.75(s,                                           O--C.sub.2 H.sub.5  3H)                                                       12 2,5-(CH.sub.3).sub.2 -4-C(C.sub.2 H.sub.5)═N--  3.8(s, 3H);                                           3.75(s,                                           O-Allyl  3H)                                                                  13 2-Cl  3.8(s, 3H); 3.75(s,                                                      3H)                                                                         14 4-Cl  3.8(s, 3H); 3.75(s,                                                      3H)                                                                         15 2-CH.sub.3 -4-Cl  3.8(s, 3H); 3.75(s,                                          3H)                                                                         16 2-Cl-4-CH.sub.3  3.8(s, 3H); 3.75(s,                                           3H)                                                                         17 2-Cl-5-CH.sub.3  3.8(s, 3H); 3.75(s,                                           3H)                                                                         18 2,5-(CH.sub.3).sub.2 -4-C(CH.sub.3)═N--  3.8(s, 3H); 3.75(s,                                            O-Allyl  3H)                                   19 2,5-(CH.sub.3).sub.2 -4-C(C.sub.2 H.sub.5)═N--  3.8(s, 3H);                                           3.75(s,                                           O-(trans-CH.sub.2 --CH═CHCl)  3H)                                       ______________________________________                                    

                  TABLE 54                                                         ______________________________________                                         4  STR216##                                                                       - I: R.sup.1 = CH.sub.3                                                       II: R.sup.1 = C.sub.2 H.sub.5                                                  No.            B                                                             ______________________________________                                         1            2-Pyridyl                                                           2 3-Trifluormethyl-2-pyridyl                                                   3 5-Trifluormethyl-2-pyridyl                                                   4 3,5-Bis-(trifluoromethyl)-2-pyridyl                                          5 3,5-Dichloro-2-pyridyl                                                       6 3-Chloro-5-trifluoromethyl-2-pyridyl                                         7 3,5-Dichloro-2-pyridyl                                                       8 2-Chloro-4-trifluoromethylphenyl                                             9 2-Benzothiazolyl                                                             10  5-Chloro-4-methyl-2-benzimidazolyl                                         11  2-Benzoxazolyl                                                             12  1-Methyl-5-trifluoromethylimi-                                              dazo[5,4-a]-pyridin-2-yl                                                      13  5-Chloro-2-pyrimidinyl                                                     14  4-Methyl-5-phenyl-2-thiazolin-2-yl                                         15  4-Methyl-5-phenyl-2-oxazolin-2-yl                                          16  7-Trifluoromethyl-4-quinolinyl                                           ______________________________________                                    

                  TABLE 55                                                         ______________________________________                                         Selected physical data of some compounds                                       5  STR217##                                                                      No.      X.sub.m  mp (° C.)                                                                         .sup.1 H-NMR(ppm) or IR(cm.sup.-1)               ______________________________________                                         1      H                3.75(s, 3H); 3.65(s, 3H)                                 2 4-OCH.sub.3 3.8(s, 3H); 3.75(s, 3H);                                           3.65(s, 3H)                                                                  3 4-CH.sub.3 3.75(s, 3H); 3.65(s, 3H)                                          4 4-Cl 3.75(s, 3H); 3.65(s, 3H)                                                5 4-CF.sub.3 3.75(s, 3H); 3.65(s, 3H)                                          6 3,5-(CF.sub.3).sub.2 3.75(s, 3H); 3.65(s, 3H)                                7 2,4-Cl.sub.2 3.75(s, 3H); 3.65(s, 3H)                                        8 3,4-Cl.sub.2 3.75(s, 3H); 3.65(s, 3H)                                      ______________________________________                                    

Example 6

O-Methyl-N-(2-methylphenyl)-N-propionyl-hydroxylamine (Table 21, No. 1)

a) N-(2-Methylphenyl)-N-propionyl-hydroxylamine

At 25 to 30° C., 12.5 g (0.135 mol) of propionyl Chloroide and then 10.7 g (0.135 mol) of pyridine are dripped into 30 g of N-(2-methylphenyl)-hydroxylamine (crude product, prepared according to Bamberger et al., Anm. Chem. 316 (1901), 278; content approx. 80%=0.2 mol) in 500 ml of methylene Chloroide. The mixture is stirred for 30 minutes at room temperature, and is then extracted with dilute hydroChloroic acid and water. The organic phase is dried over MgSO₄ and evaporated down. The residue is purified by column chromatography with mixtures of cyclohexane and ethyl acetate. There is obtained 22.7 g (0.127 mol=63%) of the title compound as a yellow oil.

¹ H-NMR (COCl₃ ; δ in ppm): 9.4 (s, broad, 1H, OH); 7.2 (m, 4H, phenyl); 2.4 (s, 3H, CH₃); 2.1 (q, broad, 2H, CH₂); 1.1 (t, 3H, I=7 Hz, CH₃)

b) O-Methyl-N-(2-methylphenyl)-N-propionyl-hydroxylamine (Table 21, No. 1)

At 25 to 30° C., a solution of 22.7 g (0.127 mol) (Example 6a) of N-(2-methylphenyl)-N-propionyl-hydroxylamine in 50 ml of dimethylformamide is dripped into a stirred mixture of 3.4 g (0.14 mol) of NaH in 150 ml of dimethylformamide. After completion of gas evolution (15 mins) 18.4 g (0.13 mol) of methyl iodide is added and the mixture is stirred overnight at room temperature. The reaction mixture is then diluted with water and the aqueous phase is extracted three times with methyl tert-butyl ether. The combined organic phases are extracted with water, dried over MgSO₄ and evaporated down. The residue is purified by column chromatography with mixtures of cyclohexane and ethyl acetate. There is obtained 18 g (0.081 mol=64%) of the title compound as a yellow oil.

¹ H-NMR (COCl₃ ; δ in ppm): 7.2 (m, 4H, phenyl); 3.7 (s, broad, 3H, OCH₃); 2.6 (s, very broad, 2H, CH₂); 2.3 (s, 3H, CH₃); 1.2 (s, broad, 3H, CH₃)

Example 7

O-Methyl-N-(2-bromomethylphenyl)-N-propionyl-hydroxylamine (Table 21, No. 2)

A mixture of 10 g (51.8 mmol) of the hydroxylamine derivative from Example 1, 11 g (61 mmol) of N-bromosuccinimide and 0.1 g of azoisobutyrodinitrile in 100 ml of CCl₄ is refluxed. One drop of bromine is added and the mixture is refluxed for a further 2.5 hours. The reaction mixture is cooled to room temperature, washed with water, dried over MgSO₄ and evaporated down. The residue is purified by column chromatography with mixtures of cyclohexane and ethyl acetate. There is obtained in this sequence 3.4 g (7.9 mmol=15%) of O-methyl-N-(2-bromomethylphenyl)-d-(α,α-dibromopropionyl)-hydroxylamine, 3.8 g (10.8 mmol=21%) of O-methyl-N-(2-bromomethylphenyl)-N-(α-bromopropionyl)-hydroxylamine, 2.3 g (8.5 g (8.5 mmol=16%) of the title compound and 3.5 g of starting material, each as brown oils.

a) O-Methyl-N-(2-bromomethylphenyl)-N-(α,α-dibromopropionyl)-hydroxylamine

7.55 (m, 1H, phenyl); 7.4 (m, 3H, phenyl); 4.5 (s, 2H, CH₂, Br); 3.8 (s, 3H, OCH₃); 2.75 (s, 3H, CH₃)

b) O-Methyl-N-(2-bromomethylphenyl)-N-(α-bromopropionyl)-hydroxylamine

7.5 (s, broad, 1H, phenyl); 7.4 (s, broad, 3H, phenyl); 5.15 (s, broad, 1H, CH--Br); 4.5 (dd, broad, 2H, CH₂ --Br); 3.8 (s, 3H, OCH₃); 1.85 (s, broad, 3H, CH₃)

c) O-Methyl-N-(2-bromomethylphenyl)-N-propionyl-hydroxylamine

7.5 (m, 1H, phenyl); 7.35 (m, 3H, phenyl); 4.5 (s, broad, 2H, CH₂ --Br); 3.75 (s, 3H, OCH₃); 2.55 (s, very broad, CH₂); 1.2 (t, 3H, I=7 Hz, CH₃)

Example 8

O-Methyl-N-(2-(2'-methylphenyloxymethyl)-phenyl)-N-propionyl-hydroxylamine (Table 21, No. 3)

0.12 g (5 mmol) of sodium hydride is added to a solution of 0.4 g (3.7 mmol) of o-cresol in 5 ml of dimethylformamide. Upon completion of gas evolution, 1 g (3.6 mmol) of the benzyl bromide from Example 2c is added and the mixture is stirred for 2 hours at room temperature. The reaction mixture is diluted with water and extracted three times with methyl tert-butyl ether. The combined organic phases are washed with water, dried over MgSO₄ and evaporated down. The residue is chromatographed with mixtures of cyclohexane and ethyl acetate using Al₂ O₃ and silica gel. There is obtained 0.4 g (1.33 mmol=37%) of the title compound as a yellow oil.

¹ H-NMR (COCl₃ ; δ in ppm): 7.7 (d, broad, 1H, phenyl); 7.35 (m, 3H, phenyl); 7.1 (m, 2H, phenyl); 6.85 (t, broad, 2H, phenyl); 5.05 (s, 2H, OCH₃); 3.7 (s, 3H, OCH₃); 2.55 (s, very broad, 2H, CH₂); 2.3 (s, 3H, CH₃); 1.2 (t, broad, 3H, CH₃)

Example 9

N-Methyl-N'-methoxy-N'-2-methylphenylurea (Table 21, No. 5)

a) Phenyl N-hydroxy-N-(2-methylphenyl)-carbamate

A mixture of 2.5 g (20 mmol) of N-(2-methylphenyl)-hydroxylamine (crude product, obtained according to Bamberger et al., Anm. Chem. 316 (1901), 278), 3.5 g (25 mmol) of K₂ CO₃ and 3.5 g (22 mmol) of phenyl Chlorooformate in 20 ml of CH₂ Cl₂ is stirred for 2 hours at room temperature. The reaction mixture is then extracted with water, dried over MgSO₄ and evaporated down. The residue is purified by column chromatography with mixtures of cyclohexane and ethyl acetate. There is obtained 2.0 g (8.2 mmol=42%) of the title compound as a colorless solid (mp=98° C.).

¹ H-NMR (COCl₃ ; δ in ppm): 7-7.6 (m, 10H, phenyl, OH); 2.35 (s, 3H, CH₃)

b) Phenyl N-methoxy-N-(2-methylphenyl)-carbamate

A mixture of 2.0 g (8.2 mmol) of the phenyl carbamate from Example 4a, 2 g (15 mmol) of K₂ CO₃ and 1.3 g (10 mmol) of dimethyl sulfate in 20 ml of acetone is stirred for 3 hours at room temperature. The reaction mixture is then filtered and evaporated down, and the residue is purified by column chromatography with mixtures of cyclohexane and ethyl acetate. There is obtained 1.5 g (5.8 mmol=71%) of the title compound as a colorless oil, which slowly crystallizes (mp=60° C.).

¹ H-NMR (COCl₃ ; δ in ppm): 7.1-7.5 (m, 9H, phenyl); 3.8 (s, 3H, OCH₃); 2.4 (s, 3H, CH₃)

c) N-Methyl-N'-methoxy-N'-2-methylphenylurea (Table 21, No. 5)

1.5 g (5.8 mmol) of the phenyl carbamate from Example 4b in 20 ml of 40% strength aqueous methylamine solution is stirred for 1 hour at 50° C. The reaction mixture is then cooled and extracted with CH₂ Cl₂. The combined organic phases are dried over MgCO₄ and evaporated down. The residue is purified by column chromatography with mixtures of cyclohexane and ethyl acetate. There is obtained 0.6 g (3.1 mmol=53%) of the title compound as a colorless solid (mp=99° C.).

¹ H-NMR (COCl₃ ; δ in ppm): 7.2 (m, 4H, phenyl); 5.9 (s, broad, 1H, NH); 3.6 (s, 3H, OCH₃); 2.9 (d, 3H, I=approx. 2 Hz, N--CH₃); 2.3 (s, 3H, CH₃)

Example 18

N-Methyl-N'-methoxy-N'-(2-2',5'-dimethylphenoxymethyl)-phenyl)-urea

a) Phenyl N-methoxy-N-(2-bromomethylphenyl)-carbamate

A mixture of 125 g (0.486 mol) of methyl N-methoxy-N-(2-methylphenyl)-carbamate (Example 4b), 88 g (0.494 mol) of N-bromosuccinimide and 1 g of azoisobutyrodinitrile (AIBN) in 800 ml of CCl₄ is refluxed for about 12 hours. 10 g of N-bromosuccinimide is then added and the mixture is refluxed for about 4 hours. The reaction mixture is extracted with water and sodium thiosulfate solution, and the organic phase is dried over MgSO₄ and evaporated down under reduced pressure. The residue crystallizes, is stirred with hexane/methyl tert-butyl ether and suction dried. There is obtained 107 g (63%) of the title compound as a colorless solid.

¹ H-NMR (CDCl₃ ; δ in ppm): 7.1-7.6 (m, 9H, phenyl); 4.65 (s, 2H, CH₂ Br); 3.9 (s, 3H, OCH₃)

b) Phenyl N-methoxy-N-(2-(2',5'-dimethylphenoxymethyl)-phenyl)-carbamate

A mixture of 7 g (20 mmol) of the bromide of Example 5a and 3.3 g (22 mmol) of sodium iodide in 50 ml of acetone is refluxed for 30 minutes. The precipitated solid is then filtered off and the organic phase is evaporated down under reduced pressure. The crude product obtained is the iodide corresponding to Example 5a, which is used in the next reaction without any further purification.

The crude product obtained above is dissolved in 100 ml of dimethylformamide, 3 g (21.6 mmol) of K₂ CO₃ and 7.3 g (60 mmol) of 2,5-dimethylphenol are added and the mixture is stirred overnight at room temperature. The reaction mixture is then diluted with water and the aqueous phase is extracted three times with methyl tert-butyl ether. The combined organic phases are extracted with water, dried over MgSO₄ and evaporated down. The residue is purified by column chromatography using methylene chloride/cyclohexane (1:2) over Al₂ O₃. There is obtained 7.3 g (94%) of the title compound as a yellow oil.

¹ H-NMR (CDCl₃ ; δ in PPM): 7.7 (d, broad, 1H, phenyl); 7-7.6 (m, 9H, phenyl); 6.7 (m, 2H, phenyl); 5.2 (s, 2H, OCH₂); 3.85 (s, 3H, OCH₃); 2.3 (s, 6H, 2×CH₃).

c) N-Methyl-N'-methoxy-N'-(2-(2',5'-dimethylphenoxymethyl)-phenyl)-urea (Table 1, No. V.71)

A mixture of 3.4 g (8.8 mmol) of the phenyl carbamate of Example 5b and 20 ml of 40% strength aqueous methylamine solution is stirred for 2 hours at 50° C. The mixture is allowed to cool and is then extracted with methylene chloride. The organic phase is evaporated down and the residue is purified by column chromatography with mixtures of cyclohexane/ethyl acetate. There is obtained 1 g (36%) of the title compound as a colorless solid (mp=101° C.).

¹ H-NMR (CDCl₃ ; δ in PPM): 7.75 (m, 1H, phenyl); 6.6-7.4 (m, 6H, phenyl); 6.0 (s, broad, NH); 5.15 (s, 2H, OCH₂); 3.65 (s, 3H, OCH₃); 2.9 (d, 3H, N--CH₃); 2.3 (s, 3H, CH₃); 2.25 (s, 3H, CH₃).

The compounds listed in the tables below may be prepared analogously. Compound I.1 from Table 15 has for instance the following formula ##STR218##

                  TABLE 15                                                         ______________________________________                                            -      I: R.sup.1 = CH.sub.3, Z = CH.sub.3                                    II: R.sup.1 = CH.sub.2 --CH.sub.3, Z = CH.sub.3                                III: R.sup.1 = CH.sub.3, Z = C.sub.2 H.sub.5                                   IV: R.sup.1 = CH.sub.2 --CH.sub.3, Z = C.sub.2 H.sub.5                         V: R.sup.1 = CH.sub.3, Z = NHCH.sub.3                                          VI: R.sup.1 = CH.sub.2 --CH.sub.3, Z = NHCH.sub.3                            No.     Xm                                                                     ______________________________________                                          1      H                                                                         2 2-F                                                                          3 3-F                                                                          4 4-F                                                                          5 2,4-F.sub.2                                                                  6 2,4,6-F.sub.3                                                                7 2,3,4,5,6-F.sub.5                                                            8 2,3-F.sub.2                                                                  9 2-Cl                                                                         10 3-Cl                                                                        11 4-Cl                                                                        12 2,3-Cl.sub.2                                                                13 2,4-Cl.sub.2                                                                14 2,5-Cl.sub.2                                                                15 2,6-Cl.sub.2                                                                16 3,4-Cl.sub.2                                                                17 3,5-Cl.sub.2                                                                18 2,3,4-Cl.sub.3                                                              19 2,3,5-Cl.sub.3                                                              20 2,3,6-Cl.sub.3                                                              21 2,4,5-Cl.sub.3                                                              22 2,4,6-Cl.sub.3                                                              23 3,4,5-Cl.sub.3                                                              24 2,3,4,6-Cl.sub.4                                                            25 2,3,5,6-Cl.sub.4                                                            26 2,3,4,5,6-Cl.sub.5                                                          27 2-Br                                                                        28 3-Br                                                                        29 4-Br                                                                        30 2,4-Br.sub.2                                                                31 2,5-Br.sub.2                                                                32 2,6-Br.sub.2                                                                33 2,4,6-Br.sub.3                                                              34 2,3,4,5,6-Br.sub.5                                                          35 2-I                                                                         36 3-I                                                                         37 4-I                                                                         38 2,4-I.sub.2                                                                 39 2-Cl, 3-F                                                                   40 2-Cl, 4-F                                                                   41 2-Cl, 5-F                                                                   42 2-Cl, 6-F                                                                   43 2-Cl, 3-Br                                                                  44 2-Cl, 4-Br                                                                  45 2-Cl, 5-Br                                                                  46 2-Cl, 6-Br                                                                  47 2-Br, 3-Cl                                                                  48 2-Br, 4-Cl                                                                  49 2-Br, 5-Cl                                                                  50 2-Br, 3-F                                                                   51 2-Br, 4-F                                                                   52 2-Br, 5-F                                                                   53 2-Br, 6-F                                                                   54 2-F, 3-Cl                                                                   55 2-F, 4-Cl                                                                   56 2-F, 5-Cl                                                                   57 3-Cl, 4-F                                                                   58 3-Cl, 5-F                                                                   59 3-Cl, 4-Br                                                                  60 3-Cl, 5-Br                                                                  61 3-F, 4-Cl                                                                   62 3-F, 4-Br                                                                   63 3-Br, 4-Cl                                                                  64 3-Br, 4-F                                                                   65 2,6-Cl.sub.2, 4-Br                                                          66 2-CH.sub.3                                                                  67 3-CH.sub.3                                                                  68 4-CH.sub.3                                                                  69 2,3-(CH.sub.3).sub.2                                                        70 2,4-(CH.sub.3).sub.2                                                        71 2,5-(CH.sub.3).sub.2                                                        72 2,6-(CH.sub.3).sub.2                                                        73 3,4-(CH.sub.3).sub.2                                                        74 3,5-(CH.sub.3).sub.2                                                        75 2,3,5-(CH.sub.3).sub.3                                                      76 2,3,4-(CH.sub.3).sub.3                                                      77 2,3,6-(CH.sub.3).sub.3                                                      78 2,4,5-(CH.sub.3).sub.3                                                      79 2,4,6-(CH.sub.3).sub.3                                                      80 3,4,5-(CH.sub.3).sub.3                                                      81 2,3,4,6-(CH.sub.3).sub.4                                                    82 2,3,5,6-(CH.sub.3).sub.4                                                    83 2,3,4,5,6-(CH.sub.3).sub.5                                                  84 2-C.sub.2 H.sub.5                                                           85 3-C.sub.2 H.sub.5                                                           86 4-C.sub.2 H.sub.5                                                           87 2,4-(C2H5).sub.2                                                            88 2,6-(C.sub.2 H.sub.5).sub.2                                                 89 3,5-(C.sub.2 H.sub.5).sub.2                                                 90 2,4,6-(C.sub.2 H.sub.5).sub.3                                               91 2-n-C.sub.3 H.sub.7                                                         92 3-n-C.sub.3 H.sub.7                                                         93 4-n-C.sub.3 H.sub.7                                                         94 2-i-C.sub.3 H.sub.7                                                         95 3-i-C.sub.3 H.sub.7                                                         96 4-i-C.sub.3 H.sub.7                                                         97 2,4-(i-C.sub.3 H.sub.7).sub.2                                               98 2,6-(i-C.sub.3 H.sub.7).sub.2                                               99 3,5-(i-C.sub.3 H.sub.7).sub.2                                              100 2,4,6-(i-C.sub.3 H.sub.7).sub.3                                            101 2-s-C.sub.4 H.sub.9                                                        102 3-s-C.sub.4 H.sub.9                                                        103 4-s-C.sub.4 H.sub.9                                                        104 2-t-C.sub.4 H.sub.9                                                        105 3-t-C.sub.4 H.sub.9                                                        106 4-t-C.sub.4 H.sub.9                                                        107 2,3-(t-C.sub.4 H.sub.9).sub.2                                              108 2,4-(t-C.sub.4 H.sub.9).sub.2                                              109 2,5-(t-C.sub.4 H.sub.9).sub.2                                              110 2,6-(t-C.sub.4 H.sub.9).sub.2                                              111 3,4-(t-C.sub.4 H.sub.9).sub.2                                              112 2,4,6-(t-C.sub.4 H.sub.9).sub.3                                            113 4-n-C.sub.9 H.sub.19                                                       114 4-n-C.sub.12 H.sub.25                                                      115 4-n-C.sub.15 H.sub.31                                                      116 4-(1,1,3,3-Tetramethylbutyl)                                               117 4-(2,4,4-Trimethylpropyl)                                                  118 2-t-C.sub.4 H.sub.9, 4-CH.sub.3                                            119 2-t-C.sub.4 H.sub.9, 5-CH.sub.3                                            120 2,6-(t-C.sub.4 H.sub.9).sub.2, 4-CH.sub.3                                  121 2-CH.sub.3, 4-t-C.sub.4 H.sub.9                                            122 2-CH.sub.3, 6-t-C.sub.4 H.sub.9                                            123 2-CH.sub.3, 4-i-C.sub.3 H.sub.7                                            124 2-CH.sub.3, 5-i-C.sub.3 H.sub.7                                            125 3-CH.sub.3, 4-i-C.sub.3 H.sub.7                                            126 2-i-C.sub.3 H.sub.7, 5-CH.sub.3                                            127 2,4-(t-C.sub.4 H.sub.9).sub.2, 6-i-C.sub.3 H.sub.7                         128 2-Allyl                                                                    129 3-Allyl                                                                    130 4-Allyl                                                                    131 2-Allyl, 6-CH.sub.3                                                        132 2-cyclo-C.sub.6 H.sub.11                                                   133 3-cyclo-C.sub.6 H.sub.11                                                   134 4-cyclo-C.sub.6 H.sub.11                                                   135 2,4-(cyclo-C.sub.6 H.sub.11), 6-CH.sub.3                                   136 2-CH.sub.3, 4-cyclo-C.sub.6 H.sub.11                                       137 2-CH.sub.2 --C.sub.6 H.sub.5                                               138 3-CH.sub.2 --C.sub.6 H.sub.5                                               139 4-CH.sub.2 --C.sub.6 H.sub.5                                               140 2-CH.sub.2 --C.sub.6 H.sub.5, 4-CH.sub.3                                   141 2-CH.sub.3, 4-CH.sub.2 --C.sub.6 H.sub.5                                   142 2-C.sub.6 H.sub.5                                                          143 3-C.sub.6 H.sub.5                                                          144 4-C.sub.6 H.sub.5                                                          145 4-(2-i-C.sub.3 H.sub.7 --C.sub.6 H.sub.4)                                  146 4-C.sub.6 H.sub.5, 2,6-(CH.sub.3).sub.2                                    147 2-Cl, 4-C.sub.6 H.sub.5                                                    148 2-Br, 4-C.sub.6 H.sub.5                                                    149 2-C.sub.6 H.sub.5, 4-Cl                                                    150 2-C.sub.6 H.sub.5, 4-Br                                                    151 2-CH.sub.2 C.sub.6 H.sub.5, 4-Cl                                           152 2-CH.sub.2 C.sub.6 H.sub.5, 4-Br                                           153 2-Cl, 4-CH.sub.2 C.sub.6 H.sub.5                                           154 2-Br, 4-CH.sub.2 C.sub.6 H.sub.5                                           155 2-cyclo-C.sub.6 H.sub.11, 4-Cl                                             156 2-cyclo-C.sub.6 H.sub.11, 4-Br                                             157 2-Cl, 4-cyclo-C.sub.6 H.sub.11                                             158 2-Br, 4-cyclo-C.sub.6 H.sub.11                                             159 2-OCH.sub.3                                                                160 3-OCH.sub.3                                                                161 4-OCH.sub.3                                                                162 2-OC.sub.2 H.sub.5                                                         163 3-O--C.sub.2 H.sub.5                                                       164 4-O--C.sub.2 H.sub.5                                                       165 2-O-n-C.sub.3 H.sub.7                                                      166 3-O-n-C.sub.3 H.sub.7                                                      167 4-O-n-C.sub.3 H.sub.7                                                      168 2-O-i-C.sub.3 H.sub.7                                                      169 3-O-i-C.sub.3 H.sub.7                                                      170 4-O-i-C.sub.3 H.sub.7                                                      171 2-O-n-C.sub.6 H.sub.13                                                     172 3-O-n-C.sub.6 H.sub.13                                                     173 4-O-n-C6H13                                                                174 2-O-n-C.sub.8 H.sub.17                                                     175 3-O-n-C.sub.8 H.sub.17                                                     176 4-O-n-C.sub.8 H.sub.17                                                     177 2-O--CH.sub.2 C.sub.6 H.sub.5                                              178 3-O--CH.sub.2 C.sub.6 H.sub.5                                              179 4-O--CH.sub.2 C.sub.6 H.sub.5                                              180 2-O--(CH.sub.2).sub.3 C.sub.6 H.sub.5                                      181 3-O--(CH.sub.2).sub.3 C.sub.6 H.sub.5                                      182 4-O--(CH.sub.2).sub.3 C.sub.6 H.sub.5                                      183 2,4-(OCH.sub.3).sub.2                                                      184 2-CF.sub.3                                                                 185 3-CF.sub.3                                                                 186 4-CF.sub.3                                                                 187 2-OCF.sub.3                                                                188 3-OCF.sub.3                                                                189 4-OCF.sub.3                                                                190 3-OCH.sub.2 CHF.sub.2                                                      191 2-NO.sub.2                                                                 192 3-NO.sub.2                                                                 193 4-NO.sub.2                                                                 194 2-CN                                                                       195 3-CN                                                                       196 4-CN                                                                       197 2-CH.sub.3, 3-Cl                                                           198 2-CH.sub.3, 4-Cl                                                           199 2-CH.sub.3, 5-Cl                                                           200 2-CH.sub.3, 6-Cl                                                           201 2-CH.sub.3, 3-F                                                            202 2-CH.sub.3, 4-F                                                            203 2-CH.sub.3, 5-F                                                            204 2-CH.sub.3, 6-F                                                            205 2-CH.sub.3, 3-Br                                                           206 2-CH.sub.3, 4-Br                                                           207 2-CH.sub.3, 5-Br                                                           208 2-CH.sub.3, 6-Br                                                           209 2-Cl, 3-CH.sub.3                                                           210 2-Cl, 4-CH.sub.3                                                           211 2-Cl, 5-CH.sub.3                                                           212 2-F, 3-CH.sub.3                                                            213 2-F, 4-CH.sub.3                                                            214 2-F, 5-CH.sub.3                                                            215 2-Br, 3-CH.sub.3                                                           216 2-Br, 4-CH.sub.3                                                           217 2-Br, 5-CH.sub.3                                                           218 3-CH.sub.3, 4-Cl                                                           219 3-CH.sub.3, 5-Cl                                                           220 3-CH.sub.3, 4-F                                                            221 3-CH.sub.3, 5-F                                                            222 3-CH.sub.3, 4-Br                                                           223 3-CH.sub.3, 5-Br                                                           224 3-F, 4-CH.sub.3                                                            225 3-Cl, 4-CH.sub.3                                                           226 3-Br, 4-CH.sub.3                                                           227 2-Cl, 4,5-(CH.sub.3).sub.2                                                 228 2-Br, 4,5-(CH.sub.3).sub.2                                                 229 2-Cl, 3,5-(CH.sub.3).sub.2                                                 230 2-Br, 3,5-(CH.sub.3).sub.2                                                 231 2,6-Cl.sub.2, 4-CH.sub.3                                                   232 2,6-F.sub.2, 4-CH.sub.3                                                    233 2,6-Br.sub.2, 4-CH.sub.3                                                   234 2,4-Br.sub.2, 6-CH.sub.3                                                   235 2,4-F.sub.2, 6-CH.sub.3                                                    236 2,4-Br.sub.2, 6-CH.sub.3                                                   237 2,6-(CH.sub.3).sub.2, 4-F                                                  238 2,6-(CH.sub.3).sub.2, 4-Cl                                                 239 2,6-(CH.sub.3).sub.2, 4-Br                                                 240 3,5-(CH.sub.3).sub.2, 4-F                                                  241 3,5-(CH.sub.3).sub.2, 4-Cl                                                 242 3,5-(CH.sub.3).sub.2, 4-Br                                                 243 2,3,6-(CH.sub.3).sub.3, 4-F                                                244 2,3,6-(CH.sub.3).sub.3, 4-Cl                                               245 2,3,6-(CH.sub.3).sub.3, 4-Br                                               246 2,4-(CH.sub.3).sub.2, 6-F                                                  247 2,4-(CH.sub.3).sub.2, 6-Cl                                                 248 2,4-(CH.sub.3).sub.2, 6-Br                                                 249 2-i-C.sub.3 H.sub.7, 4-Cl, 5-CH.sub.3                                      250 2-Cl, 4-NO2                                                                251 2-NO2, 4-Cl                                                                252 2-OCH.sub.3, 5-NO.sub.2                                                    253 2,4-Cl2, 5-NO2                                                             254 2,4-Cl2, 6-NO2                                                             255 2,6-Cl2, 4-NO2                                                             256 2,6-Br2, 4-NO2                                                             257 2,6-I2, 4-NO2                                                              258 2-CH3, 5-i-C3H7, 4-Cl                                                      259 2-CO.sub.2 CH.sub.3                                                        260 3-CO2CH3                                                                   261 4-CO2CH3                                                                   262 2-CO2(C2H5)                                                                263 3-CO.sub.2 (C.sub.2 H.sub.5)                                               264 4-CO.sub.2 (C.sub.2 H.sub.5)                                               265 2-CO.sub.2 (n-C.sub.3 H.sub.7)                                             266 3-CO.sub.2 (n-C.sub.3 H.sub.7)                                             267 4-CO.sub.2 (n-C.sub.3 H.sub.7)                                             268 2-CO.sub.2 (i-C.sub.3 H.sub.7)                                             269 3-CO.sub.2 (i-C.sub.3 H.sub.7)                                             270 4-CO.sub.2 (i-C.sub.3 H.sub.7)                                             271 2-CO.sub.2 (n-C.sub.6 H.sub.13)                                            272 3-CO.sub.2 (n-C.sub.6 H.sub.13)                                            273 4-CO.sub.2 (n-C.sub.6 H.sub.13)                                            274 2-CH.sub.2 --OCH.sub.3                                                     275 3-CH.sub.2 --OCH.sub.3                                                     276 4-CH.sub.2 --OCH.sub.3                                                     277 2-CH.sub.2 O(C.sub.2 H.sub.5)                                              278 3-CH.sub.2 O(C.sub.2 H.sub.5)                                              279 4-CH.sub.2 O(C.sub.2 H.sub.5)                                              280 2-CH.sub.2 O(n-C.sub.3 H.sub.7)                                            281 3-CH.sub.2 O(n-C.sub.3 H.sub.7)                                            282 4-CH.sub.2 O(n-C.sub.3 H.sub.7)                                            283 2-CH.sub.2 O(i-C.sub.3 H.sub.7)                                            284 3-CH.sub.2 O(i-C.sub.3 H.sub.7)                                            285 4-CH.sub.2 O(i-C.sub.3 H.sub.7)                                            286 2-CHO                                                                      287 3-CHO                                                                      288 4-CHO                                                                      289 2-CO--CH.sub.3                                                             290 3-CO--CH.sub.3                                                             291 4-CO--CH.sub.3                                                             292 2-CO--CH.sub.2 --CH.sub.3                                                  293 3-CO--CH.sub.2 --CH.sub.3                                                  294 4-CO--CH.sub.2 --CH.sub.3                                                  295 2-CO--CH.sub.2 --CH.sub.2 --CH.sub.3                                       296 3-CO--CH.sub.2 --CH.sub.2 --CH.sub.3                                       297 4-CO--CH.sub.2 --CH.sub.2 --CH.sub.3                                       298 2-CO--CH(CH.sub.3)--CH.sub.3                                               299 3-CO--CH(CH.sub.3)--CH.sub.3                                               300 4-CO--CH(CH.sub.3)--CH.sub.3                                               301 2-Me-4-CHO                                                                 302 2-Me-4-CH.sub.3 --CO                                                       303 2-Me-4-CH.sub.3 --CH.sub.2 --CO                                            304 2-Me-4-CH.sub.3 --CH.sub.2 --CH.sub.2 --CO                                 305 2-Me-4-CH.sub.3 --CH(CH.sub.3)--CO                                         306 2,5-Me.sub.2 -4-CHO                                                        307 2,5-Me.sub.2 -4-CH.sub.3 --CO                                              308 2,5-Me.sub.2 -4-CH.sub.3 --CH.sub.2 --CO                                   309 2,5-Me.sub.2 -4-CH.sub.3 --CH.sub.2 --CH.sub.2 --CO                        310 2,5-Me.sub.2 -4-CH.sub.3 --CH(CH.sub.3)--CO                                311 2-Cl-4-CHO                                                                 312 2-Cl-4-CH.sub.3 --CO                                                       313 2-Cl-4-CH.sub.3 --CH.sub.2 --CO                                            314 2-Cl-4-CH.sub.3 --CH(CH.sub.3)--CO                                         315 2,5-Cl.sub.2 -4-CHO                                                        316 2,5-Cl.sub.2 -4-CH.sub.3 --CO                                              317 2,5-Cl.sub.2 -4-CH.sub.3 --CH.sub.2 --CO                                   318 2,5-Cl.sub.2 -4-CH.sub.3 --CH.sub.2 --CH.sub.2 --CO                        319 2,5-Cl.sub.2 -4-CH.sub.3 -- --CH(CH.sub.3)--CO                             320 2-C(═NOCH.sub.3)--CH.sub.3                                             321 3-C(═NOCH.sub.3)--CH.sub.3                                             322 4-C(═NOCH.sub.3)--CH.sub.3                                             323 2-C(═NOC.sub.2 H.sub.5)--CH.sub.3                                      324 3-C(═NOC.sub.2 H.sub.5)--CH.sub.3                                      325 4-C(═NOC.sub.2 H.sub.5)--CH.sub.3                                      326 2-C(═NO-n-C.sub.3 H.sub.7)--CH.sub.3                                   327 3-C(═NO-n-C.sub.3 H.sub.7)--CH.sub.3                                   328 4-C(═NO-n-C.sub.3 H.sub.7)--CH.sub.3                                   329 2-C(═NO-i-C.sub.3 H.sub.7)--CH.sub.3                                   330 3-C(═NO-i-C.sub.3 H.sub.7)--CH.sub.3                                   331 4-C(═NO-i-C.sub.3 H.sub.7)--CH.sub.3                                   332 2-C(═NO-Allyl)-CH.sub.3                                                333 3-C(═NO-Allyl)-CH.sub.3                                                334 4-C(═NO-Allyl)-CH.sub.3                                                335 2-C(═NO-trans-Chloroallyl)-CH.sub.3                                    336 3-C(═NO-trans-Chloroallyl)-CH.sub.3                                    337 4-C(═NO-trans-Chloroallyl)-CH.sub.3                                    338 2-C(═NO-Propargyl)-CH.sub.3                                            339 3-C(═NO-Propargyl)-CH.sub.3                                            340 4-C(═NO-Propargyl)-CH.sub.3                                            341 2-C(═NO-n-C.sub.4 H.sub.9)--CH.sub.3                                   342 3-C(═NO-n-C.sub.4 H.sub.9)--CH.sub.3                                   343 4-C(═NO-n-C.sub.4 H.sub.9)--CH.sub.3                                   344 2-C(═NO--CH.sub.2 --C.sub.6 H.sub.5)--CH.sub.3                         345 3-C(═NO--CH.sub.2 --C.sub.6 H.sub.5)--CH.sub.3                         346 4-C(═NO--CH.sub.2 --C.sub.6 H.sub.5)--CH.sub.3                         347 2-CH.sub.3 -4-CH═NOCH.sub.3                                            348 2-CH.sub.3 -4-CH═NOC.sub.2 H.sub.5                                     349 2-CH.sub.3 -4-CH═NO-n-C.sub.3 H.sub.7                                  350 2-CH.sub.3 -4-CH═NO-i-C.sub.3 H.sub.7                                  351 2-CH.sub.3 -4-CH═NO-Allyl                                              352 2-CH.sub.3 -4-CH═NO-(trans-Chloroallyl)                                353 2-CH.sub.3 -4-CH═NO-Propargyl                                          354 2-CH.sub.3 -4-CH═NO-n-C.sub.4 H.sub.9                                  355 2-CH.sub.3 -4-CH═NO--CH.sub.2 --C.sub.6 H.sub.5                        356 2-CH.sub.3 -4-(CH.sub.3 --C═NOCH.sub.3)                                357 2-CH.sub.3 -4-(CH.sub.3 --C═NOC.sub.2 H.sub.5)                         358 2-CH.sub.3 -4-(CH.sub.3 --C═NO-n-C.sub.3 H.sub.7)                      359 2-CH.sub.3 -4-(CH.sub.3 --C═NO-i-C.sub.3 H.sub.7)                      360 2-CH.sub.3 -4-(CH.sub.3 --C═NO-Allyl)                                  361 2-CH3-4-(CH3--C═NO-trans-Chloroallyl)                                  362 2-CH.sub.3 -4-(CH.sub.3 --C═NO-Propargyl)                              363 2-CH.sub.3 -4-(CH.sub.3 --C═NO-n-C.sub.4 H.sub.9)                      364 2-CH.sub.3 -4-(CH.sub.3 --C═NO--CH.sub.2 --C.sub.6 H.sub.5)                   365 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C═NO--CH.sub.3)                       366 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C═NO--C.sub.2 H.sub.5)                367 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C═NO-n-C.sub.3 H.sub.7)        368 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C═NO-i-C.sub.3 H.sub.7                       369 2-CH3-4-(C2H5--C═NO-Allyl)                                      370 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C═NO-trans-Chloroallyl)                      371 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C═NO-Propargyl)                       372 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C═NO-n-C.sub.4 H.sub.9)        373 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C═NO--CH.sub.2 --C.sub.6                    H.sub.5)                                                                 374 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C═NOCH.sub.3)                      375 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C═NOC.sub.2 H.sub.5)                      376 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C═NO-n-C.sub.3                    H.sub.7)                                                                 377 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C═NO-i-C.sub.3 H.sub.7)                   378 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C═NO-Allyl)                 379 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C═NO-trans-Chloroallyl)                   380 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C═NO-Proparyl)                     381 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C═NO-n-C.sub.4                    H.sub.9)                                                                 382 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C═NO--CH.sub.2 --C.sub.6                 H.sub.5)                                                                 383 2-C.sub.6 H.sub.5                                                          384 3-C.sub.6 H.sub.5                                                          385 4-C.sub.6 H.sub.5                                                          386 2-(2'-F--C.sub.6 H.sub.4)                                                  387 2-(3'-F--C.sub.6 H.sub.4)                                                  388 2-(4'-F--C.sub.6 H.sub.4)                                                  389 3-(2'-F--C.sub.6 H.sub.4)                                                  390 3-(3'-F--C.sub.6 H.sub.4)                                                  391 3-(4'-F--C.sub.6 H.sub.4)                                                  392 4-(2'-F--C.sub.6 H.sub.4)                                                  393 4-(3'-F--C.sub.6 H.sub.4)                                                  394 4-(4'-F--C.sub.6 H.sub.4)                                                  395 2-(2'-Cl--C.sub.6 H.sub.4)                                                 396 2-(3'-Cl--C.sub.6 H.sub.4)                                                 397 2-(4'-Cl--C.sub.6 H.sub.4)                                                 398 3-(2'-Cl--C.sub.6 H.sub.4)                                                 399 3-(3'-Cl--C.sub.6 H.sub.4)                                                 400 3-(4'-Cl--C.sub.6 H.sub.4)                                                 401 4-(2'-Cl--C.sub.6 H.sub.4)                                                 402 4-(3'-Cl--C.sub.6 H.sub.4)                                                 403 4-(4'-Cl--C.sub.6 H.sub.4)                                                 405 2-(2'-CH.sub.3 --C.sub.6 H.sub.4)                                          406 2-(3'-CH.sub.3 --C.sub.6 H.sub.4)                                          407 2-(4'-CH.sub.3 --C.sub.6 H.sub.4)                                          408 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)                                          409 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)                                          410 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)                                          411 4-(2'-CH.sub.3 --C.sub.6 H.sub.4)                                          412 4-(3'-CH.sub.3 --C.sub.6 H.sub.4)                                          413 4-(4'-CH.sub.3 --C.sub.6 H.sub.4)                                          414 2-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                      415 2-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                      416 2-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                      417 3-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                      418 3-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                      419 3-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                      420 4-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                      421 4-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                      422 4-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                      423 2-(2'-(CH.sub.3 --C(═NOAllyl))-C.sub.6 H.sub.4)                        424 2-(3'-(CH.sub.3 --C(═NOAllyl))-C.sub.6 H.sub.4)                        425 2-(4'-(CH.sub.3 --C(═NOAllyl))-C.sub.6 H.sub.4)                        426 3-(2'-(CH.sub.3 --C(═NOAllyl))-C.sub.6 H.sub.4)                        427 3-(3'-(CH.sub.3 --C(═NOAllyl))-C.sub.6 H.sub.4)                        428 3-(4'-(CH.sub.3 --C(═NOAllyl))-C.sub.6 H.sub.4)                        429 4-(2'-(CH.sub.3 --C(═NOAllyl))-C.sub.6 H.sub.4)                        430 4-(3'-(CH.sub.3 --C(═NOAllyl))-C.sub.6 H.sub.4)                        431 4-(4'-(CH.sub.3 --C(═NOAllyl))-C.sub.6 H.sub.4)                        432 2-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                                 433 2-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                                 434 2-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                                 435 3-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                                 436 3-(3'-CH3O2C--C.sub.6 H.sub.4)                                             437 3-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                                 438 4-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                                 439 4-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                                 440 4-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                                 441 2-(2'-CH.sub.3 O--C.sub.6 H.sub.4)                                         442 2-(3'-CH.sub.3 O--C.sub.6 H.sub.4)                                         443 2-(4'-CH.sub.3 O--C.sub.6 H.sub.4)                                         444 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)                                         445 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)                                         446 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)                                         447 4-(2'-CH.sub.3 O--C.sub.6 H.sub.4)                                         448 4-(3'-CH.sub.3 O--C.sub.6 H.sub.4)                                         449 4-(4'-CH.sub.3 O--C.sub.6 H.sub.4)                                         450 2-(2'-O.sub.2 N--C.sub.6 H.sub.4)                                          451 2-(3'-O.sub.2 N--C.sub.6 H.sub.4)                                          452 2-(4'-O.sub.2 N--C.sub.6 H.sub.4)                                          453 3-(2'-O.sub.2 N--C.sub.6 H.sub.4)                                          454 3-(3'-O.sub.2 N--C.sub.6 H.sub.4)                                          455 3-(4'-O.sub.2 N--C.sub.6 H.sub.4)                                          456 4-(2'-O.sub.2 N--C.sub.6 H.sub.4)                                          457 4-(3'-O.sub.2 N--C.sub.6 H.sub.4)                                          458 4-(4'-O.sub.2 N--C.sub.6 H.sub.4)                                          459 2-(2'-NC--C.sub.6 H.sub.4)                                                 460 2-(3'-NC--C.sub.6 H.sub.4)                                                 461 2-(4'-NC--C.sub.6 H.sub.4)                                                 462 3-(2'-NC--C.sub.6 H.sub.4)                                                 463 3-(3'-NC--C.sub.6 H.sub.4)                                                 464 3-(4'-NC--C.sub.6 H.sub.4)                                                 465 4-(2'-NC--C.sub.6 H.sub.4)                                                 466 4-(3'-NC--C.sub.6 H.sub.4)                                                 467 4-(4'-NC--C.sub.6 H.sub.4)                                                 468 2-(2'-CF.sub.3 --C.sub.6 H.sub.4)                                          469 2-(3'-CF.sub.3 --C.sub.6 H.sub.4)                                          470 2-(4'-CF.sub.3 --C.sub.6 H.sub.4)                                          471 3-(2'-CF.sub.3 --C.sub.6 H.sub.4)                                          472 3-(3'-CF.sub.3 --C.sub.6 H.sub.4)                                          473 3-(4'-CF.sub.3 --C.sub.6 H.sub.4)                                          474 4-(2'-CF.sub.3 --C.sub.6 H.sub.4)                                          475 4-(3'-CF.sub.3 --C.sub.6 H.sub.4)                                          476 4-(4'-CF.sub.3 --C.sub.6 H.sub.4)                                          477 2-O--C.sub.6 H.sub.5                                                       475 3-O--C6H5                                                                  476 4-O--C6H5                                                                  478 2-O-(2'-F--C.sub.6 H.sub.4)                                                479 2-O-(3'-F--C.sub.6 H.sub.4)                                                480 2-O-(4'-F--C.sub.6 H.sub.4)                                                481 3-O-(2'-F--C.sub.6 H.sub.4)                                                482 3-O-(3'-F--C.sub.6 H.sub.4)                                                483 3-O-(4'-F--C.sub.6 H.sub.4)                                                484 4-O-(2'-F--C.sub.6 H.sub.4)                                                485 4-O-(3'-F--C.sub.6 H.sub.4)                                                486 4-O-(4'-F--C.sub.6 H.sub.4)                                                487 2-O-(2'-Cl--C.sub.6 H.sub.4)                                               488 2-O-(3'-Cl--C.sub.6 H.sub.4)                                               489 2-O-(4'-Cl--C.sub.6 H.sub.4)                                               490 3-O-(2'-Cl--C.sub.6 H.sub.4)                                               491 3-O-(3'-Cl--C.sub.6 H.sub.4)                                               492 3-O-(4'-Cl--C.sub.6 H.sub.4)                                               493 3-O-(4'-Cl--C.sub.6 H.sub.4)                                               494 4-O-(2'-Cl--C.sub.6 H.sub.4)                                               495 4-O-(3'-Cl--C.sub.6 H.sub.4)                                               496 4-O-(4'-Cl--C.sub.6 H.sub.4)                                               497 2-O-(2'-CH.sub.3 --C.sub.6 H.sub.4)                                        498 2-O-(3'-CH.sub.3 --C.sub.6 H.sub.4)                                        499 2-O-(4'-CH.sub.3 --C.sub.6 H.sub.4)                                        500 3-O-(2'-CH.sub.3 --C.sub.6 H.sub.4)                                        501 3-O-(3'-CH.sub.3 --C.sub.6 H.sub.4)                                        502 3-O-(4'-CH.sub.3 --C.sub.6 H.sub.4)                                        503 4-O-(2'-CH.sub.3 --C.sub.6 H.sub.4)                                        504 4-O-(3'-CH.sub.3 --C.sub.6 H.sub.4)                                        505 4-O-(4'-CH.sub.3 --C.sub.6 H.sub.4)                                        506 2-O-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                    507 2-O-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                    508 2-O-(4'-CH3--CO--C6H4)                                                     509 3-O-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                    510 3-O-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                    511 3-O-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                    512 4-O-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                    513 4-O-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                    514 4-O-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                    515 2-O-(2'-(CH.sub.3 --C(═NOAllyl))-C.sub.6 H.sub.4)                      516 2-O-(3'-(CH.sub.3 --C(═NOAllyl))-C.sub.6 H.sub.4)                      517 2-O-(4'-(CH.sub.3 --C(═NOAllyl))-C.sub.6 H.sub.4)                      518 3-O-(2'-(CH.sub.3 --C(═NOAllyl))-C.sub.6 H.sub.4)                      519 3-O-(3'-(CH.sub.3 --C(═NOAllyl))-C.sub.6 H.sub.4)                      520 3-O-(4'-(CH.sub.3 --C(═NOAllyl))-C.sub.6 H.sub.4)                      521 4-O-(2'-(CH.sub.3 --C(═NOAllyl))-C.sub.6 H.sub.4)                      522 4-O-(3'-(CH.sub.3 --C(═NOAllyl))-C.sub.6 H.sub.4)                      523 4-O-(4'-(CH.sub.3 --C(═NOAllyl))-C.sub.6 H.sub.4)                      524 2-O-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                               525 2-O-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                               526 2-O-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                               527 3-O-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                               528 3-O-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                               529 3-O-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                               530 4-O-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                               531 4-O-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                               532 4-O-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                               533 2-O-(2'-CH.sub.3 O--C.sub.6 H.sub.4)                                       534 2-O-(3'-CH.sub.3 O--C.sub.6 H.sub.4)                                       535 2-O-(4'-CH.sub.3 O--C.sub.6 H.sub.4)                                       536 3-O-(2'-CH.sub.3 O--C.sub.6 H.sub.4)                                       537 3-O-(3'-CH.sub.3 O--C.sub.6 H.sub.4)                                       538 3-O-(4'-CH.sub.3 O--C.sub.6 H.sub.4)                                       539 4-O-(2'-CH.sub.3 O--C.sub.6 H.sub.4)                                       540 4-O-(3'-CH.sub.3 O--C.sub.6 H.sub.4)                                       541 4-O-(4'-CH.sub.3 O--C.sub.6 H.sub.4)                                       542 2-O-(2'-O.sub.2 N--C.sub.6 H.sub.4)                                        543 2-O-(3'-O.sub.2 N--C.sub.6 H.sub.4)                                        544 2-O-(4'-O.sub.2 N--C.sub.6 H.sub.4)                                        545 3-O-(2'-O2N--C.sub.6 H.sub.4)                                              546 3-O-(3'-O.sub.2 N--C.sub.6 H.sub.4)                                        547 3-O-(4'-O.sub.2 N--C.sub.6 H.sub.4)                                        548 4-O-(2'-O.sub.2 N--C.sub.6 H.sub.4)                                        549 4-O-(3'-O.sub.2 N--C.sub.6 H.sub.4)                                        550 4-O-(4'-O.sub.2 N--C.sub.6 H.sub.4)                                        551 2-O-(2'-NC--C.sub.6 H.sub.4)                                               552 2-O-(3'-NC--C.sub.6 H.sub.4)                                               553 2-O-(4'-NC--C.sub.6 H.sub.4)                                               554 3-O-(2'-NC--C.sub.6 H.sub.4)                                               555 3-O-(3'-NC--C.sub.6 H.sub.4)                                               556 3-O-(4'-NC--C.sub.6 H.sub.4)                                               557 4-O-(2'-NC--C.sub.6 H.sub.4)                                               558 4-O-(3'-NC--C.sub.6 H.sub.4)                                               559 4-O-(4'-NC--C.sub.6 H.sub.4)                                               560 2-O-(2'-CF.sub.3 --C.sub.6 H.sub.4)                                        561 2-O-(3'-CF.sub.3 --C.sub.6 H.sub.4)                                        562 2-O-(4'-CF.sub.3 --C.sub.6 H.sub.4)                                        563 3-O-(2'-CF.sub.3 --C.sub.6 H.sub.4)                                        564 3-O-(3'-CF.sub.3 --C.sub.6 H.sub.4)                                        565 3-O-(4'-CF.sub.3 --C.sub.6 H.sub.4)                                        566 4-O-(2'-CF.sub.3 --C.sub.6 H.sub.4)                                        567 4-O-(3'-CF.sub.3 --C.sub.6 H.sub.4)                                        568 4-O-(4'-CF.sub.3 --C.sub.6 H.sub.4)                                        569 2-Pyridinyl-2'                                                             570 2-Pyridinyl-3'                                                             571 2-Pyridinyl-4'                                                             572 3-Pyridinyl-2'                                                             573 3-Pyridinyl-3'                                                             574 3-Pyridinyl-4'                                                             575 4-Pyridinyl-2'                                                             576 4-Pyridinyl-3'                                                             577 4-Pyridinyl-4'                                                             578 2-Pyrimidinyl-2'                                                           579 2-Pyrimidinyl-3'                                                           580 2-Pyrimidinyl-4'                                                           581 3-Pyrimidinyl-2'                                                           582 3-Pyrimidinyl-3'                                                           583 3-Pyrimidinyl-4'                                                           584 4-Pyrimidinyl-2'                                                           585 4-Pyrimidinyl-3'                                                           586 4-Pyrimidinyl-4'                                                           587 2-Pyrazolyl-1'                                                             588 2-Pyrazolyl-3'                                                             589 2-Pyrazolyl-4'                                                             590 3-Pyrazolyl-1'                                                             591 3-Pyrazolyl-3'                                                             592 3-Pyrazolyl-4'                                                             593 4-Pyrazolyl-1'                                                             594 4-Pyrazolyl-3'                                                             595 4-Pyrazolyl-4'                                                             596 2-Isoxazolyl-3'                                                            597 2-Isoxazolyl-4'                                                            598 2-Isoxazolyl-5'                                                            599 3-Isoxazolyl-3'                                                            600 3-Isoxazolyl-4'                                                            601 3-Isoxazolyl-5'                                                            602 4-Isoxazolyl-3'                                                            603 4-Isoxazolyl-4'                                                            604 4-Isoxazolyl-5'                                                            605 2-Isothiazolyl-3'                                                          606 2-Isothiazolyl-4'                                                          607 2-Isothiazolyl-5'                                                          608 3-Isothiazolyl-3'                                                          609 3-Isothiazolyl-4'                                                          610 3-Isothiazolyl-5'                                                          611 4-Isothiazolyl-3'                                                          612 4-Isothiazolyl-4'                                                          613 4-Isothiazolyl-5'                                                          614 2-Imidazolyl-1'                                                            615 2-Imidazolyl-2'                                                            616 2-Imidazolyl-4'                                                            617 3-Imidazolyl-1'                                                            618 3-Imidazolyl-2'                                                            619 3-Imidazolyl-4'                                                            620 4-Imidazolyl-1'                                                            621 4-Imidazolyl-2'                                                            622 4-Imidazolyl-4'                                                            623 2-Oxazolyl-2'                                                              624 2-Oxazolyl-4'                                                              625 2-Oxazolyl-5'                                                              626 3-Oxazolyl-2'                                                              627 3-Oxazolyl-4'                                                              628 3-Oxazolyl-5'                                                              629 4-Oxazolyl-2'                                                              630 4-Oxazolyl-4'                                                              631 4-Oxazolyl-5'                                                              632 2-Thiazolyl-2'                                                             633 2-Thiazolyl-4'                                                             634 2-Thiazolyl-5'                                                             635 3-Thiazolyl-2'                                                             636 3-Thiazolyl-4'                                                             637 3-Thiazolyl-5'                                                             638 4-Thiazolyl-2                                                              639 4-Thiazolyl-4'                                                             640 4-Thiazolyl-5'                                                             641 2-CH.sub.3 -4-(CH.sub.3 --C═N--O--CH.sub.2 --CH.sub.2 --OCH.sub.             3)                                                                       642 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C═N--O--CH.sub.2 --CH.sub.2                 --OCH.sub.3)                                                             643 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C═N--O--CH.sub.2 --CH.sub.2              --OCH.sub.3)                                                             644 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C═N--OCH.sub.3)                     645 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C═N--OC.sub.2 H.sub.5)                     646 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C═N--O-n-C.sub.3                   H.sub.7)                                                                 647 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C═N--O-i-C.sub.3 H.sub.7)                  648 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C═N--O-Allyl)                       649 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C═N--O-trans-Chloroall             yl)                                                                      650 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C═N--O-Propargyl)                   651 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C═N--O-n-C.sub.4 H.sub.9)                  652 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C═N--O--CH.sub.2                   --C.sub.6 H.sub.5)                                                       653 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C═N--OCH.sub.3)                     654 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C═N--OC.sub.2 H.sub.5)                     655 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C═N--O-n-C.sub.3                   H.sub.7)                                                                 656 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C═N--O-i-C.sub.3 H.sub.7)                  657 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C═N--O-Allyl)                       658 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C═N--O-trans-Chloroall             yl)                                                                      659 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C═N--O-Propargyl)                   660 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C═N--O-n-C.sub.4 H.sub.9)                  661 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C═N--O--CH.sub.2                   --C.sub.6 H.sub.5)                                                       662 2-O-n-C.sub.4 H.sub.9                                                      663 2-O-i-C.sub.4 H.sub.9                                                      664 2-O-s-C.sub.4 H.sub.9                                                      665 2-O-t-C.sub.4 H.sub.9                                                      666 2-Neopentyloxy                                                             667 3-O-n-C.sub.4 H.sub.9                                                      668 3-O-i-C.sub.4 H.sub.9                                                      669 3-O-s-C.sub.4 H.sub.9                                                      670 3-O-t-C.sub.4 H.sub.9                                                      671 3-Neopentyloxy                                                             672 4-O-n-C.sub.4 H.sub.9                                                      673 4-O-i-C.sub.4 H.sub.9                                                      674 4-O-s-C.sub.4 H.sub.9                                                      675 4-O-t-C.sub.4 H.sub.9                                                      676 4-Neopentyloxy                                                             677 3-CH.sub.3 -4-OCH.sub.3                                                    678 3-CH.sub.3 -4-OC.sub.2 H.sub.5                                             679 3-CH.sub.3 -4-O-n-C.sub.3 H.sub.7                                          680 3-CH.sub.3 -4-O-n-C.sub.4 H.sub.9                                          681 3-CH.sub.3 -4-O-i-C.sub.4 H.sub.9                                          682 3-CH.sub.3 -4-O-s-C.sub.4 H.sub.9                                          683 3-CH.sub.3 -4-O-t-C.sub.4 H.sub.9                                          684 3-CH.sub.3 -4-Neopentyloxy                                                 685 2-CH.sub.3 -3-oCH.sub.3                                                    686 2-CH.sub.3 -4-OCH.sub.3                                                    687 2-CH.sub.3 -5-OCH.sub.3                                                    688 2-CH.sub.3 -6-OCH.sub.3                                                    689 3-CH.sub.3 -4-OCH.sub.3                                                    690 3-CH.sub.3 -5-OCH.sub.3                                                    691 3-CH.sub.3 -6-OCH.sub.3                                                    692 4-CH.sub.3 -5-O--CH.sub.3                                                  693 4-CH.sub.3 -6-O--CH.sub.3                                                  694 4-CH.sub.3 -6-OCH.sub.3                                                    695 2-CH.sub.3 -3-O-i-C.sub.3 H.sub.7                                          696 2-CH.sub.3 -4-O-i-C.sub.3 H.sub.7                                          697 2-CH.sub.3 -5-O-i-C.sub.3 H.sub.7                                          698 2-CH.sub.3 -6-O-i-C.sub.3 H.sub.7                                          699 3-CH.sub.3 -4-O-i-C.sub.3 H.sub.7                                          700 3-CH.sub.3 -5-O-i-C.sub.3 H.sub.7                                          701 3-CH.sub.3 -6-O-i-C.sub.3 H.sub.7                                          702 4-CH.sub.3 -5-O-i-C.sub.3 H.sub.7                                          703 4-CH.sub.3 -6-O-i-C.sub.3 H.sub.7                                          704 5-CH.sub.3 -6-O-i-C.sub.3 H.sub.7                                          705 2-Cl-3-OCH.sub.3                                                           706 2-Cl-4-OCH.sub.3                                                           707 2-Cl-5-OCH.sub.3                                                           708 2-Cl-6-OCH.sub.3                                                           709 3-Cl-4-OCH.sub.3                                                           710 3-Cl-5-OCH.sub.3                                                           711 3-Cl-6-OCH.sub.3                                                           712 4-Cl-5-OCH.sub.3                                                           713 4-Cl-6-OCH.sub.3                                                           714 5-Cl-6-OCH.sub.3                                                         ______________________________________                                    

                  TABLE 16                                                         ______________________________________                                         1  STR219##                                                                       -      I: R.sup.1 = CH.sub.3, Z = CH.sub.3                                    II: R.sup.1 = CH.sub.2 --CH.sub.3, Z = CH.sub.3                                III: R.sup.1 = CH.sub.3, Z = C.sub.2 H.sub.5                                   IV: R.sup.1 = CH.sub.2 --CH.sub.3, Z = C.sub.2 H.sub.5                         V: R.sup.1 = CH.sub.3, Z = NHCH.sub.3                                          VI: R.sup.1 = CH.sub.2 --CH.sub.3, Z = NHCH.sub.3                            No.       B                                                                    ______________________________________                                          1        Pyrrolyl-3                                                              2 N-CH.sub.3 -Pyrrolyl-3                                                       3 N-C.sub.6 H.sub.5 -Pyrrolyl-3                                                4 N-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrrolyl-3                                 5 N-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrrolyl-3                                 6 N-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrrolyl-3                                 7 N-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrrolyl-3                                8 N-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrrolyl-3                                9 N-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrrolyl-3                                10 N-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrrolyl-3                                11 N-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrrolyl-3                                12 N-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrrolyl-3                                13 N-(4'-CN-C.sub.6 H.sub.4)-Pyrrolyl-3                                        14 N-(3'-CN-C.sub.6 H.sub.4)-Pyrrolyl-3                                        15 N-(2'-CN-C.sub.6 H.sub.4)-Pyrrolyl-3                                        16 N-(4'-Cl--C.sub.6 H.sub.4)-Pyrrolyl-3                                       17 N-(3'-Cl--C.sub.6 H.sub.4)-Pyrrolyl-3                                       18 N-(2'-Cl--C.sub.6 H.sub.4)-Pyrrolyl-3                                       19 Pyrrolyl-2                                                                  20 N-CH.sub.3 -Pyrrolyl-2                                                      21 N-C.sub.6 H.sub.5 -Pyrrolyl-2                                               22 N-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrrolyl-2                                23 N-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrrolyl-2                                24 N-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrrolyl-2                                25 N-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrrolyl-2                               26 N-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrrolyl-2                               27 N-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrrolyl-2                               28 N-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrrolyl-2                                29 N-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrrolyl-2                                30 N-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrrolyl-2                                31 N-(4'-CN--C.sub.6 H.sub.4)-Pyrrolyl-2                                       32 N-(3'-CN--C.sub.6 H.sub.4)-Pyrrolyl-2                                       33 N-(2'-CN--C.sub.6 H.sub.4)-Pyrrolyl-2                                       34 N-(4'-Cl--C.sub.6 H.sub.4)-Pyrrolyl-2                                       35 N-(3'-Cl--C.sub.6 H.sub.4)-Pyrrolyl-2                                       36 N-(2'-Cl--C.sub.6 H.sub.4)-Pyrrolyl-2                                       37 Furyl-2                                                                     38 5-CH.sub.3 -Furyl-2                                                         39 5-C.sub.6 H.sub.5 -Furyl-2                                                  40 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Furyl-2                                   41 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Furyl-2                                   42 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Furyl-2                                   43 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Furyl-2                                  44 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Furyl-2                                  45 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Furyl-2                                  46 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Furyl-2                                   47 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Furyl-2                                   48 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Furyl-2                                   49 5-(4'-CN--C.sub.6 H.sub.4)-Furyl-2                                          50 5-(3'-CN--C.sub.6 H.sub.4)-Furyl-2                                          51 5-(2'-CN--C.sub.6 H.sub.4)-Furyl-2                                          52 5-(4'-Cl--C.sub.6 H.sub.4)-Furyl-2                                          53 5-(3'-Cl--C.sub.6 H.sub.4)-Furyl-2                                          54 5-(2'-Cl--C.sub.6 H.sub.4)-Furyl-2                                          55 4-CH.sub.3 -Furyl-2                                                         56 4-C.sub.6 H.sub.5 -Furyl-2                                                  57 4-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Furyl-2                                   58 4-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Furyl-2                                   59 4-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Furyl-2                                   60 4-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Furyl-2                                  61 4-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Furyl-2                                  62 4-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Furyl-2                                  63 4-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Furyl-2                                   64 4-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Furyl-2                                   65 4-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Furyl-2                                   66 4-(4'-CN--C.sub.6 H.sub.4)-Furyl-2                                          67 4-(3'-CN--C.sub.6 H.sub.4)-Furyl-2                                          68 4-(2'-CN--C.sub.6 H.sub.4)-Furyl-2                                          69 4-(4'-Cl--C.sub.6 H.sub.4)-Furyl-2                                          70 4-(3'-Cl--C.sub.6 H.sub.4)-Furyl-2                                          71 4-(2'-Cl--C.sub.6 H.sub.4)-Furyl-2                                          72 Thienyl-2                                                                   73 5-CH.sub.3 -Thienyl-2                                                       74 5-C.sub.6 H.sub.5 -Thienyl-2                                                75 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-2                                 76 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-2                                 77 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-2                                 78 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-2                                79 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-2                                80 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-2                                81 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-2                                 82 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-2                                 83 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-2                                 84 5-(4'-CN--C.sub.6 H.sub.4)-Thienyl-2                                        85 5-(3'-CN--C.sub.6 H.sub.4)-Thienyl-2                                        86 5-(2'-CN--C.sub.6 H.sub.4)-Thienyl-2                                        87 5-(4'-Cl--C.sub.6 H.sub.4)-Thienyl-2                                        88 5-(3'-Cl--C.sub.6 H.sub.4)-Thienyl-2                                        89 5-(2'-Cl--C.sub.6 H.sub.4)-Thienyl-2                                        90 4-CH.sub.3 -Thienyl-2                                                       91 4-C.sub.6 H.sub.5 -Thienyl-2                                                92 4-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-2                                 93 4-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-2                                 94 4-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-2                                 95 4-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-2                                96 4-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-2                                97 4-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-2                                98 4-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-2                                 99 4-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-2                                100 4-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-2                                101 4-(4'-CN--C.sub.6 H.sub.4)-Thienyl-2                                       102 4-(3'-CN--C.sub.6 H.sub.4)-Thienyl-2                                       103 4-(2'-CN--C.sub.6 H.sub.4)-Thienyl-2                                       104 4-(4'-Cl--C.sub.6 H.sub.4)-Thienyl-2                                       105 4-(3'-Cl--C.sub.6 H.sub.4)-Thienyl-2                                       106 4-(2'-Cl--C.sub.6 H.sub.4)-Thienyl-2                                       107 Thienyl-3                                                                  108 5-CH.sub.3 -Thienyl-3                                                      109 5-C.sub.6 H.sub.5 -Thienyl-3                                               110 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-3                                111 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-3                                112 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-3                                113 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-3                               114 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-3                               115 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-3                               116 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-3                                117 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-3                                118 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-3                                119 5-(4'-CN--C.sub.6 H.sub.4)-Thienyl-3                                       120 5-(3'-CN--C.sub.6 H.sub.4)-Thienyl-3                                       121 5-(2'-CN--C.sub.6 H.sub.4)-Thienyl-3                                       122 5-(4'-Cl--C.sub.6 H.sub.4)-Thienyl-3                                       123 5-(3'-Cl--C.sub.6 H.sub.4)-Thienyl-3                                       124 5-(2'-Cl--C.sub.6 H.sub.4)-Thienyl-3                                       125 Pyrazolyl-4                                                                126 N-CH.sub.3 -Pyrazolyl-4                                                    127 N-C.sub.6 H.sub.5 -Pyrazolyl-4                                             128 N-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrazolyl-4                              129 N-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrazolyl-4                              130 N-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrazolyl-4                              131 N-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrazolyl-4                             132 N-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrazolyl-4                             133 N-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrazolyl-4                             134 N-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrazolyl-4                              135 N-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrazolyl-4                              136 N-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrazolyl-4                              137 N-(4'-CN--C.sub.6 H.sub.4)-Pyrazolyl-4                                     138 N-(3'-CN--C.sub.6 H.sub.4)-Pyrazolyl-4                                     139 N-(2'-CN--C6H.sub.4)-Pyrazolyl-4                                           140 N-(4'-Cl--C.sub.6 H.sub.4)-Pyrazolyl-4                                     141 N-(3'-Cl--C.sub.6 H.sub.4)-Pyrazolyl-4                                     142 N-(2'-Cl--C.sub.6 H.sub.4)-Pyrazolyl-4                                     143 3-CH.sub.3 --N-Methylpyrazolyl-4                                           144 3-C.sub.6 H.sub.5 --N-Methylpyrazolyl-4                                    145 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)--N-Methylpyrazolyl-4                     146 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)--N-Methylpyrazolyl-4                     147 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)--N-Methylpyrazolyl-4                     148 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)--N-Methylpyrazolyl-4                    149 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)--N-Methylpyrazolyl-4                    150 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)--N-Methylpyrazolyl-4                    151 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)--N-Methylpyrazolyl-4                     152 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)--N-Methylpyrazolyl-4                     153 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)--N-Methylpyrazolyl-4                     154 3-(4'-CN--C.sub.6 H.sub.4)--N-Methylpyrazolyl-4                            155 3-(3'-CN--C.sub.6 H.sub.4)--N-Methylpyrazolyl-4                            156 3-(2'-CN--C.sub.6 H.sub.4)--N-Methylpyrazolyl-4                            157 3-(4'-Cl--C.sub.6 H.sub.4)--N-Methylpyrazolyl-4                            158 3-(3'-Cl--C.sub.6 H.sub.4)--N-Methylpyrazolyl-4                            159 3-(2'-Cl--C.sub.6 H.sub.4)--N-Methylpyrazolyl-4                            160 Isoxazolyl-5                                                               161 3-CH.sub.3 -Isoxazolyl-5                                                   162 3-C.sub.6 H.sub.5 -Isoxazolyl-5                                            163 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Isoxazolyl-5                             164 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Isoxazolyl-5                             165 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Isoxazolyl-5                             166 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Isoxazolyl-5                            167 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Isoxazolyl-5                            168 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Isoxazolyl-5                            169 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Isoxazolyl-5                             170 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Isoxazolyl-5                             171 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Isoxazolyl-5                             172 3-(4'-CN--C.sub.6 H.sub.4)-Isoxazolyl-5                                    173 3-(3'-CN--C.sub.6 H.sub.4)-Isoxazolyl-5                                    174 3-(2'-CN--C.sub.6 H.sub.4)-Isoxazolyl-5                                    175 3-(4'-Cl--C.sub.6 H.sub.4)-Isoxazolyl-5                                    176 3-(3'-Cl--C.sub.6 H.sub.4)-Isoxazolyl-5                                    177 3-(2'-Cl--C.sub.6 H.sub.4)-Isoxazolyl-5                                    178 4-Chloroisoxazolyl-5                                                       179 3-CH.sub.3 -4-Chloroisoxazolyl-5                                           180 3-C.sub.6 H.sub.5 -4-Chloroisoxazolyl-5                                    181 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                     182 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                     183 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                     184 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                    185 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                    186 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                    187 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                     188 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                     189 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                     190 3-(4'-CN--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                            191 3-(3'-CN--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                            192 3-(2'-CN--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                            193 3-(4'-Cl--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                            194 3-(3'-Cl--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                            195 3-(2'-Cl--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                            196 Isoxazolyl-3                                                               197 5-CH.sub.3 -Isoxazolyl-3                                                   198 5-C.sub.6 H.sub.5 -Isoxazolyl-3                                            199 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Isoxazolyl-3                             200 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Isoxazolyl-3                             201 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Isoxazolyl-3                             202 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Isoxazolyl-3                            203 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Isoxazolyl-3                            204 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Isoxazolyl-3                            205 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Isoxazolyl-3                             206 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Isoxazolyl-3                             207 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Isoxazolyl-3                             208 5-(4'-CN--C.sub.6 H.sub.4)-Isoxazolyl-3                                    209 5-(3'-CN--C.sub.6 H.sub.4)-Isoxazolyl-3                                    210 5-(2'-CN--C.sub.6 H.sub.4)-Isoxazolyl-3                                    211 5-(4'-Cl--C.sub.6 H.sub.4)-Isoxazolyl-3                                    212 5-(3'-Cl--C.sub.6 H.sub.4)-Isoxazolyl-3                                    213 5-(2'-Cl--C.sub.6 H.sub.4)-Isoxazolyl-3                                    214 Isothiazolyl-5                                                             215 3-CH.sub.3 -Isothiazolyl-5                                                 216 3-C.sub.6 H.sub.5 -Isothiazolyl-5                                          217 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Isothiazolyl-5                           218 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Isothiazolyl-5                           219 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Isothiazolyl-5                           220 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Isothiazolyl-5                          221 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Isothiazolyl-5                          222 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Isothiazolyl-5                          223 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Isothiazolyl-5                           224 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Isothiazolyl-5                           225 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Isothiazolyl-5                           226 3-(4'-CN--C.sub.6 H.sub.4)-Isothiazolyl-5                                  227 3-(3'-CN--C.sub.6 H.sub.4)-Isothiazolyl-5                                  228 3-(2'-CN--C.sub.6 H.sub.4)-Isothiazolyl-5                                  229 3-(4'-Cl--C.sub.6 H.sub.4)-Isothiazolyl-5                                  230 3-(3'-Cl--C.sub.6 H.sub.4)-Isothiazolyl-5                                  231 3-(2'-Cl--C.sub.6 H.sub.4)-Isothiazolyl-5                                  232 Oxazolyl-4                                                                 233 2-CH.sub.3 -Oxazolyl-4                                                     234 2-C.sub.6 H.sub.5 -Oxazolyl-4                                              235 2-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Oxazolyl-4                               236 2-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Oxazolyl-4                               237 2-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Oxazolyl-4                               238 2-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Oxazolyl-4                              239 2-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Oxazolyl-4                              240 2-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Oxazolyl-4                              241 2-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Oxazolyl-4                               242 2-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Oxazolyl-4                               243 2-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Oxazolyl-4                               244 2-(4'-CN--C.sub.6 H.sub.4)-Oxazolyl-4                                      245 2-(3'-CN--C.sub.6 H.sub.4)-Oxazolyl-4                                      246 2-(2'-CN--C.sub.6 H.sub.4)-Oxazolyl-4                                      247 2-(4'-Cl--C.sub.6 H.sub.4)-Oxazolyl-4                                      248 2-(3'-Cl--C.sub.6 H.sub.4)-Oxazolyl-4                                      249 2-(2'-Cl--C.sub.6 H.sub.4)-Oxazolyl-4                                      250 Thiazolyl-4                                                                251 2-CH.sub.3 -Thiazolyl-4                                                    252 2-C.sub.6 H.sub.5 -Thiazolyl-4                                             253 2-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Thiazolyl-4                              254 2-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Thiazolyl-4                              255 2-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Thiazolyl-4                              256 2-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Thiazolyl-4                             267 2-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Thiazolyl-4                             258 2-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Thiazolyl-4                             259 2-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Thiazolyl-4                              260 2-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Thiazolyl-4                              261 2-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Thiazolyl-4                              262 2-(4'-CN--C.sub.6 H.sub.4)-Thiazolyl-4                                     263 2-(3'-CN--C.sub.6 H.sub.4)-Thiazolyl-4                                     264 2-(2'-CN--C.sub.6 H.sub.4)-Thiazolyl-4                                     265 2-(4'-Cl--C.sub.6 H.sub.4)-Thiazolyl-4                                     266 2-(3'-Cl--C.sub.6 H.sub.4)-Thiazolyl-4                                     267 2-(2'-Cl--C.sub.6 H.sub.4)-Thiazolyl-4                                     268 N-CH.sub.3 -1,2,4-Triazolyl-5                                              269 3-CH.sub.3 --N--CH.sub.3 -1,2,4-Triazolyl-5                                270 3-C.sub.6 H.sub.5 --N--CH.sub.3 -1,2,4-Triazolyl-5                         271 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5                   272 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triaz               olyl-5                                                                 273 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5                   274 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Tria               zolyl-5                                                                275 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5                  276 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Tria               zolyl-5                                                                277 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5                   278 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triaz               olyl-5                                                                 279 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5                   280 3-(4'-CN--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5        281 3-(3'-CN--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5                 282 3-(2'-CN--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5                 283 3-(4'-Cl--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5                 284 3-(3'-Cl--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5                 285 3-(2'-Cl--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5                 286 1,3,4-Oxadiazolyl-2                                                        287 5-CH.sub.3 -1,3,4-Oxadiazolyl-2                                            288 5-C.sub.6 H.sub.5 -1,3,4-Oxadiazolyl-2                                     289 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                      290 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                      291 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                      292 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                     293 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                     294 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                     295 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                      296 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                      297 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                      298 5-(4'-CN--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                             299 5-(3'-CN--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                             300 5-(2'-CN--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                             301 5-(4'-Cl--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                             302 5-(3'-Cl--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                             303 5-(2'-Cl--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                             304 1,2,4-Oxadiazolyl-3                                                        305 5-CH.sub.3 -1,2,4-Oxadiazolyl-3                                            306 5-C.sub.6 H.sub.5 -1,2,4-Oxadiazolyl-3                                     307 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                      308 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                      309 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                      310 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                     311 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                     312 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                     313 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                      314 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                      315 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                      316 5-(4'-CN--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                             317 5-(3'-CN--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                             318 5-(2'-CN--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                             319 5-(4'-Cl--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                             320 5-(3'-Cl--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                             321 5-(2'-Cl--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                             322 1,2,4-Oxadiazolyl-5                                                        323 3-CH.sub.3 -1,2,4-Oxadiazolyl-5                                            324 3-C.sub.6 H.sub.5 -1,2,4-Oxadiazolyl-5                                     325 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                      326 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                      327 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                      328 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                     329 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                     330 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                     331 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                      332 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                      333 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                      334 3-(4'-CN--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                             335 3-(3'-CN--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                             336 3-(2'-CN--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                             337 3-(4'-Cl--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                             338 3-(3'-Cl--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                             339 3-(2'-Cl--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                             340 1,2,4-Thiadiazolyl-3                                                       341 5-CH.sub.3 -1,2,4-Thiadiazolyl-3                                           342 5-C.sub.6 H.sub.5 -1,2,4-Thiadiazolyl-3                                    343 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                     344 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                     345 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                     346 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                    347 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                    348 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                    349 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                     350 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                     351 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                     352 5-(4'-CN--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                            353 5-(3'-CN--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                            354 5-(2'-CN--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                            355 5-(4'-Cl--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                            356 5-(3'-Cl--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                            357 5-(2'-Cl--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                            358 1,3,4-Thiadiazolyl-2                                                       359 5-CH.sub.3 -1,3,4-Thiadiazolyl-2                                           360 5-C.sub.6 H.sub.5 -1,3,4-Thiadiazolyl-2                                    361 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                     362 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                     363 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                     364 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                    365 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                    366 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                    367 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                     368 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                     369 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                     370 5-(4'-CN--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                            371 5-(3'-CN--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                            372 5-(2'-CN--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                            373 5-(4'-Cl--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                            374 5-(3'-Cl--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                            375 5-(2'-Cl--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                            376 Pyridinyl-2                                                                377 Pyridinyl-4                                                                378 Pyridazinyl-3                                                              379 Pyridazinyl-4                                                              380 Pyridazinyl-2                                                              381 Pyrimidinyl-4                                                              382 Pyrimidinyl-5                                                              383 Pyrimidinyl-2                                                              384 Pyridinyl-3                                                                385 1-Naphthyl                                                                 386 2-Naphthyl                                                               ______________________________________                                    

                  TABLE 17                                                         ______________________________________                                         1  STR220##                                                                       -      I: R.sup.1 = CH.sub.3, Z = CH.sub.3                                    II: R.sup.1 = CH.sub.2 --CH.sub.3, Z = CH.sub.3                                III: R.sup.1 = CH.sub.3, Z = C.sub.2 H.sub.5                                   IV: R.sup.1 = CH.sub.2 --CH.sub.3, Z = C.sub.2 H.sub.5                         V: R.sup.1 = CH.sub.3, Z = NHCH.sub.3                                          VI: R.sup.1 = CH.sub.2 --CH.sub.3, Z = NHCH.sub.3                            No.     X.sub.m                                                                ______________________________________                                          1      H                                                                         2 2-F                                                                          3 3-F                                                                          4 4-F                                                                          5 2,4-F.sub.2                                                                  6 2,4,6-F.sub.3                                                                7 2,3,4,5,6-F.sub.5                                                            8 2,3-F.sub.2                                                                  9 2-Cl                                                                         10 3-Cl                                                                        11 4-Cl                                                                        12 2,3-Cl.sub.2                                                                13 2,4-Cl.sub.2                                                                14 2,5-Cl.sub.2                                                                15 2,6-Cl.sub.2                                                                16 3,4-Cl.sub.2                                                                17 3,5-Cl.sub.2                                                                18 2,3,4-Cl.sub.3                                                              19 2,3,5-Cl.sub.3                                                              20 2,3,6-Cl.sub.3                                                              21 2,4,5-Cl.sub.3                                                              22 2,4,6-Cl.sub.3                                                              23 3,4,5-Cl.sub.3                                                              24 2,3,4,6-Cl.sub.4                                                            25 2,3,5,6-Cl.sub.4                                                            26 2,3,4,5,6-Cl.sub.5                                                          27 2-Br                                                                        28 3-Br                                                                        29 4-Br                                                                        30 2,4-Br.sub.2                                                                31 2,5-Br.sub.2                                                                32 2,6-Br.sub.2                                                                33 2,4,6-Br.sub.3                                                              34 2,3,4,5,6-Br.sub.5                                                          35 2-I                                                                         36 3-I                                                                         37 4-I                                                                         38 2,4-I.sub.2                                                                 39 2-Cl, 3-F                                                                   40 2-Cl, 4-F                                                                   41 2-Cl, 5-F                                                                   42 2-Cl, 6-F                                                                   43 2-Cl, 3-Br                                                                  44 2-Cl, 4-Br                                                                  45 2-Cl, 5-Br                                                                  46 2-Cl, 6-Br                                                                  47 2-Br, 3-Cl                                                                  48 2-Br, 4-Cl                                                                  49 2-Br, 5-Cl                                                                  50 2-Br, 3-F                                                                   51 2-Br, 4-F                                                                   52 2-Br, 5-F                                                                   53 2-Br, 6-F                                                                   54 2-F, 3-Cl                                                                   55 2-F, 4-Cl                                                                   56 2-F, 5-Cl                                                                   57 3-Cl, 4-F                                                                   58 3-Cl, 5-F                                                                   59 3-Cl, 4-Br                                                                  60 3-Cl, 5-Br                                                                  61 3-F, 4-Cl                                                                   62 3-F, 4-Br                                                                   63 3-Br, 4-Cl                                                                  64 3-Br, 4-F                                                                   65 2,6-Cl.sub.2, 4-Br                                                          66 2-CH.sub.3                                                                  67 3-CH.sub.3                                                                  68 4-CH.sub.3                                                                  69 2,3-(CH.sub.3).sub.2                                                        70 2,4-(CH.sub.3).sub.2                                                        71 2,5-(CH.sub.3).sub.2                                                        72 2,6-(CH.sub.3).sub.2                                                        73 3,4-(CH.sub.3).sub.2                                                        74 3,5-(CH.sub.3).sub.2                                                        75 2,3,5-(CH.sub.3).sub.3                                                      76 2,3,4-(CH.sub.3).sub.3                                                      77 2,3,6-(CH.sub.3).sub.3                                                      78 2,4,5-(CH.sub.3).sub.3                                                      79 2,4,6-(CH.sub.3).sub.3                                                      80 3,4,5-(CH.sub.3).sub.3                                                      81 2,3,4,6-(CH.sub.3).sub.4                                                    82 2,3,5,6-(CH.sub.3).sub.4                                                    83 2,3,4,5,6-(CH.sub.3).sub.5                                                  84 2-C.sub.2 H.sub.5                                                           85 3-C.sub.2 H.sub.5                                                           86 4-C.sub.2 H.sub.5                                                           87 2,4-(C.sub.2 H.sub.5).sub.2                                                 88 2,6-(C.sub.2 H.sub.5).sub.2                                                 89 3,5-(C.sub.2 H.sub.5).sub.2                                                 90 2,4,6-(C2H5)3                                                               91 2-n-C.sub.3 H.sub.7                                                         92 3-n-C.sub.3 H.sub.7                                                         93 4-n-C.sub.3 H.sub.7                                                         94 2-i-C.sub.3 H.sub.7                                                         95 3-i-C.sub.3 H.sub.7                                                         96 4-i-C.sub.3 H.sub.7                                                         97 2,4-(i-C.sub.3 H.sub.7).sub.2                                               98 2,6-(i-C.sub.3 H.sub.7).sub.2                                               99 3,5-(i-C.sub.3 H.sub.7).sub.2                                              100 2,4,6-(i-C.sub.3 H.sub.7).sub.3                                            101 2-s-C.sub.4 H.sub.9                                                        102 3-s-C.sub.4 H.sub.9                                                        103 4-s-C.sub.4 H.sub.9                                                        104 2-t-C.sub.4 H.sub.9                                                        105 3-t-C.sub.4 H.sub.9                                                        106 4-t-C.sub.4 H.sub.9                                                        107 2,3-(t-C.sub.4 H.sub.9).sub.2                                              108 2,4-(t-C.sub.4 H.sub.9).sub.2                                              109 2,5-(t-C.sub.4 H.sub.9).sub.2                                              110 2,6-(t-C.sub.4 H.sub.9).sub.2                                              111 3,4-(t-C.sub.4 H.sub.9).sub.2                                              112 2,4,6-(t-C.sub.4 H.sub.9).sub.3                                            113 4-n-C.sub.9 H.sub.19                                                       114 4-n-C.sub.12 H.sub.25                                                      115 4-n-C.sub.15 H.sub.31                                                      116 4-(1,1,3,3-Tetramethylbutyl)                                               117 4-(2,4,4-Trimethylpropyl)                                                  118 2-t-C.sub.4 H.sub.9, 4-CH.sub.3                                            119 2-t-C.sub.4 H.sub.9, 5-CH.sub.3                                            120 2,6-(t-C.sub.4 H.sub.9), 4-CH.sub.3                                        121 2-CH.sub.3, 4-t-C.sub.4 H.sub.9                                            122 2-CH.sub.3, 6-t-C.sub.4 H.sub.9                                            123 2-CH.sub.3, 4-i-C.sub.3 H.sub.7                                            124 2-CH.sub.3, 5-i-C.sub.3 H.sub.7                                            125 3-CH.sub.3, 4-i-C.sub.3 H.sub.7                                            126 2-i-C.sub.3 H.sub.7, 5-CH.sub.3                                            127 2,4-(t-C.sub.4 H.sub.9), 6-i-C.sub.3 H.sub.7                               128 2-Allyl                                                                    129 3-Allyl                                                                    130 4-Allyl                                                                    131 2-Allyl, 6-CH.sub.3                                                        132 2-cyclo-C.sub.6 H.sub.11                                                   133 3-cyclo-C.sub.6 H.sub.11                                                   134 4-cyclo-C.sub.6 H.sub.11                                                   135 2,4-(cyclo-C.sub.6 H.sub.11), 6-CH.sub.3                                   136 2-CH.sub.3, 4-cyclo-C.sub.6 H.sub.11                                       137 2-CH.sub.2 --C.sub.6 H.sub.5                                               138 3-CH.sub.2 --C.sub.6 H.sub.5                                               139 4-CH.sub.2 --C.sub.6 H.sub.5                                               140 2-CH.sub.2 --C.sub.6 H.sub.5, 4-CH.sub.3                                   141 2-CH.sub.3, 4-CH.sub.2 --C.sub.6 H.sub.5                                   142 2-C.sub.6 H.sub.5                                                          143 3-C.sub.6 H.sub.5                                                          144 4-C.sub.6 H.sub.5                                                          145 4-(2-i-C.sub.3 H.sub.7 --C.sub.6 H.sub.4)                                  146 4-C.sub.6 H.sub.5, 2,6-(CH.sub.3).sub.2                                    147 2-Cl, 4-C.sub.6 H.sub.5                                                    148 2-Br, 4-C.sub.6 H.sub.5                                                    149 2-C.sub.6 H.sub.5, 4-Cl                                                    150 2-C.sub.6 H.sub.5, 4-Br                                                    151 2-CH.sub.2 C.sub.6 H.sub.5, 4-Cl                                           152 2-CH.sub.2 C.sub.6 H.sub.5, 4-Br                                           153 2-Cl, 4-CH.sub.2 C.sub.6 H.sub.5                                           154 2-Br, 4-CH.sub.2 C.sub.6 H.sub.5                                           155 2-cyclo-C.sub.6 H.sub.11, 4-Cl                                             156 2-cyclo-C.sub.6 H.sub.11, 4-Br                                             157 2-Cl, 4-cyclo-C.sub.6 H.sub.11                                             158 2-Br, 4-cyclo-C.sub.6 H.sub.11                                             159 2-OCH.sub.3                                                                160 3-OCH.sub.3                                                                161 4-OCH.sub.3                                                                162 2-OC.sub.2 H.sub.5                                                         163 3-O--C.sub.2 H.sub.5                                                       164 4-O--C.sub.2 H.sub.5                                                       165 2-O-n-C.sub.3 H.sub.7                                                      166 3-O-n-C.sub.3 H.sub.7                                                      167 4-C-n-C.sub.3 H.sub.7                                                      168 2-O-i-C.sub.3 H.sub.7                                                      169 3-O-i-C.sub.3 H.sub.7                                                      170 4-O-i-C.sub.3 H.sub.7                                                      171 2-O-n-C.sub.6 H.sub.13                                                     172 3-O-n-C.sub.6 H.sub.13                                                     173 4-O-n-C.sub.6 H.sub.13                                                     174 2-O-n-C.sub.8 H.sub.17                                                     175 3-O-n-C.sub.8 H.sub.17                                                     176 4-O-n-C.sub.8 H.sub.17                                                     177 2-O--CH.sub.2 C.sub.6 H.sub.5                                              178 3-O--CH.sub.2 C.sub.6 H.sub.5                                              179 4-O--CH.sub.2 C.sub.6 H.sub.5                                              180 2-O--(CH.sub.2).sub.3 C.sub.6 H.sub.5                                      181 3-O--(CH.sub.2).sub.3 C.sub.6 H.sub.5                                      182 4-O--(CH.sub.2).sub.3 C.sub.6 H.sub.5                                      183 2,4-(OCH.sub.3).sub.2                                                      184 2-CF.sub.3                                                                 185 3-CF.sub.3                                                                 186 4-CF.sub.3                                                                 187 2-OCF.sub.3                                                                188 3-OCF.sub.3                                                                189 4-OCF.sub.3                                                                190 3-OCH.sub.2 CHF.sub.2                                                      191 2-NO.sub.2                                                                 192 3-NO.sub.2                                                                 193 4-NO.sub.2                                                                 194 2-CN                                                                       195 3-CN                                                                       196 4-CN                                                                       197 2-CH.sub.3, 3-Cl                                                           198 2-CH.sub.3, 4-Cl                                                           199 2-CH.sub.3, 5-Cl                                                           200 2-CH.sub.3, 6-Cl                                                           201 2-CH.sub.3, 3-F                                                            202 2-CH.sub.3, 4-F                                                            203 2-CH.sub.3, 5-F                                                            204 2-CH.sub.3, 6-F                                                            205 2-CH.sub.3, 3-Br                                                           206 2-CH.sub.3, 4-Br                                                           207 2-CH.sub.3, 5-Br                                                           208 2-CH.sub.3, 6-Br                                                           209 2-Cl, 3-CH.sub.3                                                           210 2-Cl, 4-CH3                                                                211 2-Cl, 5-CH3                                                                212 2-F, 3-CH.sub.3                                                            213 2-F, 4-CH.sub.3                                                            214 2-F, 5-CH.sub.3                                                            215 2-Br, 3-CH.sub.3                                                           216 2-Br, 4-CH.sub.3                                                           217 2-Br, 5-CH.sub.3                                                           218 3-CH.sub.3, 4-Cl                                                           219 3-CH.sub.3, 5-Cl                                                           220 3-CH.sub.3, 4-F                                                            221 3-CH.sub.3, 5-F                                                            222 3-CH.sub.3, 4-Br                                                           223 3-CH.sub.3, 5-Br                                                           224 3-F, 4-CH.sub.3                                                            225 3-Cl, 4-CH3                                                                226 3-Br, 4-CH3                                                                227 2-Cl, 4,5-(CH.sub.3).sub.2                                                 228 2-Br, 4,5-(CH.sub.3).sub.2                                                 229 2-Cl, 3,5-(CH.sub.3).sub.2                                                 230 2-Br, 3,5-(CH.sub.3).sub.2                                                 231 2,6-Cl.sub.2, 4-CH.sub.3                                                   232 2,6-F.sub.2, 4-CH.sub.3                                                    233 2,6-Br.sub.2, 4-CH.sub.3                                                   234 2,4-Br.sub.2, 6-CH.sub.3                                                   235 2,4-F.sub.2, 6-CH.sub.3                                                    236 2,4-Br.sub.2, 6-CH.sub.3                                                   237 2,6-(CH.sub.3).sub.2, 4-F                                                  238 2,6-(CH.sub.3).sub.2, 4-Cl                                                 239 2,6-(CH.sub.3).sub.2, 4-Br                                                 240 3,5-(CH.sub.3).sub.2, 4-F                                                  241 3,5-(CH.sub.3).sub.2, 4-Cl                                                 242 3,5-(CH.sub.3).sub.2, 4-Br                                                 243 2,3,6-(CH.sub.3).sub.3, 4-F                                                244 2,3,6-(CH.sub.3).sub.3, 4-Cl                                               245 2,3,6-(CH.sub.3).sub.3, 4-Br                                               246 2,4-(CH.sub.3).sub.2, 6-F                                                  247 2,4-(CH.sub.3).sub.2, 6-Cl                                                 248 2,4-(CH.sub.3).sub.2, 6-Br                                                 249 2-i-C.sub.3 H.sub.7, 4-Cl, 5-CH.sub.3                                      250 2-Cl, 4-NO.sub.2                                                           251 2-NO.sub.2, 4-Cl                                                           252 2-OCH.sub.3, 5-NO.sub.2                                                    253 2,4-Cl.sub.2, 5-NO.sub.2                                                   254 2,4-Cl.sub.2, 6-NO.sub.2                                                   255 2,6-Cl.sub.2, 4-NO.sub.2                                                   256 2,6-Br.sub.2, 4-NO.sub.2                                                   257 2,6-I.sub.2, 4-NO.sub.2                                                    258 2-CH.sub.3, 5-i-C.sub.3 H.sub.7, 4-Cl                                      259 2-CO.sub.2 CH.sub.3                                                        260 3-CO.sub.2 CH.sub.3                                                        261 4-CO.sub.2 CH.sub.3                                                        262 2-CO.sub.2 (C.sub.2 H.sub.5)                                               263 3-CO.sub.2 (C.sub.2 H.sub.5)                                               264 4-CO.sub.2 (C.sub.2 H.sub.5)                                               265 2-CO.sub.2 (n-C.sub.3 H.sub.7)                                             266 3-CO.sub.2 (n-C.sub.3 H.sub.7)                                             267 4-CO.sub.2 (n-C.sub.3 H.sub.7)                                             268 2-CO.sub.2 (i-C.sub.3 H.sub.7)                                             269 3-CO.sub.2 (i-C.sub.3 H.sub.7)                                             270 4-CO.sub.2 (i-C.sub.3 H.sub.7)                                             271 2-CO.sub.2 (n-C.sub.6 H.sub.13)                                            272 3-CO.sub.2 (n-C.sub.6 H.sub.13)                                            273 4-CO.sub.2 (n-C.sub.6 H.sub.13)                                            274 2-CH.sub.2 --OCH.sub.3                                                     275 3-CH.sub.2 --OCH.sub.3                                                     276 4-CH.sub.2 --OCH.sub.3                                                     277 2-CH.sub.2 O(C.sub.2 H.sub.5)                                              278 3-CH.sub.2 O(C.sub.2 H.sub.5)                                              279 4-CH.sub.2 O(C.sub.2 H.sub.5)                                              280 2-CH.sub.2 O(n-C.sub.3 H.sub.7)                                            281 3-CH.sub.2 O(n-C.sub.3 H.sub.7)                                            282 4-CH.sub.2 O(n-C.sub.3 H.sub.7)                                            283 2-CH.sub.2 O(i-C.sub.3 H.sub.7)                                            284 3-CH.sub.2 O(i-C.sub.3 H.sub.7)                                            285 4-CH.sub.2 O(i-C.sub.3 H.sub.7)                                            286 2-CHO                                                                      287 3-CHO                                                                      288 4-CHO                                                                      289 2-CO--CH.sub.3                                                             290 3-CO--CH.sub.3                                                             291 4-CO--CH.sub.3                                                             292 2-CO--CH.sub.2 --CH.sub.3                                                  293 3-CO--CH.sub.2 --CH.sub.3                                                  294 4-CO--CH.sub.2 --CH.sub.3                                                  295 2-CO--CH.sub.2 --CH.sub.2 --CH.sub.3                                       296 3-CO--CH.sub.2 --CH.sub.2 --CH.sub.3                                       297 4-CO--CH.sub.2 --CH.sub.2 --CH.sub.3                                       298 2-CO--CH(CH.sub.3)--CH.sub.3                                               299 3-CO--CH(CH.sub.3)--CH.sub.3                                               300 4-CO--CH(CH.sub.3)--CH.sub.3                                               301 2-Me-4-CHO                                                                 302 2-Me-4-CH.sub.3 --CO                                                       303 2-Me-4-CH.sub.3 --CH.sub.2 --CO                                            304 2-Me-4-CH.sub.3 --CH.sub.2 --CH.sub.2 --CO                                 305 2-Me-4-CH.sub.3 --CH(CH.sub.3)--CO                                         306 2,5-Me.sub.2 -4-CHO                                                        307 2,5-Me.sub.2 -4-CH.sub.3 --CO                                              308 2,5-Me.sub.2 -4-CH.sub.3 --CH.sub.2 --CO                                   309 2,5-Me.sub.2 -4-CH.sub.3 --CH.sub.2 --CH.sub.2 --CO                        310 2,5-Me.sub.2 -4-CH.sub.3 --CH(CH.sub.3)--CO                                311 2-Cl-4-CHO                                                                 312 2-Cl-4-CH.sub.3 --CO                                                       313 2-Cl-4-CH.sub.3 --CH.sub.2 --CO                                            314 2-Cl-4-CH.sub.3 --CH(CH.sub.3)--CO                                         315 2,5-Cl.sub.2 -4-CHO                                                        316 2,5-Cl.sub.2 -4-CH.sub.3 --CO                                              317 2,5-Cl.sub.2 -4-CH.sub.3 --CH.sub.2 --CO                                   318 2,5-Cl.sub.2 -4-CH.sub.3 --CH.sub.2 --CH.sub.2 --CO                        319 2,5-Cl.sub.2 -4-CH.sub.3 -- --CH(CH.sub.3)--CO                             320 2-C(═NOCH.sub.3)--CH.sub.3                                             321 3-C(═NOCH.sub.3)--CH.sub.3                                             322 4-C(═NOCH.sub.3)--CH.sub.3                                             323 2-C(═NOC.sub.2 H.sub.5)--CH.sub.3                                      324 3-C(═NOC.sub.2 H.sub.5)--CH.sub.3                                      325 4-C(═NOC.sub.2 H.sub.5)--CH.sub.3                                      326 2-C(═NO-n-C.sub.3 H.sub.7)--CH.sub.3                                   327 3-C(═NO-n-C.sub.3 H.sub.7)--CH.sub.3                                   328 4-C(═NO-n-C.sub.3 H.sub.7)--CH.sub.3                                   329 2-C(═NO-i-C.sub.3 H.sub.7)--CH.sub.3                                   330 3-C(═NO-i-C.sub.3 H.sub.7)--CH.sub.3                                   331 4-C(═NO-i-C.sub.3 H.sub.7)--CH.sub.3                                   332 2-C(═NO-Allyl)-CH.sub.3                                                333 3-C(═NO-Allyl)-CH.sub.3                                                334 4-C(═NO-Allyl)-CH.sub.3                                                335 2-C(═NO-trans-Chloroallyl)-CH.sub.3                                    336 3-C(═NO-trans-Chloroallyl)-CH.sub.3                                    337 4-C(═NO-trans-Chloroallyl)-CH.sub.3                                    338 2-C(═NO-Propargyl)-CH.sub.3                                            339 3-C(═NO-Propargyl)-CH.sub.3                                            340 4-C(═NO-Propargyl)-CH.sub.3                                            341 2-C(═NO-n-C.sub.4 H.sub.9)--CH.sub.3                                   342 3-C(═NO-n-C.sub.4 H.sub.9)--CH.sub.3                                   343 4-C(═NO-n-C.sub.4 H.sub.9)--CH.sub.3                                   344 2-C(═NO--CH.sup.2 --C.sup.6 H.sup.5)--CH.sub.3                         345 3-C(═NO--CH.sub.2 --C.sub.6 H.sub.5)--CH.sub.3                         346 4-C(═NO--CH.sub.2 --C.sub.6 H.sub.5)--CH.sub.3                         347 2-CH.sub.3 -4-CH═NOCH.sub.3                                            348 2-CH.sub.3 -4-CH═NOC.sub.2 H.sub.5                                     349 2-CH.sub.3 -4-CH═NO-n-C.sub.3 H.sub.7                                  350 2-CH.sub.3 -4-CH═NO-i-C.sub.3 H.sub.7                                  351 2-CH.sub.3 -4-CH═NO-Allyl                                              352 2-CH.sub.3 -4-CH═NO-(trans-Chloroallyl)                                353 2-CH.sub.3 -4-CH═NO-Propargyl                                          354 2-CH.sub.3 -4-CH═NO-n-C.sub.4 H.sub.9                                  355 2-CH.sub.3 -4-CH═NO--CH.sub.2 --C.sub.6 H.sub.5                        356 2-CH.sub.3 -4-(CH.sub.3 --C═NOCH.sub.3)                                357 2-CH.sub.3 -4-(CH.sub.3 --C═NOC.sub.2 H.sub.5)                         358 2-CH.sub.3 -4-(CH.sub.3 --C═NO-n-C.sub.3 H.sub.7)                      359 2-CH.sub.3 -4-(CH.sub.3 --C═NO-i-C.sub.3 H.sub.7)                      360 2-CH.sub.3 -4-(CH.sub.3 --C═NO-Allyl)                                  361 2-CH.sub.3 -4-(CH.sub.3 --C═NO-trans-Chloroallyl)                      362 2-CH.sub.3 -4-(CH.sub.3 --C═NO-Propargyl)                              363 2-CH.sub.3 -4-(CH.sub.3 --C═NO-n-C.sub.4 H.sub.9)                      364 2-CH.sub.3 -4-(CH.sub.3 --C═NO--CH.sub.2 --C.sub.6 H.sub.5)                   365 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C═NO--CH.sub.3)                       366 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C═NO--C.sub.2 H.sub.5)                367 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C═NO-n-C.sub.3 H.sub.7)        368 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C═NO-i-C.sub.3 H.sub.7                       369 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C═NO-Allyl)                    370 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C═NO-trans-Chloroallyl)                      371 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C═NO-Propargyl)                       372 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C═NO-n-C.sub.4 H.sub.9)        373 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C═NO--CH.sub.2 --C.sub.6                    H.sub.5)                                                                 374 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C═NOCH.sub.3)                      375 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C═NOC.sub.2 H.sub.5)                      376 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C═NO-n-C.sub.3                    H.sub.7)                                                                 377 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C═NO-i-C.sub.3 H.sub.7)                   378 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C═NO-Allyl                  379 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C═NO-trans-Chloroallyl)                   380 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C═NO-Proparyl)                     381 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C═NO-n-C.sub.4                    H.sub.9)                                                                 382 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C═NO--CH.sub.2 --C.sub.6                 H.sub.5)                                                                 383 2-C.sub.6 H.sub.5                                                          384 3-C6H5                                                                     385 4-C6H5                                                                     386 2-(2'-F--C6H4)                                                             387 2-(3'-F--C.sub.6 H.sub.4)                                                  388 2-(4'-F--C.sub.6 H.sub.4)                                                  389 3-(2'-F--C.sub.6 H.sub.4)                                                  390 3-(3'-F--C.sub.6 H.sub.4)                                                  391 3-(4'-F--C.sub.6 H.sub.4)                                                  392 4-(2'-F--C.sub.6 H.sub.4)                                                  393 4-(3'-F--C.sub.6 H.sub.4)                                                  394 4-(4'-F--C.sub.6 H.sub.4)                                                  395 2-(2'-Cl--C.sub.6 H.sub.4)                                                 396 2-(3'-Cl--C.sub.6 H.sub.4)                                                 397 2-(4'-Cl--C.sub.6 H.sub.4)                                                 398 3-(2'-Cl--C.sub.6 H.sub.4)                                                 399 3-(3'-Cl--C.sub.6 H.sub.4)                                                 400 3-(4'-Cl--C.sub.6 H.sub.4)                                                 401 4-(2'-Cl--C.sub.6 H.sub.4)                                                 402 4-(3'-Cl--C.sub.6 H.sub.4)                                                 403 4-(4'-Cl--C.sub.6 H.sub.4)                                                 405 2-(2'-CH.sub.3 --C.sub.6 H.sub.4)                                          406 2-(3'-CH.sub.3 --C.sub.6 H.sub.4)                                          407 2-(4'-CH.sub.3 --C.sub.6 H.sub.4)                                          408 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)                                          409 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)                                          410 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)                                          411 4-(2'-CH.sub.3 --C.sub.6 H.sub.4)                                          412 4-(3'-CH.sub.3 --C.sub.6 H.sub.4)                                          413 4-(4'-CH.sub.3 --C.sub.6 H.sub.4)                                          414 2-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                      415 2-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                      416 2-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                      417 3-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                      418 3-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                      419 3-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                      420 4-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                      421 4-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                      422 4-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                      423 2-(2'-(CH.sub.3 --C(═NOAllyl))-C.sub.6 H.sub.4)                        424 2-(3'-(CH.sub.3 --C(═NOAllyl))-C.sub.6 H.sub.4)                        425 2-(4'-(CH.sub.3 --C(═NOAllyl))-C.sub.6 H.sub.4)                        426 3-(2'-(CH.sub.3 --C(═NOAllyl))-C.sub.6 H.sub.4)                        427 3-(3'-(CH.sub.3 --C(═NOAllyl))-C.sub.6 H.sub.4)                        428 3-(4'-(CH.sub.3 --C(═NOAllyl))-C.sub.6 H.sub.4)                        429 4-(2'-(CH.sub.3 --C(═NOAllyl))-C.sub.6 H.sub.4)                        430 4-(3'-(CH.sub.3 --C(═NOAllyl))-C.sub.6 H.sub.4)                        431 4-(4'-(CH.sub.3 --C(═NOAllyl))-C.sub.6 H.sub.4)                        432 2-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                                 433 2-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                                 434 2-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                                 435 3-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                                 436 3-(3'-CH.sub.3 O.sub.2 C--C6H4)                                            437 3-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                                 438 4-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                                 439 4-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                                 440 4-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                                 441 2-(2'-CH.sub.3 O--C.sub.6 H.sub.4)                                         442 2-(3'-CH.sub.3 O--C.sub.6 H.sub.4)                                         443 2-(4'-CH.sub.3 O--C.sub.6 H.sub.4)                                         444 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)                                         445 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)                                         446 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)                                         447 4-(2'-CH.sub.3 O--C.sub.6 H.sub.4)                                         448 4-(3'-CH.sub.3 O--C.sub.6 H.sub.4)                                         449 4-(4'-CH.sub.3 O--C.sub.6 H.sub.4)                                         450 2-(2'-O.sub.2 N--C.sub.6 H.sub.4)                                          451 2-(3'-O.sub.2 N--C.sub.6 H.sub.4)                                          452 2-(4'-O.sub.2 N--C.sub.6 H.sub.4)                                          453 3-(2'-O.sub.2 N--C.sub.6 H.sub.4)                                          454 3-(3'-O.sub.2 N--C.sub.6 H.sub.4)                                          455 3-(4'-O.sub.2 N--C.sub.6 H.sub.4)                                          456 4-(2'-O.sub.2 N--C.sub.6 H.sub.4)                                          457 4-(3'-O.sub.2 N--C.sub.6 H.sub.4)                                          458 4-(4'-O.sub.2 N--C.sub.6 H.sub.4)                                          459 2-(2'-NC--C.sub.6 H.sub.4)                                                 460 2-(3'-NC--C.sub.6 H.sub.4)                                                 461 2-(4'-NC--C.sub.6 H.sub.4)                                                 462 3-(2'-NC--C.sub.6 H.sub.4)                                                 463 3-(3'-NC--C.sub.6 H.sub.4)                                                 464 3-(4'-NC--C.sub.6 H.sub.4)                                                 465 4-(2'-NC--C.sub.6 H.sub.4)                                                 466 4-(3'-NC--C.sub.6 H.sub.4)                                                 467 4-(4'-NC--C.sub.6 H.sub.4)                                                 468 2-(2'-CF.sub.3 --C.sub.6 H.sub.4)                                          469 2-(3'-CF.sub.3 --C.sub.6 H.sub.4)                                          470 2-(4'-CF.sub.3 --C.sub.6 H.sub.4)                                          471 3-(2'-CF.sub.3 --C.sub.6 H.sub.4)                                          472 3-(3'-CF.sub.3 --C.sub.6 H.sub.4)                                          473 3-(4'-CF.sub.3 --C6H4)                                                     474 4-(2'-CF.sub.3 --C.sub.6 H.sub.4)                                          475 4-(3'-CF.sub.3 --C.sub.6 H.sub.4)                                          476 4-(4'-CF.sub.3 --C.sub.6 H.sub.4)                                          477 2-O--C.sub.6 H.sub.5                                                       475 3-O--C6H5                                                                  476 4-O--C6H5                                                                  478 2-O-(2'-F--C6H4)                                                           479 2-O-(3'-F--C.sub.6 H.sub.4)                                                480 2-O-(4'-F--C.sub.6 H.sub.4)                                                481 3-O-(2'-F--C.sub.6 H.sub.4)                                                482 3-O-(3'-F--C.sub.6 H.sub.4)                                                483 3-O-(4'-F--C.sub.6 H.sub.4)                                                484 4-O-(2'-F--C.sub.6 H.sub.4)                                                485 4-O-(3'-F--C.sub.6 H.sub.4)                                                486 4-O-(4'-F--C.sub.6 H.sub.4)                                                487 2-O-(2'-Cl--C.sub.6 H.sub.4)                                               488 2-O-(3'-Cl--C.sub.6 H.sub.4)                                               489 2-O-(4'-Cl--C.sub.6 H.sub.4)                                               490 3-O-(2'-Cl--C.sub.6 H.sub.4)                                               491 3-O-(3'-Cl--C.sub.6 H.sub.4)                                               492 3-O-(4'-Cl--C.sub.6 H.sub.4)                                               493 3-O-(4'-Cl--C.sub.6 H.sub.4)                                               494 4-O-(2'-Cl--C.sub.6 H.sub.4)                                               495 4-O-(3'-Cl--C.sub.6 H.sub.4)                                               496 4-O-(4'-Cl--C.sub.6 H.sub.4)                                               497 2-O-(2'-CH.sub.3 --C.sub.6 H.sub.4)                                        498 2-O-(3'-CH.sub.3 --C.sub.6 H.sub.4)                                        499 2-O-(4'-CH.sub.3 --C.sub.6 H.sub.4)                                        500 3-O-(2'-CH.sub.3 --C.sub.6 H.sub.4)                                        501 3-O-(3'-CH.sub.3 --C.sub.6 H.sub.4)                                        502 3-O-(4'-CH.sub.3 --C.sub.6 H.sub.4)                                        503 4-O-(2'-CH.sub.3 --C.sub.6 H.sub.4)                                        504 4-O-(3'-CH.sub.3 --C.sub.6 H.sub.4)                                        505 4-O-(4'-CH.sub.3 --C.sub.6 H.sub.4)                                        506 2-O-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                    507 2-O-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                    508 2-O-(4'-CH.sub.3 --CO--C6H4)                                               509 3-O-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                    510 3-O-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                    511 3-O-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                    512 4-O-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                    513 4-O-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                    514 4-O-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                    515 2-O-(2'-(CH.sub.3 --C(═NOAllyl))-C.sub.6 H.sub.4)                      516 2-O-(3'-(CH.sub.3 --C(═NOAllyl))-C.sub.6 H.sub.4)                      517 2-O-(4'-(CH.sub.3 --C(═NOAllyl))-C.sub.6 H.sub.4)                      518 3-O-(2'-(CH.sub.3 --C(═NOAllyl))-C.sub.6 H.sub.4)                      519 3-O-(3'-(CH.sub.3 --C(═NOAllyl))-C.sub.6 H.sub.4)                      520 3-O-(4'-(CH.sub.3 --C(═NOAllyl))-C.sub.6 H.sub.4)                      521 4-O-(2'-(CH.sub.3 --C(═NOAllyl))-C.sub.6 H.sub.4)                      522 4-O-(3'-(CH.sub.3 --C(═NOAllyl))-C.sub.6 H.sub.4)                      523 4-O-(4'-(CH.sub.3 --C(═NOAllyl))-C.sub.6 H.sub.4)                      524 2-O-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                               525 2-O-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                               526 2-O-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                               527 3-O-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                               528 3-O-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                               529 3-O-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                               530 4-O-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                               531 4-O-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                               532 4-O-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                               533 2-O-(2'-CH.sub.3 O--C.sub.6 H.sub.4)                                       534 2-O-(3'-CH.sub.3 O--C.sub.6 H.sub.4)                                       535 2-O-(4'-CH.sub.3 O--C.sub.6 H.sub.4)                                       536 3-O-(2'-CH.sub.3 O--C.sub.6 H.sub.4)                                       537 3-O-(3'-CH.sub.3 O--C.sub.6 H.sub.4)                                       538 3-O-(4'-CH.sub.3 O--C.sub.6 H.sub.4)                                       539 4-O-(2'-CH.sub.3 O--C.sub.6 H.sub.4)                                       540 4-O-(3'-CH.sub.3 O--C.sub.6 H.sub.4)                                       541 4-O-(4'-CH.sub.3 O--C.sub.6 H.sub.4)                                       542 2-O-(2'-O.sub.2 N--C.sub.6 H.sub.4)                                        543 2-O-(3'-O.sub.2 N--C.sub.6 H.sub.4)                                        544 2-O-(4'-O.sub.2 N--C.sub.6 H.sub.4)                                        545 3-O-(2'-O.sub.2 N--C6H4)                                                   546 3-O-(3'-O.sub.2 N--C.sub.6 H.sub.4)                                        547 3-O-(4'-O.sub.2 N--C.sub.6 H.sub.4)                                        548 4-O-(2'-O.sub.2 N--C.sub.6 H.sub.4)                                        549 4-O-(3'-O.sub.2 N--C.sub.6 H.sub.4)                                        550 4-O-(4'-O.sub.2 N--C.sub.6 H.sub.4)                                        551 2-O-(2'-NC--C.sub.6 H.sub.4)                                               552 2-O-(3'-NC--C.sub.6 H.sub.4)                                               553 2-O-(4'-NC--C.sub.6 H.sub.4)                                               554 3-O-(2'-NC--C.sub.6 H.sub.4                                                555 3-O-(3'-NC--C.sub.6 H.sub.4)                                               556 3-O-(4'-NC--C.sub.6 H.sub.4)                                               557 4-O-(2'-NC--C.sub.6 H.sub.4)                                               558 4-O-(3'-NC--C.sub.6 H.sub.4)                                               559 4-O-(4'-NC--C.sub.6 H.sub.4)                                               560 2-O-(2'-CF.sub.3 --C.sub.6 H.sub.4)                                        561 2-O-(3'-CF.sub.3 --C.sub.6 H.sub.4)                                        562 2-O-(4'-CF.sub.3 --C.sub.6 H.sub.4)                                        563 3-O-(2'-CF.sub.3 --C.sub.6 H.sub.4)                                        564 3-O-(3'-CF.sub.3 --C.sub.6 H.sub.4)                                        565 3-O-(4'-CF.sub.3 --C.sub.6 H.sub.4)                                        566 4-O-(2'-CF.sub.3 --C.sub.6 H.sub.4)                                        567 4-O-(3'-CF.sub.3 --C.sub.6 H.sub.4)                                        568 4-O-(4'-CF.sub.3 --C.sub.6 H.sub.4)                                        569 2-Pyridinyl-2'                                                             570 2-Pyridinyl-3'                                                             571 2-Pyridinyl-4'                                                             572 3-Pyridinyl-2'                                                             573 3-Pyridinyl-3'                                                             574 3-Pyridinyl-4'                                                             575 4-Pyridinyl-2'                                                             576 4-Pyridinyl-3'                                                             577 4-Pyridinyl-4'                                                             578 2-Pyrimidinyl-2'                                                           579 2-Pyrimidinyl-3'                                                           580 2-Pyrimidinyl-4'                                                           581 3-Pyrimidinyl-2'                                                           582 3-Pyrimidinyl-3'                                                           583 3-Pyrimidinyl-4'                                                           584 4-Pyrimidinyl-2'                                                           585 4-Pyrimidinyl-3'                                                           586 4-Pyrimidinyl-4'                                                           587 2-Pyrazolyl-1'                                                             588 2-Pyrazolyl-3'                                                             589 2-Pyrazolyl-4'                                                             590 3-Pyrazolyl-1'                                                             591 3-Pyrazolyl-3'                                                             592 3-Pyrazolyl-4'                                                             593 4-Pyrazolyl-1'                                                             594 4-Pyrazolyl-3'                                                             595 4-Pyrazolyl-4'                                                             596 2-Isoxazolyl-3'                                                            597 2-Isoxazolyl-4'                                                            598 2-Isoxazolyl-5'                                                            599 3-Isoxazolyl-3'                                                            600 3-Isoxazolyl-4'                                                            601 3-Isoxazolyl-5'                                                            602 4-Isoxazolyl-3'                                                            603 4-Isoxazolyl-4'                                                            604 4-Isoxazolyl-5'                                                            605 2-Isothiazolyl-3'                                                          606 2-Isothiazolyl-4'                                                          607 2-Isothiazolyl-5'                                                          608 3-Isothiazolyl-3'                                                          609 3-Isothiazolyl-4'                                                          610 3-Isothiazolyl-5'                                                          611 4-Isothiazolyl-3'                                                          612 4-Isothiazolyl-4'                                                          613 4-Isothiazolyl-5'                                                          614 2-Imidazolyl-1'                                                            615 2-Imidazolyl-2'                                                            616 2-Imidazolyl-4'                                                            617 3-Imidazolyl-1'                                                            618 3-Imidazolyl-2'                                                            619 3-Imidazolyl-4'                                                            620 4-Imidazolyl-1'                                                            621 4-Imidazolyl-2'                                                            622 4-Imidazolyl-4'                                                            623 2-Oxazolyl-2'                                                              624 2-Oxazolyl-4'                                                              625 2-Oxazolyl-5'                                                              626 3-Oxazolyl-2'                                                              627 3-Oxazolyl-4'                                                              628 3-Oxazolyl-5'                                                              629 4-Oxazolyl-2'                                                              630 4-Oxazolyl-4'                                                              631 4-Oxazolyl-5'                                                              632 2-Thiazolyl-2'                                                             633 2-Thiazolyl-4'                                                             634 2-Thiazolyl-5'                                                             635 3-Thiazolyl-2'                                                             636 3-Thiazolyl-4'                                                             637 3-Thiazolyl-5'                                                             638 4-Thiazolyl-2'                                                             639 4-Thiazolyl-4'                                                             640 4-Thiazolyl-5'                                                             641 2-CH.sub.3 -4-(CH.sub.3 --C═N--O--CH.sub.2 --CH.sub.2 --OCH.sub.             3)                                                                       642 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C═N--O--CH.sub.2 --CH.sub.2                 --OCH.sub.3)                                                             643 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C═N--O--CH.sub.2 --CH.sub.2              --OCH.sub.3)                                                             644 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C═N--OCH.sub.3)                     645 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C═N--OC.sub.2 H.sub.5)                     646 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C═N--O-n-C.sub.3                   H.sub.7)                                                                 647 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C═N--O-i-C.sub.3 H.sub.7)                  648 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C═N--O-Allyl)                       649 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C═N--O-trans-Chloroall             yl)                                                                      650 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C═N--O-Propargyl)                   651 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C═N--O-n-C.sub.4 H.sub.9)                  652 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C═N--O--CH.sub.2                   --C.sub.6 H.sub.5)                                                       653 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C═N--OCH.sub.3)                     654 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C═N--OC.sub.2 H.sub.5)                     655 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C═N--O-n-C.sub.3                   H.sub.7)                                                                 656 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C═N--O-i-C.sub.3 H.sub.7)                  657 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C═N--O-Allyl)                       658 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C═N--O-trans-Chloroall             yl)                                                                      659 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C═N--O-Propargyl)                   660 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C═N--O-n-C.sub.4 H.sub.9)                  661 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C═N--O--CH.sub.2                   --C.sub.6 H.sub.5)                                                       662 2-O-n-C.sub.4 H.sub.9                                                      663 2-O-i-C.sub.4 H.sub.9                                                      664 2-O-s-C.sub.4 H.sub.9                                                      665 2-O-t-C.sub.4 H.sub.9                                                      666 2-Neopentyloxy                                                             667 3-O-n-C.sub.4 H.sub.9                                                      668 3-O-i-C.sub.4 H.sub.9                                                      669 3-O-s-C.sub.4 H.sub.9                                                      670 3-o-t-C.sub.4 H.sub.9                                                      671 3-Neopentyloxy                                                             672 4-O-n-C.sub.4 H.sub.9                                                      673 4-O-i-C.sub.4 H.sub.9                                                      674 4-O-s-C.sub.4 H.sub.9                                                      675 4-O-t-C.sub.4 H.sub.9                                                      676 4-Neopentyloxy                                                             677 3-CH.sub.3 -4-OCH.sub.3                                                    678 3-CH.sub.3 -4-OC.sub.2 H.sub.5                                             679 3-CH.sub.3 -4-O-n-C.sub.3 H.sub.7                                          680 3-CH.sub.3 -4-O-n-C.sub.4 H.sub.9                                          681 3-CH.sub.3 -4-O-i-C.sub.4 H.sub.9                                          682 3-CH.sub.3 -4-O-s-C.sub.4 H.sub.9                                          683 3-CH.sub.3 -4-O-t-C.sub.4 H.sub.9                                          684 3-CH.sub.3 -4-Neopentyloxy                                                 685 2-CH.sub.3 -3-OCH.sub.3                                                    686 2-CH.sub.3 -4-OCH.sub.3                                                    687 2-CH.sub.3 -5-OCH.sub.3                                                    688 2-CH.sub.3 -6-OCH.sub.3                                                    689 3-CH.sub.3 -4-OCH.sub.3                                                    690 3-CH.sub.3 -5-OCH.sub.3                                                    691 3-CH.sub.3 -6-OCH.sub.3                                                    692 4-CH.sub.3 -5-O--CH.sub.3                                                  693 4-CH.sub.3 -6-O--CH.sub.3                                                  694 4-CH.sub.3 -6-OCH.sub.3                                                    695 2-CH.sub.3 -3-O-i-C.sub.3 H.sub.7                                          696 2-CH.sub.3 -4-O-i-C.sub.3 H.sub.7                                          697 2-CH.sub.3 -5-O-i-C.sub.3 H.sub.7                                          698 2-CH.sub.3 -6-O-i-C.sub.3 H.sub.7                                          699 3-CH.sub.3 -4-O-i-C.sub.3 H.sub.7                                          700 3-CH.sub.3 -5-O-i-C.sub.3 H.sub.7                                          701 3-CH.sub.3 -6-O-i-C.sub.3 H.sub.7                                          702 4-CH.sub.3 -5-O-i-C.sub.3 H.sub.7                                          703 4-CH.sub.3 -6-O-i-C.sub.3 H.sub.7                                          704 5-CH.sub.3 -6-O-i-C.sub.3 H.sub.7                                          705 2-Cl-3-OCH.sub.3                                                           706 2-Cl-4-OCH.sub.3                                                           707 2-Cl-5-OCH.sub.3                                                           708 2-Cl-6-OCH.sub.3                                                           709 3-Cl-4-OCH.sub.3                                                           710 3-Cl-5-OCH.sub.3                                                           711 3-Cl-6-OCH.sub.3                                                           712 4-Cl-5-OCH.sub.3                                                           713 4-Cl-6-OCH.sub.3                                                           714 5-Cl-6-OCH.sub.3                                                         ______________________________________                                    

                  TABLE 18                                                         ______________________________________                                         2  STR221##                                                                       -      I: R.sup.1 = CH.sub.3, Z = CH.sub.3                                    II: R.sup.1 = CH.sub.2 --CH.sub.3, Z = CH.sub.3                                III: R.sup.1 = CH.sub.3, Z = C.sub.2 H.sub.5                                   IV: R.sup.1 = CH.sub.2 --CH.sub.3, Z = C.sub.2 H.sub.5                         V: R.sup.1 = CH.sub.3, Z = NHCH.sub.3                                          VI: R.sup.1 = CH.sub.2 --CH.sub.3, Z = NHCH.sub.3                            No.       B                                                                    ______________________________________                                          1        Pyrrolyl-3                                                              2 N--CH.sub.3 -Pyrrolyl-3                                                      3 N--C.sub.6 H.sub.5 -Pyrrolyl-3                                               4 N-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrrolyl-3                                 5 N-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrrolyl-3                                 6 N-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrrolyl-3                                 7 N-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrrolyl-3                                8 N-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrrolyl-3                                9 N-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrrolyl-3                                10 N-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrrolyl-3                                11 N-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrrolyl-3                                12 N-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrrolyl-3                                13 N-(4'-CN--C.sub.6 H.sub.4)-Pyrrolyl-3                                       14 N-(3'-CN--C.sub.6 H.sub.4)-Pyrrolyl-3                                       15 N-(2'-CN--C.sub.6 H.sub.4)-Pyrrolyl-3                                       16 N-(4'-Cl--C.sub.6 H.sub.4)-Pyrrolyl-3                                       17 N-(3'-Cl--C.sub.6 H.sub.4)-Pyrrolyl-3                                       18 N-(2'-Cl--C.sub.6 H.sub.4)-Pyrrolyl-3                                       19 Pyrrolyl-2                                                                  20 N--CH.sub.3 -Pyrrolyl-2                                                     21 N--C.sub.6 H.sub.5 -Pyrrolyl-2                                              22 N-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrrolyl-2                                23 N-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrrolyl-2                                24 N-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrrolyl-2                                25 N-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrrolyl-2                               26 N-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrrolyl-2                               27 N-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrrolyl-2                               28 N-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrrolyl-2                                29 N-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrrolyl-2                                30 N-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrrolyl-2                                31 N-(4'-CN--C.sub.6 H.sub.4)-Pyrrolyl-2                                       32 N-(3'-CN--C.sub.6 H.sub.4)-Pyrrolyl-2                                       33 N-(2'-CN--C.sub.6 H.sub.4)-Pyrrolyl-2                                       34 N-(4'-Cl--C.sub.6 H.sub.4)-Pyrrolyl-2                                       35 N-(3'-Cl--C.sub.6 H.sub.4)-Pyrrolyl-2                                       36 N-(2'-Cl--C.sub.6 H.sub.4)-Pyrrolyl-2                                       37 Furyl-2                                                                     38 5-CH.sub.3 -Furyl-2                                                         39 5-C.sub.6 H.sub.5 -Furyl-2                                                  40 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Furyl-2                                   41 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Furyl-2                                   42 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Furyl-2                                   43 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Furyl-2                                  44 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Furyl-2                                  45 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Furyl-2                                  46 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Furyl-2                                   47 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Furyl-2                                   48 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Furyl-2                                   49 5-(4'-CN--C.sub.6 H.sub.4)-Furyl-2                                          50 5-(3'-CN--C.sub.6 H.sub.4)-Furyl-2                                          51 5-(2'-CN--C.sub.6 H.sub.4)-Furyl-2                                          52 5-(4'-Cl--C.sub.6 H.sub.4)-Furyl-2                                          53 5-(3'-Cl--C.sub.6 H.sub.4)-Furyl-2                                          54 5-(2'-Cl--C.sub.6 H.sub.4)-Furyl-2                                          55 4-CH.sub.3 -Furyl-2                                                         56 4-C.sub.6 H.sub.5 -Furyl-2                                                  57 4-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Furyl-2                                   58 4-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Furyl-2                                   59 4-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Furyl-2                                   60 4-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Furyl-2                                  61 4-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Furyl-2                                  62 4-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Furyl-2                                  63 4-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Furyl-2                                   64 4-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Furyl-2                                   65 4-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Furyl-2                                   66 4-(4'-CN--C.sub.6 H.sub.4)-Furyl-2                                          67 4-(3'-CN--C.sub.6 H.sub.4)-Furyl-2                                          68 4-(2'-CN--C.sub.6 H.sub.4)-Furyl-2                                          69 4-(4'-Cl--C.sub.6 H.sub.4)-Furyl-2                                          70 4-(3'-Cl--C.sub.6 H.sub.4)-Furyl-2                                          71 4-(2'-Cl--C.sub.6 H.sub.4)-Furyl-2                                          72 Thienyl-2                                                                   73 5-CH.sub.3 -Thienyl-2                                                       74 5-C.sub.6 H.sub.5 -Thienyl-2                                                75 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-2                                 76 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-2                                 77 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-2                                 78 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-2                                79 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-2                                80 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-2                                81 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-2                                 82 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-2                                 83 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-2                                 84 5-(4'-CN--C.sub.6 H.sub.4)-Thienyl-2                                        85 5-(3'-CN--C.sub.6 H.sub.4)-Thienyl-2                                        86 5-(2'-CN--C.sub.6 H.sub.4)-Thienyl-2                                        87 5-(4'-Cl--C.sub.6 H.sub.4)-Thienyl-2                                        88 5-(3'-Cl--C.sub.6 H.sub.4)-Thienyl-2                                        89 5-(2'-Cl--C.sub.6 H.sub.4)-Thienyl-2                                        90 4-CH.sub.3 -Thienyl-2                                                       91 4-C.sub.6 H.sub.5 -Thienyl-2                                                92 4-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-2                                 93 4-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-2                                 94 4-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-2                                 95 4-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-2                                96 4-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-2                                97 4-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-2                                98 4-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-2                                 99 4-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-2                                100 4-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-2                                101 4-(4'-CN--C.sub.6 H.sub.4)-Thienyl-2                                       102 4-(3'-CN--C.sub.6 H.sub.4)-Thienyl-2                                       103 4-(2'-CN--C.sub.6 H.sub.4)-Thienyl-2                                       104 4-(4'-Cl--C.sub.6 H.sub.4)-Thienyl-2                                       105 4-(3'-Cl--C.sub.6 H.sub.4)-Thienyl-2                                       106 4-(2'-Cl--C.sub.6 H.sub.4)-Thienyl-2                                       107 Thienyl-3                                                                  108 5-CH.sub.3 -Thienyl-3                                                      109 5-C.sub.6 H.sub.5 -Thienyl-3                                               110 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-3                                111 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-3                                112 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-3                                113 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-3                               114 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-3                               115 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-3                               116 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-3                                117 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-3                                118 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-3                                119 5-(4'-CN--C.sub.6 H.sub.4)-Thienyl-3                                       120 5-(3'-CN--C.sub.6 H.sub.4)-Thienyl-3                                       121 5-(2'-CN--C.sub.6 H.sub.4)-Thienyl-3                                       122 5-(4'-Cl--C.sub.6 H.sub.4)-Thienyl-3                                       123 5-(3'-Cl--C.sub.6 H.sub.4)-Thienyl-3                                       124 5-(2'-Cl--C.sub.6 H.sub.4)-Thienyl-3                                       125 Pyrazolyl-4                                                                126 N--CH.sub.3 -Pyrazolyl-4                                                   127 N--C.sub.6 H.sub.5 -Pyrazolyl-4                                            128 N-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrazolyl-4                              129 N-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrazolyl-4                              130 N-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrazolyl-4                              131 N-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrazolyl-4                             132 N-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrazolyl-4                             133 N-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrazolyl-4                             134 N-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrazolyl-4                              135 N-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrazolyl-4                              136 N-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrazolyl-4                              137 N-(4'-CN--C.sub.6 H.sub.4)-Pyrazolyl-4                                     138 N-(3'-CN--C.sub.6 H.sub.4)-Pyrazolyl-4                                     139 N-(2'-CN--C.sub.6 H.sub.4)-Pyrazolyl-4                                     140 N-(4'-Cl--C.sub.6 H.sub.4)-Pyrazolyl-4                                     141 N-(3'-Cl--C.sub.6 H.sub.4)-Pyrazolyl-4                                     142 N-(2'-Cl--C.sub.6 H.sub.4)-Pyrazolyl-4                                     143 3-CH.sub.3 --N-Methylpyrazolyl-4                                           144 3-C.sub.6 H.sub.5 --N-Methylpyrazolyl-4                                    145 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)--N-Methylpyrazolyl-4                     146 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)--N-Methylpyrazolyl-4                     147 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)--N-Methylpyrazolyl-4                     148 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)--N-Methylpyrazolyl-4                    149 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)--N-Methylpyrazolyl-4                    150 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)--N-Methylpyrazolyl-4                    151 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)--N-Methylpyrazolyl-4                     152 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)--N-Methylpyrazolyl-4                     153 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)--N-Methylpyrazolyl-4                     154 3-(4'-CN--C.sub.6 H.sub.4)--N-Methylpyrazolyl-4                            155 3-(3'-CN--C.sub.6 H.sub.4)--N-Methylpyrazolyl-4                            156 3-(2'-CN--C.sub.6 H.sub.4)--N-Methylpyrazolyl-4                            157 3-(4'-Cl--C.sub.6 H.sub.4)--N-Methylpyrazolyl-4                            158 3-(3'-Cl--C.sub.6 H.sub.4)--N-Methylpyrazolyl-4                            159 3-(2'-Cl--C.sub.6 H.sub.4)--N-Methylpyrazolyl-4                            160 Isoxazolyl-5                                                               161 3-CH.sub.3 -Isoxazolyl-5                                                   162 3-C.sub.6 H.sub.5 -Isoxazolyl-5                                            163 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Isoxazolyl-5                             164 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Isoxazolyl-5                             165 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Isoxazolyl-5                             166 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Isoxazolyl-5                            167 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Isoxazolyl-5                            168 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Isoxazolyl-5                            169 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Isoxazolyl-5                             170 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Isoxazolyl-5                             171 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Isoxazolyl-5                             172 3-(4'-CN--C.sub.6 H.sub.4)-Isoxazolyl-5                                    173 3-(3'-CN--C.sub.6 H.sub.4)-Isoxazolyl-5                                    174 3-(2'-CN--C.sub.6 H.sub.4)-Isoxazolyl-5                                    175 3-(4'-Cl--C.sub.6 H.sub.4)-Isoxazolyl-5                                    176 3-(3'-Cl--C.sub.6 H.sub.4)-Isoxazolyl-5                                    177 3-(2'-Cl--C.sub.6 H.sub.4)-Isoxazolyl-5                                    178 4-Chloroisoxazolyl-5                                                       179 3-CH.sub.3 -4-Chloroisoxazolyl-5                                           180 3-C.sub.6 H.sub.5 -4-Chloroisoxazolyl-5                                    181 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                     182 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                     183 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                     184 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                    185 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                    186 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                    187 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                     188 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                     189 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                     190 3-(4'-CN--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                            191 3-(3'-CN--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                            192 3-(2'-CN--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                            193 3-(4'-Cl--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                            194 3-(3'-Cl--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                            195 3-(2'-Cl--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                            196 Isoxazolyl-3                                                               197 5-CH.sub.3 -Isoxazolyl-3                                                   198 5-C.sub.6 H.sub.5 -Isoxazolyl-3                                            199 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Isoxazolyl-3                             200 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Isoxazolyl-3                             201 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Isoxazolyl-3                             202 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Isoxazolyl-3                            203 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Isoxazolyl-3                            204 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Isoxazolyl-3                            205 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Isoxazolyl-3                             206 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Isoxazolyl-3                             207 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Isoxazolyl-3                             208 5-(4'-CN--C.sub.6 H.sub.4)-Isoxazolyl-3                                    209 5-(3'-CN--C.sub.6 H.sub.4)-Isoxazolyl-3                                    210 5-(2'-CN--C.sub.6 H.sub.4)-Isoxazolyl-3                                    211 5-(4'-Cl--C.sub.6 H.sub.4)-Isoxazolyl-3                                    212 5-(3'-Cl--C.sub.6 H.sub.4)-Isoxazolyl-3                                    213 5-(2'-Cl--C.sub.6 H.sub.4)-Isoxazolyl-3                                    214 Isothiazolyl-5                                                             215 3-CH.sub.3 -Isothiazolyl-5                                                 216 3-C.sub.6 H.sub.5 -Isothiazolyl-5                                          217 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Isothiazolyl-5                           218 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Isothiazolyl-5                           219 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Isothiazolyl-5                           220 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Isothiazolyl-5                          221 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Isothiazolyl-5                          222 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Isothiazolyl-5                          223 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Isothiazolyl-5                           224 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Isothiazolyl-5                           225 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Isothiazolyl-5                           226 3-(4'-CN--C.sub.6 H.sub.4)-Isothiazolyl-5                                  227 3-(3'-CN--C.sub.6 H.sub.4)-Isothiazolyl-5                                  228 3-(2'-CN--C.sub.6 H.sub.4)-Isothiazolyl-5                                  229 3-(4'-Cl--C.sub.6 H.sub.4)-Isothiazolyl-5                                  230 3-(3'-Cl--C.sub.6 H.sub.4)-Isothiazolyl-5                                  231 3-(2'-Cl--C.sub.6 H.sub.4)-Isothiazolyl-5                                  232 Oxazolyl-4                                                                 233 2-CH.sub.3 -Oxazolyl-4                                                     234 2-C.sub.6 H.sub.5 -Oxazolyl-4                                              235 2-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Oxazolyl-4                               236 2-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Oxazolyl-4                               237 2-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Oxazolyl-4                               238 2-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Oxazolyl-4                              239 2-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Oxazolyl-4                              240 2-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Oxazolyl-4                              241 2-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Oxazolyl-4                               242 2-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Oxazolyl-4                               243 2-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Oxazolyl-4                               244 2-(4'-CN--C.sub.6 H.sub.4)-Oxazolyl-4                                      245 2-(3'-CN--C.sub.6 H.sub.4)-Oxazolyl-4                                      246 2-(2'-CN--C.sub.6 H.sub.4)-Oxazolyl-4                                      247 2-(4'-Cl--C.sub.6 H.sub.4)-Oxazolyl-4                                      248 2-(3'-Cl--C.sub.6 H.sub.4)-Oxazolyl-4                                      249 2-(2'-Cl--C.sub.6 H.sub.4)-Oxazolyl-4                                      250 Thiazolyl-4                                                                251 2-CH.sub.3 -Thiazolyl-4                                                    252 2-C.sub.6 H.sub.5 -Thiazolyl-4                                             253 2-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Thiazolyl-4                              254 2-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Thiazolyl-4                              255 2-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Thiazolyl-4                              256 2-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Thiazolyl-4                             267 2-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Thiazolyl-4                             258 2-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Thiazolyl-4                             259 2-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Thiazolyl-4                              260 2-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Thiazolyl-4                              261 2-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Thiazolyl-4                              262 2-(4'-CN--C.sub.6 H.sub.4)-Thiazolyl-4                                     263 2-(3'-CN--C.sub.6 H.sub.4)-Thiazolyl-4                                     264 2-(2'-CN--C.sub.6 H.sub.4)-Thiazolyl-4                                     265 2-(4'-Cl--C.sub.6 H.sub.4)-Thiazolyl-4                                     266 2-(3'-Cl--C.sub.6 H.sub.4)-Thiazolyl-4                                     267 2-(2'-Cl--C.sub.6 H.sub.4)-Thiazolyl-4                                     268 N--CH.sub.3 -1,2,4-Triazolyl-5                                             269 3-CH.sub.3 --N--CH.sub.3 -1,2,4-Triazolyl-5                                270 3-C.sub.6 H.sub.5 --N--CH.sub.3 -1,2,4-Triazolyl-5                         271 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5                   272 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triaz               olyl-5                                                                 273 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5                   274 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Tria               zolyl-5                                                                275 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5                  276 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Tria               zolyl-5                                                                277 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5                   278 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triaz               olyl-5                                                                 279 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5                   280 3-(4'-CN--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5        281 3-(3'-CN--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-.5                         282 3-(2'-CN--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5        283 3-(4'-Cl--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5                 284 3-(3'-Cl--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5                 285 3-(2'-Cl--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5                 286 1,3,4-Oxadiazolyl-2                                                        287 5-CH.sub.3 -1,3,4-Oxadiazolyl-2                                            288 5-C.sub.6 H.sub.5 -1,2,3-Oxadiazolyl-2                                     289 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                      290 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                      291 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                      292 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                     293 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                     294 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                     295 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                      296 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                      297 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                      298 5-(4'-CN--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                             299 5-(3'-CN--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                             300 5-(2'-CN--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                             301 5-(4'-Cl--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                             302 5-(3'-Cl--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                             303 5-(2'-Cl--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                             304 1,2,4-Oxadiazolyl-3                                                        305 5-CH.sub.3 -1,2,4-Oxadiazolyl-3                                            306 5-C.sub.6 H.sub.5 -1,2,4-Oxadiazolyl-3                                     307 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                      308 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                      309 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                      310 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                     311 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                     312 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                     313 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                      314 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                      315 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                      316 5-(4'-CN--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                             317 5-(3'-CN--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                             318 5-(2'-CN--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                             319 5-(4'-Cl--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                             320 5-(3'-Cl--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                             321 5-(2'-Cl--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                             322 1,2,4-Oxadiazolyl-5                                                        323 3-CH.sub.3 -1,2,4-Oxadiazolyl-5                                            324 3-C.sub.6 H.sub.5 -1,2,4-Oxadiazolyl-5                                     325 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                      326 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                      327 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                      328 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                     329 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                     330 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                     331 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                      332 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                      333 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                      334 3-(4'-CN--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                             335 3-(3'-CN--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                             336 3-(2'-CN--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                             337 3-(4'-Cl--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                             338 3-(3'-Cl--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                             339 3-(2'-Cl--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                             340 1,2,4-Thiadiazolyl-3                                                       341 5-CH.sub.3 -1,2,4-Thiadiazolyl-3                                           342 5-C.sub.6 H.sub.5 -1,2,4-Thiadiazolyl-3                                    343 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                     344 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                     345 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                     346 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                    347 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                    348 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                    349 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                     350 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                     351 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                     352 5-(4'-CN--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                            353 5-(3'-CN--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                            354 5-(2'-CN--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                            355 5-(4'-Cl--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                            356 5-(3'-Cl--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                            357 5-(2'-Cl--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                            358 1,3,4-Thiadiazolyl-2                                                       359 5-CH.sub.3 -1,3,4-Thiadiazolyl-2                                           360 5-C.sub.6 H.sub.5 -1,3,4-Thiadiazolyl-2                                    361 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                     362 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                     363 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                     364 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                    365 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                    366 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                    367 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                     368 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                     369 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                     370 5-(4'-CN--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                            371 5-(3'-CN--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                            372 5-(2'-CN--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                            373 5-(4'-Cl--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                            374 5-(3'-Cl--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                            375 5-(2'-Cl--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                            376 Pyridinyl-2                                                                377 Pyridinyl-4                                                                378 Pyridazinyl-3                                                              379 Pyridazinyl-4                                                              380 Pyridazinyl-2                                                              381 Pyrimidinyl-4                                                              382 Pyrimidinyl-5                                                              383 Pyrimidinyl-2                                                              384 Pyridinyl-3                                                                385 1-Naphthyl                                                                 386 2-Naphthyl                                                               ______________________________________                                    

                  TABLE 19                                                         ______________________________________                                         1  STR222##                                                                       -      I: R.sup.1 = CH.sub.3, Z = CH.sub.3                                    II: R.sup.1 = CH.sub.2 --CH.sub.3, Z = CH.sub.3                                III: R.sup.1 = CH.sub.3, Z = C.sub.2 H.sub.5                                   IV: R.sup.1 = CH.sub.2 --CH.sub.3, Z = C.sub.2 H.sub.5                         V: R.sup.1 = CH.sub.3, Z = NHCH.sub.3                                          VI: R.sup.1 = CH.sub.2 --CH.sub.3, Z = NHCH.sub.3                            No.       X.sub.m                                                              ______________________________________                                          1        H                                                                       2 2-F                                                                          3 3-F                                                                          4 4-F                                                                          5 2,4-F.sub.2                                                                  6 2,4,6-F.sub.3                                                                7 2,3,4,5,6-F.sub.5                                                            8 2,3-F.sub.2                                                                  9 2-Cl                                                                         10 3-Cl                                                                        11 4-Cl                                                                        12 2,3-Cl.sub.2                                                                13 2,4-Cl.sub.2                                                                14 2,5-Cl.sub.2                                                                15 2,6-Cl.sub.2                                                                16 3,4-Cl.sub.2                                                                17 3,5-Cl.sub.2                                                                18 2,3,4-Cl.sub.3                                                              19 2,3,5-Cl.sub.3                                                              20 2,3,6-Cl.sub.3                                                              21 2,4,5-Cl.sub.3                                                              22 2,4,6-Cl.sub.3                                                              23 3,4,5-Cl.sub.3                                                              24 2,3,4,6-Cl.sub.4                                                            25 2,3,5,6-Cl.sub.4                                                            26 2,3,4,5,6-Cl.sub.5                                                          27 2-Br                                                                        28 3-Br                                                                        29 4-Br                                                                        30 2,4-Br.sub.2                                                                31 2,5-Br.sub.2                                                                32 2,6-Br.sub.2                                                                33 2,4,6-Br.sub.3                                                              34 2,3,4,5,6-Br.sub.5                                                          35 2-I                                                                         36 3-I                                                                         37 4-I                                                                         38 2,4-I.sub.2                                                                 39 2-Cl, 3-F                                                                   40 2-Cl, 4-F                                                                   41 2-Cl, 5-F                                                                   42 2-Cl, 6-F                                                                   43 2-Cl, 3-Br                                                                  44 2-Cl, 4-Br                                                                  45 2-Cl, 5-Br                                                                  46 2-Cl, 6-Br                                                                  47 2-Br, 3-Cl                                                                  48 2-Br, 4-Cl                                                                  49 2-Br, 5-Cl                                                                  50 2-Br, 3-F                                                                   51 2-Br, 4-F                                                                   52 2-Br, 5-F                                                                   53 2-Br, 6-F                                                                   54 2-F, 3-Cl                                                                   55 2-F, 4-Cl                                                                   56 2-F, 5-Cl                                                                   57 3-Cl, 4-F                                                                   58 3-Cl, 5-F                                                                   59 3-Cl, 4-Br                                                                  60 3-Cl, 5-Br                                                                  61 3-F, 4-Cl                                                                   62 3-F, 4-Br                                                                   63 3-Br, 4-Cl                                                                  64 3-Br, 4-F                                                                   65 2,6-Cl.sub.2, 4-Br                                                          66 2-CH.sub.3                                                                  67 3-CH.sub.3                                                                  68 4-CH.sub.3                                                                  69 2,3-(CH.sub.3).sub.2                                                        70 2,4-(CH.sub.3).sub.2                                                        71 2,5-(CH.sub.3).sub.2                                                        72 2,6-(CH.sub.3).sub.2                                                        73 3,4-(CH.sub.3).sub.2                                                        74 3,5-(CH.sub.3).sub.2                                                        75 2,3,5-(CH.sub.3).sub.3                                                      76 2,3,4-(CH.sub.3).sub.3                                                      77 2,3,6-(CH.sub.3).sub.3                                                      78 2,4,5-(CH.sub.3).sub.3                                                      79 2,4,6-(CH.sub.3).sub.3                                                      80 3,4,5-(CH.sub.3).sub.3                                                      81 2,3,4,6-(CH.sub.3).sub.4                                                    82 2,3,5,6-(CH.sub.3).sub.4                                                    83 2,3,4,5,6-(CH.sub.3).sub.5                                                  84 2-C.sub.2 H.sub.5                                                           85 3-C.sub.2 H.sub.5                                                           86 4-C.sub.2 H.sub.5                                                           87 2,4-(C.sub.2 H.sub.5).sub.2                                                 88 2,6-(C.sub.2 H.sub.5).sub.2                                                 89 3,5-(C.sub.2 H.sub.5).sub.2                                                 90 2,4,6-(C.sub.2 H.sub.5).sub.3                                               91 2-n-C.sub.3 H.sub.7                                                         92 3-n-C.sub.3 H.sub.7                                                         93 4-n-C.sub.3 H.sub.7                                                         94 2-i-C.sub.3 H.sub.7                                                         95 3-i-C.sub.3 H.sub.7                                                         96 4-i-C.sub.3 H.sub.7                                                         97 2,4-(i-C.sub.3 H.sub.7).sub.2                                               98 2,6-(i-C.sub.3 H.sub.7).sub.2                                               99 3,5-(i-C.sub.3 H.sub.7).sub.2                                              100 2,4,6-(i-C.sub.3 H.sub.7).sub.3                                            101 2-s-C.sub.4 H.sub.9                                                        102 3-s-C.sub.4 H.sub.9                                                        103 4-s-C.sub.4 H.sub.9                                                        104 2-t-C.sub.4 H.sub.9                                                        105 3-t-C.sub.4 H.sub.9                                                        106 4-t-C.sub.4 H.sub.9                                                        107 2,3-(t-C.sub.4 H.sub.9).sub.2                                              108 2,4-(t-C.sub.4 H.sub.9).sub.2                                              109 2,5-(t-C.sub.4 H.sub.9).sub.2                                              110 2,6-(t-C.sub.4 H.sub.9).sub.2                                              111 3,4-(t-C.sub.4 H.sub.9).sub.2                                              112 2,4,6-(t-C.sub.4 H.sub.9).sub.3                                            113 4-n-C.sub.9 H.sub.19                                                       114 4-n-C.sub.12 H.sub.25                                                      115 4-n-C.sub.15 H.sub.31                                                      116 4-(1,1,3,3-Tetramethylbutyl)                                               117 4-(2,4,4-Trimethylpropyl)                                                  118 2-t-C.sub.4 H.sub.9, 4-CH.sub.3                                            119 2-t-C.sub.4 H.sub.9, 5-CH.sub.3                                            120 2,6-(t-C4H9)2, 4-CH3                                                       121 2-CH.sub.3, 4-t-C.sub.4 H.sub.9                                            122 2-CH.sub.3, 6-t-C.sub.4 H.sub.9                                            123 2-CH.sub.3, 4-i-C.sub.3 H.sub.7                                            124 2-CH.sub.3, 5-i-C.sub.3 H.sub.7                                            125 3-CH.sub.3, 4-i-C.sub.3 H.sub.7                                            126 2-i-C.sub.3 H.sub.7, 5-CH.sub.3                                            127 2,4-(t-C.sub.4 H.sub.9).sub.2, 6-i-C.sub.3 H.sub.7                         128 2-Allyl                                                                    129 3-Allyl                                                                    130 4-Allyl                                                                    131 2-Allyl, 6-CH.sub.3                                                        132 2-cyclo-C.sub.6 H.sub.11                                                   133 3-cyclo-C.sub.6 H.sub.11                                                   134 4-cyclo-C.sub.6 H.sub.11                                                   135 2,4-(cyclo-C.sub.6 H.sub.11).sub.2, 6-CH.sub.3                             136 2-CH.sub.3, 4-cyclo-C.sub.6 H.sub.11                                       137 2-CH.sub.2 --C.sub.6 H.sub.5                                               138 3-CH.sub.2 --C.sub.6 H.sub.5                                               139 4-CH.sub.2 --C.sub.6 H.sub.5                                               140 2-CH.sub.2 --C.sub.6 H.sub.5, 4-CH.sub.3                                   141 2-CH.sub.3, 4-CH.sub.2 --C.sub.6 H.sub.5                                   142 2-C.sub.6 H.sub.5                                                          143 3-C.sub.6 H.sub.5                                                          144 4-C.sub.6 H.sub.5                                                          145 4-(2-i-C.sub.3 H.sub.7 --C.sub.6 H.sub.4)                                  146 4-C.sub.6 H.sub.5, 2,6-(CH.sub.3).sub.2                                    147 2-Cl, 4-C.sub.6 H.sub.5                                                    148 2-Br, 4-C.sub.6 H.sub.5                                                    149 2-C.sub.6 H.sub.5, 4-Cl                                                    150 2-C.sub.6 H.sub.5, 4-Br                                                    151 2-CH.sub.2 C.sub.6 H.sub.5, 4-Cl                                           152 2-CH.sub.2 C.sub.6 H.sub.5, 4-Br                                           153 2-Cl, 4-CH.sub.2 C.sub.6 H.sub.5                                           154 2-Br, 4-CH.sub.2 C.sub.6 H.sub.5                                           155 2-cyclo-C.sub.6 H.sub.11, 4-Cl                                             156 2-cyclo-C.sub.6 H.sub.11, 4-Br                                             157 2-Cl, 4-cyclo-C.sub.6 H.sub.11                                             158 2-Br, 4-cyclo-C6H11                                                        159 2-OCH.sub.3                                                                160 3-OCH.sub.3                                                                161 4-OCH.sub.3                                                                162 2-OC.sub.2 H.sub.5                                                         163 3-O--C.sub.2 H.sub.5                                                       164 4-O--C.sub.2 H.sub.5                                                       165 2-O-n-C.sub.3 H.sub.7                                                      166 3-O-n-C.sub.3 H.sub.7                                                      167 4-O-n-C.sub.3 H.sub.7                                                      168 2-O-i-C.sub.3 H.sub.7                                                      169 3-O-i-C.sub.3 H.sub.7                                                      170 4-O-i-C.sub.3 H.sub.7                                                      171 2-O-n-C.sub.6 H.sub.13                                                     172 3-O-n-C.sub.6 H.sub.13                                                     173 4-O-n-C.sub.6 H.sub.13                                                     174 2-O-n-C.sub.8 H.sub.17                                                     175 3-O-n-C.sub.8 H.sub.17                                                     176 4-O-n-C.sub.8 H.sub.17                                                     177 2-O--CH.sub.2 C.sub.6 H.sub.5                                              178 3-O--CH.sub.2 C.sub.6 H.sub.5                                              179 4-O--CH.sub.2 C.sub.6 H.sub.5                                              180 2-O--(CH.sub.2).sub.3 C.sub.6 H.sub.5                                      181 3-O--(CH.sub.2).sub.3 C.sub.6 H.sub.5                                      182 4-O--(CH.sub.2).sub.3 C.sub.6 H.sub.5                                      183 2,4-(OCH.sub.3).sub.2                                                      184 2-CF.sub.3                                                                 185 3-CF.sub.3                                                                 186 4-CF.sub.3                                                                 187 2-OCF.sub.3                                                                188 3-OCF.sub.3                                                                189 4-OCF.sub.3                                                                190 3-OCH.sub.2 CHF.sub.2                                                      191 2-NO.sub.2                                                                 192 3-NO.sub.2                                                                 193 4-NO.sub.2                                                                 194 2-CN                                                                       195 3-CN                                                                       196 4-CN                                                                       197 2-CH.sub.3, 3-Cl                                                           198 2-CH.sub.3, 4-Cl                                                           199 2-CH.sub.3, 5-Cl                                                           200 2-CH.sub.3, 6-Cl                                                           201 2-CH.sub.3, 3-F                                                            202 2-CH.sub.3, 4-F                                                            203 2-CH.sub.3, 5-F                                                            204 2-CH.sub.3, 6-F                                                            205 2-CH.sub.3, 3-Br                                                           206 2-CH.sub.3, 4-Br                                                           297 2-CH.sub.3, 5-Br                                                           208 2-CH.sub.3, 6-Br                                                           209 2-Cl, 3-CH.sub.3                                                           210 2-Cl, 4-CH.sub.3                                                           211 2-Cl, 5-CH.sub.3                                                           212 2-F, 3-CH.sub.3                                                            213 2-F, 4-CH.sub.3                                                            214 2-F, 5-CH.sub.3                                                            215 2-Br, 3-CH.sub.3                                                           216 2-Br, 4-CH.sub.3                                                           217 2-Br, 5-CH.sub.3                                                           218 3-CH.sub.3, 4-Cl                                                           219 3-CH.sub.3, 5-Cl                                                           220 3-CH.sub.3, 4-F                                                            221 3-CH.sub.3, 5-F                                                            222 3-CH.sub.3, 4-Br                                                           223 3-CH.sub.3, 5-Br                                                           224 3-F, 4-CH.sub.3                                                            225 3-Cl, 4-CH.sub.3                                                           226 3-Br, 4-CH.sub.3                                                           227 2-Cl, 4,5-(CH.sub.3).sub.2                                                 228 2-Br, 4,5-(CH.sub.3).sub.2                                                 229 2-Cl, 3,5-(CH.sub.3).sub.2                                                 230 2-Br, 3,5-(CH.sub.3).sub.2                                                 231 2,6-Cl.sub.2, 4-CH.sub.3                                                   232 2,6-F.sub.2, 4-CH.sub.3                                                    233 2,6-Br.sub.2, 4-CH.sub.3                                                   234 2,4-Br.sub.2, 6-CH.sub.3                                                   235 2,4-F.sub.2, 6-CH.sub.3                                                    236 2,4-Br.sub.2, 6-CH.sub.3                                                   237 2,6-(CH.sub.3).sub.2, 4-F                                                  238 2,6-(CH.sub.3).sub.2, 4-Cl                                                 239 2,6-(CH.sub.3).sub.2, 4-Br                                                 240 3,5-(CH.sub.3).sub.2, 4-F                                                  241 3,5-(CH.sub.3).sub.2, 4-Cl                                                 242 3,5-(CH.sub.3).sub.2, 4-Br                                                 243 2,3,6-(CH.sub.3).sub.3, 4-F                                                244 2,3,6-(CH.sub.3).sub.3, 4-Cl                                               245 2,3,6-(CH.sub.3).sub.3, 4-Br                                               246 2,4-(CH.sub.3).sub.2, 6-F                                                  247 2,4-(CH.sub.3).sub.2, 6-Cl                                                 248 2,4-(CH.sub.3).sub.2, 6-Br                                                 249 2-i-C.sub.3 H.sub.7, 4-Cl, 5-CH.sub.3                                      250 2-Cl, 4-NO.sub.2                                                           251 2-NO.sub.2, 4-Cl                                                           252 2-OCH.sub.3, 5-NO.sub.2                                                    253 2,4-Cl.sub.2, 5-NO.sub.2                                                   254 2,4-Cl.sub.2, 6-NO.sub.2                                                   255 2,6-Cl.sub.2, 4-NO.sub.2                                                   256 2,6-Br.sub.2, 4-NO.sub.2                                                   257 2,6-I.sub.2, 4-NO.sub.2                                                    258 2-CH.sub.3, 5-i-C.sub.3 H.sub.7, 4-Cl                                      259 2-CO.sub.2 CH.sub.3                                                        260 3-CO.sub.2 CH.sub.3                                                        261 4-CO.sub.2 CH.sub.3                                                        262 2-CO.sub.2 (C.sub.2 H.sub.5)                                               263 3-CO.sub.2 (C.sub.2 H.sub.5)                                               264 4-CO.sub.2 (C.sub.2 H.sub.5)                                               265 2-CO.sub.2 (n-C.sub.3 H.sub.7)                                             266 3-CO.sub.2 (n-C.sub.3 H.sub.7)                                             267 4-CO.sub.2 (n-C.sub.3 H.sub.7)                                             268 2-CO.sub.2 (i-C.sub.3 H.sub.7)                                             269 3-CO.sub.2 (i-C.sub.3 H.sub.7)                                             270 4-CO.sub.2 (i-C.sub.3 H.sub.7)                                             271 2-CO.sub.2 (n-C.sub.6 H.sub.13)                                            272 3-CO.sub.2 (n-C.sub.6 H.sub.13)                                            273 4-CO.sub.2 (n-C.sub.6 H.sub.13)                                            274 2-CH.sub.2 --OCH.sub.3                                                     275 3-CH.sub.2 --OCH.sub.3                                                     276 4-CH2--OCH.sub.3                                                           277 2-CH.sub.2 O(C.sub.2 H.sub.5)                                              278 3-CH.sub.2 C(C.sub.2 H.sub.5)                                              279 4-CH.sub.2 O(C.sub.2 H.sub.5)                                              280 2-CH.sub.2 O(n-C.sub.3 H.sub.7)                                            281 3-CH.sub.2 O (n-C.sub.3 H.sub.7)                                           282 4-CH.sub.2 O(n-C.sub.3 H.sub.7)                                            283 2-CH.sub.2 O(i-C.sub.3 H.sub.7)                                            284 3-CH.sub.2 O(i-C.sub.3 H.sub.7)                                            285 4-CH.sub.2 O(i-C.sub.3 H.sub.7)                                            286 2-CHO                                                                      287 3-CHO                                                                      288 4-CHO                                                                      289 2-CO--CH.sub.3                                                             290 3-CO--CH.sub.3                                                             291 4-CO--CH.sub.3                                                             292 2-CO--CH.sub.2 --CH.sub.3                                                  293 3-CO--CH.sub.2 --CH.sub.3                                                  294 4-CO--CH.sub.2 --CH.sub.3                                                  295 2-CO--CH.sub.2 --CH.sub.2 --CH.sub.3                                       296 3-CO--CH.sub.2 --CH.sub.2 --CH.sub.3                                       297 4-CO--CH.sub.2 --CH.sub.2 --CH.sub.3                                       298 2-CO--CH(CH.sub.3)--CH.sub.3                                               299 3-CO--CH(CH.sub.3)--CH.sub.3                                               300 4-CO--CH(CH.sub.3)--CH.sub.3                                               301 2-Me-4-CHO                                                                 302 2-Me-4-CH.sub.3 --CO                                                       303 2-Me-4-CH.sub.3 --CH.sub.2 --CO                                            304 2-Me-4-CH.sub.3 --CH.sub.2 --CH.sub.2 --CO                                 305 2-Me-4-CH.sub.3 --CH(CH.sub.3)--CO                                         306 2,5-Me.sub.2 -4-CHO                                                        307 2,5-Me.sub.2 -4-CH.sub.3 --CO                                              308 2,5-Me.sub.2 -4-CH.sub.3 --CH.sub.2 --CO                                   309 2,5-Me.sub.2 -4-CH.sub.3 --CH.sub.2 --CH.sub.2 --CO                        310 2,5-Me.sub.2 -4-CH.sub.3 --CH(CH.sub.3)--CO                                311 2-Cl-4-CHO                                                                 312 2-Cl-4-CH.sub.3 --CO                                                       313 2-Cl-4-CH.sub.3 --CH.sub.2 --CO                                            314 2-Cl-4-CH.sub.3 --CH(CH.sub.3)--CO                                         315 2,5-Cl.sub.2 -4-CHO                                                        316 2,5-Cl.sub.2 -4-CH.sub.3 --CO                                              317 2,5-Cl.sub.2 -4-CH.sub.3 --CH.sub.2 --CO                                   318 2,5-Cl.sub.2 -4-CH.sub.3 --CH.sub.2 --CH.sub.2 --CO                        319 2,5-Cl.sub.2 -4-CH.sub.3 --CH(CH.sub.3)--CO                                320 2-C(═NOCH.sub.3)--CH.sub.3                                             321 3-C(═NOCH.sub.3)--CH.sub.3                                             322 4-C(═NOCH.sub.3)--CH.sub.3                                             323 2-C(═NOC.sub.2 H.sub.5)--CH.sub.3                                      324 3-C(═NOC.sub.2 H.sub.5)--CH.sub.3                                      325 4-C(═NCC.sub.2 H.sub.5)--CH.sub.3                                      326 2-C(═NO-n-C.sub.3 H.sub.7)--CH.sub.3                                   327 3-C(═NO-n-C.sub.3 H.sub.7)--CH.sub.3                                   328 4-C(═NO-n-C.sub.3 H.sub.7)--CH.sub.3                                   329 2-C(═NO-i-C.sub.3 H.sub.7)--CH.sub.3                                   330 3-C(═NO-i-C.sub.3 H.sub.7)--CH.sub.3                                   331 4-C(═NO-i-C.sub.3 H.sub.7)--CH.sub.3                                   332 2-C(═NO-Allyl)-CH.sub.3                                                333 3-C(═NO-Allyl)-CH.sub.3                                                334 4-C(═NO-Allyl)-CH.sub.3                                                335 2-C(═NO-trans-Chloroallyl)-CH.sub.3                                    336 3-C(═NO-trans-Chloroallyl)-CH.sub.3                                    337 4-C(═NO-trans-Chloroallyl)-CH.sub.3                                    338 2-C(═NO-Propargyl)-CH.sub.3                                            339 3-C(═NO-Propargyl)-CH.sub.3                                            340 4-C(═NO-Propargyl)-CH.sub.3                                            341 2-C(═NO-n-C.sub.4 H.sub.9)--CH.sub.3                                   342 3-C(═NO-n-C.sub.4 H.sub.9)--CH.sub.3                                   343 4-C(═NO-n-C.sub.4 H.sub.9)--CH.sub.3                                   344 2-C(═NO--CH.sub.2 --C.sub.6 H.sub.5)--CH.sub.3                         345 3-C(═NO--CH.sub.2 --C.sub.6 H.sub.5)--CH.sub.3                         346 4-C(═NO--CH.sub.2 --C.sub.6 H.sub.5)--CH.sub.3                         347 2-CH.sub.3 -4-CH═NOCH.sub.3                                            348 2-CH.sub.3 -4-CH═NOC.sub.2 H.sub.5                                     349 2-CH.sub.3 -4-CH═NO-n-C.sub.3 H.sub.7                                  350 2-CH.sub.3 -4-CH═NO-i-C.sub.3 H.sub.7                                  351 2-CH.sub.3 -4-CH═NO-Allyl                                              352 2-CH.sub.3 -4-CH═NO-(trans-Chloroallyl)                                353 2-CH.sub.3 -4-CH═NO-Propargyl                                          354 2-CH.sub.3 -4-CH═NO-n-C.sub.4 H.sub.9                                  355 2-CH.sub.3 -4-CH═NO--CH.sub.2 --C.sub.6 H.sub.5                        356 2-CH.sub.3 -4-(CH.sub.3 --C═NOCH.sub.3)                                357 2-CH.sub.3 -4-(CH.sub.3 --C═NOC.sub.2 H.sub.5)                         358 2-CH.sub.3 -4-(CH.sub.3 --C═NO-n-C.sub.3 H.sub.7)                      359 2-CH.sub.3 -4-(CH.sub.3 --C═NO-i-C.sub.3 H.sub.7)                      360 2-CH.sub.3 -4-(CH.sub.3 --C═NO-Allyl)                                  361 2-CH.sub.3 -4-(CH.sub.3 --C═NO-trans-Chloroallyl)                      362 2-CH.sub.3 -4-(CH.sub.3 --C═NO-Propargyl)                              363 2-CH.sub.3 -4-(CH.sub.3 --C═NO-n-C.sub.4 H.sub.9)                      364 2-CH.sub.3 -4-(CH.sub.3 --C═NO--CH.sub.2 --C.sub.6 H.sub.5)                     365 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C═NO--CH.sub.3)                       366 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C═NO--C.sub.2                        H.sub.5)                                                               367 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C═NO-n-C.sub.3 H.sub.7)                        368 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C═NO-i-C.sub.3                       H.sub.7                                                                369 2-CH3-4-(C2H5--C═NO-Allyl)                                             370 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C═No-trans-Chloroallyl)                        371 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C═NO-Propargyl)                       372 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C═NO-n-C.sub.4                       H.sub.9)                                                               373 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C═NO--CH.sub.2 --C.sub.6                      H.sub.5)                                                               374 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C═NOCH.sub.3)                      375 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C═NOC.sub.2 H.sub.5)                        376 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C═NO-n-C.sub.3                    H.sub.7)                                                               377 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C═NO-i-C.sub.3 H.sub.7)                     378 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C═NO-Allyl)                        379 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C═NO-trans-Chloroal               lyl)                                                                   380 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C═NO-Proparyl)                     381 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C═NO-n-C.sub.4 H.sub.9)                     382 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C═NO--CH.sub.2                    --C.sub.6 H.sub.5)                                                     383 2-C.sub.6 H.sub.5                                                          384 3-C6H5                                                                     385 4-C6H5                                                                     386 2-(2'-F--C.sub.6 H.sub.4)                                                  387 2-(3'-F--C.sub.6 H.sub.4)                                                  388 2-(4'-F--C.sub.6 H.sub.4)                                                  389 3-(2'-F--C.sub.6 H.sub.4)                                                  390 3-(3'-F--C.sub.6 H.sub.4)                                                  391 3-(4'-F--C.sub.6 H.sub.4)                                                  392 4-(2'-F--C.sub.6 H.sub.4)                                                  393 4-(3'-F--C.sub.6 H.sub.4)                                                  394 4-(4'-F--C.sub.6 H.sub.4)                                                  395 2-(2'-Cl--C.sub.6 H.sub.4)                                                 396 2-(3'-Cl--C.sub.6 H.sub.4)                                                 397 2-(4'-Cl--C.sub.6 H.sub.4)                                                 398 3-(2'-Cl--C6H4)                                                            399 3-(3'-Cl--C.sub.6 H.sub.4)                                                 400 3-(4'-Cl--C.sub.6 H.sub.4)                                                 401 4-(2'-Cl--C.sub.6 H.sub.4)                                                 402 4-(3'-Cl--C.sub.6 H.sub.4)                                                 403 4-(4'-Cl--C.sub.6 H.sub.4)                                                 405 2-(2'-CH.sub.3' --C.sub.6 H.sub.4)                                         406 2-(3'-CH.sub.3' --C.sub.6 H.sub.4)                                         407 2-(4'-CH.sub.3' --C.sub.6 H.sub.4)                                         408 3-(2'-CH.sub.3' --C.sub.6 H.sub.4)                                         409 3-(3'-CH.sub.3' --C.sub.6 H.sub.4)                                         410 3-(4'-CH.sub.3' --C.sub.6 H.sub.4)                                         411 4-(2'-CH.sub.3' --C.sub.6 H.sub.4)                                         412 4-(3'-CH.sub.3' --C.sub.6 H.sub.4)                                         413 4-(4'-CH.sub.3' --C.sub.6 H.sub.4)                                         414 2-(2'-CH.sub.3' --CO--C.sub.6 H.sub.4)                                     415 2-(3'-CH.sub.3' --CO--C.sub.6 H.sub.4)                                     416 2-(4'-CH.sub.3' --CO--C.sub.6 H.sub.4)                                     417 3-(2'-CH.sub.3' --CO--C.sub.6 H.sub.4)                                     418 3-(3'-CH.sub.3' --CO--C.sub.6 H.sub.4)                                     419 3-(4'-CH.sub.3' --CO--C.sub.6 H.sub.4)                                     420 4-(2'-CH.sub.3' --CO--C.sub.6 H.sub.4)                                     421 4-(3'-CH.sub.3' --CO--C.sub.6 H.sub.4)                                     422 4-(4'-CH.sub.3' --CO--C.sub.6 H.sub.4)                                     423 2-(2'-(CH.sub.3' --C(═NOAllyl))-C.sub.6 H.sub.4)                       424 2-(3'-(CH.sub.3' --C(═NOAllyl))-C.sub.6 H.sub.4)                       425 2-(4'-(CH.sub.3' --C(.═NOAllyl))-C.sub.6 H.sub.4)                      426 3-(2'-(CH.sub.3' --C(═NOAllyl))-C.sub.6 H.sub.4)                       427 3-(3'-(CH.sub.3' --C(═NOAllyl))-C.sub.6 H.sub.4)                       428 3-(4'-(CH.sub.3' --C(═NOAllyl))-C.sub.6 H.sub.4)                       429 4-(2'-(CH.sub.3' --C(═NOAllyl))-C.sub.6 H.sub.4)                       430 4-(3'-(CH.sub.3' --C(═NOAllyl))-C.sub.6 H.sub.4)                       431 4-(4'-(CH.sub.3' --C(═NOAllyl))-C.sub.6 H.sub.4)                       432 2-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                                 433 2-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                                 434 2-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                                 435 3-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                                 436 3-(3'-CH3O2C--C6H4)                                                        437 3-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                                 438 4-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                                 439 4-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                                 440 4-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                                 441 2-(2'-CH.sub.3 O--C.sub.6 H.sub.4)                                         442 2-(3'-CH.sub.3 O--C.sub.6 H.sub.4)                                         443 2-(4'-CH.sub.3 O--C.sub.6 H.sub.4)                                         444 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)                                         445 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)                                         446 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)                                         447 4-(2'-CH.sub.3 O--C.sub.6 H.sub.4)                                         448 4-(3'-CH.sub.3 O--C.sub.6 H.sub.4)                                         449 4-(4'-CH.sub.3 O--C.sub.6 H.sub.4)                                         450 2-(2'-O.sub.2 N--C.sub.6 H.sub.4)                                          451 2-(3'-O.sub.2 N--C.sub.6 H.sub.4)                                          452 2-(4'-O.sub.2 N--C.sub.6 H.sub.4)                                          453 3-(2'-O.sub.2 N--C.sub.6 H.sub.4)                                          454 3-(3'-O.sub.2 N--C.sub.6 H.sub.4)                                          455 3-(4'-O.sub.2 N--C.sub.6 H.sub.4)                                          456 4-(2'-O.sub.2 N--C.sub.6 H.sub.4)                                          457 4-(3'-O.sub.2 N--C.sub.6 H.sub.4)                                          458 4-(4'-O.sub.2 N--C.sub.6 H.sub.4)                                          459 2-(2'-NC--C.sub.6 H.sub.4)                                                 460 2-(3'-NC--C.sub.6 H.sub.4)                                                 461 2-(4'-NC--C.sub.6 H.sub.4)                                                 462 3-(2'-NC--C.sub.6 H.sub.4)                                                 463 3-(3'-NC--C.sub.6 H.sub.4)                                                 464 3-(4'-NC--C.sub.6 H.sub.4)                                                 465 4-(2'-NC--C.sub.6 H.sub.4)                                                 466 4-(3'-NC--C.sub.6 H.sub.4)                                                 467 4-(4'-NC--C.sub.6 H.sub.4)                                                 468 2-(2'-CF.sub.3 --C.sub.6 H.sub.4)                                          469 2-(3'-CF.sub.3 --C.sub.6 H.sub.4)                                          470 2-(4'-CF.sub.3 --C.sub.6 H.sub.4)                                          471 3-(2'-CF.sub.3 --C.sub.6 H.sub.4)                                          472 3-(3'-CF.sub.3 --C.sub.6 H.sub.4)                                          473 3-(4'-CF.sub.3 --C.sub.6 H.sub.4)                                          474 4-(2'-CF.sub.3 --C.sub.6 H.sub.4)                                          475 4-(3'-CF.sub.3 --C.sub.6 H.sub.4)                                          476 4-(4'-CF.sub.3 --C.sub.6 H.sub.4)                                          477 2-O--C.sub.6 H.sub.5                                                       475 3-O--C6H5                                                                  476 4-O--C6H5                                                                  478 2-O-(2'-F--C6H4)                                                           479 2-O-(3'-F--C.sub.6 H.sub.4)                                                480 2-O-(4'-F--C.sub.6 H.sub.4)                                                481 3-O-(2'-F--C.sub.6 H.sub.4)                                                482 3-O-(3'-F--C.sub.6 H.sub.4)                                                483 3-O-(4'-F--C.sub.6 H.sub.4)                                                484 4-O-(2'-F--C.sub.6 H.sub.4)                                                485 4-O-(3'-F--C.sub.6 H.sub.4)                                                486 4-O-(4'-F--C.sub.6 H.sub.4)                                                487 2-O-(2'-Cl--C.sub.6 H.sub.4)                                               488 2-O-(3'-Cl--C.sub.6 H.sub.4)                                               489 2-O-(4'-Cl--C.sub.6 H.sub.4)                                               490 3-O-(2'-Cl--C.sub.6 H.sub.4)                                               491 3-O-(3'-Cl--C.sub.6 H.sub.4)                                               492 3-O-(4'-Cl--C.sub.6 H.sub.4)                                               493 3-O-(4'-Cl--C.sub.6 H.sub.4)                                               494 4-O-(2'-Cl--C.sub.6 H.sub.4)                                               495 4-O-(3'-Cl--C.sub.6 H.sub.4)                                               496 4-O-(4'-Cl--C.sub.6 H.sub.4)                                               497 2-O-(2'-CH.sub.3 --C.sub.6 H.sub.4)                                        498 2-O-(3'-CH.sub.3 --C.sub.6 H.sub.4)                                        499 2-O-(4'-CH.sub.3 --C.sub.6 H.sub.4)                                        500 3-O-(2'-CH.sub.3 --C.sub.6 H.sub.4)                                        501 3-O-(3'-CH.sub.3 --C.sub.6 H.sub.4)                                        502 3-O-(4'-CH.sub.3 --C.sub.6 H.sub.4)                                        503 4-O-(2'-CH.sub.3 --C.sub.6 H.sub.4)                                        504 4-O-(3'-CH.sub.3 --C.sub.6 H.sub.4)                                        505 4-O-(4'-CH.sub.3 --C.sub.6 H.sub.4)                                        506 2-O-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                    507 2-O-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                    508 2-O-(4'-CH3--CO--C6H4)                                                     509 3-O-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                    510 3-O-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                    511 3-O-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                    512 4-O-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                    513 4-O-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                    514 4-O-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                    515 2-O-(2'-(CH.sub.3 --C(═NOAllyl))-C.sub.6 H.sub.4)                      516 2-O-(3'-(CH.sub.3 --C(═NOAllyl))-C.sub.6 H.sub.4)                      517 2-O-(4'-(CH.sub.3 --C(═NOAllyl))-C.sub.6 H.sub.4)                      518 3-O-(2'-(CH.sub.3 --C(═NOAllyl))-C.sub.6 H.sub.4)                      519 3-O-(3'-(CH.sub.3 --C(═NOAllyl))-C.sub.6 H.sub.4)                      520 3-O-(4'-(CH.sub.3 --C(═NOAllyl))-C.sub.6 H.sub.4)                      521 4-O-(2'-(CH.sub.3 --C(═NOAllyl))-C.sub.6 H.sub.4)                      522 4-O-(3'-(CH.sub.3 --C(═NOAllyl))-C.sub.6 H.sub.4)                      523 4-O-(4'-(CH.sub.3 --C(═NOAllyl))-C.sub.6 H.sub.4)                      524 2-O-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                               525 2-O-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                               526 2-O-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                               527 3-O-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                               528 3-O-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                               529 3-O-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                               530 4-O-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                               531 4-O-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                               532 4-O-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                               533 2-O-(2'-CH.sub.3 O--C.sub.6 H.sub.4)                                       534 2-O-(3'-CH.sub.3 O--C.sub.6 H.sub.4)                                       535 2-O-(4'-CH.sub.3 O--C.sub.6 H.sub.4)                                       536 3-O-(2'-CH.sub.3 O--C.sub.6 H.sub.4)                                       537 3-O-(3'-CH.sub.3 O--C.sub.6 H.sub.4)                                       538 3-O-(4'-CH.sub.3 O--C.sub.6 H.sub.4)                                       539 4-O-(2'-CH.sub.3 O--C.sub.6 H.sub.4)                                       540 4-O-(3'-CH.sub.3 O--C.sub.6 H.sub.4)                                       541 4-O-(4'-CH.sub.3 O--C.sub.6 H.sub.4)                                       542 2-O-(2'-O.sub.2 N--C.sub.6 H.sub.4)                                        543 2-O-(3'-O.sub.2 N--C.sub.6 H.sub.4)                                        544 2-O-(4'-O.sub.2 N--C.sub.6 H.sub.4)                                        545 3-O-(2'-O2N--C6H4)                                                         546 3-O-(3'-O.sub.2 N--C.sub.6 H.sub.4)                                        547 3-O-(4'-O.sub.2 N--C.sub.6 H.sub.4)                                        548 4-O-(2'-O.sub.2 N--C.sub.6 H.sub.4)                                        549 4-O-(3'-O.sub.2 N--C.sub.6 H.sub.4)                                        550 4-O-(4'-O.sub.2 N--C.sub.6 H.sub.4)                                        551 2-O-(2'-NC--C.sub.6 H.sub.4)                                               552 2-O-(3'-NC--C.sub.6 H.sub.4)                                               553 2-O-(4'-NC--C.sub.6 H.sub.4)                                               554 3-O-(2'-NC--C.sub.6 H.sub.4)                                               555 3-O-(3'-NC--C.sub.6 H.sub.4)                                               556 3-O-(4'-NC--C.sub.6 H.sub.4)                                               557 4-O-(2'-NC--C.sub.6 H.sub.4)                                               558 4-O-(3'-NC--C.sub.6 H.sub.4)                                               559 4-O-(4'-NC--C.sub.6 H.sub.4)                                               560 2-O-(2'-CF.sub.3 --C.sub.6 H.sub.4)                                        561 2-O-(3'-CF.sub.3 --C.sub.6 H.sub.4)                                        562 2-O-(4'-CF.sub.3 --C.sub.6 H.sub.4)                                        563 3-O-(2'-CF.sub.3 --C.sub.6 H.sub.4)                                        564 3-O-(3'-CF.sub.3 --C.sub.6 H.sub.4)                                        565 3-O-(4'-CF.sub.3 --C.sub.6 H.sub.4)                                        566 4-O-(2'-CF.sub.3 --C.sub.6 H.sub.4)                                        567 4-O-(3'-CF.sub.3 --C.sub.6 H.sub.4)                                        568 4-O-(4'-CF.sub.3 --C.sub.6 H.sub.4)                                        569 2-Pyridinyl-2'                                                             570 2-Pyridinyl-3'                                                             571 2-Pyridinyl-4'                                                             572 3-Pyridinyl-2'                                                             573 3-Pyridinyl-3'                                                             574 3-Pyridinyl-4'                                                             575 4-Pyridinyl-2'                                                             576 4-Pyridinyl-3'                                                             577 4-Pyridinyl-4'                                                             578 2-Pyrimidinyl-2'                                                           579 2-Pyrimidinyl-3'                                                           580 2-Pyrimidinyl-4'                                                           581 3-Pyrimidinyl-2'                                                           582 3-Pyrimidinyl-3'                                                           583 3-Pyrimidinyl-4'                                                           584 4-Pyrimidinyl-2'                                                           585 4-Pyrimidinyl-3'                                                           586 4-Pyrimidinyl-4'                                                           587 2-Pyrazolyl-1'                                                             588 2-Pyrazolyl-3'                                                             589 2-Pyrazolyl-4'                                                             590 3-Pyrazolyl-1'                                                             591 3-Pyrazolyl-3'                                                             592 3-Pyrazolyl-4'                                                             593 4-Pyrazolyl-1'                                                             594 4-Pyrazolyl-3'                                                             595 4-Pyrazolyl-4'                                                             596 2-Isoxazolyl-3'                                                            597 2-Isoxazolyl-4'                                                            598 2-Isoxazolyl-5'                                                            599 3-Isoxazolyl-3'                                                            600 3-Isoxazolyl-4'                                                            601 3-Isoxazolyl-5'                                                            602 4-Isoxazolyl-3'                                                            603 4-Isoxazolyl-4'                                                            604 4-Isoxazolyl-5'                                                            605 2-Isothiazolyl-3'                                                          606 2-Isothiazolyl-4'                                                          607 2-Isothiazolyl-5'                                                          608 3-Isothiazolyl-3'                                                          609 3-Isothiazolyl-4'                                                          610 3-Isothiazolyl-5'                                                          611 4-Isothiazolyl-3'                                                          612 4-Isothiazolyl-4'                                                          613 4-Isothiazolyl-5'                                                          614 2-Imidazolyl-1'                                                            615 2-Imidazolyl-2'                                                            616 2-Imidazolyl-4'                                                            617 3-Imidazolyl-1'                                                            618 3-Imidazolyl-2'                                                            619 3-Imidazolyl-4'                                                            620 4-Imidazolyl-1'                                                            621 4-Imidazolyl-2'                                                            622 4-Imidazolyl-4'                                                            623 2-Oxazolyl-2'                                                              624 2-Oxazolyl-4'                                                              625 2-Oxazolyl-5'                                                              626 3-Oxazolyl-2'                                                              627 3-Oxazolyl-4'                                                              628 3-Oxazolyl-5'                                                              629 4-Oxazolyl-2'                                                              630 4-Oxazolyl-4'                                                              631 4-Oxazolyl-5'                                                              632 2-Thiazolyl-2'                                                             633 2-Thiazolyl-4'                                                             634 2-Thiazolyl-5'                                                             635 3-Thiazolyl-2'                                                             636 3-Thiazolyl-4'                                                             637 3-Thiazolyl-5'                                                             638 4-Thiazolyl-2'                                                             639 4-Thiazolyl-4'                                                             640 4-Thiazolyl-5'                                                           ______________________________________                                    

                  TABLE 20                                                         ______________________________________                                         1  STR223##                                                                       - I: R.sup.1 = CH.sub.3, Z = CH.sub.3 II: R.sup.1 = CH.sub.2 --CH.sub.3     , Z = CH.sub.3 III: R.sup.1 = CH.sub.3, Z = C.sub.2 H.sub.5 IV: R.sup.1 =      CH.sub.2 --CH.sub.3, Z = C.sub.2 H.sub.5 V: R.sup.1 = CH.sub.3, Z =            NHCH.sub.3 VI: R.sup.1 = CH.sub.2 --CH.sub.3, Z = NHCH.sub.3                     No.        B                                                                 ______________________________________                                         1        Pyrrolyl-3                                                              2 N-CH.sub.3 -Pyrrolyl-3                                                       3 N-C.sub.6 H.sub.5 -Pyrrolyl-3                                                4 N-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrrolyl-3                                 5 N-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrrolyl-3                                 6 N-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrrolyl-3                                 7 N-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrrolyl-3                                8 N-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrrolyl-3                                9 N-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrrolyl-3                                10 N-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrrolyl-3                                11 N-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrrolyl-3                                12 N-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrrolyl-3                                13 N-(4'-CN--C.sub.6 H.sub.4)-Pyrrolyl-3                                       14 N-(3'-CN--C.sub.6 H.sub.4)-Pyrrolyl-3                                       15 N-(2'-CN--C.sub.6 H.sub.4)-Pyrrolyl-3                                       16 N-(4'-Cl--C.sub.6 H.sub.4)-Pyrrolyl-3                                       17 N-(3'-Cl--C.sub.6 H.sub.4)-Pyrrolyl-3                                       18 N-(2'-Cl--C.sub.6 H.sub.4)-Pyrrolyl-3                                       19 Pyrrolyl-2                                                                  20 N-CH.sub.3 -Pyrrolyl-2                                                      21 N-C.sub.6 H.sub.5 -Pyrrolyl-2                                               22 N-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrrolyl-2                                23 N-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrrolyl-2                                24 N-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrrolyl-2                                25 N-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrrolyl-2                               26 N-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrrolyl-2                               27 N-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrrolyl-2                               28 N-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrrolyl-2                                29 N-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrrolyl-2                                30 N-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrrolyl-2                                31 N-(4'-CN--C.sub.6 H.sub.4)-Pyrrolyl-2                                       32 N-(3'-CN--C.sub.6 H.sub.4)-Pyrrolyl-2                                       33 N-(2'-CN--C.sub.6 H.sub.4)-Pyrrolyl-2                                       34 N-(4'-Cl--C.sub.6 H.sub.4)-Pyrrolyl-2                                       35 N-(3'-Cl--C.sub.6 H.sub.4)-Pyrrolyl-2                                       36 N-(2'-Cl--C.sub.6 H.sub.4)-Pyrrolyl-2                                       37 Furyl-2                                                                     38 5-CH.sub.3 -Furyl-2                                                         39 5-C.sub.6 H.sub.5 -Furyl-2                                                  40 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Furyl-2                                   41 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Furyl-2                                   42 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Furyl-2                                   43 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Furyl-2                                  44 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Furyl-2                                  45 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Furyl-2                                  46 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Furyl-2                                   47 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Furyl-2                                   48 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Furyl-2                                   49 5-(4'-CN--C.sub.6 H.sub.4)-Furyl-2                                          50 5-(3'-CN--C.sub.6 H.sub.4)-Furyl-2                                          51 5-(2'-CN--C.sub.6 H.sub.4)-Furyl-2                                          52 5-(4'-Cl--C.sub.6 H.sub.4)-Furyl-2                                          53 5-(3'-Cl--C.sub.6 H.sub.4)-Furyl-2                                          54 5-(2'-Cl--C.sub.6 H.sub.4)-Furyl-2                                          55 4-CH.sub.3 -Furyl-2                                                         56 4-C.sub.6 H.sub.5 -Furyl-2                                                  57 4-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Furyl-2                                   58 4-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Furyl-2                                   59 4-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Furyl-2                                   60 4-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Furyl-2                                  61 4-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Furyl-2                                  62 4-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Furyl-2                                  63 4-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Furyl-2                                   64 4-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Furyl-2                                   65 4-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Furyl-2                                   66 4-(4'-CN--C.sub.6 H.sub.4)-Furyl-2                                          67 4-(3'-CN--C.sub.6 H.sub.4)-Furyl-2                                          68 4-(2'-CN--C.sub.6 H.sub.4)-Furyl-2                                          69 4-(4'-Cl--C.sub.6 H.sub.4)-Furyl-2                                          70 4-(3'-Cl--C.sub.6 H.sub.4)-Furyl-2                                          71 4-(2'-Cl--C.sub.6 H.sub.4)-Furyl-2                                          72 Thienyl-2                                                                   73 5-CH.sub.3 -Thienyl-2                                                       74 5-C.sub.6 H.sub.5 -Thienyl-2                                                75 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-2                                 76 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-2                                 77 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-2                                 78 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-2                                79 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-2                                80 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-2                                81 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-2                                 82 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-2                                 83 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-2                                 84 5-(4'-CN--C.sub.6 H.sub.4)-Thienyl-2                                        85 5-(3'-CN--C.sub.6 H.sub.4)-Thienyl-2                                        86 5-(2'-CN--C.sub.6 H.sub.4)-Thienyl-2                                        87 5-(4'-Cl--C.sub.6 H.sub.4)-Thienyl-2                                        88 5-(3'-Cl--C.sub.6 H.sub.4)-Thienyl-2                                        89 5-(2'-Cl--C.sub.6 H.sub.4)-Thienyl-2                                        90 4-CH.sub.3 -Thienyl-2                                                       91 4-C.sub.6 H.sub.5 -Thienyl-2                                                92 4-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-2                                 93 4-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-2                                 94 4-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-2                                 95 4-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-2                                96 4-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-2                                97 4-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-2                                98 4-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-2                                 99 4-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-2                                 100 4-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-2                                101 4-(4'-CN--C.sub.6 H.sub.4)-Thienyl-2                                       102 4-(3'-CN--C.sub.6 H.sub.4)-Thienyl-2                                       103 4-(2'-CN--C.sub.6 H.sub.4)-Thienyl-2                                       104 4-(4'-Cl--C.sub.6 H.sub.4)-Thienyl-2                                       105 4-(3'-Cl--C.sub.6 H.sub.4)-Thienyl-2                                       106 4-(2'-Cl--C.sub.6 H.sub.4)-Thienyl-2                                       107 Thienyl-3                                                                  108 5-CH.sub.3 -Thienyl-3                                                      109 5-C.sub.6 H.sub.5 -Thienyl-3                                               110 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-3                                111 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-3                                112 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-3                                113 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-3                               114 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-3                               115 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-3                               116 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-3                                117 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-3                                118 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-3                                119 5-(4'-CN--C.sub.6 H.sub.4)-Thienyl-3                                       120 5-(3'-CN--C.sub.6 H.sub.4)-Thienyl-3                                       121 5-(2'-CN--C.sub.6 H.sub.4)-Thienyl-3                                       122 5-(4'-Cl--C.sub.6 H.sub.4)-Thienyl-3                                       123 5-(3'-Cl--C.sub.6 H.sub.4)-Thienyl-3                                       124 5-(2'-Cl--C.sub.6 H.sub.4)-Thienyl-3                                       125 Pyrazolyl-4                                                                126 N-CH.sub.3 -Pyrazolyl-4                                                    127 N-C.sub.6 H.sub.5 -Pyrazolyl-4                                             128 N-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrazolyl-4                              129 N-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrazolyl-4                              130 N-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrazolyl-4                              131 N-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrazolyl-4                             132 N-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrazolyl-4                             133 N-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrazolyl-4                             134 N-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrazolyl-4                              135 N-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrazolyl-4                              136 N-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrazolyl-4                              137 N-(4'-CN--C.sub.6 H.sub.4)-Pyrazolyl-4                                     138 N-(3'-CN--C.sub.6 H.sub.4)-Pyrazolyl-4                                     139 N-(2'-CN--C.sub.6 H.sub.4)-Pyrazolyl-4                                     140 N-(4'-Cl--C.sub.6 H.sub.4)-Pyrazolyl-4                                     141 N-(3'-Cl--C.sub.6 H.sub.4)-Pyrazolyl-4                                     142 N-(2'-Cl--C.sub.6 H.sub.4)-Pyrazolyl-4                                     143 3-CH.sub.3 --N-Methylpyrazolyl-4                                           144 3-C.sub.6 H.sub.5 --N-Methylpyrazolyl-4                                    145 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)-N-Methylpyrazolyl-4                      146 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)-N-Methylpyrazolyl-4                      147 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)-N-Methylpyrazolyl-4                      148 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-N-Methylpyrazolyl-4                     149 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-N-Methylpyrazolyl-4                     150 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-N-Methylpyrazolyl-4                     151 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)-N-Methylpyrazolyl-4                      152 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)-N-Methylpyrazolyl-4                      153 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)-N-Methylpyrazolyl-4                      154 3-(4'-CN--C.sub.6 H.sub.4)-N-Methylpyrazolyl-4                             155 3-(3'-CN--C.sub.6 H.sub.4)-N-Methylpyrazolyl-4                             156 3-(2'-CN--C.sub.6 H.sub.4)-N-Methylpyrazolyl-4                             157 3-(4'-Cl--C.sub.6 H.sub.4)-N-Methylpyrazolyl-4                             158 3 (3'-Cl--C.sub.6 H.sub.4)-N-Methylpyrazolyl-4                             159 3-(2'-Cl--C.sub.6 H.sub.4)-N-Methylpyrazolyl-4                             160 Isoxazolyl-5                                                               161 3-CH.sub.3 -Isoxazolyl-5                                                   162 3-C.sub.6 H.sub.5 -Isoxazolyl-5                                            163 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Isoxazolyl-5                             164 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Isoxazolyl-5                             165 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Isoxazolyl-5                             166 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Isoxazolyl-5                            167 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Isoxazolyl-5                            168 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4) Isoxazolyl-5                            169 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Isoxazolyl-5                             170 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Isoxazolyl-5                             171 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Isoxazolyl-5                             172 3-(4'-CN--C.sub.6 H.sub.4)-Isoxazolyl-5                                    173 3-(3'-CN--C.sub.6 H.sub.4)-Isoxazolyl-5                                    174 3-(2'-CN--C.sub.6 H.sub.4)-Isoxazolyl-5                                    175 3-(4'-Cl--C.sub.6 H.sub.4)-Isoxazolyl-5                                    176 3-(3'-Cl--C.sub.6 H.sub.4)-Isoxazolyl-5                                    177 3-(2'-Cl--C.sub.6 H.sub.4)-Isoxazolyl-5                                    178 4-Chloroisoxazolyl-5                                                       179 3-CH.sub.3 -4-Chloroisoxazolyl-5                                           180 3-C.sub.6 H.sub.5 -4-Chloroisoxazolyl-5                                    181 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                     182 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                     183 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                     184 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                    185 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                    186 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                    187 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                     188 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                     189 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)-4-Chlorpisoxazolyl-5                     190 3-(4'-CN--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                            191 3-(3'-CN--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                            192 3-(2'-CN--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                            193 3-(4'-Cl--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                            194 3-(3'-Cl--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                            195 3-(2'-Cl--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                            196 Isoxazolyl-3                                                               197 5-CH.sub.3 -Isoxazolyl-3                                                   198 5-C.sub.6 H.sub.5 -Isoxazolyl-3                                            199 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Isoxazolyl-3                             200 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Isoxazolyl-3                             201 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Isoxazolyl-3                             202 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Isoxazolyl-3                            203 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Isoxazolyl-3                            204 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Isoxazolyl-3                            205 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Isoxazolyl-3                             206 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Isoxazolyl-3                             207 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Isoxazolyl-3                             208 5-(4'-CN--C.sub.6 H.sub.4)-Isoxazolyl-3                                    209 5-(3'-CN--C.sub.6 H.sub.4)-Isoxazolyl-3                                    210 5-(2'-CN--C.sub.6 H.sub.4)-Isoxazolyl-3                                    211 5-(4'-Cl--C.sub.6 H.sub.4)-Isoxazolyl-3                                    212 5-(3'-Cl--C.sub.6 H.sub.4)-Isoxazolyl-3                                    213 5-(2'-Cl--C.sub.6 H.sub.4)-Isoxazolyl-3                                    214 Isothiazolyl-5                                                             215 3-CH.sub.3 -Isothiazolyl-5                                                 216 3-C.sub.6 H.sub.5 -Isothiazolyl-5                                          217 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Isothiazolyl-5                           218 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Isothiazolyl-5                           219 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Isothiazolyl-5                           220 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Isothiazolyl-5                          221 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Isothiazolyl-5                          222 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Isothiazolyl-5                          223 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Isothiazolyl-5                           224 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Isothiazolyl-5                           225 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Isothiazolyl-5                           226 3-(4'-CN--C.sub.6 H.sub.4)-Isothiazolyl-5                                  227 3-(3'-CN--C.sub.6 H.sub.4)-Isothiazolyl-5                                  228 3-(2'-CN--C.sub.6 H.sub.4)-Isothiazolyl-5                                  229 3-(4'-Cl--C.sub.6 H.sub.4)-Isothiazolyl-5                                  230 3-(3'-Cl--C.sub.6 H.sub.4)-Isothiazolyl-5                                  231 3-(2'-Cl--C.sub.6 H.sub.4)-Isothiazolyl-5                                  232 Oxazolyl-4                                                                 233 2-CH.sub.3 -Oxazolyl-4                                                     234 2-C.sub.6 H.sub.5 -Oxazolyl-4                                              235 2-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Oxazolyl-4                               236 2-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Oxazolyl-4                               237 2-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Oxazolyl-4                               238 2-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Oxazolyl-4                              239 2-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Oxazolyl-4                              240 2-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Oxazolyl-4                              241 2-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Oxazolyl-4                               242 2-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Oxazolyl-4                               243 2-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Oxazolyl-4                               244 2-(4'-CN--C.sub.6 H.sub.4)-Oxazolyl-4                                      245 2-(3'-CN--C.sub.6 H.sub.4)-Oxazolyl-4                                      246 2-(2'-CN--C.sub.6 H.sub.4)-Oxazolyl-4                                      247 2-(4'-Cl--C.sub.6 H.sub.4)-Oxazolyl-4                                      248 2-(3'-Cl--C.sub.6 H.sub.4)-Oxazolyl-4                                      249 2-(2'-Cl--C.sub.6 H.sub.4)-Oxazolyl-4                                      250 Thiazolyl-4                                                                251 2-CH.sub.3 -Thiazolyl-4                                                    252 2-C.sub.6 H.sub.5 -Thiazolyl-4                                             253 2-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Thiazolyl-4                              254 2-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Thiazolyl-4                              255 2-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Thiazolyl-4                              256 2-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Thiazolyl-4                             267 2-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Thiazolyl-4                             258 2-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Thiazolyl-4                             259 2-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Thiazolyl-4                              260 2-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Thiazolyl-4                              261 2-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Thiazolyl-4                              262 2-(4'-CN--C.sub.6 H.sub.4)-Thiazolyl-4                                     263 2-(3'-CN--C.sub.6 H.sub.4)-Thiazolyl-4                                     264 2-(2'-CN--C.sub.6 H.sub.4)-Thiazolyl-4                                     265 2-(4'-Cl--C.sub.6 H.sub.4)-Thiazolyl-4                                     266 2-(3'-Cl--C.sub.6 H.sub.4)-Thiazolyl-4                                     267 2-(2'-Cl--C.sub.6 H.sub.4)-Thiazolyl-4                                     268 N--CH.sub.3 -1,2,4-Triazolyl-5                                             269 3-CH.sub.3 --N--CH.sub.3 -1,2,4-Triazolyl-5                                270 3-C.sub.6 H.sub.5 --N--CH.sub.3 -1,2,4-Triazolyl-5                         271 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)-N--CH.sub.3 -1,2,4-Triazolyl-5                   272 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)-N--CH.sub.3 -1,2,4-Triazol              yl-5                                                                    273 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)-N--CH.sub.3 -1,2,4-Triazolyl-5                   274 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-N--CH.sub.3 -1,2,4-Triazo              lyl-5                                                                   275 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-N--CH.sub.3 -1,2,4-Triazolyl-5                  276 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-N--CH.sub.3 -1,2,4-Triazo              lyl-5                                                                   277 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)-N--CH.sub.3 -1,2,4-Triazolyl-5                   278 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)-N--CH.sub.3 -1,2,4-Triazol              yl-5                                                                    279 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)-N--CH.sub.3 -1,2,4-Triazolyl-5                   280 3-(4'-CN--C.sub.6 H.sub.4)-N--CH.sub.3 -1,2,4-Triazolyl-5                  281 3-(3'-CN--C.sub.6 H.sub.4)-N--CH.sub.3 -1,2,4-Triazolyl-5                  282 3-(2'-CN--C.sub.6 H.sub.4)-N--CH.sub.3 -1,2,4-Triazolyl-5                  283 3-(4'-Cl--C.sub.6 H.sub.4)-N--CH.sub.3 -1,2,4-Triazolyl-5                  284 3-(3'-Cl--C.sub.6 H.sub.4)-N--CH.sub.3 -1,2,4-Triazolyl-5                  285 3-(2'-Cl--C.sub.6 H.sub.4)-N--CH.sub.3 -1,2,4-Triazolyl-5                  286 1,3,4-Oxadiazolyl-2                                                287 5-CH.sub.3 -1,3,4-Oxadiazolyl-2                                            288 5-C.sub.6 H.sub.5 -1,2,3-Oxadiazolyl-2                                     289 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                      290 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                      291 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                      292 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                     293 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                     294 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                     295 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                      296 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                      297 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                      298 5-(4'-CN--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                             299 5-(3'-CN--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                             300 5-(2'-CN--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                             301 5-(4'-Cl--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                             302 5-(3'-Cl--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                             303 5-(2'-Cl--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                             304 1,2,4-Oxadiazolyl-3                                                        305 5-CH.sub.3 -1,2,4-Oxadiazolyl-3                                            306 5-C.sub.6 H.sub.5 -1,2,4-Oxadiazolyl-3                                     307 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                      308 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                      309 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                      310 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                     311 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                     312 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                     313 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                      314 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                      315 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                      316 5-(4'-CN--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                             317 5-(3'-CN--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                             318 5-(2'-CN--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                             319 5-(4'-Cl--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                             320 5-(3'-Cl--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                             321 5-(2'-Cl--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                             322 1,2,4-Oxadiazolyl-5                                                        323 3-CH.sub.3 -1,2,4-Oxadiazolyl-5                                            324 3-C.sub.6 H.sub.5 -1,2,4-Oxadiazolyl-5                                     325 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                      326 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                      327 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                      328 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                     329 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                     330 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                     331 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                      332 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                      333 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                      334 3-(4'-CN--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                             335 3-(3'-CN--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                             336 3-(2'-CN--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                             337 3-(4'-Cl--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                             338 3-(3'-Cl--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                             339 3-(2'-Cl--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                             340 1,2,4-Thiadiazolyl-3                                                       341 5-CH.sub.3 -1,2,4-Thiadiazolyl-3                                           342 5-C.sub.6 H.sub.5 -1,2,4-Thiadiazolyl-3                                    343 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                     344 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                     345 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                     346 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                    347 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                    348 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                    349 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                     350 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                     351 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                     352 5-(4'-CN--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                            353 5-(3'-CN--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                            354 5-(2'-CN--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                            355 5-(4'-Cl--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                            356 5-(3'-Cl--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                            357 5-(2'-Cl--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                            358 1,3,4-Thiadiazolyl-2                                                       359 5-CH.sub.3 -1,3,4-Thiadiazolyl-2                                           360 5-C.sub.6 H.sub.5 1,3,4-Thiadiazolyl-2                                     361 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                     362 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                     363 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                     364 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                    365 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                    366 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                    367 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                     368 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                     369 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                     370 5-(4'-CN--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                            371 5-(3'-CN--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                            372 5-(2'-CN--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                            373 5-(4'-Cl--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                            374 5-(3'-Cl--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                            375 5-(2'-Cl--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                            376 Pyridinyl-2                                                                377 Pyridinyl-4                                                                378 Pyridazinyl-3                                                              379 Pyridazinyl-4                                                              380 Pyridazinyl-2                                                              381 Pyrimidinyl-4                                                              382 Pyrimidinyl-5                                                              383 Pyrimidinyl-2                                                              384 Pyridinyl-3                                                              ______________________________________                                    

                                      TABLE 21                                     __________________________________________________________________________     Selected physical data of some compounds                                       No.                                                                               Compound                    .sup.1 H--NMR (ppm)                                                                     m.p.                                   __________________________________________________________________________       1                                                                                                                    2  3,7(s, broad, 3H); 1,2(s,                                                   broad, 3H)                                - 2                                                                                                                 3  3,75(s, 3H): 1,2(t, 3H)                                                       - 3                                                                          4  3,7(s, 3H); 1,2(t, 3H)                                                        - 4                                                                          5  3,95(s, 3H); 3,7(s, 3H);                                                    1,2(t, 3H)                                - 5                                                                                                                 6  3,6(s, 3H); 2,9(d, 3H)                                                        - 6                                                                          7   123 9##                               - 7                                                                                                                 8   118 0##                               - 8                                                                                                                 9  3.7(s, 3H); 2.55 (s, very                                                   broad, 2H)                             __________________________________________________________________________

                  TABLE 56                                                         ______________________________________                                         Selected physical data of some compounds                                       0  STR232##                                                                       -                             .sup.1 H--NMR (ppm) or                          No. X.sub.m mp (° C.) IR (cm.sup.-1)                                  ______________________________________                                         1    H                90                                                         2 2-CH.sub.3 80                                                                3 2,5-(CH.sub.3).sub.2 101                                                     4 2-CH.sub.3 -4-C(CH.sub.3)═N--OCH.sub.3  3.95(s, 3H); 3.65(s,                                              3H); 2.9(d, 3H)                               5 2,5-(CH.sub.3).sub.2 -4-C(CH.sub.3)═N--  3.65(s, 3H); 2.9(d,                                            O-Allyl  3H)                                  ______________________________________                                    

                  TABLE 22                                                         ______________________________________                                         1  STR233##                                                                      No.       X        Z        A                                                ______________________________________                                         1       H        CH.sub.3   --CH.sub.2 O--                                       2 H CH.sub.3 --CH.sub.2 O--N═C(CH.sub.3)--                                 3 H CH.sub.3 --CH═CH--                                                     4 H NH.sub.2 --CH.sub.2 O--                                                    5 H NH.sub.2 --CH.sub.2 O--N═C(CH.sub.3)--                                 6 H NH.sub.2 --CH═CH--                                                     7 H N(CH.sub.3).sub.2 --CH.sub.2 O--                                           8 H N(CH.sub.3).sub.2 --CH.sub.2 O--N═C(CH.sub.3)--                        9 H N(CH.sub.3).sub.2 --CH═CH--                                            10 H CCl.sub.3 --CH.sub.2 O--                                                  11 H CCl.sub.3 --CH.sub.2 O--N═C(CH.sub.3)--                               12 H CCl.sub.3 --CH═CH--                                                   13 H CF.sub.3 --CH.sub.2 O--                                                   14 H CF.sub.3 --CH.sub.2 O--N═C(CH.sub.3)--                                15 H CF.sub.3 --CH═CH--                                                    16 CH.sub.3 CH.sub.3 --CH.sub.2 O--                                            17 CH.sub.3 CH.sub.3 --CH.sub.2 O--N═C(CH.sub.3)--                         18 CH.sub.3 CH.sub.3 --CH═CH--                                             19 CH.sub.3 NH.sub.2 --CH.sub.2 O--                                            20 CH.sub.3 NH.sub.2 --CH.sub.2 O--N═C(CH.sub.3)--                         21 CH.sub.3 NH.sub.2 --CH═CH--                                             22 CH.sub.3 N(CH.sub.3).sub.2 --CH.sub.2 O--                                   23 CH.sub.3 N(CH.sub.3).sub.2 --CH.sub.2 O--N═C(CH.sub.3)--                                           24 CH.sub.3 N(CH.sub.3).sub.2 --CH═CH--                                    25 CH.sub.3 CCl.sub.3 --CH.sub.2 O--                                           26 CH.sub.3 CCl.sub.3 --CH.sub.2 O--N═C(C                                 H.sub.3)--                                           27 CH.sub.3 CCl.sub.3 --CH═CH--                                            28 CH.sub.3 CF.sub.3 --CH.sub.2 O--                                            29 CH.sub.3 CF.sub.3 --CH.sub.2 O--N═C(CH.sub.3)--                         30 CH.sub.3 CF.sub.3 --CH═CH--                                             31 Cl CH.sub.3 --CH.sub.2 O--                                                  32 Cl CH.sub.3 --CH.sub.2 O--N--C(CH.sub.3)--                                  33 Cl CH.sub.3 --CH═CH--                                                   34 Cl NH.sub.2 --CH.sub.2 O--                                                  35 Cl NH.sub.2 --CH.sub.2 O--N═C(CH.sub.3)--                               36 Cl NH.sub.2 --CH═CH--                                                   37 Cl N(CH.sub.3).sub.2 --CH.sub.2 O--                                         38 Cl N(CH.sub.3).sub.2 --CH.sub.2 O--N═C(CH.sub.3)--                      39 Cl N(CH.sub.3).sub.2 --CH═CH--                                          40 Cl CCl.sub.3 --CH.sub.2 O--                                                 41 Cl CCl.sub.3 --CH.sub.2 O--N═C(CH.sub.3)--                              42 Cl CCl.sub.3 --CH═CH--                                                  43 Cl CF.sub.3 --CH.sub.2 O--                                                  44 Cl CF.sub.3 --CH.sub.2 O--N═C(CH.sub.3)--                               45 Cl CF.sub.3 --CH═CH--                                                 ______________________________________                                    

                  TABLE 23                                                         ______________________________________                                         2  STR234##                                                                       - I: R.sup.1 = CH.sub.3, Z = CH.sub.3 II: R.sup.1 = CH.sub.2 --CH.sub.3     ,Z = CH.sub.3 III: R.sup.1 = CH.sub.3, Z = C.sub.2 H.sub.5 IV: R.sup.1 =       CH.sub.2 --CH.sub.3, Z = C.sub.2 H.sub.5 V: R.sup.1 = CH.sub.3, Z =            NHCH.sub.3 VI: R.sup.1 = CH.sub.2 --CH.sub.3, Z = NHCH.sub.3                     No.             B                                                            ______________________________________                                         1             2-Pyridyl                                                          2 3-Trifluoromethyl-2-pyridyl                                                  3 5-Trifluoromethyl-2-pyridyl                                                  4 3,5-Bis-(trifluoromethyl)-2-pyridyl                                          5 3,5-Dichloro-2-pyridyl                                                       6 3-Chloro-5-trifluoromethyl-2-pyridyl                                         7 3,5-Dichloro-2-pyridyl                                                       8 2-Chloro-4-trifluormethylphenyl                                              9 2-Benzothiazolyl                                                             10 5-Chloro-4-methyl-2-benzimidazolyl                                          11 2-Benzoxazolyl                                                              12 1-Methyl-5-trifluoromethylimi-                                               dazo[5,4-a]-pyridin-2-yl                                                      13 5-Chloro-2-pyrimidinyl                                                      14 4-Methyl-5-phenyl-2-thiazolin-2-yl                                          15 4-Methyl-5-phenyl-2-oxazolin-2-yl                                           16 7-Trifluoromethyl-4-quinolinyl                                            ______________________________________                                    

Example 10

N-(2,6-Dimethylphenyl)-N-methoxycarbonyl-O-methyl-hydroxylamine (Table 30, No. 1)

a) N-(2,6-Dimethylphenyl)-N-methoxycarbonyl-hydroxylamine

At 0 to 5° C., 7.0 g (70 mmol) of methyl chloroformate is added dropwise to 11.3 g (80 mmol) of N-2,6-dimethylphenyl-hydroxylamine (prepared analogously to Bamberger et al., Ann. Chem. 316 (1901), 278) and 12.5 g (90 mmol) of K₂ CO₃ in 30 ml of methylene chloride. The mixture is stirred for 30 mins at 0-5° C., the insoluble solid is filtered off and the filtrate is evaporated down under reduced pressure. The residue is purified by column chromatography with mixtures of cyclohexand and ethyl acetate. There is obtained 1.4 g (7.2 mmol=9%) of the title compound as a dark oil.

¹ H-NMR (CDCl₃ ; δ in ppm): 8.85 (s, broad, 1H, OH); 7.1 (m, 3H, phenyl); 3.75 (s, 3H, OCH₃); 2.3 (s, 6H, 2×CH₃)

b) N-(2,6-Dimethylphenyl)-N-methoxycarbonyl-O-methylhydroxylamine (Table 7, No. 1)

A mixture of 1.4 g (7.2 mmol) of N-(2,6-dimethylphenyl)-N-methoxycarbonyl-hydroxylamine (Example 1a), 1.3 g (9 mmol) of K₂ CO₃ and 10 g (8 mmol) of dimethyl sulfate in 10 ml of acetone is stirred overnight at room temperature. The reaction mixture is then diluted with CH₂ Cl₂ and stirred with dilute NH₃ solution. The phases are then separated and the organic phase is extracted another twice with water. The organic phase is dried over MgSO₄ and evaporated down, and the residue is purified by column chromatography with mixtures of cyclohexane and ethyl acetate. There is obtained 1.2 g (6 mmol=83%) of the title compound as a colorless solid (mp=81° C.).

¹ H-NMR (CDCl₃ ; δ in ppm): 7.1 (m, 3H, phenyl); 3.75 (s, broad, 6H, 2×OCH₃); 2.3 (s, 3H, CH₃)

The compounds listed in the following tables may be prepared similarly. Compound I, No. 1 from Table 24, No. 1 has for example the following formula: ##STR235##

                  TABLE 24                                                         ______________________________________                                            -       a I: R.sup.1 = CH.sub.3, X = CH.sub.3                                 b II: R.sup.1 = CH.sub.2 --CH.sub.3, X = CH.sub.3                              c III: R.sup.1 = CH.sub.3, X = Cl                                              b IV: R.sup.1 = CH.sub.2 --CH.sub.3, X = Cl                                  No.     T.sub.m                                                                ______________________________________                                          1      H                                                                         2 2-F                                                                          3 3-F                                                                          4 4-F                                                                          5 2,4-F.sub.2                                                                  6 2,4,6-F.sub.3                                                                7 2,3,4,5,6-F.sub.5                                                            8 2,3-F.sub.2                                                                  9 2-Cl                                                                         10 3-Cl                                                                        11 4-Cl                                                                        12 2,3-Cl.sub.2                                                                13 2,4-Cl.sub.2                                                                14 2,5-Cl.sub.2                                                                15 2,6-Cl.sub.2                                                                16 3,4-Cl.sub.2                                                                17 3,5-Cl.sub.2                                                                18 2,3,4-Cl.sub.3                                                              19 2,3,5-Cl.sub.3                                                              20 2,3,6-Cl.sub.3                                                              21 2,4,5-Cl.sub.3                                                              22 2,4,6-Cl.sub.3                                                              23 3,4,5-Cl.sub.3                                                              24 2,3,4,6-Cl.sub.4                                                            25 2,3,5,6-Cl.sub.4                                                            26 2,3,4,5,6-Cl.sub.5                                                          27 2-Br                                                                        28 3-Br                                                                        29 4-Br                                                                        30 2,4-Br.sub.2                                                                31 2,5-Br.sub.2                                                                32 2,6-Br.sub.2                                                                33 2,4,6-Br.sub.3                                                              34 2,3,4,5,6-Br.sub.5                                                          35 2-I                                                                         36 3-I                                                                         37 4-I                                                                         38 2,4-I.sub.2                                                                 39 2-Cl, 3-F                                                                   40 2-Cl, 4-F                                                                   41 2-Cl, 5-F                                                                   42 2-Cl, 6-F                                                                   43 2-Cl, 3-Br                                                                  44 2-Cl, 4-Br                                                                  45 2-Cl, 5-Br                                                                  46 2-Cl, 6-Br                                                                  47 2-Br, 3-Cl                                                                  48 2-Br, 4-Cl                                                                  49 2-Br, 5-Cl                                                                  50 2-Br, 3-F                                                                   51 2-Br, 4-F                                                                   52 2-Br, 5-F                                                                   53 2-Br, 6-F                                                                   54 2-F, 3-Cl                                                                   55 2-F, 4-Cl                                                                   56 2-F, 5-Cl                                                                   57 3-Cl, 4-F                                                                   58 3-Cl, 5-F                                                                   59 3-Cl, 4-Br                                                                  60 3-Cl, 5-Br                                                                  61 3-F, 4-Cl                                                                   62 3-F, 4-Br                                                                   63 3-Br, 4-Cl                                                                  64 3-Br, 4-F                                                                   65 2,6-Cl.sub.2, 4-Br                                                          66 2-CH.sub.3                                                                  67 3-CH.sub.3                                                                  68 4-CH.sub.3                                                                  69 2,3-(CH.sub.3).sub.2                                                        70 2,4-(CH.sub.3).sub.2                                                        71 2,5-(CH.sub.3).sub.2                                                        72 2,6-(CH.sub.3).sub.2                                                        73 3,4-(CH.sub.3).sub.2                                                        74 3,5-(CH.sub.3).sub.2                                                        75 2,3,5-(CH.sub.3).sub.3                                                      76 2,3,4-(CH.sub.3).sub.3                                                      77 2,3,6-(CH.sub.3).sub.3                                                      78 2,4,5-(CH.sub.3).sub.3                                                      79 2,4,6-(CH.sub.3).sub.3                                                      80 3,4,5-(CH.sub.3).sub.3                                                      81 2,3,4,6-(CH.sub.3).sub.4                                                    82 2,3,5,6-(CH.sub.3).sub.4                                                    83 2,3,4,5,6-(CH.sub.3).sub.5                                                  84 2-C.sub.2 H.sub.5                                                           85 3-C.sub.2 H.sub.5                                                           86 4-C.sub.2 H.sub.5                                                           87 2,4-(C2H5).sub.2                                                            88 2,6-(C.sub.2 H.sub.5).sub.2                                                 89 3,5-(C.sub.2 H.sub.5).sub.2                                                 90 2,4,6-(C.sub.2 H.sub.5).sub.3                                               91 2-n-C.sub.3 H.sub.7                                                         92 3-n-C.sub.3 H.sub.7                                                         93 4-n-C.sub.3 H.sub.7                                                         94 2-i-C.sub.3 H.sub.7                                                         95 3-i-C.sub.3 H.sub.7                                                         96 4-i-C.sub.3 H.sub.7                                                         97 2,4-(i-C.sub.3 H.sub.7).sub.2                                               98 2,6-(i-C.sub.3 H.sub.7).sub.2                                               99 3,5-(i-C.sub.3 H.sub.7).sub.2                                              100 2,4,6-(i-C.sub.3 H.sub.7).sub.3                                            101 2-s-C.sub.4 H.sub.9                                                        102 3-s-C.sub.4 H.sub.9                                                        103 4-s-C.sub.4 H.sub.9                                                        104 2-t-C.sub.4 H.sub.9                                                        105 3-t-C.sub.4 H.sub.9                                                        106 4-t-C.sub.4 H.sub.9                                                        107 2,3-(t-C.sub.4 H.sub.9).sub.2                                              108 2,4-(t-C.sub.4 H.sub.9).sub.2                                              109 2,5-(t-C.sub.4 H.sub.9).sub.2                                              110 2,6-(t-C.sub.4 H.sub.9).sub.2                                              111 3,4-(t-C.sub.4 H.sub.9).sub.2                                              112 2,4,6-(t-C.sub.4 H.sub.9).sub.3                                            113 4-n-C.sub.9 H.sub.19                                                       114 4-n-C.sub.12 H.sub.25                                                      115 4-n-C.sub.15 H.sub.31                                                      116 4-(1,1,3,3-Tetramethylbutyl)                                               117 4-(2,4,4-Trimethylpropyl)                                                  118 2-t-C.sub.4 H.sub.9, 4-CH.sub.3                                            119 2-t-C.sub.4 H.sub.9, 5-CH.sub.3                                            120 2,6-(t-C.sub.4 H.sub.9).sub.2, 4-CH.sub.3                                  121 2-CH.sub.3, 4-t-C.sub.4 H.sub.9                                            122 2-CH.sub.3, 6-t-C.sub.4 H.sub.9                                            123 2-CH.sub.3, 4-i-C.sub.3 H.sub.7                                            124 2-CH.sub.3, 5-i-C.sub.3 H.sub.7                                            125 3-CH.sub.3, 4-i-C.sub.3 H.sub.7                                            126 2-i-C.sub.3 H.sub.7, 5-CH.sub.3                                            127 2,4-(t-C.sub.4 H.sub.9).sub.2, 6-i-C.sub.3 H.sub.7                         128 2-Allyl                                                                    129 3-Allyl                                                                    130 4-Allyl                                                                    131 2-Allyl, 6-CH.sub.3                                                        132 2-cyclo-C.sub.6 H.sub.11                                                   133 3-cyclo-C.sub.6 H.sub.11                                                   134 4-cyclo-C.sub.6 H.sub.11                                                   135 2,4-(cyclo-C.sub.6 H.sub.11).sub.2, 6-CH.sub.3                             136 2-CH.sub.3, 4-cyclo-C.sub.6 H.sub.11                                       137 2-CH.sub.2 --C.sub.6 H.sub.5                                               138 3-CH.sub.2 --C.sub.6 H.sub.5                                               139 4-CH.sub.2 --C.sub.6 H.sub.5                                               140 2-CH.sub.2 --C.sub.6 H.sub.5, 4-CH.sub.3                                   141 2-CH.sub.3, 4-CH.sub.2 --C.sub.6 H.sub.5                                   142 2-C.sub.6 H.sub.5                                                          143 3-C.sub.6 H.sub.5                                                          144 4-C.sub.6 H.sub.5                                                          145 4-(2-i-C.sub.3 H.sub.7 --C.sub.6 H.sub.4)                                  146 4-C.sub.6 H.sub.5, 2,6-(CH.sub.3).sub.2                                    147 2-Cl, 4-C.sub.6 H.sub.5                                                    148 2-Br, 4-C.sub.6 H.sub.5                                                    149 2-C.sub.6 H.sub.5, 4-Cl                                                    150 2-C.sub.6 H.sub.5, 4-Br                                                    151 2-CH.sub.2 C.sub.6 H.sub.5, 4-Cl                                           152 2-CH.sub.2 C.sub.6 H.sub.5, 4-Br                                           153 2-Cl, 4-CH.sub.2 C.sub.6 H.sub.5                                           154 2-Br, 4-CH.sub.2 C.sub.6 H.sub.5                                           155 2-cyclo-C.sub.6 H.sub.11, 4-Cl                                             156 2-cyclo-C.sub.6 H.sub.11, 4-Br                                             157 2-Cl, 4-cyclo-C.sub.6 H.sub.11                                             158 2-Br, 4-cyclo-C.sub.6 H.sub.11                                             159 2-OCH.sub.3                                                                160 3-OCH.sub.3                                                                161 4-OCH.sub.3                                                                162 2-OC.sub.2 H.sub.5                                                         163 3-O--C.sub.2 H.sub.5                                                       164 4-O--C.sub.2 H.sub.5                                                       165 2-O-n-C.sub.3 H.sub.7                                                      166 3-O-n-C.sub.3 H.sub.7                                                      167 4-O-n-C.sub.3 H.sub.7                                                      168 2-O-i-C.sub.3 H.sub.7                                                      169 3-O-i-C.sub.3 H.sub.7                                                      170 4-O-i-C.sub.3 H.sub.7                                                      171 2-O-n-C.sub.6 H.sub.13                                                     172 3-O-n-C.sub.6 H.sub.13                                                     173 4-O-n-C.sub.6 H.sub.13                                                     174 2-O-n-C.sub.8 H.sub.17                                                     175 3-O-n-C.sub.8 H.sub.17                                                     176 4-O-n-C.sub.8 H.sub.17                                                     177 2-O--CH.sub.2 C.sub.6 H.sub.5                                              178 3-O--CH.sub.2 C.sub.6 H.sub.5                                              179 4-O--CH.sub.2 C.sub.6 H.sub.5                                              180 2-O--(CH.sub.2).sub.3 C.sub.6 H.sub.5                                      181 3-O--(CH.sub.2).sub.3 C.sub.6 H.sub.5                                      182 4-O--(CH.sub.2).sub.3 C.sub.6 H.sub.5                                      183 2,4-(OCH.sub.3).sub.2                                                      184 2-CF.sub.3                                                                 185 3-CF.sub.3                                                                 186 4-CF.sub.3                                                                 187 2-OCF.sub.3                                                                188 3-OCF.sub.3                                                                189 4-OCF.sub.3                                                                190 3-OCH.sub.2 CHF.sub.2                                                      191 2-NO.sub.2                                                                 192 3-NO.sub.2                                                                 193 4-NO.sub.2                                                                 194 2-CN                                                                       195 3-CN                                                                       196 4-CN                                                                       197 2-CH.sub.3, 3-Cl                                                           198 2-CH.sub.3, 4-Cl                                                           199 2-CH.sub.3, 5-Cl                                                           200 2-CH.sub.3, 6-Cl                                                           201 2-CH.sub.3, 3-F                                                            202 2-CH.sub.3, 4-F                                                            203 2-CH.sub.3, 5-F                                                            204 2-CH.sub.3, 6-F                                                            205 2-CH.sub.3, 3-Br                                                           206 2-CH.sub.3, 4-Br                                                           207 2-CH.sub.3, 5-Br                                                           208 2-CH.sub.3, 6-Br                                                           209 2-Cl, 3-CH.sub.3                                                           210 2-Cl, 4-CH.sub.3                                                           211 2-Cl, 5-CH.sub.3                                                           212 2-F, 3-CH.sub.3                                                            213 2-F, 4-CH.sub.3                                                            214 2-F, 5-CH.sub.3                                                            215 2-Br, 3-CH.sub.3                                                           216 2-Br, 4-CH.sub.3                                                           217 2-Br, 5-CH.sub.3                                                           218 3-CH3, 4-Cl                                                                219 3-CH.sub.3, 5-Cl                                                           220 3-CH.sub.3, 4-F                                                            221 3-CH.sub.3, 5-F                                                            222 3-CH.sub.3, 4-Br                                                           223 3-CH.sub.3, 5-Br                                                           224 3-F, 4-CH.sub.3                                                            225 3-Cl, 4-CH.sub.3                                                           226 3-Br, 4-CH.sub.3                                                           227 2-Cl, 4,5-(CH.sub.3).sub.2                                                 228 2-Br, 4,5-(CH.sub.3).sub.2                                                 229 2-Cl, 3,5-(CH.sub.3).sub.2                                                 230 2-Br, 3,5-(CH.sub.3).sub.2                                                 231 2,6-Cl.sub.2, 4-CH.sub.3                                                   232 2,6-F.sub.2, 4-CH.sub.3                                                    233 2,6-Br.sub.2, 4-CH.sub.3                                                   234 2,4-Br.sub.2, 6-CH.sub.3                                                   235 2,4-F.sub.2, 6-CH.sub.3                                                    236 2,4-Br.sub.2, 6-CH.sub.3                                                   237 2,6-(CH.sub.3).sub.2, 4-F                                                  238 2,6-(CH.sub.3).sub.2, 4-Cl                                                 239 2,6-(CH.sub.3).sub.2, 4-Br                                                 240 3,5-(CH.sub.3).sub.2, 4-F                                                  241 3,5-(CH.sub.3).sub.2, 4-Cl                                                 242 3,5-(CH.sub.3).sub.2, 4-Br                                                 243 2,3,6-(CH.sub.3).sub.3, 4-F                                                244 2,3,6-(CH.sub.3).sub.3, 4-Cl                                               245 2,3,6-(CH.sub.3).sub.3, 4-Br                                               246 2,4-(CH.sub.3).sub.2, 6-F                                                  247 2,4-(CH.sub.3).sub.2, 6-Cl                                                 248 2,4-(CH.sub.3).sub.2, 6-Br                                                 249 2-i-C.sub.3 H.sub.7, 4-Cl, 5-CH.sub.3                                      250 2-Cl, 4-NO2                                                                251 2-NO2, 4-Cl                                                                252 2-OCH.sub.3, 5-NO.sub.2                                                    253 2,4-Cl2, 5-NO2                                                             254 2,4-Cl2, 6-NO2                                                             255 2,6-Cl2, 4-NO2                                                             256 2,6-Br2, 4-NO2                                                             257 2,6-I2, 4-NO2                                                              258 2-CH3, 5-i-C3H7, 4-Cl                                                      259 2-CO.sub.2 CH.sub.3                                                        260 3-CO2CH3                                                                   261 4-CO2CH3                                                                   262 2-CO2(C2H5)                                                                263 3-CO.sub.2 (C.sub.2 H.sub.5)                                               264 4-CO.sub.2 (C.sub.2 H.sub.5)                                               265 2-CO.sub.2 (n-C.sub.3 H.sub.7)                                             266 3-CO.sub.2 (n-C.sub.3 H.sub.7)                                             267 4-CO.sub.2 (n-C.sub.3 H.sub.7)                                             268 2-CO.sub.2 (i-C.sub.3 H.sub.7)                                             269 3-CO.sub.2 (i-C.sub.3 H.sub.7)                                             270 4-CO.sub.2 (i-C.sub.3 H.sub.7)                                             271 2-CO.sub.2 (n-C.sub.6 H.sub.13)                                            272 3-CO.sub.2 (n-C.sub.6 H.sub.13)                                            273 4-CO.sub.2 (n-C.sub.6 H.sub.13)                                            274 2-CH.sub.2 --OCH.sub.3                                                     275 3-CH.sub.2 --OCH.sub.3                                                     276 4-CH.sub.2 --OCH.sub.3                                                     277 2-CH.sub.2 O(C.sub.2 H.sub.5)                                              278 3-CH.sub.2 O(C.sub.2 H.sub.5)                                              279 4-CH.sub.2 O(C.sub.2 H.sub.5)                                              280 2-CH.sub.2 O(n-C.sub.3 H.sub.7)                                            281 3-CH.sub.2 O(n-C.sub.3 H.sub.7)                                            282 4-CH.sub.2 O(n-C.sub.3 H.sub.7)                                            283 2-CH.sub.2 O(i-C.sub.3 H.sub.7)                                            284 3-CH.sub.2 O(i-C.sub.3 H.sub.7)                                            285 4-CH.sub.2 O(i-C.sub.3 H.sub.7)                                            286 2-CHO                                                                      287 3-CHO                                                                      288 4-CHO                                                                      289 2-CO--CH.sub.3                                                             290 3-CO--CH.sub.3                                                             291 4-CO--CH.sub.3                                                             292 2-CO--CH.sub.2 --CH.sub.3                                                  293 3-CO--CH.sub.2 --CH.sub.3                                                  294 4-CO--CH.sub.2 --CH.sub.3                                                  295 2-CO--CH.sub.2 --CH.sub.2 --CH.sub.3                                       296 3-CO--CH.sub.2 --CH.sub.2 --CH.sub.3                                       297 4-CO--CH.sub.2 --CH.sub.2 --CH.sub.3                                       298 2-CO--CH(CH.sub.3)--CH.sub.3                                               299 3-CO--CH(CH.sub.3)--CH.sub.3                                               300 4-CO--CH(CH.sub.3)--CH.sub.3                                               301 2-Me-4-CHO                                                                 302 2-Me-4-CH.sub.3 --CO                                                       303 2-Me-4-CH.sub.3 --CH.sub.2 --CO                                            304 2-Me-4-CH.sub.3 --CH.sub.2 --CH.sub.2 --CO                                 305 2-Me-4-CH.sub.3 --CH(CH.sub.3)--CO                                         306 2,5-Me.sub.2 -4-CHO                                                        307 2,5-Me.sub.2 -4-CH.sub.3 --CO                                              308 2,5-Me.sub.2 -4-CH.sub.3 --CH.sub.2 --CO                                   309 2,5-Me.sub.2 -4-CH.sub.3 --CH.sub.2 --CH.sub.2 --CO                        310 2,5-Me.sub.2 -4-CH.sub.3 --CH(CH.sub.3)--CO                                311 2-Cl-4-CHO                                                                 312 2-Cl-4-CH.sub.3 --CO                                                       313 2-Cl-4-CH.sub.3 --CH.sub.2 --CO                                            314 2-Cl-4-CH.sub.3 --CH(CH.sub.3)--CO                                         315 2,5-Cl.sub.2 -4-CHO                                                        316 2,5-Cl.sub.2 -4-CH.sub.3 --CO                                              317 2,5-Cl.sub.2 -4-CH.sub.3 --CH.sub.2 --CO                                   318 2,5-Cl.sub.2 -4-CH.sub.3 --CH.sub.2 --CH.sub.2 --CO                        319 2,5-Cl.sub.2 -4-CH.sub.3 --CH(CH.sub.3)--CO                                320 2-C(═NOCH.sub.3)--CH.sub.3                                             321 3-C(═NOCH.sub.3)--CH.sub.3                                             322 4-C(═NOCH.sub.3)--CH.sub.3                                             323 2-C(═NOC.sub.2 H.sub.5)--CH.sub.3                                      324 3-C(═NOC.sub.2 H.sub.5)--CH.sub.3                                      325 4-C(═NOC.sub.2 H.sub.5)--CH.sub.3                                      326 2-C(═NO-n-C.sub.3 H.sub.7)--CH.sub.3                                   327 3-C(═NO-n-C.sub.3 H.sub.7)--CH.sub.3                                   328 4-C(═NO-n-C.sub.3 H.sub.7)--CH.sub.3                                   329 2-C(═NO-i-C.sub.3 H.sub.7)--CH.sub.3                                   330 3-C(═NO-i-C.sub.3 H.sub.7)--CH.sub.3                                   331 4-C(═NO-i-C.sub.3 H.sub.7)--CH.sub.3                                   332 2-C(═NO-Allyl)-CH.sub.3                                                333 3-C(═NO-Allyl)-CH.sub.3                                                334 4-C(═NO-Allyl)-CH.sub.3                                                335 2-C(═NO-trans-Chloroallyl)-CH.sub.3                                    336 3-C(═NO-trans-Chloroallyl)-CH.sub.3                                    337 4-C(═NO-trans-Chloroallyl)-CH.sub.3                                    338 2-C(═NO-Propargyl)-CH.sub.3                                            339 3-C(═NO-Propargyl)-CH.sub.3                                            340 4-C(═NO-Propargyl)-CH.sub.3                                            341 2-C(═NO-n-C.sub.4 H.sub.9)--CH.sub.3                                   342 3-C(═NO-n-C.sub.4 H.sub.9)--CH.sub.3                                   343 4-C(═NO-n-C.sub.4 H.sub.9)--CH.sub.3                                   344 2-C(═NO--CH.sub.2 --C.sub.6 H.sub.5)--CH.sub.3                         345 3-C(═NO--CH.sub.2 --C.sub.6 H.sub.5)--CH.sub.3                         346 4-C(═NO--CH.sub.2 --C.sub.6 H.sub.5)--CH.sub.3                         347 2-CH.sub.3 -4-CH═NOCH.sub.3                                            348 2-CH.sub.3 -4-CH═NOC.sub.2 H.sub.5                                     349 2-CH.sub.3 -4-CH═NO-n-C.sub.3 H.sub.7                                  350 2-CH.sub.3 -4-CH═NO-i-C.sub.3 H.sub.7                                  351 2-CH.sub.3 -4-CH═NO-Allyl                                              352 2-CH.sub.3 -4-CH═NO-(trans-Chloroallyl)                                353 2-CH.sub.3 -4-CH═NO-Propargyl                                          354 2-CH.sub.3 -4-CH═NO-n-C.sub.4 H.sub.9                                  355 2-CH.sub.3 -4-CH═NO--CH.sub.2 --C.sub.6 H.sub.5                        356 2-CH.sub.3 -4-(CH.sub.3 --C═NOCH.sub.3)                                357 2-CH.sub.3 -4-(CH.sub.3 --C═NOC.sub.2 H.sub.5)                         358 2-CH.sub.3 -4-(CH.sub.3 --C═NO-n-C.sub.3 H.sub.7)                      359 2-CH.sub.3 -4-(CH.sub.3 --C═NO-i-C.sub.3 H.sub.7)                      360 2-CH.sub.3 -4-(CH.sub.3 --C═NO-Allyl)                                  361 2-CH3-4-(CH3--C═NO-trans-Chloroallyl)                                  362 2-CH.sub.3 -4-(CH.sub.3 --C═NO-Propargyl)                              363 2-CH.sub.3 -4-(CH.sub.3 --C═NO-n-C.sub.4 H.sub.9)                      364 2-CH.sub.3 -4-(CH.sub.3 --C═NO--CH.sub.2 --C.sub.6 H.sub.5)                   365 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C═NO--CH.sub.3)                       366 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C═NO--C.sub.2 H.sub.5)                367 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C═NO-n-C.sub.3 H.sub.7)        368 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C═NO-i-C.sub.3 H.sub.7                       369 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C═NO-Allyl)                    370 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C═NO-trans-Chloroallyl)                      371 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C═NO-Propargyl)                       372 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C═NO-n-C.sub.4 H.sub.9)        373 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C═NO--CH.sub.2 --C.sub.6                    H.sub.5)                                                                 374 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C═NOCH.sub.3)                      375 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C═NOC.sub.2 H.sub.5)                      376 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C═NO-n-C.sub.3                    H.sub.7)                                                                 377 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C═NO-i-C.sub.3 H.sub.7)                   378 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C═NO-Allyl)                 379 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C═NO-trans-Chloroallyl)                   380 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C═NO-Proparyl)                     381 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C═NO-n-C.sub.4                    H.sub.9)                                                                 382 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C═NO--CH.sub.2 --C.sub.6                 H.sub.5)                                                                 383 2-C.sub.6 H.sub.5                                                          384 3-C.sub.6 H.sub.5                                                          385 4-C.sub.6 H.sub.5                                                          386 2-(2'-F--C.sub.6 H.sub.4)                                                  387 2-(3'-F--C.sub.6 H.sub.4)                                                  388 2-(4'-F--C.sub.6 H.sub.4)                                                  389 3-(2'-F--C.sub.6 H.sub.4)                                                  390 3-(3'-F--C.sub.6 H.sub.4)                                                  391 3-(4'-F--C.sub.6 H.sub.4)                                                  392 4-(2'-F--C.sub.6 H.sub.4)                                                  393 4-(3'-F--C.sub.6 H.sub.4)                                                  394 4-(4'-F--C.sub.6 H.sub.4)                                                  395 2-(2'-Cl--C.sub.6 H.sub.4)                                                 396 2-(3'-Cl--C.sub.6 H.sub.4)                                                 397 2-(4'-Cl--C.sub.6 H.sub.4)                                                 398 3-(2'-Cl--C.sub.6 H.sub.4)                                                 399 3-(3'-Cl--C.sub.6 H.sub.4)                                                 400 3-(4'-Cl--C.sub.6 H.sub.4)                                                 401 4-(2'-Cl--C.sub.6 H.sub.4)                                                 402 4-(3'-Cl--C.sub.6 H.sub.4)                                                 403 4-(4'-Cl--C.sub.6 H.sub.4)                                                 405 2-(2'-CH.sub.3 --C.sub.6 H.sub.4)                                          406 2-(3'-CH.sub.3 --C.sub.6 H.sub.4)                                          407 2-(4'-CH.sub.3 --C.sub.6 H.sub.4)                                          408 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)                                          409 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)                                          410 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)                                          411 4-(2'-CH.sub.3 --C.sub.6 H.sub.4)                                          412 4-(3'-CH.sub.3 --C.sub.6 H.sub.4)                                          413 4-(4'-CH.sub.3 --C.sub.6 H.sub.4)                                          414 2-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                      415 2-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                      416 2-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                      417 3-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                      418 3-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                      419 3-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                      420 4-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                      421 4-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                      422 4-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                      423 2-(2'-(CH.sub.3 --C(═NOAllyl))-C.sub.6 H.sub.4)                        424 2-(3'-(CH.sub.3 --C(═NOAllyl))-C.sub.6 H.sub.4)                        425 2-(4'-(CH.sub.3 --C(═NOAllyl))-C.sub.6 H.sub.4)                        426 3-(2'-(CH.sub.3 --C(═NOAllyl))-C.sub.6 H.sub.4)                        427 3-(3'-(CH.sub.3 --C(═NOAllyl))-C.sub.6 H.sub.4)                        428 3-(4'-(CH.sub.3 --C(═NOAllyl))-C.sub.6 H.sub.4)                        429 4-(2'-(CH.sub.3 --C(═NOAllyl))-C.sub.6 H.sub.4)                        430 4-(3'-(CH.sub.3 --C(═NOAllyl))-C.sub.6 H.sub.4)                        431 4-(4'-(CH.sub.3 --C(═NOAllyl))-C.sub.6 H.sub.4)                        432 2-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                                 433 2-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                                 434 2-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                                 435 3-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                                 436 3-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                                 437 3-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                                 438 4-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                                 439 4-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                                 440 4-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                                 441 2-(2'-CH.sub.3 O--C.sub.6 H.sub.4)                                         442 2-(3'-CH.sub.3 O--C.sub.6 H.sub.4)                                         443 2-(4'-CH.sub.3 O--C.sub.6 H.sub.4)                                         444 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)                                         445 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)                                         446 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)                                         447 4-(2'-CH.sub.3 O--C.sub.6 H.sub.4)                                         448 4-(3'-CH.sub.3 O--C.sub.6 H.sub.4)                                         449 4-(4'-CH.sub.3 O--C.sub.6 H.sub.4)                                         450 2-(2'-O.sub.2 N--C.sub.6 H.sub.4)                                          451 2-(3'-O.sub.2 N--C.sub.6 H.sub.4)                                          452 2-(4'-O.sub.2 N--C.sub.6 H.sub.4)                                          453 3-(2'-O.sub.2 N--C.sub.6 H.sub.4)                                          454 3-(3'-O.sub.2 N--C.sub.6 H.sub.4)                                          455 3-(4'-O.sub.2 N--C.sub.6 H.sub.4)                                          456 4-(2'-O.sub.2 N--C.sub.6 H.sub.4)                                          457 4-(3'-O.sub.2 N--C.sub.6 H.sub.4)                                          458 4-(4'-O.sub.2 N--C.sub.6 H.sub.4)                                          459 2-(2'-NC--C.sub.6 H.sub.4)                                                 460 2-(3'-NC--C.sub.6 H.sub.4)                                                 461 2-(4'-NC--C.sub.6 H.sub.4)                                                 462 3-(2'-NC--C.sub.6 H.sub.4)                                                 463 3-(3'-NC--C.sub.6 H.sub.4)                                                 464 3-(4'-NC--C.sub.6 H.sub.4)                                                 465 4-(2'-NC--C.sub.6 H.sub.4)                                                 466 4-(3'-NC--C.sub.6 H.sub.4)                                                 467 4-(4'-NC--C.sub.6 H.sub.4)                                                 468 2-(2'-CF.sub.3 --C.sub.6 H.sub.4)                                          469 2-(3'-CF.sub.3 --C.sub.6 H.sub.4)                                          470 2-(4'-CF.sub.3 --C.sub.6 H.sub.4)                                          471 3-(2'-CF.sub.3 --C.sub.6 H.sub.4)                                          472 3-(3'-CF.sub.3 --C.sub.6 H.sub.4)                                          473 3-(4'-CF.sub.3 --C.sub.6 H.sub.4)                                          474 4-(2'-CF.sub.3 --C.sub.6 H.sub.4)                                          475 4-(3'-CF.sub.3 --C.sub.6 H.sub.4)                                          476 4-(4'-CF.sub.3 --C.sub.6 H.sub.4)                                          477 2-O--C.sub.6 H.sub.5                                                       475 3-O--C6H5                                                                  476 4-O--C6H5                                                                  478 2-O-(2'-F--C.sub.6 H.sub.4)                                                479 2-O-(3'-F--C.sub.6 H.sub.4)                                                480 2-O-(4'-F--C.sub.6 H.sub.4)                                                481 3-O-(2'-F--C.sub.6 H.sub.4)                                                482 3-O-(3'-F--C.sub.6 H.sub.4)                                                483 3-O-(4'-F--C.sub.6 H.sub.4)                                                484 4-O-(2'-F--C.sub.6 H.sub.4)                                                485 4-O-(3'-F--C.sub.6 H.sub.4)                                                486 4-O-(4'-F--C.sub.6 H.sub.4)                                                487 2-O-(2'-Cl--C.sub.6 H.sub.4)                                               488 2-O-(3'-Cl--C.sub.6 H.sub.4)                                               489 2-O-(4'-Cl--C.sub.6 H.sub.4)                                               490 3-O-(2'-Cl--C.sub.6 H.sub.4)                                               491 3-O-(3'-Cl--C.sub.6 H.sub.4)                                               492 3-O-(4'-Cl--C.sub.6 H.sub.4)                                               493 3-O-(4'-Cl--C.sub.6 H.sub.4)                                               494 4-O-(2'-Cl--C.sub.6 H.sub.4)                                               495 4-O-(3'-Cl--C.sub.6 H.sub.4)                                               496 4-O-(4'-Cl--C.sub.6 H.sub.4)                                               497 2-O-(2'-CH.sub.3 --C.sub.6 H.sub.4)                                        498 2-O-(3'-CH.sub.3 --C.sub.6 H.sub.4)                                        499 2-O-(4'-CH.sub.3 --C.sub.6 H.sub.4)                                        500 3-O-(2'-CH.sub.3 --C.sub.6 H.sub.4)                                        501 3-O-(3'-CH.sub.3 --C.sub.6 H.sub.4)                                        502 3-O-(4'-CH.sub.3 --C.sub.6 H.sub.4)                                        503 4-O-(2'-CH.sub.3 --C.sub.6 H.sub.4)                                        504 4-O-(3'-CH.sub.3 --C.sub.6 H.sub.4)                                        505 4-O-(4'-CH.sub.3 --C.sub.6 H.sub.4)                                        506 2-O-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                    507 2-O-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                    508 2-O-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                    509 3-O-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                    510 3-O-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                    511 3-O-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                    512 4-O-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                    513 4-O-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                    514 4-O-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                    515 2-O-(2'-(CH.sub.3 --C(═NOAllyl))-C.sub.6 H.sub.4)                      516 2-O-(3'-(CH.sub.3 --C(═NOAllyl))-C.sub.6 H.sub.4)                      517 2-O-(4'-(CH.sub.3 --C(═NOAllyl))-C.sub.6 H.sub.4)                      518 3-O-(2'-(CH.sub.3 --C(═NOAllyl))-C.sub.6 H.sub.4)                      519 3-O-(3'-(CH.sub.3 --C(═NOAllyl))-C.sub.6 H.sub.4)                      520 3-O-(4'-(CH.sub.3 --C(═NOAllyl))-C.sub.6 H.sub.4)                      521 4-O-(2'-(CH.sub.3 --C(═NOAllyl))-C.sub.6 H.sub.4)                      522 4-O-(3'-(CH.sub.3 --C(═NOAllyl))-C.sub.6 H.sub.4)                      523 4-O-(4'-(CH.sub.3 --C(═NOAllyl))-C.sub.6 H.sub.4)                      524 2-O-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                               525 2-O-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                               526 2-O-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                               527 3-O-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                               528 3-O-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                               529 3-O-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                               530 4-O-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                               531 4-O-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                               532 4-O-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                               533 2-O-(2'-CH.sub.3 O--C.sub.6 H.sub.4)                                       534 2-O-(3'-CH.sub.3 O--C.sub.6 H.sub.4)                                       535 2-O-(4'-CH.sub.3 O--C.sub.6 H.sub.4)                                       536 3-O-(2'-CH.sub.3 O--C.sub.6 H.sub.4)                                       537 3-O-(3'-CH.sub.3 O--C.sub.6 H.sub.4)                                       538 3-O-(4'-CH.sub.3 O--C.sub.6 H.sub.4)                                       539 4-O-(2'-CH.sub.3 O--C.sub.6 H.sub.4)                                       540 4-O-(3'-CH.sub.3 O--C.sub.6 H.sub.4)                                       541 4-O-(4'-CH.sub.3 O--C.sub.6 H.sub.4)                                       542 2-O-(2'-O.sub.2 N--C.sub.6 H.sub.4)                                        543 2-O-(3'-O.sub.2 N--C.sub.6 H.sub.4)                                        544 2-O-(4'-O.sub.2 N--C.sub.6 H.sub.4)                                        545 3-O-(2'-O.sub.2 N--C.sub.6 H.sub.4)                                        546 3-O-(3'-O.sub.2 N--C.sub.6 H.sub.4)                                        547 3-O-(4'-O.sub.2 N--C.sub.6 H.sub.4)                                        548 4-O-(2'-O.sub.2 N--C.sub.6 H.sub.4)                                        549 4-O-(3'-O.sub.2 N--C.sub.6 H.sub.4)                                        550 4-O-(4'-O.sub.2 N--C.sub.6 H.sub.4)                                        551 2-O-(2'-NC--C.sub.6 H.sub.4)                                               552 2-O-(3'-NC--C.sub.6 H.sub.4)                                               553 2-O-(4'-NC--C.sub.6 H.sub.4)                                               554 3-O-(2'-NC--C.sub.6 H.sub.4)                                               555 3-O-(3'-NC--C.sub.6 H.sub.4)                                               556 3-O-(4'-NC--C.sub.6 H.sub.4)                                               557 4-O-(2'-NC--C.sub.6 H.sub.4)                                               558 4-O-(3'-NC--C.sub.6 H.sub.4)                                               559 4-O-(4'-NC--C.sub.6 H.sub.4)                                               560 2-O-(2'-CF.sub.3 --C.sub.6 H.sub.4)                                        561 2-O-(3'-CF.sub.3 --C.sub.6 H.sub.4)                                        562 2-O-(4'-CF.sub.3 --C.sub.6 H.sub.4)                                        563 3-O-(2'-CF.sub.3 --C.sub.6 H.sub.4)                                        564 3-O-(3'-CF.sub.3 --C.sub.6 H.sub.4)                                        565 3-O-(4'-CF.sub.3 --C.sub.6 H.sub.4)                                        566 4-O-(2'-CF.sub.3 --C.sub.6 H.sub.4)                                        567 4-O-(3'-CF.sub.3 --C.sub.6 H.sub.4)                                        568 4-O-(4'-CF.sub.3 --C.sub.6 H.sub.4)                                        569 2-Pyridinyl-2'                                                             570 2-Pyridinyl-3'                                                             571 2-Pyridinyl-4'                                                             572 3-Pyridinyl-2'                                                             573 3-Pyridinyl-3'                                                             574 3-Pyridinyl-4'                                                             575 4-Pyridinyl-2'                                                             576 4-Pyridinyl-3'                                                             577 4-Pyridinyl-4'                                                             578 2-Pyrimidinyl-2'                                                           579 2-Pyrimidinyl-3'                                                           580 2-Pyrimidinyl-4'                                                           581 3-Pyrimidinyl-2'                                                           582 3-Pyrimidinyl-3'                                                           583 3-Pyrimidinyl-4'                                                           584 4-Pyrimidinyl-2'                                                           585 4-Pyrimidinyl-3'                                                           586 4-Pyrimidinyl-4'                                                           587 2-Pyrazolyl-1'                                                             588 2-Pyrazolyl-3'                                                             589 2-Pyrazolyl-4'                                                             590 3-Pyrazolyl-1'                                                             591 3-Pyrazolyl-3'                                                             592 3-Pyrazolyl-4'                                                             593 4-Pyrazolyl-1'                                                             594 4-Pyrazolyl-3'                                                             595 4-Pyrazolyl-4'                                                             596 2-Isoxazolyl-3'                                                            597 2-Isoxazolyl-4'                                                            598 2-Isoxazolyl-5'                                                            599 3-Isoxazolyl-3'                                                            600 3-Isoxazolyl-4'                                                            601 3-Isoxazolyl-5'                                                            602 4-Isoxazolyl-3'                                                            603 4-Isoxazolyl-4'                                                            604 4-Isoxazolyl-5'                                                            605 2-Isothiazolyl-3'                                                          606 2-Isothiazolyl-4'                                                          607 2-Isothiazdlyl-5'                                                          608 3-Isothiazolyl-3'                                                          609 3-Isothiazolyl-4'                                                          610 3-Isothiazolyl-5'                                                          611 4-Isothiazolyl-3'                                                          612 4-Isothiazolyl-4'                                                          613 4-Isothiazolyl-5'                                                          614 2-Imidazolyl-1'                                                            615 2-Imidazolyl-2'                                                            616 2-Imidazolyl-4'                                                            617 3-Imidazolyl-1'                                                            618 3-Imidazolyl-2'                                                            619 3-Imidazolyl-4'                                                            620 4-Imidazolyl-1'                                                            621 4-Imidazolyl-2'                                                            622 4-Imidazolyl-4'                                                            623 2-Oxazolyl-2'                                                              624 2-Oxazolyl-4'                                                              625 2-Oxazolyl-5'                                                              626 3-Oxazolyl-2'                                                              627 3-Oxazolyl-4'                                                              628 3-Oxazolyl-5'                                                              629 4-Oxazolyl-2'                                                              630 4-oxazolyl-4'                                                              631 4-Oxazolyl-5'                                                              632 2-Thiazolyl-2'                                                             633 2-Thiazolyl-4'                                                             634 2-Thiazolyl-5                                                              635 3-Thiazolyl-2'                                                             636 3-Thiazolyl-4'                                                             637 3-Thiazolyl-5'                                                             638 4-Thiazolyl-2'                                                             639 4-Thiazolyl-4'                                                             640 4-Thiazolyl-5'                                                             641 2-CH.sub.3 -4-(CH.sub.3 --C═N-O--CH.sub.2 --CH.sub.2 --OCH.sub.3             )                                                                        642 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C═N-O--CH.sub.2 --CH.sub.2                  --OCH.sub.3)                                                             643 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C═N--O--CH.sub.2 --CH.sub.2              --OCH.sub.3)                                                             644 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C═N--OCH.sub.3)                     645 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C═N--OC.sub.2 H.sub.5)                     646 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C═N--O-n-C.sub.3                   H.sub.7)                                                                 647 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C═N--O-i-C.sub.3 H.sub.7)                  648 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C═N--O-Allyl)                       649 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C═N--O-trans-Chloroall             yl)                                                                      650 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C═N--O-Propargyl)                   651 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C═N--O-n-C.sub.4 H.sub.9)                  652 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C═N--O--CH.sub.2                   --C.sub.6 H.sub.5)                                                       653 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C═N--OCH.sub.3)                     654 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C═N--OC.sub.2 H.sub.5)                     655 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C═N--O-n-C.sub.3                   H.sub.7)                                                                 656 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C═N--O-i-C.sub.3 H.sub.7)                  657 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C═N--O-Allyl)                       658 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C═N--O-trans-Chloroall             yl)                                                                      659 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C═N--O-Propargyl)                   660 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C═N--O-n-C.sub.4 H.sub.9)                  661 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C═N--O--CH.sub.2                   --C.sub.6 H.sub.5)                                                       662 2-O-n-C.sub.4 H.sub.9                                                      663 2-O-i-C.sub.4 H.sub.9                                                      664 2-O-s-C.sub.4 H.sub.9                                                      665 2-O-t-C.sub.4 H.sub.9                                                      666 2-Neopentyloxy                                                             667 3-O-n-C.sub.4 H.sub.9                                                      668 3-O-i-C.sub.4 H.sub.9                                                      669 3-O-s-C.sub.4 H.sub.9                                                      670 3-O-t-C.sub.4 H.sub.9                                                      671 3-Neopentyloxy                                                             672 4-O-n-C.sub.4 H.sub.9                                                      673 4-O-i-C.sub.4 H.sub.9                                                      674 4-O-s-C.sub.4 H.sub.9                                                      675 4-O-t-C.sub.4 H.sub.9                                                      676 4-Neopentyloxy                                                             677 3-CH.sub.3 -4-OCH.sub.3                                                    678 3-CH.sub.3 -4-OC.sub.2 H.sub.5                                             679 3-CH.sub.3 -4-O-n-C.sub.3 H.sub.7                                          680 3-CH.sub.3 -4-O-n-C.sub.4 H.sub.9                                          681 3-CH.sub.3 -4-O-i-C.sub.4 H.sub.9                                          682 3-CH.sub.3 -4-O-s-C.sub.4 H.sub.9                                          683 3-CH.sub.3 -4-O-t-C.sub.4 H.sub.9                                          684 3-CH.sub.3 -4-Neopentyloxy                                                 685 2-CH.sub.3 -3-OCH.sub.3                                                    686 2-CH.sub.3 -4-OCH.sub.3                                                    687 2-CH.sub.3 -5-OCH.sub.3                                                    688 2-CH.sub.3 -6-OCH.sub.3                                                    689 3-CH.sub.3 -4-OCH.sub.3                                                    690 3-CH.sub.3 -5-OCH.sub.3                                                    691 3-CH.sub.3 -6-OCH.sub.3                                                    692 4-CH.sub.3 -5-O--CH.sub.3                                                  693 4-CH.sub.3 -6-O--CH.sub.3                                                  694 4-CH.sub.3 -6-OCH.sub.3                                                    695 2-CH.sub.3 -3-O-i-C.sub.3 H.sub.7                                          696 2-CH.sub.3 -4-O-i-C.sub.3 H.sub.7                                          697 2-CH.sub.3 -5-O-i-C.sub.3 H.sub.7                                          698 2-CH.sub.3 -6-O-i-C.sub.3 H.sub.7                                          699 3-CH.sub.3 -4-O-i-C.sub.3 H.sub.7                                          700 3-CH.sub.3 -5-O-i-C.sub.3 H.sub.7                                          701 3-CH.sub.3 -6-O-i-C.sub.3 H.sub.7                                          702 4-CH.sub.3 -5-O-i-C.sub.3 H.sub.7                                          703 4-CH.sub.3 -6-O-i-C.sub.3 H.sub.7                                          704 5-CH.sub.3 -6-O-i-C.sub.3 H.sub.7                                          705 2-Cl-3-OCH.sub.3                                                           706 2-Cl-4-OCH.sub.3                                                           707 2-Cl-5-OCH.sub.3                                                           708 2-Cl-6-OCH.sub.3                                                           709 3-Cl-4-OCH.sub.3                                                           710 3-Cl-5-OCH.sub.3                                                           711 3-Cl-6-QCH.sub.3                                                           712 4-Cl-5-OCH.sub.3                                                           713 4-Cl-6-OCH.sub.3                                                           714 5-Cl-6-OCH.sub.3                                                         ______________________________________                                    

                  TABLE 25                                                         ______________________________________                                                            1   I: R.sup.1 = CH.sub.3, X = CH.sub.3 II: R.sup.1 =                          CH.sub.2 --CH.sub.3, X = CH.sub.3 III: R.sup.1 =                               CH.sub.3, X = Cl IV: R.sup.1 = CH.sub.2 --CH.sub.3, X                          = Cl                                                           -                                                                           No.       B                                                                    ______________________________________                                         1         Pyrrolyl-3                                                             2 N--CH.sub.3 -Pyrrolyl-3                                                      3 N--C.sub.6 H.sub.5 -Pyrrolyl-3                                               4 N-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrrolyl-3                                 5 N-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrrolyl-3                                 6 N-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrrolyl-3                                 7 N-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrrolyl-3                                8 N-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrrolyl-3                                9 N-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrrolyl-3                                10 N-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrrolyl-3                                11 N-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrrolyl-3                                12 N-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrrolyl-3                                13 N-(4'-CN--C.sub.6 H.sub.4)-Pyrrolyl-3                                       14 N-(3'-CN--C.sub.6 H.sub.4)-Pyrrolyl-3                                       15 N-(2'-CN--C.sub.6 H.sub.4)-Pyrrolyl-3                                       16 N-(4'-Cl--C.sub.6 H.sub.4)-Pyrrolyl-3                                       17 N-(3'-Cl--C.sub.6 H.sub.4)-Pyrrolyl-3                                       18 N-(2'-Cl--C.sub.6 H.sub.4)-Pyrrolyl-3                                       19 Pyrrolyl-2                                                                  20 N--CH.sub.3 -Pyrrolyl-2                                                     21 N--C.sub.6 H.sub.5 -Pyrrolyl-2                                              22 N-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrrolyl-2                                23 N-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrrolyl-2                                24 N-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrrolyl-2                                25 N-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrrolyl-2                               26 N-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrrolyl-2                               27 N-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrrolyl-2                               28 N-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrrolyl-2                                29 N-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrrolyl-2                                30 N-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrrolyl-2                                31 N-(4'-CN--C.sub.6 H.sub.4)-Pyrrolyl-2                                       32 N-(3'-CN--C.sub.6 H.sub.4)-Pyrrolyl-2                                       33 N-(2'-CN--C.sub.6 H.sub.4)-Pyrrolyl-2                                       34 N-(4'-Cl--C.sub.6 H.sub.4)-Pyrrolyl-2                                       35 N-(3'-Cl--C.sub.6 H.sub.4)-Pyrrolyl-2                                       36 N-(2'-Cl--C.sub.6 H.sub.4)-Pyrrolyl-2                                       37 Furyl-2                                                                     38 5-CH.sub.3 -Furyl-2                                                         39 5-C.sub.6 H.sub.5 -Furyl-2                                                  40 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Furyl-2                                   41 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Furyl-2                                   42 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Furyl-2                                   43 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Furyl-2                                  44 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Furyl-2                                  45 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Furyl-2                                  46 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Furyl-2                                   47 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Furyl-2                                   48 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Furyl-2                                   49 5-(4'-CN--C.sub.6 H.sub.4)-Furyl-2                                          50 5-(3'-CN--C.sub.6 H.sub.4)-Furyl-2                                          51 5-(2'-CN--C.sub.6 H.sub.4)-Furyl-2                                          52 5-(4'-Cl--C.sub.6 H.sub.4)-Furyl-2                                          53 5-(3'-Cl--C.sub.6 H.sub.4)-Furyl-2                                          54 5-(2'-Cl--C.sub.6 H.sub.4)-Furyl-2                                          55 4-CH.sub.3 -Furyl-2                                                         56 4-C.sub.6 H.sub.5 -Furyl-2                                                  57 4-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Furyl-2                                   58 4-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Furyl-2                                   59 4-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Furyl-2                                   60 4-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Furyl-2                                  61 4-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Furyl-2                                  62 4-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Furyl-2                                  63 4-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Furyl-2                                   64 4-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Furyl-2                                   65 4-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Furyl-2                                   66 4-(4'-CN--C.sub.6 H.sub.4)-Furyl-2                                          67 4-(3'-CN--C.sub.6 H.sub.4)-Furyl-2                                          68 4-(2'-CN--C.sub.6 H.sub.4)-Furyl-2                                          69 4-(4'-Cl--C.sub.6 H.sub.4)-Furyl-2                                          70 4-(3'-Cl--C.sub.6 H.sub.4)-Furyl-2                                          71 4-(2'-Cl--C.sub.6 H.sub.4)-Furyl-2                                          72 Thienyl-2                                                                   73 5-CH.sub.3 -Thienyl-2                                                       74 5-C.sub.6 H.sub.5 -Thienyl-2                                                75 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-2                                 76 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-2                                 77 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-2                                 78 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-2                                79 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-2                                80 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-2                                81 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-2                                 82 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-2                                 83 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-2                                 84 5-(4'-CN--C.sub.6 H.sub.4)-Thienyl-2                                        85 5-(3'-CN--C.sub.6 H.sub.4)-Thienyl-2                                        86 5-(2'-CN--C.sub.6 H.sub.4)-Thienyl-2                                        87 5-(4'-Cl--C.sub.6 H.sub.4)-Thienyl-2                                        88 5-(3'-Cl--C.sub.6 H.sub.4)-Thienyl-2                                        89 5-(2'-Cl--C.sub.6 H.sub.4)-Thienyl-2                                        90 4-CH.sub.3 -Thienyl-2                                                       91 4-C.sub.6 H.sub.5 -Thienyl-2                                                92 4-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-2                                 93 4-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-2                                 94 4-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-2                                 95 4-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-2                                96 4-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-2                                97 4-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-2                                98 4-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-2                                 99 4-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-2                                 100 4-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-2                                101 4-(4'-CN--C.sub.6 H.sub.4)-Thienyl-2                                       102 4-(3'-CN--C.sub.6 H.sub.4)-Thienyl-2                                       103 4-(2'-CN--C.sub.6 H.sub.4)-Thienyl-2                                       104 4-(4'-Cl--C.sub.6 H.sub.4)-Thienyl-2                                       105 4-(3'-Cl--C.sub.6 H.sub.4)-Thienyl-2                                       106 4-(2'-Cl--C.sub.6 H.sub.4)-Thienyl-2                                       107 Thienyl-3                                                                  108 5-CH.sub.3 -Thienyl-3                                                      109 5-C.sub.6 H.sub.5 -Thienyl-3                                               110 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-3                                111 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-3                                112 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-3                                113 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-3                               114 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-3                               115 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-3                               116 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-3                                117 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-3                                118 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-3                                119 5-(4'-CN--C.sub.6 H.sub.4)-Thienyl-3                                       120 5-(3'-CN--C.sub.6 H.sub.4)-Thienyl-3                                       121 5-(2'-CN--C.sub.6 H.sub.4)-Thienyl-3                                       122 5-(4'-Cl--C.sub.6 H.sub.4)-Thienyl-3                                       123 5-(3'-Cl--C.sub.6 H.sub.4)-Thienyl-3                                       124 5-(2'-Cl--C.sub.6 H.sub.4)-Thienyl-3                                       125 Pyrazolyl-4                                                                126 N--CH.sub.3 -Pyrazolyl-4                                                   127 N--C.sub.6 H.sub.5 -Pyrazolyl-4                                            128 N-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrazolyl-4                              129 N-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrazolyl-4                              130 N-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrazolyl-4                              131 N-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrazolyl-4                             132 N-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrazolyl-4                             133 N-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrazolyl-4                             134 N-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrazolyl-4                              135 N-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrazolyl-4                              136 N-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrazolyl-4                              137 N-(4'-CN--C.sub.6 H.sub.4)-Pyrazolyl-4                                     138 N-(3'-CN--C.sub.6 H.sub.4)-Pyrazolyl-4                                     139 N-(2'-CN--C.sub.6 H.sub.4)-Pyrazolyl-4                                     140 N-(4'-Cl--C.sub.6 H.sub.4)-Pyrazolyl-4                                     141 N-(3'-Cl--C.sub.6 H.sub.4)-Pyrazolyl-4                                     142 N-(2'-Cl--C.sub.6 H.sub.4)-Pyrazolyl-4                                     143 3-CH.sub.3 --N-Methylpyrazolyl-4                                           144 3-C.sub.6 H.sub.5 --N-Methylpyrazolyl-4                                    145 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)-N-Methylpyrazolyl-4                      146 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)-N-Methylpyrazolyl-4                      147 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)-N-Methylpyrazolyl-4                      148 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-N-Methylpyrazolyl-4                     149 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-N-Methylpyrazolyl-4                     150 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-N-Methylpyrazolyl-4                     151 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)-N-Methylpyrazolyl-4                      152 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)-N-Methylpyrazolyl-4                      153 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)-N-Methylpyrazolyl-4                      154 3-(4'-CN--C.sub.6 H.sub.4)-N-Methylpyrazolyl-4                             155 3-(3'-CN--C.sub.6 H.sub.4)-N-Methylpyrazolyl-4                             156 3-(2'-CN--C.sub.6 H.sub.4)-N-Methylpyrazolyl-4                             157 3-(4'-Cl--C.sub.6 H.sub.4)-N-Methylpyrazolyl-4                             158 3-(3'-Cl--C.sub.6 H.sub.4)-N-Methylpyrazolyl-4                             159 3-(2'-Cl--C.sub.6 H.sub.4)-N-Methylpyrazolyl-4                             160 Isoxazolyl-5                                                               161 3-CH.sub.3 -Isoxazolyl-5                                                   162 3-C.sub.6 H.sub.5 -Isoxazolyl-5                                            163 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Isoxazolyl-5                             164 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Isoxazolyl-5                             165 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Isoxazolyl-5                             166 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Isoxazolyl-5                            167 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Isoxazolyl-5                            168 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Isoxazolyl-5                            169 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Isoxazolyl-5                             170 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Isoxazolyl-5                             171 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Isoxazolyl-5                             172 3-(4'-CN--C.sub.6 H.sub.4)-Isoxazolyl-5                                    173 3-(3'-CN--C.sub.6 H.sub.4)-Isoxazolyl-5                                    174 3-(2'-CN--C.sub.6 H.sub.4)-Isoxazolyl-5                                    175 3-(4'-Cl--C.sub.6 H.sub.4)-Isoxazolyl-5                                    176 3-(3'-Cl--C.sub.6 H.sub.4)-Isoxazolyl-5                                    177 3-(2'-Cl--C.sub.6 H.sub.4)-Isoxazolyl-5                                    178 4-Chloroisoxazolyl-5                                                       179 3-CH.sub.3 -4-Chloroisoxazolyl-5                                           180 3-C.sub.6 H.sub.5 -4-Chloroisoxazolyl-5                                    181 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                     182 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                     183 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                     184 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                    185 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                    186 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                    187 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                     188 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                     189 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                     190 3-(4'-CN--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                            191 3-(3'-CN--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                            192 3-(2'-CN--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                            193 3-(4'-Cl--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                            194 3-(3'-Cl--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                            195 3-(2'-Cl--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                            196 Isoxazolyl-3                                                               197 5-CH.sub.3 -Isoxazolyl-3                                                   198 5-C.sub.6 H.sub.5 -Isoxazolyl-3                                            199 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Isoxazolyl-3                             200 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Isoxazolyl-3                             201 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Isoxazolyl-3                             202 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Isoxazolyl-3                            203 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Isoxazolyl-3                            204 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Isoxazolyl-3                            205 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Isoxazolyl-3                             206 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Isoxazolyl-3                             207 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Isoxazolyl-3                             208 5-(4'-CN--C.sub.6 H.sub.4)-Isoxazolyl-3                                    209 5-(3'-CN--C.sub.6 H.sub.4)-Isoxazolyl-3                                    210 5-(2'-CN--C.sub.6 H.sub.4)-Isoxazolyl-3                                    211 5-(4'-Cl--C.sub.6 H.sub.4)-Isoxazolyl-3                                    212 5-(3'-Cl--C.sub.6 H.sub.4)-Isoxazolyl-3                                    213 5-(2'-Cl--C.sub.6 H.sub.4)-Isoxazolyl-3                                    214 Isothiazolyl-5                                                             215 3-CH.sub.3 -Isothiazolyl-5                                                 216 3-C.sub.6 H.sub.5 -Isothiazolyl-5                                          217 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Isothiazolyl-5                           218 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Isothiazolyl-5                           219 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Isothiazolyl-5                           220 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Isothiazolyl-5                          221 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Isothiazolyl-5                          222 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Isothiazolyl-5                          223 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Isothiazolyl-5                           224 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Isothiazolyl-5                           225 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Isothiazolyl-5                           226 3-(4'-CN--C.sub.6 H.sub.4)-Isothiazolyl-5                                  227 3-(3'-CN--C.sub.6 H.sub.4)-Isothiazolyl-5                                  228 3-(2'-CN--C.sub.6 H.sub.4)-Isothiazolyl-5                                  229 3-(4'-Cl--C.sub.6 H.sub.4)-Isothiazolyl-5                                  230 3-(3'-Cl--C.sub.6 H.sub.4)-Isothiazolyl-5                                  231 3-(2'-Cl--C.sub.6 H.sub.4)-Isothiazolyl-5                                  232 Oxazolyl-4                                                                 233 2-CH.sub.3 -Oxazolyl-4                                                     234 2-C.sub.6 H.sub.5 -Oxazolyl-4                                              235 2-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Oxazolyl-4                               236 2-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Oxazolyl-4                               237 2-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Oxazolyl-4                               238 2-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Oxazolyl-4                              239 2-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Oxazolyl-4                              240 2-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Oxazolyl-4                              241 2-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Oxazolyl-4                               242 2-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Oxazolyl-4                               243 2-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Oxazolyl-4                               244 2-(4'-CN--C.sub.6 H.sub.4)-Oxazolyl-4                                      245 2-(3'-CN--C.sub.6 H.sub.4)-Oxazolyl-4                                      246 2-(2'-CN--C.sub.6 H.sub.4)-Oxazolyl-4                                      247 2-(4'-Cl--C.sub.6 H.sub.4)-Oxazolyl-4                                      248 2-(3'-Cl--C.sub.6 H.sub.4)-Oxazolyl-4                                      249 2-(2'-Cl--C.sub.6 H.sub.4)-Oxazolyl-4                                      250 Thiazolyl-4                                                                251 2-CH.sub.3 -Thiazolyl-4                                                    252 2-C.sub.6 H.sub.5 -Thiazolyl-4                                             253 2-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Thiazolyl-4                              254 2-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Thiazolyl-4                              255 2-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Thiazolyl-4                              256 2-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Thiazolyl-4                             267 2-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Thiazolyl-4                             258 2-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Thiazolyl-4                             259 2-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Thiazolyl-4                              260 2-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Thiazolyl-4                              261 2-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Thiazolyl-4                              262 2-(4'-CN--C.sub.6 H.sub.4)-Thiazolyl-4                                     263 2-(3'-CN--C.sub.6 H.sub.4)-Thiazolyl-4                                     264 2-(2'-CN--C.sub.6 H.sub.4)-Thiazolyl-4                                     265 2-(4'-Cl--C.sub.6 H.sub.4)-Thiazolyl-4                                     266 2-(3'-Cl--C.sub.6 H.sub.4)-Thiazolyl-4                                     267 2-(2'-Cl--C.sub.6 H.sub.4)-Thiazolyl-4                                     268 N--CH.sub.3 -1,2,4-Triazolyl-5                                             269 3-CH.sub.3 --N--CH.sub.3 -1,2,4-Triazolyl-5                                270 3-C.sub.6 H.sub.5 --N--CH.sub.3 -1,2,4-Triazolyl-5                         271 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5                   272 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triaz               olyl-5                                                                 273 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5                   274 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Tria               zolyl-5                                                                275 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5                  276 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Tria               zolyl-5                                                                277 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5                   278 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triaz               olyl-5                                                                 279 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5                   280 3-(4'-CN--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5        281 3-(3'-CN--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5                 282 3-(2'-CN--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5                 283 3-(4'-Cl--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5                 284 3-(3'-Cl--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5                 285 3-(2'-Cl--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5                 286 1,3,4-Oxadiazolyl-2                                                        287 5-CH.sub.3 -1,3,4-Oxadiazolyl-2                                            288 5-C.sub.6 H.sub.5 -1,3,4-Oxadiazolyl-2                                     289 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                      290 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                      291 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                      292 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                     293 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                     294 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                     295 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                      296 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                      297 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                      298 5-(4'-CN--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                             299 5-(3'-CN--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                             300 5-(2'-CN--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                             301 5-(4'-Cl--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                             302 5-(3'-Cl--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                             303 5-(2'-Cl--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                             304 1,2,4-Oxadiazolyl-3                                                        305 5-CH.sub.3 -1,2,4-Oxadiazolyl-3                                            306 5-C.sub.6 H.sub.5 -1,2,4-Oxadiazolyl-3                                     307 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                      308 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                      309 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                      310 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                     311 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                     312 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                     313 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                      314 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                      315 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                      316 5-(4'-CN--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                             317 5-(3'-CN--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                             318 5-(2'-CN--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                             319 5-(4'-Cl--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                             320 5-(3'-Cl--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                             321 5-(2'-Cl--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                             322 1,2,4-Oxadiazolyl-5                                                        323 3-CH.sub.3 -1,2,4-Oxadiazolyl-5                                            324 3-C.sub.6 H.sub.5 -1,2,4-Oxadiazolyl-5                                     325 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                      326 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                      327 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                      328 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                     329 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                     330 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                     331 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                      332 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                      333 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                      334 3-(4'-CN--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                             335 3-(3'-CN--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                             336 3-(2'-CN--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                             337 3-(4'-Cl--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                             338 3-(3'-Cl--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                             339 3-(2'-Cl--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                             340 1,2,4-Thiadiazolyl-3                                                       341 5-CH.sub.3 -1,2,4-Thiadiazolyl-3                                           342 5-C.sub.6 H.sub.5 -1,2,4-Thiadiazolyl-3                                    343 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                     344 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                     345 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                     346 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                    347 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                    348 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                    349 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                     350 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                     351 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                     352 5-(4'-CN--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                            353 5-(3'-CN--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                            354 5-(2'-CN--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                            355 5-(4'-Cl--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                            356 5-(3'-Cl--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                            357 5-(2'-Cl--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                            358 1,3,4-Thiadiazolyl-2                                                       359 5-CH.sub.3 -1,3,4-Thiadiazolyl-2                                           360 5-C.sub.6 H.sub.5 -1,3,4-Thiadiazolyl-2                                    361 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                     362 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                     363 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                     364 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                    365 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                    366 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                    367 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                     368 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                     369 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                     370 5-(4'-CN--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                            371 5-(3'-CN--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                            372 5-(2'-CN--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                            373 5-(4'-Cl--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                            374 5-(3'-Cl--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                            375 5-(2'-Cl--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                            376 Pyridinyl-2                                                                377 Pyridinyl-4                                                                378 Pyridazinyl-3                                                              379 Pyridazinyl-4                                                              380 Pyridazinyl-2                                                              381 Pyrimidinyl-4                                                              382 Pyrimidinyl-5                                                              383 Pyrimidinyl-2                                                              384 Pyridinyl-3                                                                385 1-Naphthyl                                                                 386 2-Naphthyl                                                               ______________________________________                                    

                  TABLE 26                                                         ______________________________________                                         1  STR237##                                                                       - I: R.sup.1 = CH.sub.3, X = CH.sub.3                                         II: R.sup.1 = CH.sub.2 --CH.sub.3, X = CH.sub.3                                III: R.sup.1 = CH.sub.3, X = Cl                                                IV: R.sup.1 = CH.sub.2 --CH.sub.3, X = Cl                                      No.        T.sub.m                                                           ______________________________________                                          1       H                                                                        2 2-F                                                                          3 3-F                                                                          4 4-F                                                                          5 2,4-F.sub.2                                                                  6 2,4,6-F.sub.3                                                                7 2,3,4,5,6-F.sub.5                                                            8 2,3-F.sub.2                                                                  9 2-Cl                                                                         10 3-Cl                                                                        11 4-Cl                                                                        12 2,3-Cl.sub.2                                                                13 2,4-Cl.sub.2                                                                14 2,5-Cl.sub.2                                                                15 2,6-Cl.sub.2                                                                16 3,4-Cl.sub.2                                                                17 3,5-Cl.sub.2                                                                18 2,3,4-Cl.sub.3                                                              19 2,3,5-Cl.sub.3                                                              20 2,3,6-Cl.sub.3                                                              21 2,4,5-Cl.sub.3                                                              22 2,4,6-Cl.sub.3                                                              23 3,4,5-Cl.sub.3                                                              24 2,3,4,6-Cl.sub.4                                                            25 2,3,5,6-Cl.sub.4                                                            26 2,3,4,5,6-Cl.sub.5                                                          27 2-Br                                                                        28 3-Br                                                                        29 4-Br                                                                        30 2,4-Br.sub.2                                                                31 2,5-Br.sub.2                                                                32 2,6-Br.sub.2                                                                33 2,4,6-Br.sub.3                                                              34 2,3,4,5,6-Br.sub.5                                                          35 2-I                                                                         36 3-I                                                                         37 4-I                                                                         38 2,4-I.sub.2                                                                 39 2-Cl, 3-F                                                                   40 2-Cl, 4-F                                                                   41 2-Cl, 5-F                                                                   42 2-Cl, 6-F                                                                   43 2-Cl, 3-Br                                                                  44 2-Cl, 4-Br                                                                  45 2-Cl, 5-Br                                                                  46 2-Cl, 6-Br                                                                  47 2-Br, 3-Cl                                                                  48 2-Br, 4-Cl                                                                  49 2-Br, 5-Cl                                                                  50 2-Br, 3-F                                                                   51 2-Br, 4-F                                                                   52 2-Br, 5-F                                                                   53 2-Br, 6-F                                                                   54 2-F, 3-Cl                                                                   55 2-F, 4-Cl                                                                   56 2-F, 5-Cl                                                                   57 3-Cl, 4-F                                                                   58 3-Cl, 5-F                                                                   59 3-Cl, 4-Br                                                                  60 3-Cl, 5-Br                                                                  61 3-F, 4-Cl                                                                   62 3-F, 4-Br                                                                   63 3-Br, 4-Cl                                                                  64 3-Br, 4-F                                                                   65 2,6-Cl.sub.2, 4-Br                                                          66 2-CH.sub.3                                                                  67 3-CH.sub.3                                                                  68 4-CH.sub.3                                                                  69 2,3-(CH.sub.3).sub.2                                                        70 2,4-(CH.sub.3).sub.2                                                        71 2,5-(CH.sub.3).sub.2                                                        72 2,6-(CH.sub.3).sub.2                                                        73 3,4-(CH.sub.3).sub.2                                                        74 3,5-(CH.sub.3).sub.2                                                        75 2,3,5-(CH.sub.3).sub.3                                                      76 2,3,4-(CH.sub.3).sub.3                                                      77 2,3,6-(CH.sub.3).sub.3                                                      78 2,4,5-(CH.sub.3).sub.3                                                      79 2,4,6-(CH.sub.3).sub.3                                                      80 3,4,5-(CH.sub.3).sub.3                                                      81 2,3,4,6-(CH.sub.3).sub.4                                                    82 2,3,5,6-(CH.sub.3).sub.4                                                    83 2,3,4,5,6-(CH.sub.3).sub.5                                                  84 2-C.sub.2 H.sub.5                                                           85 3-C.sub.2 H.sub.5                                                           86 4-C.sub.2 H.sub.5                                                           87 2,4-(C.sub.2 H.sub.5).sub.2                                                 88 2,6-(C.sub.2 H.sub.5).sub.2                                                 89 3,5-(C.sub.2 H.sub.5).sub.2                                                 90 2,4,6-(C.sub.2 H.sub.5).sub.3                                               91 2-n-C.sub.3 H.sub.7                                                         92 3-n-C.sub.3 H.sub.7                                                         93 4-n-C.sub.3 H.sub.7                                                         94 2-i-C.sub.3 H.sub.7                                                         95 3-i-C.sub.3 H.sub.7                                                         96 4-i-C.sub.3 H.sub.7                                                         97 2,4-(i-C.sub.3 H.sub.7).sub.2                                               98 2,6-(i-C.sub.3 H.sub.7).sub.2                                               99 3,5-(i-C.sub.3 H.sub.7).sub.2                                              100 2,4,6-(i-C.sub.3 H.sub.7).sub.3                                            101 2-s-C.sub.4 H.sub.9                                                        102 3-s-C.sub.4 H.sub.9                                                        103 4-s-C.sub.4 H.sub.9                                                        104 2-t-C.sub.4 H.sub.9                                                        105 3-t-C.sub.4 H.sub.9                                                        106 4-t-C.sub.4 H.sub.9                                                        107 2,3-(t-C.sub.4 H.sub.9).sub.2                                              108 2,4-(t-C.sub.4 H.sub.9).sub.2                                              109 2,5-(t-C.sub.4 H.sub.9).sub.2                                              110 2,6-(t-C.sub.4 H.sub.9).sub.2                                              111 3,4-(t-C.sub.4 H.sub.9).sub.2                                              112 2,4,6-(t-C.sub.4 H.sub.9).sub.3                                            113 4-n-C.sub.9 H.sub.19                                                       114 4-n-C.sub.12 H.sub.25                                                      115 4-n-C.sub.15 H.sub.31                                                      116 4-(1,1,3,3-Tetramethylbutyl)                                               117 4-(2,4,4-Trimethylpropyl)                                                  118 2-t-C.sub.4 H.sub.9, 4-CH.sub.3                                            119 2-t-C.sub.4 H.sub.9, 5-CH.sub.3                                            120 2,6-(t-C.sub.4 H.sub.9).sub.2, 4-CH.sub.3                                  121 2-CH.sub.3, 4-t-C.sub.4 H.sub.9                                            122 2-CH.sub.3, 6-t-C.sub.4 H.sub.9                                            123 2-CH.sub.3, 4-i-C.sub.3 H.sub.7                                            124 2-CH.sub.3, 5-i-C.sub.3 H.sub.7                                            125 3-CH.sub.3, 4-i-C.sub.3 H.sub.7                                            126 2-i-C.sub.3 H.sub.7, 5-CH.sub.3                                            127 2,4-(t-C.sub.4 H.sub.9).sub.2, 6-i-C.sub.3 H.sub.7                         128 2-Allyl                                                                    129 3-Allyl                                                                    130 4-Allyl                                                                    131 2-Allyl, 6-CH.sub.3                                                        132 2-cyclo-C.sub.6 H.sub.11                                                   133 3-cyclo-C.sub.6 H.sub.11                                                   134 4-cyclo-C.sub.6 H.sub.11                                                   135 2,4-(cyclo-C.sub.6 H.sub.11).sub.2, 6-CH.sub.3                             136 2-CH.sub.3, 4-cyclo-C.sub.6 H.sub.11                                       137 2-CH.sub.2 --C.sub.6 H.sub.5                                               138 3-CH.sub.2 --C.sub.6 H.sub.5                                               139 4-CH.sub.2 --C.sub.6 H.sub.5                                               140 2-CH.sub.2 --C.sub.6 H.sub.5, 4-CH.sub.3                                   141 2-CH.sub.3, 4-CH.sub.2 --C.sub.6 H.sub.5                                   142 2-C.sub.6 H.sub.5                                                          143 3-C.sub.6 H.sub.5                                                          144 4-C.sub.6 H.sub.5                                                          145 4-(2-i-C.sub.3 H.sub.7 --C.sub.6 H.sub.4)                                  146 4-C.sub.6 H.sub.5, 2,6-(CH.sub.3).sub.2                                    147 2-Cl, 4-C.sub.6 H.sub.5                                                    148 2-Br, 4-C.sub.6 H.sub.5                                                    149 2-C.sub.6 H.sub.5, 4-Cl                                                    150 2-C.sub.6 H.sub.5, 4-Br                                                    151 2-CH.sub.2 C.sub.6 H.sub.5, 4-Cl                                           152 2-CH.sub.2 C.sub.6 H.sub.5, 4-Br                                           153 2-Cl, 4-CH.sub.2 C.sub.6 H.sub.5                                           154 2-Br, 4-CH.sub.2 C.sub.6 H.sub.5                                           155 2-cyclo-C.sub.6 H.sub.11, 4-Cl                                             156 2-cyclo-C.sub.6 H.sub.11, 4-Br                                             157 2-Cl, 4-cyclo-C.sub.6 H.sub.11                                             158 2-Br, 4-cyclo-C.sub.6 H.sub.11                                             159 2-OCH.sub.3                                                                160 3-OCH.sub.3                                                                161 4-OCH.sub.3                                                                162 2-OC.sub.2 H.sub.5                                                         163 3-O--C.sub.2 H.sub.5                                                       164 4-O--C.sub.2 H.sub.5                                                       165 2-O-n-C.sub.3 H.sub.7                                                      166 3-O-n-C.sub.3 H.sub.7                                                      167 4-O-n-C.sub.3 H.sub.7                                                      168 2-O-i-C.sub.3 H.sub.7                                                      169 3-O-i-C.sub.3 H.sub.7                                                      170 4-O-i-C.sub.3 H.sub.7                                                      171 2-O-n-C.sub.6 H.sub.13                                                     172 3-O-n-C.sub.6 H.sub.13                                                     173 4-O-n-C.sub.6 H.sub.13                                                     174 2-O-n-C.sub.8 H.sub.17                                                     175 3-O-n-C.sub.8 H.sub.17                                                     176 4-O-n-C.sub.8 H.sub.17                                                     177 2-O-CH.sub.2 C.sub.6 H.sub.5                                               178 3-O-CH.sub.2 C.sub.6 H.sub.5                                               179 4-O-CH.sub.2 C.sub.6 H.sub.5                                               180 2-O-(CH.sub.2).sub.3 C.sub.6 H.sub.5                                       181 3-O-(CH.sub.2).sub.3 C.sub.6 H.sub.5                                       182 4-O-(CH.sub.2).sub.3 C.sub.6 H.sub.5                                       183 2,4-(OCH.sub.3).sub.2                                                      184 2-CF.sub.3                                                                 185 3-CF.sub.3                                                                 186 4-CF.sub.3                                                                 187 2-OCF.sub.3                                                                188 3-OCF.sub.3                                                                189 4-OCF.sub.3                                                                190 3-OCH.sub.2 CHF.sub.2                                                      191 2-NO.sub.2                                                                 192 3-NO.sub.2                                                                 193 4-NO.sub.2                                                                 194 2-CN                                                                       195 3-CN                                                                       196 4-CN                                                                       197 2-CH.sub.3, 3-Cl                                                           198 2-CH.sub.3, 4-Cl                                                           199 2-CH.sub.3, 5-Cl                                                           200 2-CH.sub.3, 6-Cl                                                           201 2-CH.sub.3, 3-F                                                            202 2-CH.sub.3, 4-F                                                            203 2-CH.sub.3, 5-F                                                            204 2-CH.sub.3, 6-F                                                            205 2-CH.sub.3, 3-Br                                                           206 2-CH.sub.3, 4-Br                                                           207 2-CH.sub.3, 5-Br                                                           208 2-CH.sub.3, 6-Br                                                           209 2-Cl, 3-CH.sub.3                                                           210 2-Cl, 4-CH.sub.3                                                           211 2-Cl, 5-CH.sub.3                                                           212 2-F, 3-CH.sub.3                                                            213 2-F, 4-CH.sub.3                                                            214 2-F, 5-CH.sub.3                                                            215 2-Br, 3-CH.sub.3                                                           216 2-Br, 4-CH.sub.3                                                           217 2-Br, 5-CH.sub.3                                                           218 3-CH.sub.3, 4-Cl                                                           219 3-CH.sub.3, 5-Cl                                                           220 3-CH.sub.3, 4-F                                                            221 3-CH.sub.3, 5-F                                                            222 3-CH.sub.3, 4-Br                                                           223 3-CH.sub.3, 5-Br                                                           224 3-F, 4-CH.sub.3                                                            225 3-Cl, 4-CH.sub.3                                                           226 3-Br, 4-CH.sub.3                                                           227 2-Cl, 4,5-(CH.sub.3).sub.2                                                 228 2-Br, 4,5-(CH.sub.3).sub.2                                                 229 2-Cl, 3,5-(CH.sub.3).sub.2                                                 230 2-Br, 3,5-(CH.sub.3).sub.2                                                 231 2,6-Cl.sub.2, 4-CH.sub.3                                                   232 2,6-F.sub.2, 4-CH.sub.3                                                    233 2,6-Br.sub.2, 4-CH.sub.3                                                   234 2,4-Br.sub.2, 6-CH.sub.3                                                   235 2,4-F.sub.2, 6-CH.sub.3                                                    236 2,4-Br.sub.2, 6-CH.sub.3                                                   237 2,6-(CH.sub.3).sub.2, 4-F                                                  238 2,6-(CH.sub.3).sub.2, 4-Cl                                                 239 2,6-(CH.sub.3).sub.2, 4-Br                                                 240 3,5-(CH.sub.3).sub.2, 4-F                                                  241 3,5-(CH.sub.3).sub.2, 4-Cl                                                 242 3,5-(CH.sub.3).sub.2, 4-Br                                                 243 2,3,6-(CH.sub.3).sub.3, 4-F                                                244 2,3,6-(CH.sub.3).sub.3, 4-Cl                                               245 2,3,6-(CH.sub.3).sub.3, 4-Br                                               246 2,4-(CH.sub.3).sub.2, 6-F                                                  247 2,4-(CH.sub.3).sub.2, 6-Cl                                                 248 2,4-(CH.sub.3).sub.2, 6-Br                                                 249 2-i-C.sub.3 H.sub.7, 4-Cl, 5-CH.sub.3                                      250 2-Cl, 4-NO.sub.2                                                           251 2-NO.sub.2, 4-Cl                                                           252 2-OCH.sub.3, 5-NO.sub.2                                                    253 2,4-Cl.sub.2, 5-NO.sub.2                                                   254 2,4-Cl.sub.2, 6-NO.sub.2                                                   255 2,6-Cl.sub.2, 4-NO.sub.2                                                   256 2,6-Br.sub.2, 4-NO.sub.2                                                   257 2,6-I.sub.2, 4-NO.sub.2                                                    258 2-CH.sub.3, 5-i-C.sub.3 H.sub.7, 4-Cl                                      259 2-CO.sub.2 CH.sub.3                                                        260 3-CO.sub.2 CH.sub.3                                                        261 4-CO.sub.2 CH.sub.3                                                        262 2-CO.sub.2 (C.sub.2 H.sub.5)                                               263 3-CO.sub.2 (C.sub.2 H.sub.5)                                               264 4-CO.sub.2 (C.sub.2 H.sub.5)                                               265 2-CO.sub.2 (n-C.sub.3 H.sub.7)                                             266 3-CO.sub.2 (n-C.sub.3 H.sub.7)                                             267 4-CO.sub.2 (n-C.sub.3 H.sub.7)                                             268 2-CO.sub.2 (i-C.sub.3 H.sub.7)                                             269 3-CO.sub.2 (i-C.sub.3 H.sub.7)                                             270 4-CO.sub.2 (i-C.sub.3 H.sub.7)                                             271 2-CO.sub.2 (n-C.sub.6 H.sub.13)                                            272 3-CO.sub.2 (n-C.sub.6 H.sub.13)                                            273 4-CO.sub.2 (n-C.sub.6 H.sub.13)                                            274 2-CH.sub.2 --OCH.sub.3                                                     275 3-CH.sub.2 --OCH.sub.3                                                     276 4-CH.sub.2 --OCH.sub.3                                                     277 2-CH.sub.2 O(C.sub.2 H.sub.5)                                              278 3-CH.sub.2 O(C.sub.2 H.sub.5)                                              279 4-CH.sub.2 O(C.sub.2 H.sub.5)                                              280 2-CH.sub.2 O(n-C.sub.3 H.sub.7)                                            281 3-CH.sub.2 O(n-C.sub.3 H.sub.7)                                            282 4-CH.sub.2 O(n-C.sub.3 H.sub.7)                                            283 2-CH.sub.2 O(i-C.sub.3 H.sub.7)                                            284 3-CH.sub.2 O(i-C.sub.3 H.sub.7)                                            285 4-CH.sub.2 O(i-C.sub.3 H.sub.7)                                            286 2-CHO                                                                      287 3-CHO                                                                      288 4-CHO                                                                      289 2-CO--CH.sub.3                                                             290 3-CO--CH.sub.3                                                             291 4-CO--CH.sub.3                                                             292 2-CO--CH.sub.2 --CH.sub.3                                                  293 3-CO--CH.sub.2 --CH.sub.3                                                  294 4-CO--CH.sub.2 --CH.sub.3                                                  295 2-CO--CH.sub.2 --CH.sub.2 --CH.sub.3                                       296 3-CO--CH.sub.2 --CH.sub.2 --CH.sub.3                                       297 4-CO--CH.sub.2 --CH.sub.2 --CH.sub.3                                       298 2-CO--CH(CH.sub.3)--CH.sub.3                                               299 3-CO--CH(CH.sub.3)--CH.sub.3                                               300 4-CO--CH(CH.sub.3)--CH.sub.3                                               301 2-Me-4-CHO                                                                 302 2-Me-4-CH.sub.3 --CO                                                       303 2-Me-4-CH.sub.3 --CH.sub.2 --CO                                            304 2-Me-4-CH.sub.3 --CH.sub.2 --CH.sub.2 --CO                                 305 2-Me-4-CH.sub.3 --CH(CH.sub.3)--CO                                         306 2,5-Me.sub.2 -4-CHO                                                        307 2,5-Me.sub.2 -4-CH.sub.3 --CO                                              308 2,5-Me.sub.2 -4-CH.sub.3 --CH.sub.2 --CO                                   309 2,5-Me.sub.2 -4-CH.sub.3 --CH.sub.2 --CH.sub.2 --CO                        310 2,5-Me.sub.2 -4-CH.sub.3 --CH(CH.sub.3)--CO                                311 2-Cl-4-CHO                                                                 312 2-Cl-4-CH.sub.3 --CO                                                       313 2-Cl-4-CH.sub.3 --CH.sub.2 --CO                                            314 2-Cl-4-CH.sub.3 --CH(CH.sub.3)--CO                                         315 2,5-Cl.sub.2 -4-CHO                                                        316 2,5-Cl.sub.2 -4-CH.sub.3 --CO                                              317 2,5-Cl.sub.2 -4-CH.sub.3 --CH.sub.2 --CO                                   318 2,5-Cl.sub.2 -4-CH.sub.3 --CH.sub.2 --CH.sub.2 --CO                        319 2,5-Cl.sub.2 -4-CH.sub.3 --CH(CH.sub.3)--CO                                320 2-C(═NOCH.sub.3)--CH.sub.3                                             321 3-C(═NOCH.sub.3)--CH.sub.3                                             322 4-C(═NOCH.sub.3)--CH.sub.3                                             323 2-C(═NOC.sub.2 H.sub.5)--CH.sub.3                                      324 3-C(═NOC.sub.2 H.sub.5)--CH.sub.3                                      325 4-C(═NOC.sub.2 H.sub.5)--CH.sub.3                                      326 2-C(═NO-n-C.sub.3 H.sub.7)--CH.sub.3                                   327 3-C(═NO-n-C.sub.3 H.sub.7)--CH.sub.3                                   328 4-C(═NO-n-C.sub.3 H.sub.7)--CH.sub.3                                   329 2-C(═NO-i-C.sub.3 H.sub.7)--CH.sub.3                                   330 3-C(═NO-i-C.sub.3 H.sub.7)--CH.sub.3                                   331 4-C(═NO-i-C.sub.3 H.sub.7)--CH.sub.3                                   332 2-C(═NO-Allyl)--CH.sub.3                                               333 3-C(═NO-Allyl)--CH.sub.3                                               334 4-C(═NO-Allyl)--CH.sub.3                                               335 2-C(═NO-trans-Chloroallyl)--CH.sub.3                                   336 3-C(═NO-trans-Chloroallyl)--CH.sub.3                                   337 4-C(═NO-trans-Chloroallyl)--CH.sub.3                                   338 2-C(═NO-Propargyl)--CH.sub.3                                           339 3-C(═NO-Propargyl)--CH.sub.3                                           340 4-C(═NO-Propargyl)--CH.sub.3                                           341 2-C(═NO-n-C.sub.4 H.sub.9)--CH.sub.3                                   342 3-C(═NO-n-C.sub.4 H.sub.9)--CH.sub.3                                   343 4-C(═NO-n-C.sub.4 H.sub.9)--CH.sub.3                                   344 2-C(═NO--CH.sub.2 --C.sub.6 H.sub.5)--CH.sub.3                         345 3-C(═NO--CH.sub.2 --C.sub.6 H.sub.5)--CH.sub.3                         346 4-C(═NO--CH.sub.2 --C.sub.6 H.sub.5)--CH.sub.3                         347 2-CH.sub.3 -4-CH═NOCH.sub.3                                            348 2-CH.sub.3 -4-CH═NOC.sub.2 H.sub.5                                     349 2-CH.sub.3 -4-CH═NO-n-C.sub.3 H.sub.7                                  350 2-CH.sub.3 -4-CH═NO-i-C.sub.3 H.sub.7                                  351 2-CH.sub.3 -4-CH═NO-Allyl                                              352 2-CH.sub.3 -4-CH═NO-(trans-Chloroallyl)                                353 2-CH.sub.3 -4-CH═NO-Propargyl                                          354 2-CH.sub.3 -4-CH═NO-n-C.sub.4 H.sub.9                                  355 2-CH.sub.3 -4-CH═NO--CH.sub.2 --C.sub.6 H.sub.5                        356 2-CH.sub.3 -4-(CH.sub.3 --C═NOCH.sub.3)                                357 2-CH.sub.3 -4-(CH.sub.3 --C═NOC.sub.2 H.sub.5)                         358 2-CH.sub.3 -4-(CH.sub.3 --C═NO-n-C.sub.3 H.sub.7)                      359 2-CH.sub.3 -4-(CH.sub.3 --C═NO-i-C.sub.3 H.sub.7)                      360 2-CH.sub.3 -4-(CH.sub.3 --C═NO-Allyl)                                  361 2-CH.sub.3 -4-(CH.sub.3 --C═NO-trans-Chloroallyl)                      362 2-CH.sub.3 -4-(CH.sub.3 --C═NO-Propargyl)                              363 2-CH.sub.3 -4-(CH.sub.3 --C═NO-n-C.sub.4 H.sub.9)                      364 2-CH.sub.3 -4-(CH.sub.3 --C═NO--CH.sub.2 --C.sub.6 H.sub.5)                    365 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C═NO--CH.sub.3)                       366 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C═NO--C.sub.2 H.sub.5)        367 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C═NO-n-C.sub.3 H.sub.7)                       368 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C═NO-i-C.sub.3                       H.sub.7)                                                                369 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C═NO-Allyl)                           370 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C═NO-trans-Chloroallyl)                       371 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C═NO-Propargyl)                       372 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C═NO-n-C.sub.4                       H.sub.9)                                                                373 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C═NO--CH.sub.2 --C.sub.6                     H.sub.5)                                                                374 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C═NOCH.sub.3)                      375 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C═NOC.sub.2 H.sub.5)                       376 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C═NO-n-C.sub.3                    H.sub.7)                                                                377 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C═NO-i-C.sub.3 H.sub.7)                    378 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C═NO-Allyl)                        379 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C═NO-trans-Chloroall              yl)                                                                     380 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C═NO-Proparyl)                     381 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C═NO-n-C.sub.4 H.sub.9)                    382 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C═NO--CH.sub.2                    --C.sub.6 H.sub.5)                                                      383 2-C.sub.6 H.sub.5                                                          384 3-C.sub.6 H.sub.5                                                          385 4-C.sub.6 H.sub.5                                                          386 2-(2'-F--C.sub.6 H.sub.4)                                                  387 2-(3'-F--C.sub.6 H.sub.4)                                                  388 2-(4'-F--C.sub.6 H.sub.4)                                                  389 3-(2'-F--C.sub.6 H.sub.4)                                                  390 3-(3'-F--C.sub.6 H.sub.4)                                                  391 3-(4'-F--C.sub.6 H.sub.4)                                                  392 4-(2'-F--C.sub.6 H.sub.4)                                                  393 4-(3'-F--C.sub.6 H.sub.4)                                                  394 4-(4'-F--C.sub.6 H.sub.4)                                                  395 2-(2'-Cl--C.sub.6 H.sub.4)                                                 396 2-(3'-Cl--C.sub.6 H.sub.4)                                                 397 2-(4'-Cl--C.sub.6 H.sub.4)                                                 398 3-(2'-Cl--C.sub.6 H.sub.4)                                                 399 3-(3'-Cl--C.sub.6 H.sub.4)                                                 400 3-(4'-Cl--C.sub.6 H.sub.4)                                                 401 4-(2'-Cl--C.sub.6 H.sub.4)                                                 402 4-(3'-Cl--C.sub.6 H.sub.4)                                                 403 4-(4'-Cl--C.sub.6 H.sub.4)                                                 405 2-(2'-CH.sub.3 --C.sub.6 H.sub.4)                                          406 2-(3'-CH.sub.3 --C.sub.6 H.sub.4)                                          407 2-(4'-CH.sub.3 --C.sub.6 H.sub.4)                                          408 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)                                          409 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)                                          410 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)                                          411 4-(2'-CH.sub.3 --C.sub.6 H.sub.4)                                          412 4-(3'-CH.sub.3 --C.sub.6 H.sub.4)                                          413 4-(4'-CH.sub.3 --C.sub.6 H.sub.4)                                          414 2-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                      415 2-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                      416 2-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                      417 3-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                      418 3-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                      419 3-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                      420 4-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                      421 4-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                      422 4-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                      423 2-(2'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                       424 2-(3'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                       425 2-(4'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                       426 3-(2'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                       427 3-(3'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                       428 3-(4'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                       429 4-(2'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                       430 4-(3'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                       431 4-(4'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                       432 2-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                                 433 2-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                                 434 2-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                                 435 3-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                                 436 3-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                                 437 3-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                                 438 4-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                                 439 4-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                                 440 4-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                                 441 2-(2'-CH.sub.3 O--C.sub.6 H.sub.4)                                         442 2-(3'-CH.sub.3 O--C.sub.6 H.sub.4)                                         443 2-(4'-CH.sub.3 O--C.sub.6 H.sub.4)                                         444 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)                                         445 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)                                         446 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)                                         447 4-(2'-CH.sub.3 O--C.sub.6 H.sub.4)                                         448 4-(3'-CH.sub.3 O--C.sub.6 H.sub.4)                                         449 4-(4'-CH.sub.3 O--C.sub.6 H.sub.4)                                         450 2-(2'-O.sub.2 N--C.sub.6 H.sub.4)                                          451 2-(3'-O.sub.2 N--C.sub.6 H.sub.4)                                          452 2-(4'-O.sub.2 N--C.sub.6 H.sub.4)                                          453 3-(2'-O.sub.2 N--C.sub.6 H.sub.4)                                          454 3-(3'-O.sub.2 N--C.sub.6 H.sub.4)                                          455 3-(4'-O.sub.2 N--C.sub.6 H.sub.4)                                          456 4-(2'-O.sub.2 N--C.sub.6 H.sub.4)                                          457 4-(3'-O.sub.2 N--C.sub.6 H.sub.4)                                          458 4-(4'-O.sub.2 N--C.sub.6 H.sub.4)                                          459 2-(2'-NC--C.sub.6 H.sub.4)                                                 460 2-(3'-NC--C.sub.6 H.sub.4)                                                 461 2-(4'-NC--C.sub.6 H.sub.4)                                                 462 3-(2'-NC--C.sub.6 H.sub.4)                                                 463 3-(3'-NC--C.sub.6 H.sub.4)                                                 464 3-(4'-NC--C.sub.6 H.sub.4)                                                 465 4-(2'-NC--C.sub.6 H.sub.4)                                                 466 4-(3'-NC--C.sub.6 H.sub.4)                                                 467 4-(4'-NC--C.sub.6 H.sub.4)                                                 468 2-(2'-CF.sub.3 --C.sub.6 H.sub.4)                                          469 2-(3'-CF.sub.3 --C.sub.6 H.sub.4)                                          470 2-(4'-CF.sub.3 --C.sub.6 H.sub.4)                                          471 3-(2'-CF.sub.3 --C.sub.6 H.sub.4)                                          472 3-(3'-CF.sub.3 --C.sub.6 H.sub.4)                                          473 3-(4'-CF.sub.3 --C.sub.6 H.sub.4)                                          474 4-(2'-CF.sub.3 --C.sub.6 H.sub.4)                                          475 4-(3'-CF.sub.3 --C.sub.6 H.sub.4)                                          476 4-(4'-CF.sub.3 --C.sub.6 H.sub.4)                                          477 2-O-C.sub.6 H.sub.5                                                        475 3-O-C.sub.6 H.sub.5                                                        476 4-O-C.sub.6 H.sub.5                                                        478 2-O-(2'-F--C.sub.6 H.sub.4)                                                479 2-O-(3'-F--C.sub.6 H.sub.4)                                                480 2-O-(4'-F--C.sub.6 H.sub.4)                                                481 3-O-(2'-F--C.sub.6 H.sub.4)                                                482 3-O-(3'-F--C.sub.6 H.sub.4)                                                483 3-O-(4'-F--C.sub.6 H.sub.4)                                                484 4-O-(2'-F--C.sub.6 H.sub.4)                                                485 4-O-(3'-F--C.sub.6 H.sub.4)                                                486 4-O-(4'-F--C.sub.6 H.sub.4)                                                487 2-O-(2'-Cl--C.sub.6 H.sub.4)                                               488 2-O-(3'-Cl--C.sub.6 H.sub.4)                                               489 2-O-(4'-Cl--C.sub.6 H.sub.4)                                               490 3-O-(2'-Cl--C.sub.6 H.sub.4)                                               491 3-O-(3'-Cl--C.sub.6 H.sub.4)                                               492 3-O-(4'-Cl--C.sub.6 H.sub.4)                                               493 3-O-(4'-Cl--C.sub.6 H.sub.4)                                               494 4-O-(2'-Cl--C.sub.6 H.sub.4)                                               495 4-O-(3'-Cl--C.sub.6 H.sub.4)                                               496 4-O-(4'-Cl--C.sub.6 H.sub.4)                                               497 2-O-(2'-CH.sub.3 --C.sub.6 H.sub.4)                                        498 2-O-(3'-CH.sub.3 --C.sub.6 H.sub.4)                                        499 2-O-(4'-CH.sub.3 --C.sub.6 H.sub.4)                                        500 3-O-(2'-CH.sub.3 --C.sub.6 H.sub.4)                                        501 3-O-(3'-CH.sub.3 --C.sub.6 H.sub.4)                                        502 3-O-(4'-CH.sub.3 --C.sub.6 H.sub.4)                                        503 4-O-(2'-CH.sub.3 --C.sub.6 H.sub.4)                                        504 4-O-(3'-CH.sub.3 --C.sub.6 H.sub.4)                                        505 4-O-(4'-CH.sub.3 --C.sub.6 H.sub.4)                                        506 2-O-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                    507 2-O-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                    508 2-O-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                    509 3-O-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                    510 3-O-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                    511 3-O-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                    512 4-O-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                    513 4-O-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                    514 4-O-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                    515 2-O-(2'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                     516 2-O-(3'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                     517 2-O-(4'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                     518 3-O-(2'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                     519 3-O-(3'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                     520 3-O-(4'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                     521 4-O-(2'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                     522 4-O-(3'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                     523 4-O-(4'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                     524 2-O-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                               525 2-O-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                               526 2-O-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                               527 3-O-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                               528 3-O-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                               529 3-O-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                               530 4-O-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                               531 4-O-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                               532 4-O-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                               533 2-O-(2'-CH.sub.3 O--C.sub.6 H.sub.4)                                       534 2-O-(3'-CH.sub.3 O--C.sub.6 H.sub.4)                                       535 2-O-(4'-CH.sub.3 O--C.sub.6 H.sub.4)                                       536 3-O-(2'-CH.sub.3 O--C.sub.6 H.sub.4)                                       537 3-O-(3'-CH.sub.3 O--C.sub.6 H.sub.4)                                       538 3-O-(4'-CH.sub.3 O--C.sub.6 H.sub.4)                                       539 4-O-(2'-CH.sub.3 O--C.sub.6 H.sub.4)                                       540 4-O-(3'-CH.sub.3 O--C.sub.6 H.sub.4)                                       541 4-O-(4'-CH.sub.3 O--C.sub.6 H.sub.4)                                       542 2-O-(2'-O.sub.2 N--C.sub.6 H.sub.4)                                        543 2-O-(3'-O.sub.2 N--C.sub.6 H.sub.4)                                        544 2-O-(4'-O.sub.2 N--C.sub.6 H.sub.4)                                        545 3-O-(2'-O.sub.2 N--C.sub.6 H.sub.4)                                        546 3-O-(3'-O.sub.2 N--C.sub.6 H.sub.4)                                        547 3-O-(4'-O.sub.2 N--C.sub.6 H.sub.4)                                        548 4-O-(2'-O.sub.2 N--C.sub.6 H.sub.4)                                        549 4-O-(3'-O.sub.2 N--C.sub.6 H.sub.4)                                        550 4-O-(4'-O.sub.2 N--C.sub.6 H.sub.4)                                        551 2-O-(2'-NC--C.sub.6 H.sub.4)                                               552 2-O-(3'-NC--C.sub.6 H.sub.4)                                               553 2-O-(4'-NC--C.sub.6 H.sub.4)                                               554 3-O-(2'-NC--C.sub.6 H.sub.4)                                               555 3-O-(3'-NC--C.sub.6 H.sub.4)                                               556 3-O-(4'-NC--C.sub.6 H.sub.4)                                               557 4-O-(2'-NC--C.sub.6 H.sub.4)                                               558 4-O-(3'-NC--C.sub.6 H.sub.4)                                               559 4-O-(4'-NC--C.sub.6 H.sub.4)                                               560 2-O-(2'-CF.sub.3 --C.sub.6 H.sub.4)                                        561 2-O-(3'-CF.sub.3 --C.sub.6 H.sub.4)                                        562 2-O-(4'-CF.sub.3 --C.sub.6 H.sub.4)                                        563 3-O-(2'-CF.sub.3 --C.sub.6 H.sub.4)                                        564 3-O-(3'-CF.sub.3 --C.sub.6 H.sub.4)                                        565 3-O-(4'-CF.sub.3 --C.sub.6 H.sub.4)                                        566 4-O-(2'-CF.sub.3 --C.sub.6 H.sub.4)                                        567 4-O-(3'-CF.sub.3 --C.sub.6 H.sub.4)                                        568 4-O-(4'-CF.sub.3 --C.sub.6 H.sub.4)                                        569 2-Pyridinyl-2'                                                             570 2-Pyridinyl-3'                                                             571 2-Pyridinyl-4'                                                             572 3-Pyridinyl-2'                                                             573 3-Pyridinyl-3'                                                             574 3-Pyridinyl-4'                                                             575 4-Pyridinyl-2'                                                             576 4-Pyridinyl-3'                                                             577 4-Pyridinyl-4'                                                             578 2-Pyrimidinyl-2'                                                           579 2-Pyrimidinyl-3'                                                           580 2-Pyrimidinyl-4'                                                           581 3-Pyrimidinyl-2'                                                           582 3-Pyrimidinyl-3'                                                           583 3-Pyrimidinyl-4'                                                           584 4-Pyrimidinyl-2'                                                           585 4-Pyrimidinyl-3'                                                           586 4-Pyrimidinyl-4'                                                           587 2-Pyrazolyl-1'                                                             588 2-Pyrazolyl-3'                                                             589 2-Pyrazolyl-4'                                                             590 3-Pyrazolyl-1'                                                             591 3-Pyrazolyl-3'                                                             592 3-Pyrazolyl-4'                                                             593 4-Pyrazolyl-1'                                                             594 4-Pyrazolyl-3'                                                             595 4-Pyrazolyl-4'                                                             596 2-Isoxazolyl-3'                                                            597 2-Isoxazolyl-4'                                                            598 2-Isoxazolyl-5'                                                            599 3-Isoxazolyl-3'                                                            600 3-Isoxazolyl-4'                                                            601 3-Isoxazolyl-5'                                                            602 4-Isoxazolyl-3'                                                            603 4-Isoxazolyl-4'                                                            604 4-Isoxazolyl-5'                                                            605 2-Isothiazolyl-3'                                                          606 2-Isothiazolyl-4'                                                          607 2-Isothiazolyl-5'                                                          608 3-Isothiazolyl-3'                                                          609 3-Isothiazolyl-4'                                                          610 3-Isothiazolyl-5'                                                          611 4-Isothiazolyl-3'                                                          612 4-Isothiazolyl-4'                                                          613 4-Isothiazolyl-5'                                                          614 2-Imidazolyl-1'                                                            615 2-Imidazolyl-2'                                                            616 2-Imidazolyl-4'                                                            617 3-Imidazolyl-1'                                                            618 3-Imidazolyl-2'                                                            619 3-Imidazolyl-4'                                                            620 4-Imidazolyl-1'                                                            621 4-Imidazolyl-2'                                                            622 4-Imidazolyl-4'                                                            623 2-Oxazolyl-2'                                                              624 2-Oxazolyl-4'                                                              625 2-Oxazolyl-5'                                                              626 3-Oxazolyl-2'                                                              627 3-Oxazolyl-4'                                                              628 3-Oxazolyl-5'                                                              629 4-Oxazolyl-2'                                                              630 4-Oxazolyl-4'                                                              631 4-Oxazolyl-5'                                                              632 2-Thiazolyl-2'                                                             633 2-Thiazolyl-4'                                                             634 2-Thiazolyl-5'                                                             635 3-Thiazolyl-2'                                                             636 3-Thiazolyl-4'                                                             637 3-Thiazolyl-5'                                                             638 4-Thiazolyl-2'                                                             639 4-Thiazolyl-4'                                                             640 4-Thiazolyl-5'                                                             641 2-CH.sub.3 -4-(CH.sub.3 --C═N--O--CH.sub.2 --CH.sub.2 --OCH.sub.              3)                                                                      642 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C═N--O--CH.sub.2 --CH.sub.2                  --OCH.sub.3)                                                            643 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C═N--O--CH.sub.2 --CH.sub.2               --OCH.sub.3)                                                            644 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C═N--OCH.sub.3)                     645 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C═N--OC.sub.2 H.sub.5)                      646 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C═N--O-n-C.sub.3                   H.sub.7)                                                                647 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C═N--O-i-C.sub.3 H.sub.7)                   648 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C═N--O-Allyl)                       649 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C═N--O-trans-Chloroal              lyl)                                                                    650 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C═N--O-Propargyl)                   651 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C═N--O-n-C.sub.4 H.sub.9)                   652 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C═N--O--CH.sub.2                   --C.sub.6 H.sub.5)                                                      653 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C═N--OCH.sub.3)                     654 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C═N--OC.sub.2 H.sub.5)                      655 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C═N--O-n-C.sub.3                   H.sub.7)                                                                656 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C═N--O-i-C.sub.3 H.sub.7)                   657 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C═N--O-Allyl)                       658 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C═N--O-trans-Chloroal              lyl)                                                                    659 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C═N--O-Propargyl)                   660 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C═N--O-n-C.sub.4 H.sub.9)                   661 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C═N--O--CH.sub.2                   --C.sub.6 H.sub.5)                                                      662 2-O-n-C.sub.4 H.sub.9                                                      663 2-O-i-C.sub.4 H.sub.9                                                      664 2-O-s-C.sub.4 H.sub.9                                                      665 2-O-t-C.sub.4 H.sub.9                                                      666 2-Neopentyloxy                                                             667 3-O-n-C.sub.4 H.sub.9                                                      668 3-O-i-C.sub.4 H.sub.9                                                      669 3-O-s-C.sub.4 H.sub.9                                                      670 3-O-t-C.sub.4 H.sub.9                                                      671 3-Neopentyloxy                                                             672 4-O-n-C.sub.4 H.sub.9                                                      673 4-O-i-C.sub.4 H.sub.9                                                      674 4-O-s-C.sub.4 H.sub.9                                                      675 4-O-t-C.sub.4 H.sub.9                                                      676 4-Neopentyloxy                                                             677 3-CH.sub.3 -4-OCH.sub.3                                                    678 3-CH.sub.3 -4-OC.sub.2 H.sub.5                                             679 3-CH.sub.3 -4-O-n-C.sub.3 H.sub.7                                          680 3-CH.sub.3 -4-O-n-C.sub.4 H.sub.9                                          681 3-CH.sub.3 -4-O-i-C.sub.4 H.sub.9                                          682 3-CH.sub.3 -4-O-s-C.sub.4 H.sub.9                                          683 3-CH.sub.3 -4-O-t-C.sub.4 H.sub.9                                          684 3-CH.sub.3 -4-Neopentyloxy                                                 685 2-CH.sub.3 -3-OCH.sub.3                                                    686 2-CH.sub.3 -4-OCH.sub.3                                                    687 2-CH.sub.3 -5-OCH.sub.3                                                    688 2-CH.sub.3 -6-OCH.sub.3                                                    689 3-CH.sub.3 -4-OCH.sub.3                                                    690 3-CH.sub.3 -5-OCH.sub.3                                                    691 3-CH.sub.3 -6-OCH.sub.3                                                    692 4-CH.sub.3 -5-O--CH.sub.3                                                  693 4-CH.sub.3 -6-O--CH.sub.3                                                  694 4-CH.sub.3 -6-OCH.sub.3                                                    695 2-CH.sub.3 -3-O-i-C.sub.3 H.sub.7                                          696 2-CH.sub.3 -4-O-i-C.sub.3 H.sub.7                                          697 2-CH.sub.3 -5-O-i-C.sub.3 H.sub.7                                          698 2-CH.sub.3 -6-O-i-C.sub.3 H.sub.7                                          699 3-CH.sub.3 -4-O-i-C.sub.3 H.sub.7                                          700 3-CH.sub.3 -5-O-i-C.sub.3 H.sub.7                                          701 3-CH.sub.3 -6-O-i-C.sub.3 H.sub.7                                          702 4-CH.sub.3 -5-O-i-C.sub.3 H.sub.7                                          703 4-CH.sub.3 -6-O-i-C.sub.3 H.sub.7                                          704 5-CH.sub.3 -6-O-i-C.sub.3 H.sub.7                                          705 2-Cl-3-OCH.sub.3                                                           706 2-Cl-4-OCH.sub.3                                                           707 2-Cl-5-OCH.sub.3                                                           708 2-Cl-6-OCH.sub.3                                                           709 3-Cl-4-OCH.sub.3                                                           710 3-Cl-5-OCH.sub.3                                                           711 3-Cl-6-OCH.sub.3                                                           712 4-Cl-5-OCH.sub.3                                                           713 4-Cl-6-OCH.sub.3                                                           714 5-Cl-6-OCH.sub.3                                                         ______________________________________                                    

                  TABLE 27                                                         ______________________________________                                         2  STR238##                                                                      I: R.sup.1 = CH.sub.3, X = CH.sub.3                                            II: R.sup.1 = CH.sub.2 --CH.sub.3, X = CH.sub.3                                III: R.sup.1 = CH.sub.3, X = Cl                                                IV: R.sup.1 = CH.sub.2 --CH.sub.3, X = Cl                                      No.         B                                                                ______________________________________                                         1         Pyrrolyl-3                                                             2 N--CH.sub.3 -Pyrrolyl-3                                                      3 N--C.sub.6 H.sub.5 -Pyrrolyl-3                                               4 N-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrrolyl-3                                 5 N-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrrolyl-3                                 6 N-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrrolyl-3                                 7 N-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrrolyl-3                                8 N-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrrolyl-3                                9 N-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrrolyl-3                                10 N-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrrolyl-3                                11 N-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrrolyl-3                                12 N-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrrolyl-3                                13 N-(4'-CN--C.sub.6 H.sub.4)-Pyrrolyl-3                                       14 N-(3'-CN--C.sub.6 H.sub.4)-Pyrrolyl-3                                       15 N-(2'-CN--C.sub.6 H.sub.4)-Pyrrolyl-3                                       16 N-(4'-Cl--C.sub.6 H.sub.4)-Pyrrolyl-3                                       17 N-(3'-Cl--C.sub.6 H.sub.4)-Pyrrolyl-3                                       18 N-(2'-Cl--C.sub.6 H.sub.4)-Pyrrolyl-3                                       19 Pyrrolyl-2                                                                  20 N--CH.sub.3 -Pyrrolyl-2                                                     21 N--C.sub.6 H.sub.5 -Pyrrolyl-2                                              22 N-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrrolyl-2                                23 N-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrrolyl-2                                24 N-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrrolyl-2                                25 N-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrrolyl-2                               26 N-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrrolyl-2                               27 N-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrrolyl-2                               28 N-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrrolyl-2                                29 N-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrrolyl-2                                30 N-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrrolyl-2                                31 N-(4'-CN--C.sub.6 H.sub.4)-Pyrrolyl-2                                       32 N-(3'-CN--C.sub.6 H.sub.4)-Pyrrolyl-2                                       33 N-(2'-CN--C.sub.6 H.sub.4)-Pyrrolyl-2                                       34 N-(4'-Cl--C.sub.6 H.sub.4)-Pyrrolyl-2                                       35 N-(3'-Cl--C.sub.6 H.sub.4)-Pyrrolyl-2                                       36 N-(2'-Cl--C.sub.6 H.sub.4)-Pyrrolyl-2                                       37 Furyl-2                                                                     38 5-CH.sub.3 -Furyl-2                                                         39 5-C.sub.6 H.sub.5 -Furyl-2                                                  40 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Furyl-2                                   41 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Furyl-2                                   42 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Furyl-2                                   43 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Furyl-2                                  44 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Furyl-2                                  45 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Furyl-2                                  46 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Furyl-2                                   47 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Furyl-2                                   48 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Furyl-2                                   49 5-(4'-CN--C.sub.6 H.sub.4)-Furyl-2                                          50 5-(3'-CN--C.sub.6 H.sub.4)-Furyl-2                                          51 5-(2'-CN--C.sub.6 H.sub.4)-Furyl-2                                          52 5-(4'-Cl--C.sub.6 H.sub.4)-Furyl-2                                          53 5-(3'-Cl--C.sub.6 H.sub.4)-Furyl-2                                          54 5-(2'-Cl--C.sub.6 H.sub.4)-Furyl-2                                          55 4-CH.sub.3 -Furyl-2                                                         56 4-C.sub.6 H.sub.5 -Furyl-2                                                  57 4-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Furyl-2                                   58 4-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Furyl-2                                   59 4-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Furyl-2                                   60 4-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Furyl-2                                  61 4-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Furyl-2                                  62 4-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Furyl-2                                  63 4-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Furyl-2                                   64 4-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Furyl-2                                   65 4-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Furyl-2                                   66 4-(4'-CN--C.sub.6 H.sub.4)-Furyl-2                                          67 4-(3'-CN--C.sub.6 H.sub.4)-Furyl-2                                          68 4-(2'-CN--C.sub.6 H.sub.4)-Furyl-2                                          69 4-(4'-Cl--C.sub.6 H.sub.4)-Furyl-2                                          70 4-(3'-Cl--C.sub.6 H.sub.4)-Furyl-2                                          71 4-(2'-Cl--C.sub.6 H.sub.4)-Furyl-2                                          72 Thienyl-2                                                                   73 5-CH.sub.3 -Thienyl-2                                                       74 5-C.sub.6 H.sub.5 -Thienyl-2                                                75 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-2                                 76 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-2                                 77 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-2                                 78 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-2                                79 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-2                                80 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-2                                81 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-2                                 82 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-2                                 83 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-2                                 84 5-(4'-CN--C.sub.6 H.sub.4)-Thienyl-2                                        85 5-(3'-CN--C.sub.6 H.sub.4)-Thienyl-2                                        86 5-(2'-CN--C.sub.6 H.sub.4)-Thienyl-2                                        87 5-(4'-Cl--C.sub.6 H.sub.4)-Thienyl-2                                        88 5-(3'-Cl--C.sub.6 H.sub.4)-Thienyl-2                                        89 5-(2'-Cl--C.sub.6 H.sub.4)-Thienyl-2                                        90 4-CH.sub.3 -Thienyl-2                                                       91 4-C.sub.6 H.sub.5 -Thienyl-2                                                92 4-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-2                                 93 4-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-2                                 94 4-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-2                                 95 4-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-2                                96 4-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-2                                97 4-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-2                                98 4-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-2                                 99 4-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-2                                 100 4-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-2                                101 4-(4'-CN--C.sub.6 H.sub.4)-Thienyl-2                                       102 4-(3'-CN--C.sub.6 H.sub.4)-Thienyl-2                                       103 4-(2'-CN--C.sub.6 H.sub.4)-Thieriyl-2                                      104 4-(4'-Cl--C.sub.6 H.sub.4)-Thienyl-2                                       105 4-(3'-Cl--C.sub.6 H.sub.4)-Thienyl-2                                       106 4-(2'-Cl--C.sub.6 H.sub.4)-Thienyl-2                                       107 Thienyl-3                                                                  108 5-CH.sub.3 -Thienyl-3                                                      109 5-C.sub.6 H.sub.5 -Thienyl-3                                               110 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-3                                111 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-3                                112 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-3                                113 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-3                               114 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-3                               115 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-3                               116 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-3                                117 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-3                                118 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-3                                119 5-(4'-CN--C.sub.6 H.sub.4)-Thienyl-3                                       120 5-(3'-CN--C.sub.6 H.sub.4)-Thienyl-3                                       121 5-(2'-CN--C.sub.6 H.sub.4)-Thienyl-3                                       122 5-(4'-Cl--C.sub.6 H.sub.4)-Thienyl-3                                       123 5-(3'-Cl--C.sub.6 H.sub.4)-Thienyl-3                                       124 5-(2'-Cl--C.sub.6 H.sub.4)-Thienyl-3                                       125 Pyrazolyl-4                                                                126 N--CH.sub.3 -Pyrazolyl-4                                                   127 N--C.sub.6 H.sub.5 -Pyrazolyl-4                                            128 N-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrazolyl-4                              129 N-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrazolyl-4                              130 N-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrazolyl-4                              131 N-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrazolyl-4                             132 N-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrazolyl-4                             133 N-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrazolyl-4                             134 N-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrazolyl-4                              135 N-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrazolyl-4                              136 N-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrazolyl-4                              137 N-(4'-CN--C.sub.6 H.sub.4)-Pyrazolyl-4                                     138 N-(3'-CN--C.sub.6 H.sub.4)-Pyrazolyl-4                                     139 N-(2'-CN--C.sub.6 H.sub.4)-Pyrazolyl-4                                     140 N-(4'-Cl--C.sub.6 H.sub.4)-Pyrazolyl-4                                     141 N-(3'-Cl--C.sub.6 H.sub.4)-Pyrazolyl-4                                     142 N-(2'-Cl--C.sub.6 H.sub.4)-Pyrazolyl-4                                     143 3-CH.sub.3 --N-Methylpyrazolyl-4                                           144 3-C.sub.6 H.sub.5 --N-Methylpyrazolyl-4                                    145 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)--N-Methylpyrazolyl-4                     146 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)--N-Methylpyrazolyl-4                     147 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)--N-Methylpyrazolyl-4                     148 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)--N-Methylpyrazolyl-4                    149 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)--N-Methylpyrazolyl-4                    150 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)--N-Methylpyrazolyl-4                    151 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)--N-Methylpyrazolyl-4                     152 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)--N-Methylpyrazolyl-4                     153 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)--N-Methylpyrazolyl-4                     154 3-(4'-CN--C.sub.6 H.sub.4)--N-Methylpyrazolyl-4                            155 3-(3'-CN--C.sub.6 H.sub.4)--N-Methylpyrazolyl-4                            156 3-(2'-CN--C.sub.6 H.sub.4)--N-Methylpyrazolyl-4                            157 3-(4'-Cl--C.sub.6 H.sub.4)--N-Methylpyrazolyl-4                            158 3-(3'-Cl--C.sub.6 H.sub.4)--N-Methylpyrazolyl-4                            159 3-(2'-Cl--C.sub.6 H.sub.4)--N-Methylpyrazolyl-4                            160 Isoxazolyl-5                                                               161 3-CH.sub.3 -Isoxazolyl-5                                                   162 3-C.sub.6 H.sub.5 -Isoxazolyl-5                                            163 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Isoxazolyl-5                             164 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Isoxazolyl-5                             165 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Isoxazolyl-5                             166 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Isoxazolyl-5                            167 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Isoxazolyl-5                            168 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Isoxazolyl-5                            169 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Isoxazolyl-5                             170 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Isoxazolyl-5                             171 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Isoxazolyl-5                             172 3-(4'-CN--C.sub.6 H.sub.4)-Isoxazolyl-5                                    173 3-(3'-CN--C.sub.6 H.sub.4)-Isoxazolyl-5                                    174 3-(2'-CN--C.sub.6 H.sub.4)-Isoxazolyl-5                                    175 3-(4'-Cl--C.sub.6 H.sub.4)-Isoxazolyl-5                                    176 3-(3'-Cl--C.sub.6 H.sub.4)-Isoxazolyl-5                                    177 3-(2'-Cl--C.sub.6 H.sub.4)-Isoxazolyl-5                                    178 4-Chloroisoxazolyl-5                                                       179 3-CH.sub.3 -4-Chloroisoxazolyl-5                                           180 3-C.sub.6 H.sub.5 -4-Chloroisoxazolyl-5                                    181 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                     182 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                     183 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                     184 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                    185 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                    186 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                    187 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                     188 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                     189 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                     190 3-(4'-CN--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                            191 3-(3'-CN--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                            192 3-(2'-CN--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                            193 3-(4'-Cl--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                            194 3-(3'-Cl--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                            195 3-(2'-Cl--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                            196 Isoxazolyl-3                                                               197 5-CH.sub.3 -Isoxazolyl-3                                                   198 5-C.sub.6 H.sub.5 -Isoxazolyl-3                                            199 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Isoxazolyl-3                             200 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Isoxazolyl-3                             201 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Isoxazolyl-3                             202 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Isoxazolyl-3                            203 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Isoxazolyl-3                            204 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Isoxazolyl-3                            205 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Isoxazolyl-3                             206 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Isoxazolyl-3                             207 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Isoxazolyl-3                             208 5-(4'-CN--C.sub.6 H.sub.4)-Isoxazolyl-3                                    209 5-(3'-CN--C.sub.6 H.sub.4)-Isoxazolyl-3                                    210 5-(2'-CN--C.sub.6 H.sub.4)-Isoxazolyl-3                                    211 5-(4'-Cl--C.sub.6 H.sub.4)-Isoxazolyl-3                                    212 5-(3'-Cl--C.sub.6 H.sub.4)-Isoxazolyl-3                                    213 5-(2'-Cl--C.sub.6 H.sub.4)-Isoxazolyl-3                                    214 Isothiazolyl-5                                                             215 3-CH.sub.3 -Isothiazolyl-5                                                 216 3-C.sub.6 H.sub.5 -Isothiazolyl-5                                          217 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Isothiazolyl-5                           218 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Isothiazolyl-5                           219 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Isothiazolyl-5                           220 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Isothiazolyl-5                          221 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Isothiazolyl-5                          222 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Isothiazolyl-5                          223 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Isothiazolyl-5                           224 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Isothiazolyl-5                           225 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Isothiazolyl-5                           226 3-(4'-CN--C.sub.6 H.sub.4)-Isothiazolyl-5                                  227 3-(3'-CN--C.sub.6 H.sub.4)-Isothiazolyl-5                                  228 3-(2'-CN--C.sub.6 H.sub.4)-Isothiazolyl-5                                  229 3-(4'-Cl--C.sub.6 H.sub.4)-Isothiazolyl-5                                  230 3-(3'-Cl--C.sub.6 H.sub.4)-Isothiazolyl-5                                  231 3-(2'-Cl--C.sub.6 H.sub.4)-Isothiazolyl-5                                  232 Oxazolyl-4                                                                 233 2-CH.sub.3 -Oxazolyl-4                                                     234 2-C.sub.6 H.sub.5 -Oxazolyl-4                                              235 2-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Oxazolyl-4                               236 2-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Oxazolyl-4                               237 2-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Oxazolyl-4                               238 2-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Oxazolyl-4                              239 2-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Oxazolyl-4                              240 2-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Oxazolyl-4                              241 2-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Oxazolyl-4                               242 2-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Oxazolyl-4                               243 2-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Oxazolyl-4                               244 2-(4'-CN--C.sub.6 H.sub.4)-Oxazolyl-4                                      245 2-(3'-CN--C.sub.6 H.sub.4)-Oxazolyl-4                                      246 2-(2'-CN--C.sub.6 H.sub.4)-Oxazolyl-4                                      247 2-(4'-Cl--C.sub.6 H.sub.4)-Oxazolyl-4                                      248 2-(3'-Cl--C.sub.6 H.sub.4)-Oxazolyl-4                                      249 2-(2'-Cl--C.sub.6 H.sub.4)-Oxazolyl-4                                      250 Thiazolyl-4                                                                251 2-CH.sub.3 -Thiazolyl-4                                                    252 2-C.sub.6 H.sub.5 -Thiazolyl-4                                             253 2-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Thiazolyl-4                              254 2-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Thiazolyl-4                              255 2-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Thiazolyl-4                              256 2-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Thiazolyl-4                             267 2-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Thiazolyl-4                             258 2-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Thiazolyl-4                             259 2-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Thiazolyl-4                              260 2-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Thiazolyl-4                              261 2-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Thiazolyl-4                              262 2-(4'-CN--C.sub.6 H.sub.4)-Thiazolyl-4                                     263 2-(3'-CN--C.sub.6 H.sub.4)-Thiazolyl-4                                     264 2-(2'-CN--C.sub.6 H.sub.4)-Thiazolyl-4                                     265 2-(4'-Cl--C.sub.6 H.sub.4)-Thiazolyl-,4                                    266 2-(3'-Cl--C.sub.6 H.sub.4)-Thiazolyl-4                                     267 2-(2'-Cl--C.sub.6 H.sub.4)-Thiazolyl-4                                     268 N--CH.sub.3 -1,2,4-Triazolyl-5                                             269 3-CH.sub.3 --N--CH.sub.3 -1,2,4-Triazolyl-5                                270 3-C.sub.6 H.sub.5 --N--CH.sub.3 -1,2,4-Triazolyl-5                         271 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5                   272 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triaz               olyl-5                                                                 273 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5                   274 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Tria               zolyl-5                                                                275 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5                  276 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Tria               zolyl-5                                                                277 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5                   278 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triaz               olyl-5                                                                 279 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5                   280 3-(4'-CN--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5        281 3-(3'-CN--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5                 282 3-(2'-CN--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5                 283 3-(4'-Cl--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5                 284 3-(3'-Cl--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5                 285 3-(2'-Cl--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5                 286 1,3,4-Oxadiazolyl-2                                                        287 5-CH.sub.3 -1,3,4-Oxadiazolyl-2                                            288 5-C.sub.6 H.sub.5 -1,2,3-Oxadiazolyl-2                                     289 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                      290 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                      291 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                      292 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                     293 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                     294 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                     295 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                      296 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                      297 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                      298 5-(4'-CN--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                             299 5-(3'-CN--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                             300 5-(2'-CN--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                             301 5-(4'-Cl--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                             302 5-(3'-Cl--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                             303 5-(2'-Cl--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                             304 1,2,4-Oxadiazolyl-3                                                        305 5-CH.sub.3 -1,2,4-Oxadiazolyl-3                                            306 5-C.sub.6 H.sub.5 -1,2,4-Oxadiazolyl-3                                     307 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                      308 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                      309 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                      310 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                     311 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                     312 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                     313 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                      314 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                      315 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                      316 5-(4'-CN--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                             317 5-(3'-CN--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                             318 5-(2'-CN--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                             319 5-(4'-Cl--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                             320 5-(3'-Cl--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                             321 5-(2'-Cl--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                             322 1,2,4-Oxadiazolyl-5                                                        323 3-CH.sub.3 -1,2,4-Oxadiazolyl-5                                            324 3-C.sub.6 H.sub.5 -1,2,4-Oxadiazolyl-5                                     325 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                      326 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                      327 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                      328 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                     329 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                     330 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                     331 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                      332 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                      333 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                      334 3-(4'-CN--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                             335 3-(3'-CN--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                             336 3-(2'-CN--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                             337 3-(4'-Cl--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                             338 3-(3'-Cl--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                             339 3-(2'-Cl--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                             340 1,2,4-Thiadiazolyl-3                                                       341 5-CH.sub.3 -1,2,4-Thiadiazolyl-3                                           342 5-C.sub.6 H.sub.5 -1,2,4-Thiadiazolyl-3                                    343 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                     344 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                     345 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                     346 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                    347 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                    348 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                    349 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                     350 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                     351 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                     352 5-(4'-CN--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                            353 5-(3'-CN--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                            354 5-(2'-CN--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                            355 5-(4'-Cl--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                            356 5-(3'-Cl--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                            357 5-(2'-Cl--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                            358 1,3,4-Thiadiazolyl-2                                                       359 5-CH.sub.3 -1,3,4-Thiadiazolyl-2                                           360 5-C.sub.6 H.sub.5 -1,3,4-Thiadiazolyl-2                                    361 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                     362 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                     363 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                     364 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                    365 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                    366 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                    367 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                     368 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                     369 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                     370 5-(4'-CN--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                            371 5-(3'-CN--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                            372 5-(2'-CN--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                            373 5-(4'-Cl--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                            374 5-(3'-Cl--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                            375 5-(2'-Cl--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                            376 Pyridinyl-2                                                                377 Pyridinyl-4                                                                378 Pyridazinyl-3                                                              379 Pyridazinyl-4                                                              380 Pyridazinyl-2                                                              381 Pyrimidinyl-4                                                              382 Pyrimidinyl-5                                                              383 Pyrimidinyl-2                                                              384 Pyridinyl-3                                                                385 1-Naphthyl                                                                 386 2-Naphthyl                                                               ______________________________________                                    

                  TABLE 28                                                         ______________________________________                                         2  STR239##                                                                       - I: R.sup.1 = CH.sub.3, X = CH.sub.3                                         II: R.sup.1 = CH.sub.2 --CH.sub.3, X = CH.sub.3                                III: R.sup.1 = CH.sub.3, X = Cl                                                IV: R.sup.1 = CH.sub.2 --CH.sub.3, X = Cl                                      No.        T.sub.m                                                           ______________________________________                                          1       H                                                                        2 2-F                                                                          3 3-F                                                                          4 4-F                                                                          5 2,4-F.sub.2                                                                  6 2,4,6-F.sub.3                                                                7 2,3,4,5,6-F.sub.5                                                            8 2,3-F.sub.2                                                                  9 2-Cl                                                                         10 3-Cl                                                                        11 4-Cl                                                                        12 2,3-Cl.sub.2                                                                13 2,4-Cl.sub.2                                                                14 2,5-Cl.sub.2                                                                15 2,6-Cl.sub.2                                                                16 3,4-Cl.sub.2                                                                17 3,5-Cl.sub.2                                                                18 2,3,4-Cl.sub.3                                                              19 2,3,5-Cl.sub.3                                                              20 2,3,6-Cl.sub.3                                                              21 2,4,5-Cl.sub.3                                                              22 2,4,6-Cl.sub.3                                                              23 3,4,5-Cl.sub.3                                                              24 2,3,4,6-Cl.sub.4                                                            25 2,3,5,6-Cl.sub.4                                                            26 2,3,4,5,6-Cl.sub.5                                                          27 2-Br                                                                        28 3-Br                                                                        29 4-Br                                                                        30 2,4-Br.sub.2                                                                31 2,5-Br.sub.2                                                                32 2,6-Br.sub.2                                                                33 2,4,6-Br.sub.3                                                              34 2,3,4,5,6-Br.sub.5                                                          35 2-I                                                                         36 3-I                                                                         37 4-I                                                                         38 2,4-I.sub.2                                                                 39 2-Cl, 3-F                                                                   40 2-Cl, 4-F                                                                   41 2-Cl, 5-F                                                                   42 2-Cl, 6-F                                                                   43 2-Cl, 3-Br                                                                  44 2-Cl, 4-Br                                                                  45 2-Cl, 5-Br                                                                  46 2-Cl, 6-Br                                                                  47 2-Br, 3-Cl                                                                  48 2-Br, 4-Cl                                                                  49 2-Br, 5-Cl                                                                  50 2-Br, 3-F                                                                   51 2-Br, 4-F                                                                   52 2-Br, 5-F                                                                   53 2-Br, 6-F                                                                   54 2-F, 3-Cl                                                                   55 2-F, 4-Cl                                                                   56 2-F, 5-Cl                                                                   57 3-Cl, 4-F                                                                   58 3-Cl, 5-F                                                                   59 3-Cl, 4-Br                                                                  60 3-Cl, 5-Br                                                                  61 3-F, 4-Cl                                                                   62 3-F, 4-Br                                                                   63 3-Br, 4-Cl                                                                  64 3-Br, 4-F                                                                   65 2,6-Cl.sub.2, 4-Br                                                          66 2-CH.sub.3                                                                  67 3-CH.sub.3                                                                  68 4-CH.sub.3                                                                  69 2,3-(CH.sub.3).sub.2                                                        70 2,4-(CH.sub.3).sub.2                                                        71 2,5-(CH.sub.3).sub.2                                                        72 2,6-(CH.sub.3).sub.2                                                        73 3,4-(CH.sub.3).sub.2                                                        74 3,5-(CH.sub.3).sub.2                                                        75 2,3,5-(CH.sub.3).sub.3                                                      76 2,3,4-(CH.sub.3).sub.3                                                      77 2,3,6-(CH.sub.3).sub.3                                                      78 2,4,5-(CH.sub.3).sub.3                                                      79 2,4,6-(CH.sub.3).sub.3                                                      80 3,4,5-(CH.sub.3).sub.3                                                      81 2,3,4,6-(CH.sub.3).sub.4                                                    82 2,3,5,6-(CH.sub.3).sub.4                                                    83 2,3,4,5,6-(CH.sub.3).sub.5                                                  84 2-C.sub.2 H.sub.5                                                           85 3-C.sub.2 H.sub.5                                                           86 4-C.sub.2 H.sub.5                                                           87 2,4-(C.sub.2 H.sub.5).sub.2                                                 88 2,6-(C.sub.2 H.sub.5).sub.2                                                 89 3,5-(C.sub.2 H.sub.5).sub.2                                                 90 2,4,6-(C.sub.2 H.sub.5).sub.3                                               91 2-n-C.sub.3 H.sub.7                                                         92 3-n-C.sub.3 H.sub.7                                                         93 4-n-C.sub.3 H.sub.7                                                         94 2-i-C.sub.3 H.sub.7                                                         95 3-i-C.sub.3 H.sub.7                                                         96 4-i-C.sub.3 H.sub.7                                                         97 2,4-(i-C.sub.3 H.sub.7).sub.2                                               98 2,6-(i-C.sub.3 H.sub.7).sub.2                                               99 3,5-(i-C.sub.3 H.sub.7).sub.2                                              100 2,4,6-(i-C.sub.3 H.sub.7).sub.3                                            101 2-s-C.sub.4 H.sub.9                                                        102 3-s-C.sub.4 H.sub.9                                                        103 4-s-C.sub.4 H.sub.9                                                        104 2-t-C.sub.4 H.sub.9                                                        105 3-t-C.sub.4 H.sub.9                                                        106 4-t-C.sub.4 H.sub.9                                                        107 2,3-(t-C.sub.4 H.sub.9).sub.2                                              108 2,4-(t-C.sub.4 H.sub.9).sub.2                                              109 2,5-(t-C.sub.4 H.sub.9).sub.2                                              110 2,6-(t-C.sub.4 H.sub.9).sub.2                                              111 3,4-(t-C.sub.4 H.sub.9).sub.2                                              112 2,4,6-(t-C.sub.4 H.sub.9).sub.3                                            113 4-n-C.sub.9 H.sub.19                                                       114 4-n-C.sub.12 H.sub.25                                                      115 4-n-C.sub.15 H.sub.31                                                      116 4-(1,1,3,3-Tetramethylbutyl)                                               117 4-(2,4,4-Trimethylpropyl)                                                  118 2-t-C.sub.4 H.sub.9, 4-CH.sub.3                                            119 2-t-C.sub.4 H.sub.9, 5-CH.sub.3                                            120 2,6-(t-C.sub.4 H.sub.9).sub.2, 4-CH.sub.3                                  121 2-CH.sub.3, 4-t-C.sub.4 H.sub.9                                            122 2-CH.sub.3, 6-t-C.sub.4 H.sub.9                                            123 2-CH.sub.3, 4-i-C.sub.3 H.sub.7                                            124 2-CH.sub.3, 5-i-C.sub.3 H.sub.7                                            125 3-CH.sub.3, 4-i-C.sub.3 H.sub.7                                            126 2-i-C.sub.3 H.sub.7, 5-CH.sub.3                                            127 2,4-(t-C.sub.4 H.sub.9).sub.2, 6-i-C.sub.3 H.sub.7                         128 2-Allyl                                                                    129 3-Allyl                                                                    130 4-Allyl                                                                    131 2-Allyl, 6-CH.sub.3                                                        132 2-cyclo-C.sub.6 H.sub.11                                                   133 3-cyclo-C.sub.6 H.sub.11                                                   134 4-cyclo-C.sub.6 H.sub.11                                                   135 2,4-(cyclo-C.sub.6 H.sub.11).sub.2, 6-CH.sub.3                             136 2-CH.sub.3, 4-cyclo-C.sub.6 H.sub.11                                       137 2-CH.sub.2 --C.sub.6 H.sub.5                                               138 3-CH.sub.2 --C.sub.6 H.sub.5                                               139 4-CH.sub.2 --C.sub.6 H.sub.5                                               140 2-CH.sub.2 --C.sub.6 H.sub.5, 4-CH.sub.3                                   141 2-CH.sub.3, 4-CH.sub.2 --C.sub.6 H.sub.5                                   142 2-C.sub.6 H.sub.5                                                          143 3-C.sub.6 H.sub.5                                                          144 4-C.sub.6 H.sub.5                                                          145 4-(2-i-C.sub.3 H.sub.7 --C.sub.6 H.sub.4)                                  146 4-C.sub.6 H.sub.5, 2,6-(CH.sub.3).sub.2                                    147 2-Cl, 4-C.sub.6 H.sub.5                                                    148 2-Br, 4-C.sub.6 H.sub.5                                                    149 2-C.sub.6 H.sub.5, 4-Cl                                                    150 2-C.sub.6 H.sub.5, 4-Br                                                    151 2-CH.sub.2 C.sub.6 H.sub.5, 4-Cl                                           152 2-CH.sub.2 C.sub.6 H.sub.5, 4-Br                                           153 2-Cl, 4-CH.sub.2 C.sub.6 H.sub.5                                           154 2-Br, 4-CH.sub.2 C.sub.6 H.sub.5                                           155 2-cyclo-C.sub.6 H.sub.11, 4-Cl                                             156 2-cyclo-C.sub.6 H.sub.11, 4-Br                                             157 2-Cl, 4-cyclo-C.sub.6 H.sub.11                                             158 2-Br, 4-cyclo-C.sub.6 H.sub.11                                             159 2-OCH.sub.3                                                                160 3-OCH.sub.3                                                                161 4-OCH.sub.3                                                                162 2-OC.sub.2 H.sub.5                                                         163 3-O--C.sub.2 H.sub.5                                                       164 4-O--C.sub.2 H.sub.5                                                       165 2-O-n-C.sub.3 H.sub.7                                                      166 3-O-n-C.sub.3 H.sub.7                                                      167 4-O-n-C.sub.3 H.sub.7                                                      168 2-O-i-C.sub.3 H.sub.7                                                      169 3-O-i-C.sub.3 H.sub.7                                                      170 4-O-i-C.sub.3 H.sub.7                                                      171 2-O-n-C.sub.6 H.sub.13                                                     172 3-O-n-C.sub.6 H.sub.13                                                     173 4-O-n-C.sub.6 H.sub.13                                                     174 2-O-n-C.sub.8 H.sub.17                                                     175 3-O-n-C.sub.8 H.sub.17                                                     176 4-O-n-C.sub.8 H.sub.17                                                     177 2-O-CH.sub.2 C.sub.6 H.sub.5                                               178 3-O-CH.sub.2 C.sub.6 H.sub.5                                               179 4-O-CH.sub.2 C.sub.6 H.sub.5                                               180 2-O-(CH.sub.2).sub.3 C.sub.6 H.sub.5                                       181 3-O-(CH.sub.2).sub.3 C.sub.6 H.sub.5                                       182 4-O-(CH.sub.2).sub.3 C.sub.6 H.sub.5                                       183 2,4-(OCH.sub.3).sub.2                                                      184 2-CF.sub.3                                                                 185 3-CF.sub.3                                                                 186 4-CF.sub.3                                                                 187 2-OCF.sub.3                                                                188 3-OCF.sub.3                                                                189 4-OCF.sub.3                                                                190 3-OCH.sub.2 CHF.sub.2                                                      191 2-NO.sub.2                                                                 192 3-NO.sub.2                                                                 193 4-NO.sub.2                                                                 194 2-CN                                                                       195 3-CN                                                                       196 4-CN                                                                       197 2-CH.sub.3, 3-Cl                                                           198 2-CH.sub.3, 4-Cl                                                           199 2-CH.sub.3, 5-Cl                                                           200 2-CH.sub.3, 6-Cl                                                           201 2-CH.sub.3, 3-F                                                            202 2-CH.sub.3, 4-F                                                            203 2-CH.sub.3, 5-F                                                            204 2-CH.sub.3, 6-F                                                            205 2-CH.sub.3, 3-Br                                                           206 2-CH.sub.3, 4-Br                                                           207 2-CH.sub.3, 5-Br                                                           208 2-CH.sub.3, 6-Br                                                           209 2-Cl, 3-CH.sub.3                                                           210 2-Cl, 4-CH.sub.3                                                           211 2-Cl, 5-CH.sub.3                                                           212 2-F, 3-CH.sub.3                                                            213 2-F, 4-CH.sub.3                                                            214 2-F, 5-CH.sub.3                                                            215 2-Br, 3-CH.sub.3                                                           216 2-Br, 4-CH.sub.3                                                           217 2-Br, 5-CH.sub.3                                                           218 3-CH.sub.3, 4-Cl                                                           219 3-CH.sub.3, 5-Cl                                                           220 3-CH.sub.3, 4-F                                                            221 3-CH.sub.3, 5-F                                                            222 3-CH.sub.3, 4-Br                                                           223 3-CH.sub.3, 5-Br                                                           224 3-F, 4-CH.sub.3                                                            225 3-Cl, 4-CH.sub.3                                                           226 3-Br, 4-CH.sub.3                                                           227 2-Cl, 4,5-(CH.sub.3).sub.2                                                 228 2-Br, 4,5-(CH.sub.3).sub.2                                                 229 2-Cl, 3,5-(CH.sub.3).sub.2                                                 230 2-Br, 3,5-(CH.sub.3).sub.2                                                 231 2,6-Cl.sub.2, 4-CH.sub.3                                                   232 2,6-F.sub.2, 4-CH.sub.3                                                    233 2,6-Br.sub.2, 4-CH.sub.3                                                   234 2,4-Br.sub.2, 6-CH.sub.3                                                   235 2,4-F.sub.2, 6-CH.sub.3                                                    236 2,4-Br.sub.2, 6-CH.sub.3                                                   237 2,6-(CH.sub.3).sub.2, 4-F                                                  238 2,6-(CH.sub.3).sub.2, 4-Cl                                                 239 2,6-(CH.sub.3).sub.2, 4-Br                                                 240 3,5-(CH.sub.3).sub.2, 4-F                                                  241 3,5-(CH.sub.3).sub.2, 4-Cl                                                 242 3,5-(CH.sub.3).sub.2, 4-Br                                                 243 2,3,6-(CH.sub.3).sub.3, 4-F                                                244 2,3,6-(CH.sub.3).sub.3, 4-Cl                                               245 2,3,6-(CH.sub.3).sub.3, 4-Br                                               246 2,4-(CH.sub.3).sub.2, 6-F                                                  247 2,4-(CH.sub.3).sub.2, 6-Cl                                                 248 2,4-(CH.sub.3).sub.2, 6-Br                                                 249 2-i-C.sub.3 H.sub.7, 4-Cl, 5-CH.sub.3                                      250 2-Cl, 4-NO.sub.2                                                           251 2-NO.sub.2, 4-Cl                                                           252 2-OCH.sub.3, 5-NO.sub.2                                                    253 2,4-Cl.sub.2, 5-NO.sub.2                                                   254 2,4-Cl.sub.2, 6-NO.sub.2                                                   255 2,6-Cl.sub.2, 4-NO.sub.2                                                   256 2,6-Br.sub.2, 4-NO.sub.2                                                   257 2,6-I.sub.2, 4-NO.sub.2                                                    258 2-CH.sub.3, 5-i-C.sub.3 H.sub.7, 4-Cl                                      259 2-CO.sub.2 CH.sub.3                                                        260 3-CO.sub.2 CH.sub.3                                                        261 4-CO.sub.2 CH.sub.3                                                        262 2-CO.sub.2 (C.sub.2 H.sub.5)                                               263 3-CO.sub.2 (C.sub.2 H.sub.5)                                               264 4-CO.sub.2 (C.sub.2 H.sub.5)                                               265 2-CO.sub.2 (n-C.sub.3 H.sub.7)                                             266 3-CO.sub.2 (n-C.sub.3 H.sub.7)                                             267 4-CO.sub.2 (n-C.sub.3 H.sub.7)                                             268 2-CO.sub.2 (i-C.sub.3 H.sub.7)                                             269 3-CO.sub.2 (i-C.sub.3 H.sub.7)                                             270 4-CO.sub.2 (i-C.sub.3 H.sub.7)                                             271 2-CO.sub.2 (n-C.sub.6 H.sub.13)                                            272 3-CO.sub.2 (n-C.sub.6 H.sub.13)                                            273 4-CO.sub.2 (n-C.sub.6 H.sub.13)                                            274 2-CH.sub.2 --OCH.sub.3                                                     275 3-CH.sub.2 --OCH.sub.3                                                     276 4-CH.sub.2 --OCH.sub.3                                                     277 2-CH.sub.2 O(C.sub.2 H.sub.5)                                              278 3-CH.sub.2 O(C.sub.2 H.sub.5)                                              279 4-CH.sub.2 O(C.sub.2 H.sub.5)                                              280 2-CH.sub.2 O(n-C.sub.3 H.sub.7)                                            281 3-CH.sub.2 O(n-C.sub.3 H.sub.7)                                            282 4-CH.sub.2 O(n-C.sub.3 H.sub.7)                                            283 2-CH.sub.2 O(i-C.sub.3 H.sub.7)                                            284 3-CH.sub.2 O(i-C.sub.3 H.sub.7)                                            285 4-CH.sub.2 O(i-C.sub.3 H.sub.7)                                            286 2-CHO                                                                      287 3-CHO                                                                      288 4-CHO                                                                      289 2-CO--CH.sub.3                                                             290 3-CO--CH.sub.3                                                             291 4-CO--CH.sub.3                                                             292 2-CO--CH.sub.2 --CH.sub.3                                                  293 3-CO--CH.sub.2 --CH.sub.3                                                  294 4-CO--CH.sub.2 --CH.sub.3                                                  295 2-CO--CH.sub.2 --CH.sub.2 --CH.sub.3                                       296 3-CO--CH.sub.2 --CH.sub.2 --CH.sub.3                                       297 4-CO--CH.sub.2 --CH.sub.2 --CH.sub.3                                       298 2-CO--CH(CH.sub.3)--CH.sub.3                                               299 3-CO--CH(CH.sub.3)--CH.sub.3                                               300 4-CO--CH(CH.sub.3)--CH.sub.3                                               301 2-Me-4-CHO                                                                 302 2-Me-4-CH.sub.3 --CO                                                       303 2-Me-4-CH.sub.3 --CH.sub.2 --CO                                            304 2-Me-4-CH.sub.3 --CH.sub.2 --CH.sub.2 --CO                                 305 2-Me-4-CH.sub.3 --CH(CH.sub.3)--CO                                         306 2,5-Me.sub.2 -4-CHO                                                        307 2,5-Me.sub.2 -4-CH.sub.3 --CO                                              308 2,5-Me.sub.2 -4-CH.sub.3 --CH.sub.2 --CO                                   309 2,5-Me.sub.2 -4-CH.sub.3 --CH.sub.2 --CH.sub.2 --CO                        310 2,5-Me.sub.2 -4-CH.sub.3 --CH(CH.sub.3)--CO                                311 2-Cl-4-CHO                                                                 312 2-Cl-4-CH.sub.3 --CO                                                       313 2-Cl-4-CH.sub.3 --CH.sub.2 --CO                                            314 2-Cl-4-CH.sub.3 --CH(CH.sub.3)--CO                                         315 2,5-Cl.sub.2 -4-CHO                                                        316 2,5-Cl.sub.2 -4-CH.sub.3 --CO                                              317 2,5-Cl.sub.2 -4-CH.sub.3 --CH.sub.2 --CO                                   318 2,5-Cl.sub.2 -4-CH.sub.3 --CH.sub.2 --CH.sub.2 --CO                        319 2,5-Cl.sub.2 -4-CH.sub.3 --CH(CH.sub.3)--CO                                320 2-C(═NOCH.sub.3)--CH.sub.3                                             321 3-C(═NOCH.sub.3)--CH.sub.3                                             322 4-C(═NOCH.sub.3)--CH.sub.3                                             323 2-C(═NOC.sub.2 H.sub.5)--CH.sub.3                                      324 3-C(═NOC.sub.2 H.sub.5)--CH.sub.3                                      325 4-C(═NOC.sub.2 H.sub.5)--CH.sub.3                                      326 2-C(═NO-n-C.sub.3 H.sub.7)--CH.sub.3                                   327 3-C(═NO-n-C.sub.3 H.sub.7)--CH.sub.3                                   328 4-C(═NO-n-C.sub.3 H.sub.7)--CH.sub.3                                   329 2-C(═NO-i-C.sub.3 H.sub.7)--CH.sub.3                                   330 3-C(═NO-i-C.sub.3 H.sub.7)--CH.sub.3                                   331 4-C(═NO-i-C.sub.3 H.sub.7)--CH.sub.3                                   332 2-C(═NO-Allyl)--CH.sub.3                                               333 3-C(═NO-Allyl)--CH.sub.3                                               334 4-C(═NO-Allyl)--CH.sub.3                                               335 2-C(═NO-trans-Chloroallyl)--CH.sub.3                                   336 3-C(═NO-trans-Chloroallyl)--CH.sub.3                                   337 4-C(═NO-trans-Chloroallyl)--CH.sub.3                                   338 2-C(═NO-Propargyl)--CH.sub.3                                           339 3-C(═NO-Propargyl)--CH.sub.3                                           340 4-C(═NO-Propargyl)--CH.sub.3                                           341 2-C(═NO-n-C.sub.4 H.sub.9)--CH.sub.3                                   342 3-C(═NO-n-C.sub.4 H.sub.9)--CH.sub.3                                   343 4-C(═NO-n-C.sub.4 H.sub.9)--CH.sub.3                                   344 2-C(═NO--CH.sub.2 --C.sub.6 H.sub.5)--CH.sub.3                         345 3-C(═NO--CH.sub.2 --C.sub.6 H.sub.5)--CH.sub.3                         346 4-C(═NO--CH.sub.2 --C.sub.6 H.sub.5)--CH.sub.3                         347 2-CH.sub.3 -4-CH═NOCH.sub.3                                            348 2-CH.sub.3 -4-CH═NOC.sub.2 H.sub.5                                     349 2-CH.sub.3 -4-CH═NO-n-C.sub.3 H.sub.7                                  350 2-CH.sub.3 -4-CH═NO-i-C.sub.3 H.sub.7                                  351 2-CH.sub.3 -4-CH═NO-Allyl                                              352 2-CH.sub.3 -4-CH═NO-(trans-Chloroallyl)                                353 2-CH.sub.3 -4-CH═NO-Propargyl                                          354 2-CH.sub.3 -4-CH═NO-n-C.sub.4 H.sub.9                                  355 2-CH.sub.3 -4-CH═NO--CH.sub.2 --C.sub.6 H.sub.5                        356 2-CH.sub.3 -4-(CH.sub.3 --C═NOCH.sub.3)                                357 2-CH.sub.3 -4-(CH.sub.3 --C═NOC.sub.2 H.sub.5)                         358 2-CH.sub.3 -4-(CH.sub.3 --C═NO-n-C.sub.3 H.sub.7)                      359 2-CH.sub.3 -4-(CH.sub.3 --C═NO-i-C.sub.3 H.sub.7)                      360 2-CH.sub.3 -4-(CH.sub.3 --C═NO-Allyl)                                  361 2-CH.sub.3 -4-(CH.sub.3 --C═NO-trans-Chloroallyl)                      362 2-CH.sub.3 -4-(CH.sub.3 --C═NO-Propargyl)                              363 2-CH.sub.3 -4-(CH.sub.3 --C═NO-n-C.sub.4 H.sub.9)                      364 2-CH.sub.3 -4-(CH.sub.3 --C═NO--CH.sub.2 --C.sub.6 H.sub.5)                    365 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C═NO--CH.sub.3)                       366 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C═NO--C.sub.2 H.sub.5)        367 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C═NO-n-C.sub.3 H.sub.7)                       368 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C═NO-i-C.sub.3                       H.sub.7)                                                                369 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C═NO-Allyl)                           370 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C═NO-trans-Chloroallyl)                       371 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C═NO-Propargyl)                       372 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C═NO-n-C.sub.4                       H.sub.9)                                                                373 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C═NO--CH.sub.2 --C.sub.6                     H.sub.5)                                                                374 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C═NOCH.sub.3)                      375 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C═NOC.sub.2 H.sub.5)                       376 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C═NO-n-C.sub.3                    H.sub.7)                                                                377 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C═NO-i-C.sub.3 H.sub.7)                    378 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C═NO-Allyl)                        379 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C═NO-trans-Chloroall              yl)                                                                     380 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C═NO-Proparyl)                     381 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C═NO-n-C.sub.4 H.sub.9)                    382 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C═NO--CH.sub.2                    --C.sub.6 H.sub.5)                                                      383 2-C.sub.6 H.sub.5                                                          384 3-C.sub.6 H.sub.5                                                          385 4-C.sub.6 H.sub.5                                                          386 2-(2'-F--C.sub.6 H.sub.4)                                                  387 2-(3'-F--C.sub.6 H.sub.4)                                                  388 2-(4'-F--C.sub.6 H.sub.4)                                                  389 3-(2'-F--C.sub.6 H.sub.4)                                                  390 3-(3'-F--C.sub.6 H.sub.4)                                                  391 3-(4'-F--C.sub.6 H.sub.4)                                                  392 4-(2'-F--C.sub.6 H.sub.4)                                                  393 4-(3'-F--C.sub.6 H.sub.4)                                                  394 4-(4'-F--C.sub.6 H.sub.4)                                                  395 2-(2'-Cl--C.sub.6 H.sub.4)                                                 396 2-(3'-Cl--C.sub.6 H.sub.4)                                                 397 2-(4'-Cl--C.sub.6 H.sub.4)                                                 398 3-(2'-Cl--C.sub.6 H.sub.4)                                                 399 3-(3'-Cl--C.sub.6 H.sub.4)                                                 400 3-(4'-Cl--C.sub.6 H.sub.4)                                                 401 4-(2'-Cl--C.sub.6 H.sub.4)                                                 402 4-(3'-Cl--C.sub.6 H.sub.4)                                                 403 4-(4'-Cl--C.sub.6 H.sub.4)                                                 405 2-(2'-CH.sub.3 --C.sub.6 H.sub.4)                                          406 2-(3'-CH.sub.3 --C.sub.6 H.sub.4)                                          407 2-(4'-CH.sub.3 --C.sub.6 H.sub.4)                                          408 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)                                          409 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)                                          410 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)                                          411 4-(2'-CH.sub.3 --C.sub.6 H.sub.4)                                          412 4-(3'-CH.sub.3 --C.sub.6 H.sub.4)                                          413 4-(4'-CH.sub.3 --C.sub.6 H.sub.4)                                          414 2-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                      415 2-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                      416 2-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                      417 3-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                      418 3-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                      419 3-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                      420 4-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                      421 4-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                      422 4-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                      423 2-(2'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                       424 2-(3'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                       425 2-(4'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                       426 3-(2'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                       427 3-(3'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                       428 3-(4'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                       429 4-(2'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                       430 4-(3'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                       431 4-(4'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                       432 2-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                                 433 2-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                                 434 2-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                                 435 3-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                                 436 3-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                                 437 3-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                                 438 4-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                                 439 4-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                                 440 4-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                                 441 2-(2'-CH.sub.3 O--C.sub.6 H.sub.4)                                         442 2-(3'-CH.sub.3 O--C.sub.6 H.sub.4)                                         443 2-(4'-CH.sub.3 O--C.sub.6 H.sub.4)                                         444 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)                                         445 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)                                         446 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)                                         447 4-(2'-CH.sub.3 O--C.sub.6 H.sub.4)                                         448 4-(3'-CH.sub.3 O--C.sub.6 H.sub.4)                                         449 4-(4'-CH.sub.3 O--C.sub.6 H.sub.4)                                         450 2-(2'-O.sub.2 N--C.sub.6 H.sub.4)                                          451 2-(3'-O.sub.2 N--C.sub.6 H.sub.4)                                          452 2-(4'-O.sub.2 N--C.sub.6 H.sub.4)                                          453 3-(2'-O.sub.2 N--C.sub.6 H.sub.4)                                          454 3-(3'-O.sub.2 N--C.sub.6 H.sub.4)                                          455 3-(4'-O.sub.2 N--C.sub.6 H.sub.4)                                          456 4-(2'-O.sub.2 N--C.sub.6 H.sub.4)                                          457 4-(3'-O.sub.2 N--C.sub.6 H.sub.4)                                          458 4-(4'-O.sub.2 N--C.sub.6 H.sub.4)                                          459 2-(2'-NC--C.sub.6 H.sub.4)                                                 460 2-(3'-NC--C.sub.6 H.sub.4)                                                 461 2-(4'-NC--C.sub.6 H.sub.4)                                                 462 3-(2'-NC--C.sub.6 H.sub.4)                                                 463 3-(3'-NC--C.sub.6 H.sub.4)                                                 464 3-(4'-NC--C.sub.6 H.sub.4)                                                 465 4-(2'-NC--C.sub.6 H.sub.4)                                                 466 4-(3'-NC--C.sub.6 H.sub.4)                                                 467 4-(4'-NC--C.sub.6 H.sub.4)                                                 468 2-(2'-CF.sub.3 --C.sub.6 H.sub.4)                                          469 2-(3'-CF.sub.3 --C.sub.6 H.sub.4)                                          470 2-(4'-CF.sub.3 --C.sub.6 H.sub.4)                                          471 3-(2'-CF.sub.3 --C.sub.6 H.sub.4)                                          472 3-(3'-CF.sub.3 --C.sub.6 H.sub.4)                                          473 3-(4'-CF.sub.3 --C.sub.6 H.sub.4)                                          474 4-(2'-CF.sub.3 --C.sub.6 H.sub.4)                                          475 4-(3'-CF.sub.3 --C.sub.6 H.sub.4)                                          476 4-(4'-CF.sub.3 --C.sub.6 H.sub.4)                                          477 2-O-C.sub.6 H.sub.5                                                        475 3-O-C.sub.6 H.sub.5                                                        476 4-O-C.sub.6 H.sub.5                                                        478 2-O-(2'-F--C.sub.6 H.sub.4)                                                479 2-O-(3'-F--C.sub.6 H.sub.4)                                                480 2-O-(4'-F--C.sub.6 H.sub.4)                                                481 3-O-(2'-F--C.sub.6 H.sub.4)                                                482 3-O-(3'-F--C.sub.6 H.sub.4)                                                483 3-O-(4'-F--C.sub.6 H.sub.4)                                                484 4-O-(2'-F--C.sub.6 H.sub.4)                                                485 4-O-(3'-F--C.sub.6 H.sub.4)                                                486 4-O-(4'-F--C.sub.6 H.sub.4)                                                487 2-O-(2'-Cl--C.sub.6 H.sub.4)                                               488 2-O-(3'-Cl--C.sub.6 H.sub.4)                                               489 2-O-(4'-Cl--C.sub.6 H.sub.4)                                               490 3-O-(2'-Cl--C.sub.6 H.sub.4)                                               491 3-O-(3'-Cl--C.sub.6 H.sub.4)                                               492 3-O-(4'-Cl--C.sub.6 H.sub.4)                                               493 3-O-(4'-Cl--C.sub.6 H.sub.4)                                               494 4-O-(2'-Cl--C.sub.6 H.sub.4)                                               495 4-O-(3'-Cl--C.sub.6 H.sub.4)                                               496 4-O-(4'-Cl--C.sub.6 H.sub.4)                                               497 2-O-(2'-CH.sub.3 --C.sub.6 H.sub.4)                                        498 2-O-(3'-CH.sub.3 --C.sub.6 H.sub.4)                                        499 2-O-(4'-CH.sub.3 --C.sub.6 H.sub.4)                                        500 3-O-(2'-CH.sub.3 --C.sub.6 H.sub.4)                                        501 3-O-(3'-CH.sub.3 --C.sub.6 H.sub.4)                                        502 3-O-(4'-CH.sub.3 --C.sub.6 H.sub.4)                                        503 4-O-(2'-CH.sub.3 --C.sub.6 H.sub.4)                                        504 4-O-(3'-CH.sub.3 --C.sub.6 H.sub.4)                                        505 4-O-(4'-CH.sub.3 --C.sub.6 H.sub.4)                                        506 2-O-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                    507 2-O-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                    508 2-O-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                    509 3-O-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                    510 3-O-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                    511 3-O-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                    512 4-O-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                    513 4-O-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                    514 4-O-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                    515 2-O-(2'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                     516 2-O-(3'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                     517 2-O-(4'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                     518 3-O-(2'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                     519 3-O-(3'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                     520 3-O-(4'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                     521 4-O-(2'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                     522 4-O-(3'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                     523 4-O-(4'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                     524 2-O-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                               525 2-O-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                               526 2-O-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                               527 3-O-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                               528 3-O-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                               529 3-O-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                               530 4-O-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                               531 4-O-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                               532 4-O-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                               533 2-O-(2'-CH.sub.3 O--C.sub.6 H.sub.4)                                       534 2-O-(3'-CH.sub.3 O--C.sub.6 H.sub.4)                                       535 2-O-(4'-CH.sub.3 O--C.sub.6 H.sub.4)                                       536 3-O-(2'-CH.sub.3 O--C.sub.6 H.sub.4)                                       537 3-O-(3'-CH.sub.3 O--C.sub.6 H.sub.4)                                       538 3-O-(4'-CH.sub.3 O--C.sub.6 H.sub.4)                                       539 4-O-(2'-CH.sub.3 O--C.sub.6 H.sub.4)                                       540 4-O-(3'-CH.sub.3 O--C.sub.6 H.sub.4)                                       541 4-O-(4'-CH.sub.3 O--C.sub.6 H.sub.4)                                       542 2-O-(2'-O.sub.2 N--C.sub.6 H.sub.4)                                        543 2-O-(3'-O.sub.2 N--C.sub.6 H.sub.4)                                        544 2-O-(4'-O.sub.2 N--C.sub.6 H.sub.4)                                        545 3-O-(2'-O.sub.2 N--C.sub.6 H.sub.4)                                        546 3-O-(3'-O.sub.2 N--C.sub.6 H.sub.4)                                        547 3-O-(4'-O.sub.2 N--C.sub.6 H.sub.4)                                        548 4-O-(2'-O.sub.2 N--C.sub.6 H.sub.4)                                        549 4-O-(3'-O.sub.2 N--C.sub.6 H.sub.4)                                        550 4-O-(4'-O.sub.2 N--C.sub.6 H.sub.4)                                        551 2-O-(2'-NC--C.sub.6 H.sub.4)                                               552 2-O-(3'-NC--C.sub.6 H.sub.4)                                               553 2-O-(4'-NC--C.sub.6 H.sub.4)                                               554 3-O-(2'-NC--C.sub.6 H.sub.4)                                               555 3-O-(3'-NC--C.sub.6 H.sub.4)                                               556 3-O-(4'-NC--C.sub.6 H.sub.4)                                               557 4-O-(2'-NC--C.sub.6 H.sub.4)                                               558 4-O-(3'-NC--C.sub.6 H.sub.4)                                               559 4-O-(4'-NC--C.sub.6 H.sub.4)                                               560 2-O-(2'-CF.sub.3 --C.sub.6 H.sub.4)                                        561 2-O-(3'-CF.sub.3 --C.sub.6 H.sub.4)                                        562 2-O-(4'-CF.sub.3 --C.sub.6 H.sub.4)                                        563 3-O-(2'-CF.sub.3 --C.sub.6 H.sub.4)                                        564 3-O-(3'-CF.sub.3 --C.sub.6 H.sub.4)                                        565 3-O-(4'-CF.sub.3 --C.sub.6 H.sub.4)                                        566 4-O-(2'-CF.sub.3 --C.sub.6 H.sub.4)                                        567 4-O-(3'-CF.sub.3 --C.sub.6 H.sub.4)                                        568 4-O-(4'-CF.sub.3 --C.sub.6 H.sub.4)                                        569 2-Pyridinyl-2'                                                             570 2-Pyridinyl-3'                                                             571 2-Pyridinyl-4'                                                             572 3-Pyridinyl-2'                                                             573 3-Pyridinyl-3'                                                             574 3-Pyridinyl-4'                                                             575 4-Pyridinyl-2'                                                             576 4-Pyridinyl-3'                                                             577 4-Pyridinyl-4'                                                             578 2-Pyrimidinyl-2'                                                           579 2-Pyrimidinyl-3'                                                           580 2-Pyrimidinyl-4'                                                           581 3-Pyrimidinyl-2'                                                           582 3-Pyrimidinyl-3'                                                           583 3-Pyrimidinyl-4'                                                           584 4-Pyrimidinyl-2'                                                           585 4-Pyrimidinyl-3'                                                           586 4-Pyrimidinyl-4'                                                           587 2-Pyrazolyl-1'                                                             588 2-Pyrazolyl-3'                                                             589 2-Pyrazolyl-4'                                                             590 3-Pyrazolyl-1'                                                             591 3-Pyrazolyl-3'                                                             592 3-Pyrazolyl-4'                                                             593 4-Pyrazolyl-1'                                                             594 4-Pyrazolyl-3'                                                             595 4-Pyrazolyl-4'                                                             596 2-Isoxazolyl-3'                                                            597 2-Isoxazolyl-4'                                                            598 2-Isoxazolyl-5'                                                            599 3-Isoxazolyl-3'                                                            600 3-Isoxazolyl-4'                                                            601 3-Isoxazolyl-5'                                                            602 4-Isoxazolyl-3'                                                            603 4-Isoxazolyl-4'                                                            604 4-Isoxazolyl-5'                                                            605 2-Isothiazolyl-3'                                                          606 2-Isothiazolyl-4'                                                          607 2-Isothiazolyl-5'                                                          608 3-Isothiazolyl-3'                                                          609 3-Isothiazolyl-4'                                                          610 3-Isothiazolyl-5'                                                          611 4-Isothiazolyl-3'                                                          612 4-Isothiazolyl-4'                                                          613 4-Isothiazolyl-5'                                                          614 2-Imidazolyl-1'                                                            615 2-Imidazolyl-2'                                                            616 2-Imidazolyl-4'                                                            617 3-Imidazolyl-1'                                                            618 3-Imidazolyl-2'                                                            619 3-Imidazolyl-4'                                                            620 4-Imidazolyl-1'                                                            621 4-Imidazolyl-2'                                                            622 4-Imidazolyl-4'                                                            623 2-Oxazolyl-2'                                                              624 2-Oxazolyl-4'                                                              625 2-Oxazolyl-5'                                                              626 3-Oxazolyl-2'                                                              627 3-Oxazolyl-4'                                                              628 3-Oxazolyl-5'                                                              629 4-Oxazolyl-2'                                                              630 4-Oxazolyl-4'                                                              631 4-Oxazolyl-5'                                                              632 2-Thiazolyl-2'                                                             633 2-Thiazolyl-4'                                                             634 2-Thiazolyl-5'                                                             635 3-Thiazolyl-2'                                                             636 3-Thiazolyl-4'                                                             637 3-Thiazolyl-5'                                                             638 4-Thiazolyl-2'                                                             639 4-Thiazolyl-4'                                                             640 4-Thiazolyl-5'                                                           ______________________________________                                    

                  TABLE 29                                                         ______________________________________                                         1  STR240##                                                                       -       I: R.sup.1 = CH.sub.3, X = CH.sub.3                                   II: R.sup.1 = CH.sub.2 --CH.sub.3, X = CH.sub.3                                III: R.sup.1 = CH.sub.3, X = Cl                                                IV: R.sup.1 = CH.sub.2 --CH.sub.3, X = Cl                                    No.       B                                                                    ______________________________________                                          1        Pyrrolyl-3                                                              2 N-CH.sub.3 -Pyrrolyl-3                                                       3 N-C.sub.6 H.sub.4 -Pyrrolyl-3                                                4 N-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrrolyl-3                                 5 N-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrrolyl-3                                 6 N-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrrolyl-3                                 7 N-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrrolyl-3                                8 N-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrrolyl-3                                9 N-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrrolyl-3                                10 N-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrrolyl-3                                11 N-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrrolyl-3                                12 N-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrrolyl-3                                13 N-(4'-CN--C.sub.6 H.sub.4)-Pyrrolyl-3                                       14 N-(3'-CN--C.sub.6 H.sub.4)-Pyrrolyl-3                                       15 N-(2'-CN--C.sub.6 H.sub.4)-Pyrrolyl-3                                       16 N-(4'-Cl--C.sub.6 H.sub.4)-Pyrrolyl-3                                       17 N-(3'-Cl--C.sub.6 H.sub.4)-Pyrrolyl-3                                       18 N-(2'-Cl--C.sub.6 H.sub.4)-Pyrrolyl-3                                       19 Pyrrolyl-2                                                                  20 N--CH.sub.3 -Pyrrolyl-2                                                     21 N--C.sub.6 H.sub.5 -Pyrrolyl-2                                              22 N-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrrolyl-2                                23 N-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrrolyl-2                                24 N-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrrolyl-2                                25 N-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrrolyl-2                               26 N-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrrolyl-2                               27 N-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrrolyl-2                               28 N-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrrolyl-2                                29 N-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrrolyl-2                                30 N-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrrolyl-2                                31 N-(4'-CN--C.sub.6 H.sub.4)-Pyrrolyl-2                                       32 N-(3'-CN--C.sub.6 H.sub.4)-Pyrrolyl-2                                       33 N-(2'-CN--C.sub.6 H.sub.4)-Pyrrolyl-2                                       34 N-(4'-Cl--C.sub.6 H.sub.4)-Pyrrolyl-2                                       35 N-(3'-Cl--C.sub.6 H.sub.4)-Pyrrolyl-2                                       36 N-(2'-Cl--C.sub.6 H.sub.4)-Pyrrolyl-2                                       37 Furyl-2                                                                     38 5-CH.sub.3 -Furyl-2                                                         39 5-C.sub.6 H.sub.5 -Furyl-2                                                  40 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Furyl-2                                   41 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Furyl-2                                   42 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Furyl-2                                   43 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Furyl-2                                  44 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Furyl-2                                  45 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Furyl-2                                  46 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Furyl-2                                   47 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Furyl-2                                   48 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Furyl-2                                   49 5-(4'-CN--C.sub.6 H.sub.4)-Furyl-2                                          50 5-(3'-CN--C.sub.6 H.sub.4)-Furyl-2                                          51 5-(2'-CN--C.sub.6 H.sub.4)-Furyl-2                                          52 5-(4'-Cl--C.sub.6 H.sub.4)-Furyl-2                                          53 5-(3'-Cl--C.sub.6 H.sub.4)-Furyl-2                                          54 5-(2'-Cl--C.sub.6 H.sub.4)-Furyl-2                                          55 4-CH.sub.3 -Furyl-2                                                         56 4-C.sub.6 H.sub.5 -Furyl-2                                                  57 4-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Furyl-2                                   58 4-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Furyl-2                                   59 4-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Furyl-2                                   60 4-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Furyl-2                                  61 4-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Furyl-2                                  62 4-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Furyl-2                                  63 4-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Furyl-2                                   64 4-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Furyl-2                                   65 4-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Furyl-2                                   66 4-(4'-CN--C.sub.6 H.sub.4)-Furyl-2                                          67 4-(3'-CN--C.sub.6 H.sub.4)-Furyl-2                                          68 4-(2'-CN--C.sub.6 H.sub.4)-Furyl-2                                          69 4-(4'-Cl--C.sub.6 H.sub.4)-Furyl-2                                          70 4-(3'-Cl--C.sub.6 H.sub.4)-Furyl-2                                          71 4-(2'-Cl-C.sub.6 H.sub.4)-Furyl-2                                           72 Thienyl-2                                                                   73 5-CH.sub.3 -Thienyl-2                                                       74 5-C.sub.6 H.sub.4 -Thienyl-2                                                75 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-2                                 76 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-2                                 77 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-2                                 78 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-2                                79 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-2                                80 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-2                                81 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-2                                 82 s-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-2                                 83 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-2                                 84 5-(4'-CN--C.sub.6 H.sub.4)-Thienyl-2                                        85 5-(3'-CN--C.sub.6 H.sub.4)-Thienyl-2                                        86 5-(2'-CN--C.sub.6 H.sub.4)-Thienyl-2                                        87 5-(4'-Cl--C.sub.6 H.sub.4)-Thienyl-2                                        88 5-(3'-Cl--C.sub.6 H.sub.4)-Thienyl-2                                        89 5-(2'-Cl--C.sub.6 H.sub.4)-Thienyl-2                                        90 4-CH.sub.3 -Thienyl-2                                                       91 4-C.sub.6 H.sub.5 -Thienyl-2                                                92 4-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-2                                 93 4-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-2                                 94 4-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-2                                 95 4-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-2                                96 4-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-2                                97 4-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-2                                98 4-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-2                                 99 4-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-2                                100 4-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-2                                101 4-(4'-CN--C.sub.6 H.sub.4)-Thienyl-2                                       102 4-(3'-CN--C.sub.6 H.sub.4)-Thienyl-2                                       103 4-(2'-CN--C.sub.6 H.sub.4)-Thienyl-2                                       104 4-(4'-Cl--C.sub.6 H.sub.4)-Thienyl-2                                       105 4-(3'-Cl--C.sub.6 H.sub.4)-Thienyl-2                                       106 4-(2'-Cl--C.sub.6 H.sub.4)-Thienyl-2                                       107 Thienyl-3                                                                  108 5-CH.sub.3 -Thienyl-3                                                      109 5-C.sub.6 H.sub.5 -Thienyl-3                                               110 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-3                                111 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-3                                112 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-3                                113 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-3                               114 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-3                               115 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-3                               116 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-3                                117 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-3                                118 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-3                                119 5-(4'-CN--C.sub.6 H.sub.4)-Thienyl-3                                       120 5-(3'-CN--C.sub.6 H.sub.4)-Thienyl-3                                       121 5-(2'-CN--C.sub.6 H.sub.4)-Thienyl-3                                       122 5-(4'-Cl--C.sub.6 H.sub.4)-Thienyl-3                                       123 5-(3'-Cl--C.sub.6 H.sub.4)-Thienyl-3                                       124 5-(2'-Cl--C.sub.6 H.sub.4)-Thienyl-3                                       125 Pyrazolyl-4                                                                126 N--CH.sub.3 -Pyrazolyl-4                                                   127 N--C.sub.6 H.sub.5 -Pyrazolyl-4                                            128 N-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrazolyl-4                              129 N-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrazolyl-4                              130 N-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrazolyl-4                              131 N-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrazolyl-4                             132 N-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrazolyl-4                             133 N-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrazolyl-4                             134 N-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrazolyl-4                              135 N-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrazolyl-4                              136 N-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrazolyl-4                              137 N-(4'-CN--C.sub.6 H.sub.4)-Pyrazolyl-4                                     138 N-(3'-CN--C.sub.6 H.sub.4)-Pyrazolyl-4                                     139 N-(2'-CN--C.sub.6 H.sub.4)-Pyrazolyl-4                                     140 N-(4'-Cl--C.sub.6 H.sub.4)-Pyrazolyl-4                                     141 N-(3'-Cl--C.sub.6 H.sub.4)-Pyrazolyl-4                                     142 N-(2'-Cl--C.sub.6 H.sub.4)-Pyrazolyl-4                                     143 3-CH.sub.3 --N-Methylpyrazolyl-4                                           144 3-C.sub.6 H.sub.5 --N-Methylpyrazolyl-4                                    145 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)--N-Methylpyrazolyl-4                     146 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)--N-Methylpyrazolyl-4                     147 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)--N-Methylpyrazolyl-4                     148 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)--N-Methylpyrazolyl-4                    149 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)--N-Methylpyrazolyl-4                    150 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)--N-Methylpyrazolyl-4                    151 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)--N-Methylpyrazolyl-4                     152 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)--N-Methylpyrazolyl-4                     153 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)--N-Methylpyrazolyl-4                     154 3-(4'-CN--C.sub.6 H.sub.4)--N-Methylpyrazolyl-4                            155 3-(3'-CN--C.sub.6 H.sub.4)--N-Methylpyrazolyl-4                            156 3-(2'-CN--C.sub.6 H.sub.4)--N-Methylpyrazolyl-4                            157 3-(4'-Cl--C.sub.6 H.sub.4)--N-Methylpyrazolyl-4                            158 3-(3'-Cl--C.sub.6 H.sub.4)--N-Methylpyrazolyl-4                            159 3-(2'-Cl--C.sub.6 H.sub.4)--N-Methylpyrazolyl-4                            160 Isoxazolyl-5                                                               161 3-CH.sub.3 -Isoxazolyl-5                                                   162 3-C.sub.6 H.sub.5 -Isoxazolyl-5                                            163 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Isoxazolyl-5                             164 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Isoxazolyl-5                             165 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Isoxazolyl-5                             166 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Isoxazolyl-5                            167 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Isoxazolyl-5                            168 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Isoxazolyl-5                            169 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Isoxazolyl-5                             170 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Isoxazolyl-5                             171 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Isoxazolyl-5                             172 3-(4'-CN--C.sub.6 H.sub.4)-Isoxazolyl-5                                    173 3-(3'-CN--C.sub.6 H.sub.4)-Isoxazolyl-5                                    174 3-(2'-CN--C.sub.6 H.sub.4)-Isoxazolyl-5                                    175 3-(4'-Cl--C.sub.6 H.sub.4)-Isoxazolyl-5                                    176 3-(3'-Cl--C.sub.6 H.sub.4)-Isoxazolyl-5                                    177 3-(2'-Cl--C.sub.6 H.sub.4)-Isoxazolyl-5                                    178 4-Chloroisoxazolyl-5                                                       179 3-CH.sub.3 -4-Chloroisoxazolyl-5                                           180 3-C.sub.6 H.sub.5 -4-Chloroisoxazolyl-5                                    181 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                     182 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                     183 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                     184 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                    185 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                    186 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                    187 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                     188 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                     189 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                     190 3-(4'-CN--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                            191 3-(3'-CN--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                            192 3-(2'-CN--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                            193 3-(4'-Cl--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                            194 3-(3'-Cl--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                            195 3-(2'-Cl--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                            196 Isoxazolyl-3                                                               197 5-CH.sub.3 -Isoxazolyl-3                                                   198 5-C.sub.6 H.sub.5 -Isoxazolyl-3                                            199 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Isoxazolyl-3                             200 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Isoxazolyl-3                             201 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Isoxazolyl-3                             202 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Isoxazolyl-3                            203 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Isoxazolyl-3                            204 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Isoxazolyl-3                            205 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Isoxazolyl-3                             206 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Isoxazolyl-3                             207 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Isoxazolyl-3                             208 5-(4'-CN--C.sub.6 H.sub.4)-Isoxazolyl-3                                    209 5-(3'-CN--C.sub.6 H.sub.4)-Isoxazolyl-3                                    210 5-(2'-CN--C.sub.6 H.sub.4)-Isoxazolyl-3                                    211 5-(4'-Cl--C.sub.6 H.sub.4)-Isoxazolyl-3                                    212 5-(3'-Cl--C.sub.6 H.sub.4)-Isoxazolyl-3                                    213 5-(2'-Cl--C.sub.6 H.sub.4)-Isoxazolyl-3                                    214 Isothiazolyl-5                                                             215 3-CH.sub.3 -Isothiazolyl-5                                                 216 3-C.sub.6 H.sub.4 -Isothiazolyl-5                                          217 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Isothiazolyl-5                           218 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Isothiazolyl-5                           219 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Isothiazolyl-5                           220 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Isothiazolyl-5                          221 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Isothiazolyl-5                          222 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Isothiazolyl-5                          223 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Isothiazolyl-5                           224 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Isothiazolyl-5                           225 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Isothiazolyl-5                           226 3-(4'-CN--C.sub.6 H.sub.4)-Isothiazolyl-5                                  227 3-(3'-CN--C.sub.6 H.sub.4)-Isothiazolyl-5                                  228 3-(2'-CN--C.sub.6 H.sub.4)-Isothiazolyl-5                                  229 3-(4'-Cl--C.sub.6 H.sub.4)-Isothiazolyl-5                                  230 3-(3'-Cl--C.sub.6 H.sub.4)-Isothiazolyl-5                                  231 3-(2'-Cl--C.sub.6 H.sub.4)-Isothiazolyl-5                                  232 Oxazolyl-4                                                                 233 2-CH.sub.3 -Oxazolyl-4                                                     234 2-C.sub.6 H.sub.5 -Oxazolyl-4                                              235 2-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Oxazolyl-4                               236 2-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Oxazolyl-4                               237 2-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Oxazolyl-4                               238 2-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Oxazolyl-4                              239 2-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Oxazolyl-4                              240 2-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Oxazolyl-4                              241 2-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Oxazolyl-4                               242 2-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Oxazolyl-4                               243 2-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Oxazolyl-4                               244 2-(4'-CN--C.sub.6 H.sub.4)-Oxazolyl-4                                      245 2-(3'-CN--C.sub.6 H.sub.4)-Oxazolyl-4                                      246 2-(2'-CN--C.sub.6 H.sub.4)-Oxazolyl-4                                      247 2-(4'-Cl--C.sub.6 H.sub.4)-Oxazolyl-4                                      248 2-(3'-Cl--C.sub.6 H.sub.4)-Oxazolyl-4                                      249 2-(2'-Cl--C.sub.6 H.sub.4)-Oxazolyl-4                                      250 Thiazolyl-4                                                                251 2-CH.sub.3 -Thiazolyl-4                                                    252 2-C.sub.6 H.sub.5 -Thiazolyl-4                                             253 2-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Thiazolyl-4                              254 2-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Thiazolyl-4                              255 2-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Thiazolyl-4                              256 2-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Thiazolyl-4                             267 2-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Thiazolyl-4                             258 2-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Thiazolyl-4                             259 2-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Thiazolyl-4                              260 2-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Thiazolyl-4                              261 2-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Thiazolyl-4                              262 2-(4'-CN--C.sub.6 H.sub.4)-Thiazolyl-4                                     263 2-(3'-CN--C.sub.6 H.sub.4)-Thiazolyl-4                                     264 2-(2'-CN--C.sub.6 H.sub.4)-Thiazolyl-4                                     265 2-(4'-Cl--C.sub.6 H.sub.4)-Thiazolyl-4                                     266 2-(3'-Cl--C.sub.6 H.sub.4)-Thiazolyl-4                                     267 2-(2'-Cl--C.sub.6 H.sub.4)-Thiazolyl-4                                     268 N--CH.sub.3 -1,2,4-Triazolyl-5                                             269 3-CH.sub.3 --N--CH.sub.3 -1,2,4-Triazolyl-5                                270 3-C.sub.6 H.sub.5 --N--CH.sub.3 -1,2,4-Triazolyl-5                         271 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5                   272 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triaz               olyl-5                                                                 273 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5                   274 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Tria               zolyl-5                                                                275 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5                  276 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Tria               zolyl-5                                                                277 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5                   278 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triaz               olyl-5                                                                 279 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5                   280 3-(4'-CN--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5        281 3-(3'-CN--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5                 282 3-(2'-CN--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5                 283 3-(4'-Cl--C.sub.6 H.sub.4)--N--CH.sub.3 -1,214-Triazolyl-5                 284 3-(3'-Cl--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5                 285 3-(2'-Cl--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5                 286 1,3,4-Oxadiazolyl-2                                                        287 5-CH.sub.3 -1,3,4-Oxadiazolyl-2                                            288 5-C.sub.6 H.sub.5 -1,2,3-Oxadiazolyl-2                                     289 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                      290 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                      291 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                      292 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                     293 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                     294 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                     295 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                      296 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                      297 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                      298 5-(4'-CN--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                             299 5-(3'-CN--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                             300 5-(2'-CN--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                             301 5-(4'-Cl--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                             302 5-(3'-Cl--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                             303 5-(2'-Cl--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                             304 1,2,4-Oxadiazolyl-3                                                        305 5-CH.sub.3 -1,2,4-Oxadiazolyl-3                                            306 5-C.sub.6 H.sub.5 -1,2,4-Oxadiazolyl-3                                     307 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                      308 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                      309 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                      310 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                     311 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                     312 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                     313 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                      314 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                      315 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                      316 5-(4'-CN--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                             317 5-(3'-CN--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                             318 5-(2'-CN--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                             319 5-(4'-Cl--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                             320 5-(3'-Cl--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                             321 5-(2'-Cl--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                             322 1,2,4-Oxadiazolyl-5                                                        323 3-CH.sub.3 -1,2,4-Oxadiazolyl-5                                            324 3-C.sub.6 H.sub.5 -1,2,4-Oxadiazolyl-5                                     325 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                      326 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                      327 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                      328 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                     329 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                     330 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                     331 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                      332 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                      333 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                      334 3-(4'-CN--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                             335 3-(3'-CN--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                             336 3-(2'-CN--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                             337 3-(4'-Cl--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                             338 3-(3'-Cl--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                             339 3-(2'-Cl--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                             340 1,2,4-Thiadiazolyl-3                                                       341 5-CH.sub.3 -1,2,4-Thiadiazolyl-3                                           342 5-C.sub.6 H.sub.4 -1,2,4-Thiadiazolyl-3                                    343 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                     344 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                     345 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                     346 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                    347 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                    348 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                    349 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                     350 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                     351 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                     352 5-(4'-CN--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                            353 5-(3'-CN--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                            354 5-(2'-CN--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                            355 5-(4'-Cl--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                            356 5-(3'-Cl--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                            357 5-(2'-Cl--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                            358 1,3,4-Thiadiazolyl-2                                                       359 5-CH.sub.3 -1,3,4-Thiadiazolyl-2                                           360 5-C.sub.6 H.sub.5 -1,3,4-Thiadiazolyl-2                                    361 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                     362 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                     363 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                     364 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                    365 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                    366 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                    367 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                     368 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                     369 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                     370 5-(4'-CN--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                            371 5-(3'-CN--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                            372 5-(2'-CN--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                            373 5-(4'-Cl--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                            374 5-(3'-Cl--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                            375 5-(2'-Cl--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                            376 Pyridinyl-2                                                                377 Pyridinyl-4                                                                378 Pyridazinyl-3                                                              379 Pyridazinyl-4                                                              380 Pyridazinyl-2                                                              381 Pyrimidinyl-4                                                              382 Pyrimidinyl-5                                                              383 Pyrimidinyl-2                                                              384 Pyridinyl-3                                                              ______________________________________                                    

                                      TABLE 30                                     __________________________________________________________________________     Selected physical data of some compounds                                       No.                                                                               Compound                 IR (cm.sup.-1) or .sup.1 H-NMR (ppm)                                                        m.p                                   __________________________________________________________________________       1                                                                                                                     2   81 41##                              - 2                                                                                                                  3   60 42##                              - 3                                                                                                                  4  3.85(s, broad, 3H); 3.7(s,                                                  broad, 3H)                               - 4                                                                                                                  5  3.85(s, broad, 3H); 3.75(s,                                                 broad, 3H)                               - 5                                                                                                                  6  3.75(2s, broad, each 3H)                                                      - 6                                                                          7   91 46##                              - 7                                                                                                                  8  3.8(s, 3H); 3.75(s, broad,                                                  3H)                                      - 8                                                                                                                  9  3.85(s, 3H); 3.8(s, broad,         __________________________________________________________________________                                              3H)                              

                  TABLE 31                                                         ______________________________________                                         0  STR249##                                                                       -        I: R.sup.1 = CH.sub.3, X = CH.sub.3                                  II: R.sup.1 = C.sub.2 H.sub.5, X = CH.sub.3                                    III: R.sup.1 = CH.sub.3, X = Cl                                                IV: R.sup.1 = C.sub.2 H.sub.5, X = Cl                                        No.     B                                                                      ______________________________________                                         1       2-Pyridyl                                                                2 3-Trifluoromethyl-2-pyridyl                                                  3 5-Trifluoromethyl-2-pyridyl                                                  4 3,5-Bis-(trifluoromethyl)-2-pyridyl                                          5 3,5-Dichloro-2-pyridyl                                                       6 3-Chloro-5-trifluoromethyl-2-pyridyl                                         7 3,5-Dichloro-2-pyridyl                                                       8 2-Chloro-4-trifluoromethylphenyl                                             9 2-Benzothiazolyl                                                             10  5-Chloro-1-methyl-2-benzimidazolyl                                         11  2-Benzoxazolyl                                                             12  1-Methyl-5-trifluoromethylimidazo-[5,4-a]-pyridin-2-yl                     13  5-Chloro-2-pyrimidinyl                                                     14  4-Methyl-5-phenyl-2-thiazolin-2-yl                                         15  4-Methyl-5-phenyl-2-oxazolin-2-yl                                          16  7-Trifluoromethyl-4-quinolinyl                                           ______________________________________                                    

                  TABLE 57                                                         ______________________________________                                         Selected physical data of some compounds                                       1  STR250##                                                                       -                            mp   .sup.1 H-NMR (ppm)                          No. X T.sub.m (° C.) or IR (cm.sup.-1)                                ______________________________________                                         1    Cl     2-CH.sub.3           3.8(s, broad, 6H)                               2 Cl 2,5-(CH.sub.3).sub.2 3.8(s, broad, 6H)                                    3 Cl 2-CH.sub.3 -4-C(CH.sub.3)═N--OCH.sub.3 4.0(s, 3H); 3.8                                                   (s, broad, 6H)                              4 Cl 2,5-(CH.sub.3).sub.2 -4-C(CH.sub.3)═N--O- 3.8(s, broad, 6H)                                             Allyl                                        5 CH.sub.3 2-CH.sub.3 -4-C(CH.sub.3)═N--OCH.sub.3 4.0(s, 3H); 3.75                                            (s, broad, 6H)                              6 CH.sub.3 2-CH.sub.3 3.75(s, broad,                                              6H)                                                                         7 CH.sub.3 2,5-(CH.sub.3).sub.2 3.75(s, broad,                                    6H)                                                                         8 CH.sub.3 2,5-(CH.sub.3).sub.2 -4-C(CH.sub.3 ═N--O- 3.75(s, broad,          Allyl 6H)                                                                  ______________________________________                                    

Example 11

2-(2'-Methylphenoxymethyl)-trichloroacetanilide (Table 38, No. 1)

) 2-(2'-Methylphenoxymethyl)-nitrobenzene

75 g (0.347 mol) of 2-nitrobenzyl bromide, 37 g (0.342 mol) of o-cresol and 56 g (0.405 mol) of potassium carbonate in 500 ml of dimethylformamide is stirred for 5 hours at room temperature (20° C. ). The reaction mixture is diluted with water and the aqueous phase is extracted three times with ether. The ether phase is dried and evaporated down. The crystalline residue is stirred with methanol and suction filtered. There is obtained 73 g (0.300 mol=88%) of the title compound as a colorless solid. Mp=83° C.

¹ H-NMR, (CDCl₃ ; δ (ppm)): 8.15 (d, 1H, I=8 Hz, aromatic); 7.95 (d, 1H, I=8 Hz, aromatic); 7.7 (t, 1H, I=8 Hz, aromatic); 7.45 (t, 1H, I=8 Hz, aromatic); 7.15 (m, 2H, aromatic); 6.9 (m, 2H, aromatic); 5.45 (s, 2H, O--CH₂); 2.35 (s, 3H, CH₃)

b) 2-(2'-Methylphenoxymethyl)-aniline

75 g (0.308 mol) of 2-(2'-methylphenoxymethyl)-nitrobenzene (Example 11a) and 10 g of 5% Pt/C (platinum adsorbed on activated carbon) in 50 ml of methanol are stirred vigorously under a hydrogen blanket for 2 hours. A further 2 g of 5% Pt/C is added and the mixture is stirred overnight. The catalyst is filtered off and replaced by 10 g of fresh catalyst. The mixture is stirred overnight and suction filtered, and the filtrate is evaporated down under reduced pressure. The residue is purified by column chromatography with mixtures of hexane and ethyl acetate. There is obtained 61 g (0.286 mol=93%) of the title compound as a colorless solid.

Mp=56° C.

¹ H-NMR (CDCl₃ ; δ (ppm)): 7.2 (m, 4H, aromatic); 6.95 (d, 1H, I=8 Hz, aromatic); 6,9 (t, 1H, I=6 Hz, aromatic); 6.7 (m, 2H, aromatic); 5.0 (s, 2H, O--CH₂); 4.05 (s, broad, 2H, NH₂); 2.2 (s, 3H, CH₃)

c) 2-(2'-Methylphenoxymethyl)-trichloroacetanilide (Table 38, No. 1)

At 10-15° C., a solution of 6 g of 2-(2'-methylphenoxymethyl)-aniline (Example 1b) in 20 ml of CH₂ Cl₂ is added to a mixture of 6.6 g (36 mmol) of trichloroacetyl chloride and 3 g (38 mmol) of pyridine in 50 ml of CH₂ Cl₂. The mixture is stirred for 1 hour at room temperature, and then extracted with water, dried over MgSO₄ and evaporated down. The residue is suction filtered over silica gel and the filtrate which is obtained is evaporated down. The residue crystallizes and is stirred with hexane. There is obtained 7.9 g (22 mmol=78%) of the title compound as a crystalline solid (mp=128° C).

¹ H-NMR (CDCl₃ ; δ (ppm)): 9.6 (s, broad, 1H, NH); 8.1 (d, 1H, I=8 Hz, phenyl); 7.5 (t, broad, 1H, phenyl); 7.4 (d, broad, 1H, phenyl); 7.2 (m, 3H, phenyl); 6.95 (m, 2H, phenyl); 5.1 (s, 2H, OCH₂); 2.2 (s, 3H, CH₃)

Example 12

N-Methyl-N'-(2-(2'-methylphenoxymethyl)-phenyl)-urea (Table 7, No. 2)

In a laboratory autoclave, about 10 ml of methylamine is added to 2 g (5.5 mmol) of the trichloroacetanilide from Example 1c. The autoclave is then closed and the reaction mixture is heated for about 6 hours at 80° C. The reaction mixture is cooled and the autoclave opened. The methylamine is allowed to evaporate off and the solid residue is stirred with methyl tert-butyl ether. The insoluble solid is filtered off and dried under reduced pressure. There is obtained 1.4 g (5.2 mmol=94%) of the title compound as a crystalline solid (mp=144° C.).

¹ H-NMR (DMSO-d₆ ; δ (ppm)): 8.05 (s, 1H, NH); 7.8 (d, 1H, I=8 Hz, phenyl); 7.4 (d, 1H, I=8 Hz, phenyl); 6.8-7.3 (m, 6H, phenyl); 6.7 (s, 1H, NH); 5.1 (s, 2H, OCH₂); 2.65 (d, 3H, I=5 Hz, N--CH₃); 2.2 (s, 3H, CH₃)

Example 13

2-(2'-Methylphenoxymethyl)-propionyl anilide (Table 38, No. 3)

A mixture of 3 g (14.1 mmol) of the aniline from Example 11b, 1.35 g (17 mmol) of pyridine and 1.4 g (15.5 mmol) of propionyl chloride in 30 ml of methylene chloride is stirred for 1 hour at room temperature. The reaction mixture is then extracted with diluted hydrochloric acid and water, dried over MgSO₄ and evaporated down. There is obtained 3.8 g (quantitative yield) of the title compound.

¹ H-NMR (COCl₃ ; δ (ppm)): 8.25 (s, broad, 1H, NH); 8.15 (d, 1H, I=8 Hz, phenyl); 6.9-7.5 (m, 7H, phenyl); 5.1 (s, 2H, OCH₂); 2.35 (q, 2H, I=8 Hz, CH₂); 2.25 (s, 3H, CH₃); 1.2 (t, 3H, I=8 Hz, CH₃)

Example 14

N-Propionyl-2-(2'-methylphenoxymethyl)-propionyl anilide (Table 38, No. 4)

0.41 g (17.1 mmol) of sodium hydride is added in portions to 3.8 g (14 mmol) of the propionyl anilide from Example 13 in 40 ml of dimethylformamide. Upon completion of gas evolution 1.4 g (15.9 mmol) of propionyl chloride is added and the mixture is stirred overnight at room temperature. The reaction mixture is then diluted with water and the aqueous phase is extracted three times with methyl tert-butyl ether. The combined organic phases are extracted with water, dried over MgSO₄ and evaporated down. The residue is purified by column chromatography with mixtures of hexane and ethyl acetate. There is obtained 2.6 g (8 mmol=57%) of the title compound as a yellow oil.

¹ H-NMR (CDCl₃): δ (ppm): 7.6 (m, 1H, phenyl); 7.4 (m, 2H, phenyl); 7.15 (m, 3H, phenyl); 6.85 (m, 2H, phenyl); 4.85 (m, 2H, OCH₂); 2.6 (m, 4H, 2×CH₂); 2.2 (s, 3H, CH₃); 1.1 (t, 6H, I=8 Hz, 2×CH₃)

Example 15

N-Methyl-2-(2'-methylphenoxymethyl)-propionyl anilide (Table 38, No. 5)

0.45 g (19 mmol) of sodium hydride is added in portions to 4.0 g (14.8 mmol) of the propionyl anilide from Example 13 in 50 ml of dimethylformamide. Upon completion of gas evolution 3.0 g (21 mmol) of methyl iodide is added and the mixture is stirred for 2 hours at room temperature. The reaction mixture is then diluted with water and the aqueous phase is extracted three times with methyl tert-butyl ether. The combined organic phases are extracted with water, dried over MgSO₄ and evaporated down. The residue crystallizes and is stirred with hexane. There is obtained 3.7 g (11.7 mmol=90%) of the title compound as a colorless solid (mp=80° C.).

1H-NMR (CDCl₃ ; δ (ppm): 7.7 (m, 1H, phenyl); 7.4 (m, 2H, phenyl); 7.2 (m, 3H, phenyl); 6.9 (m, 2H, phenyl); 5.0 (s, 2H, OCH₂); 3.2 (s, 3H, N--CH₃); 2.2 (s, 3H, CH₃); 2.0 (m, 2H, CH₂); 1.0 (t, 3H, I=8 Hz, CH₃)

Example 19

N-Methyl-2-(2'-methylphenoxymethyl)-acetanilide

a) N-Methyl-2-(2'-methylphenoxymethyl)-aniline

A mixture of 5 g (23 mmol) of 2-(2'-methylphenoxymethyl)-aniline (Example 1b), 5 g (36 mmol) of K₂ CO₃ and 3.4 g (24 mmol) of methyl iodide in 50 ml of dimethylformamide is stirred overnight at room temperature. The reaction mixture is diluted with water and the aqueous phase is extracted three times with methyl tert-butyl ether. The combined organic phases are extracted with water, dried over MgSO₄ and evaporated down. The residue is purified chromatographically using mixtures of hexane and methylene chloride. There is obtained 3.0 g (70% purity, about 40% yield) of the title compound as a yellow oil.

¹ H-NMR (CDCl₃ ; δ in ppm): 6.6-7.4 (m, 8H, phenyl); 5.0 (s, 2H, OCH₂); 4.6 (s, broad, 1H, NH); 2.9 (d, 3H, N--CH₃); 2.2 (s, 3H, CH₃).

b) N-Methyl-2-(2'-methylphenoxymethyl)-acetanilide (Table 7, No. 9)

3 g (approx. 9.3 mmol) of N-methyl-2-(2'-methylphenoxymethyl)-aniline (from Example 5a) is added to a mixture of 1.6 g (16 mmol) of acetoanhydride and 1.3 g (16 mmol) of pyridine in 20 ml of methylene chloride. The mixture is stirred for 1 hour at room temperature and is then extracted with dilute hydrochloric acid and water. The organic phase is evaporated down and the residue is purified by column chromatography with mixtures of hexane and ethyl acetate. There is obtained 2 g (80%) of the title compound as a colorless solid (mp=76° C.).

¹ H-NMR (CDCl₃ ; δ in ppm): 7.7 (m, 1H, phenyl); 7.4 (m, 2H, phenyl); 7.2 (m, 3H, phenyl); 6.9 (m, 2H, phenyl); 5.0 (s, 2H, OCH₂); 3.25 (s, 3H, CH₃); 2.25 (s, 3H, CH₃); 1.8 (s, 3H, CH₃).

The compounds listed in the tables below may be prepared correspondingly.

Compound I from Table 32, No. 1 has for example the following structural formula: ##STR251##

The compounds described in the following tables may be prepared analogously.

                  TABLE 32                                                         ______________________________________                                         1  STR252##                                                                      I: R.sup.1 = H, Z = C.sub.2 H.sub.5                                                              VIII: R.sup.1 = H, Z = NH(CH.sub.3)                          II: R.sup.1 = CH.sub.3, Z = C.sub.2 H.sub.5 IX: R.sup.1 = CH.sub.3, Z =                          NH(CH.sub.3)                                                 III: R.sup.1 = C.sub.2 H.sub.5, Z = C.sub.2 H.sub.5 X: R.sup.1 =                                 C.sub.2 H.sub.5, Z = NH(CH.sub.3)                            IV: R.sup.1 = Allyl, Z = C.sub.2 H.sub.5 XI: R.sup.1 = Allyl, Z =                                NH(CH.sub.3)                                                 V: R.sup.1 = Propargyl, Z = C.sub.2 H.sub.5 XII: R.sup.1 = Propargyl, Z                          = NH(CH.sub.3)                                               VI: R.sup.1 = CH.sub.2 --OCH.sub.3, XIII: R.sup.1 = CH.sub.2 --OCH.sub.3                         , Z = NH(CH.sub.3)                                           Z = C.sub.2 H.sub.5                                                            VII: R.sup.1 = CO--C.sub.2 H.sub.5, Z = C.sub.2 H.sub.5 XIV: R.sup.1 =                           CO--C.sub.2 H.sub.5, Z = NH(CH.sub.3)                      No.     X.sub.m                                                                ______________________________________                                          1      H                                                                         2 2-F                                                                          3 3-F                                                                          4 4-F                                                                          5 2,4-F.sub.2                                                                  6 2,4,6-F.sub.3                                                                7 2,3,4,5,6-F.sub.5                                                            8 2,3-F.sub.2                                                                  9 2-Cl                                                                         10 3-Cl                                                                        11 4-Cl                                                                        12 2,3-Cl.sub.2                                                                13 2,4-Cl.sub.2                                                                14 2,5-Cl.sub.2                                                                15 2,6-Cl.sub.2                                                                16 3,4-Cl.sub.2                                                                17 3,5-Cl.sub.2                                                                18 2,3,4-Cl.sub.3                                                              19 2,3,5-Cl.sub.3                                                              20 2,3,6-Cl.sub.3                                                              21 2,4,5-Cl.sub.3                                                              22 2,4,6-Cl.sub.3                                                              23 3,4,5-Cl.sub.3                                                              24 2,3,4,6-Cl.sub.4                                                            25 2,3,5,6-Cl.sub.4                                                            26 2,3,4,5,6-Cl.sub.5                                                          27 2-Br                                                                        28 3-Br                                                                        29 4-Br                                                                        30 2,4-Br.sub.2                                                                31 2,5-Br.sub.2                                                                32 2,6-Br.sub.2                                                                33 2,4,6-Br.sub.3                                                              34 2,3,4,5,6-Br.sub.5                                                          35 2-I                                                                         36 3-I                                                                         37 4-I                                                                         38 2,4-I.sub.2                                                                 39 2-Cl, 3-F                                                                   40 2-Cl, 4-F                                                                   41 2-Cl, 5-F                                                                   42 2-Cl, 6-F                                                                   43 2-Cl, 3-Br                                                                  44 2-Cl, 4-Br                                                                  45 2-Cl, 5-Br                                                                  46 2-Cl, 6-Br                                                                  47 2-Br, 3-Cl                                                                  48 2-Br, 4-Cl                                                                  49 2-Br, 5-Cl                                                                  50 2-Br, 3-F                                                                   51 2-Br, 4-F                                                                   52 2-Br, 5-F                                                                   53 2-Br, 6-F                                                                   54 2-F, 3-Cl                                                                   55 2-F, 4-Cl                                                                   56 2-F, 5-Cl                                                                   57 3-Cl, 4-F                                                                   58 3-Cl, 5-F                                                                   59 3-Cl, 4-Br                                                                  60 3-Cl, 5-Br                                                                  61 3-F, 4-Cl                                                                   62 3-F, 4-Br                                                                   63 3-Br, 4-Cl                                                                  64 3-Br, 4-F                                                                   65 2,6-Cl.sub.2, 4-Br                                                          66 2-CH.sub.3                                                                  67 3-CH.sub.3                                                                  68 4-CH.sub.3                                                                  69 2,3-(CH.sub.3).sub.2                                                        70 2,4-(CH.sub.3).sub.2                                                        71 2,5-(CH.sub.3).sub.2                                                        72 2,6-(CH.sub.3).sub.2                                                        73 3,4-(CH.sub.3).sub.2                                                        74 3,5-(CH.sub.3).sub.2                                                        75 2,3,5-(CH.sub.3).sub.3                                                      76 2,3,4-(CH.sub.3).sub.3                                                      77 2,3,6-(CH.sub.3).sub.3                                                      78 2,4,5-(CH.sub.3).sub.3                                                      79 2,4,6-(CH.sub.3).sub.3                                                      80 3,4,5-(CH.sub.3).sub.3                                                      81 2,3,4,6-(CH.sub.3).sub.4                                                    82 2,3,5,6-(CH.sub.3).sub.4                                                    83 2,3,4,5,6-(CH.sub.3).sub.5                                                  84 2-C.sub.2 H.sub.5                                                           85 3-C.sub.2 H.sub.5                                                           86 4-C.sub.2 H.sub.5                                                           87 2,4-(C.sub.2 H.sub.5).sub.2                                                 88 2,6-(C.sub.2 H.sub.5).sub.2                                                 89 3,5-(C.sub.2 H.sub.5).sub.2                                                 90 2,4,6-(C.sub.2 H.sub.5).sub.3                                               91 2-n-C.sub.3 H.sub.7                                                         92 3-n-C.sub.3 H.sub.7                                                         93 4-n-C.sub.3 H.sub.7                                                         94 2-i-C.sub.3 H.sub.7                                                         95 3-i-C.sub.3 H.sub.7                                                         96 4-i-C.sub.3 H.sub.7                                                         97 2,4-(i-C.sub.3 H.sub.7).sub.2                                               98 2,6-(i-C.sub.3 H.sub.7).sub.2                                               99 3,5-(i-C.sub.3 H.sub.7).sub.2                                              100 2,4,6-(i-C.sub.3 H.sub.7).sub.3                                            101 2-s-C.sub.4 H.sub.9                                                        102 3-s-C.sub.4 H.sub.9                                                        103 4-s-C.sub.4 H.sub.9                                                        104 2-t-C.sub.4 H.sub.9                                                        105 3-t-C.sub.4 H.sub.9                                                        106 4-t-C.sub.4 H.sub.9                                                        107 2,3-(t-C.sub.4 H.sub.9).sub.2                                              108 2,4-(t-C.sub.4 H.sub.9).sub.2                                              109 2,5-(t-C.sub.4 H.sub.9).sub.2                                              110 2,6-(t-C.sub.4 H.sub.9).sub.2                                              111 3,4-(t-C.sub.4 H.sub.9).sub.2                                              112 2,4,6-(t-C.sub.4 H.sub.9).sub.3                                            113 4-n-C.sub.9 H.sub.19                                                       114 4-n-C.sub.12 H.sub.25                                                      115 4-n-C.sub.15 H.sub.31                                                      116 4-(1,1,3,3-Tetramethylbutyl)                                               117 4-(2,4,4-Trimethylpropyl)                                                  118 2-t-C.sub.4 H.sub.9, 4-CH.sub.3                                            119 2-t-C.sub.4 H.sub.9, 5-CH.sub.3                                            120 2,6-(t-C.sub.4 H.sub.9).sub.2, 4-CH.sub.3                                  121 2-CH.sub.3, 4-t-C.sub.4 H.sub.9                                            122 2-CH.sub.3, 6-t-C.sub.4 H.sub.9                                            123 2-CH.sub.3, 4-i-C.sub.3 H.sub.7                                            124 2-CH.sub.3, 5-i-C.sub.3 H.sub.7                                            125 3-CH.sub.3, 4-i-C.sub.3 H.sub.7                                            126 2-i-C.sub.3 H.sub.7, 5-CH.sub.3                                            127 2,4-(t-C.sub.4 H.sub.9).sub.2, 6-i-C.sub.3 H.sub.7                         128 2-Allyl                                                                    129 3-Allyl                                                                    130 4-Allyl                                                                    131 2-Allyl, 6-CH.sub.3                                                        132 2-cyclo-C.sub.6 H.sub.11                                                   133 3-cyclo-C.sub.6 H.sub.11                                                   134 4-cyclo-C.sub.6 H.sub.11                                                   135 2,4-(cyclo-C.sub.6 H.sub.11).sub.2, 6-CH.sub.3                             136 2-CH.sub.3, 4-cyclo-C.sub.6 H.sub.11                                       137 2-CH.sub.2 --C.sub.6 H.sub.5                                               138 3-CH.sub.2 --C.sub.6 H.sub.5                                               139 4-CH.sub.2 --C.sub.6 H.sub.5                                               140 2-CH.sub.2 --C.sub.6 H.sub.5, 4-CH.sub.3                                   141 2-CH.sub.3, 4-CH.sub.2 --C.sub.6 H.sub.5                                   142 2-C.sub.6 H.sub.5                                                          143 3-C.sub.6 H.sub.5                                                          144 4-C.sub.6 H.sub.5                                                          145 4-(2-i-C.sub.3 H.sub.7 --C.sub.6 H.sub.4)                                  146 4-C.sub.6 H.sub.5, 2,6-(CH.sub.3).sub.2                                    147 2-Cl, 4-C.sub.6 H.sub.5                                                    148 2-Br, 4-C.sub.6 H.sub.5                                                    149 2-C.sub.6 H.sub.5, 4-Cl                                                    150 2-C.sub.6 H.sub.5, 4-Br                                                    151 2-CH.sub.2 C.sub.6 H.sub.5, 4-Cl                                           152 2-CH.sub.2 C.sub.6 H.sub.5, 4-Br                                           153 2-Cl, 4-CH.sub.2 C.sub.6 H.sub.5                                           154 2-Br, 4-CH.sub.2 C.sub.6 H.sub.5                                           155 2-cyclo-C.sub.6 H.sub.11, 4-Cl                                             156 2-cyclo-C.sub.6 H.sub.11, 4-Br                                             157 2-Cl, 4-cyclo-C.sub.6 H.sub.11                                             158 2-Br, 4-cyclo-C.sub.6 H.sub.11                                             159 2-OCH.sub.3                                                                160 3-OCH.sub.3                                                                161 4-OCH.sub.3                                                                162 2-OC.sub.2 H.sub.5                                                         163 3-O--C.sub.2 H.sub.5                                                       164 4-O--C.sub.2 H.sub.5                                                       165 2-O-n-C.sub.3 H.sub.7                                                      166 3-O-n-C.sub.3 H.sub.7                                                      167 4-O-n-C.sub.3 H.sub.7                                                      168 2-O-i-C.sub.3 H.sub.7                                                      169 3-O-i-C.sub.3 H.sub.7                                                      170 4-O-i-C.sub.3 H.sub.7                                                      171 2-O-n-C.sub.6 H.sub.13                                                     172 3-O-n-C.sub.6 H.sub.13                                                     173 4-O-n-C.sub.6 H.sub.13                                                     174 2-O-n-C.sub.8 H.sub.17                                                     175 3-O-n-C.sub.8 H.sub.17                                                     176 4-O-n-C.sub.8 H.sub.17                                                     177 2-O--CH.sub.2 C.sub.6 H.sub.5                                              178 3-O--CH.sub.2 C.sub.6 H.sub.5                                              179 4-O--CH.sub.2 C.sub.6 H.sub.5                                              180 2-O--(CH.sub.2).sub.3 C.sub.6 H.sub.5                                      181 3-O--(CH.sub.2).sub.3 C.sub.6 H.sub.5                                      182 4-O--(CH.sub.2).sub.3 C.sub.6 H.sub.5                                      183 2,4-(OCH.sub.3).sub.2                                                      184 2-CF.sub.3                                                                 185 3-CF.sub.3                                                                 186 4-CF.sub.3                                                                 187 2-OCF.sub.3                                                                188 3-OCF.sub.3                                                                189 4-OCF.sub.3                                                                190 3-OCH.sub.2 CHF.sub.2                                                      191 2-NO.sub.2                                                                 192 3-NO.sub.2                                                                 193 4-NO.sub.2                                                                 194 2-CN                                                                       195 3-CN                                                                       196 4-CN                                                                       197 2-CH.sub.3, 3-Cl                                                           198 2-CH.sub.3, 4-Cl                                                           199 2-CH.sub.3, 5-Cl                                                           200 2-CH.sub.3, 6-Cl                                                           201 2-CH.sub.3, 3-F                                                            202 2-CH.sub.3, 4-F                                                            203 2-CH.sub.3, 5-F                                                            204 2-CH.sub.3, 6-F                                                            205 2-CH.sub.3, 3-Br                                                           206 2-CH.sub.3, 4-Br                                                           207 2-CH.sub.3, 5-Br                                                           208 2-CH.sub.3, 6-Br                                                           209 2-Cl, 3-CH.sub.3                                                           210 2-Cl, 4-CH.sub.3                                                           211 2-Cl, 5-CH.sub.3                                                           212 2-F, 3-CH.sub.3                                                            213 2-F, 4-CH.sub.3                                                            214 2-F, 5-CH.sub.3                                                            215 2-Br, 3-CH.sub.3                                                           216 2-Br, 4-CH.sub.3                                                           217 2-Br, 5-CH.sub.3                                                           218 3-CH.sub.3, 4-Cl                                                           219 3-CH.sub.3, 5-Cl                                                           220 3-CH.sub.3, 4-F                                                            221 3-CH.sub.3, 5-F                                                            222 3-CH.sub.3, 4-Br                                                           223 3-CH.sub.3, 5-Br                                                           224 3-F, 4-CH.sub.3                                                            225 3-Cl, 4-CH.sub.3                                                           226 3-Br, 4-CH.sub.3                                                           227 2-Cl, 4,5-(CH.sub.3).sub.2                                                 228 2-Br, 4,5-(CH.sub.3).sub.2                                                 229 2-Cl, 3,5-(CH.sub.3).sub.2                                                 230 2-Br, 3,5-(CH.sub.3).sub.2                                                 231 2,6-Cl.sub.2, 4-CH.sub.3                                                   232 2,6-F.sub.2, 4-CH.sub.3                                                    233 2,6-Br.sub.2, 4-CH.sub.3                                                   234 2,4-Br.sub.2, 6-CH.sub.3                                                   235 2,4-F.sub.2, 6-CH.sub.3                                                    236 2,4-Br.sub.2, 6-CH.sub.3                                                   237 2,6-(CH.sub.3).sub.2, 4-F                                                  238 2,6-(CH.sub.3).sub.2, 4-Cl                                                 239 2,6-(CH.sub.3).sub.2, 4-Br                                                 240 3,5-(CH.sub.3).sub.2, 4-F                                                  241 3,5-(CH.sub.3).sub.2, 4-Cl                                                 242 3,5-(CH.sub.3).sub.2, 4-Br                                                 243 2,3,6-(CH.sub.3).sub.3, 4-F                                                244 2,3,6-(CH.sub.3).sub.3, 4-Cl                                               245 2,3,6-(CH.sub.3).sub.3, 4-Br                                               246 2,4-(CH.sub.3).sub.2, 6-F                                                  247 2,4-(CH.sub.3).sub.2, 6-Cl                                                 248 2,4-(CH.sub.3).sub.2, 6-Br                                                 249 2-i-C.sub.3 H.sub.7, 4-Cl, 5-CH.sub.3                                      250 2-Cl, 4-NO.sub.2                                                           251 2-NO.sub.2, 4-Cl                                                           252 2-OCH.sub.3, 5-NO.sub.2                                                    253 2,4-Cl.sub.2, 5-NO.sub.2                                                   254 2,4-Cl.sub.2, 6-NO.sub.2                                                   255 2,6-Cl.sub.2, 4-NO.sub.2                                                   256 2,6-Br.sub.2, 4-NO.sub.2                                                   257 2,6-I.sub.2, 4-NO.sub.2                                                    258 2-CH.sub.3, 5-i-C.sub.3 H.sub.7, 4-Cl                                      259 2-CO.sub.2 CH.sub.3                                                        260 3-CO.sub.2 CH.sub.3                                                        261 4-CO.sub.2 CH.sub.3                                                        262 2-CO.sub.2 (C.sub.2 H.sub.5)                                               263 3-CO.sub.2 (C.sub.2 H.sub.5)                                               264 4-CO.sub.2 (C.sub.2 H.sub.5)                                               265 2-CO.sub.2 (n-C.sub.3 H.sub.7)                                             266 3-CO.sub.2 (n-C.sub.3 H.sub.7)                                             267 4-CO.sub.2 (n-C.sub.3 H.sub.7)                                             268 2-CO.sub.2 (i-C.sub.3 H.sub.7)                                             269 3-CO.sub.2 (i-C.sub.3 H.sub.7)                                             270 4-CO.sub.2 (i-C.sub.3 H.sub.7)                                             271 2-CO.sub.2 (n-C.sub.6 H.sub.13)                                            272 3-CO.sub.2 (n-C.sub.6 H.sub.13)                                            273 4-CO.sub.2 (n-C.sub.6 H.sub.13)                                            274 2-CH.sub.2 --OCH.sub.3                                                     275 3-CH.sub.2 --OCH.sub.3                                                     276 4-CH.sub.2 --OCH.sub.3                                                     277 2-CH.sub.2 O(C.sub.2 H.sub.5)                                              278 3-CH.sub.2 O(C.sub.2 H.sub.5)                                              279 4-CH.sub.2 O(C.sub.2 H.sub.5)                                              280 2-CH.sub.2 O(n-C.sub.3 H.sub.7)                                            281 3-CH.sub.2 O(n-C.sub.3 H.sub.7)                                            282 4-CH.sub.2 O(n-C.sub.3 H.sub.7)                                            283 2-CH.sub.2 O(i-C.sub.3 H.sub.7)                                            284 3-CH.sub.2 O(i-C.sub.3 H.sub.7)                                            285 4-CH.sub.2 O(i-C.sub.3 H.sub.7)                                            286 2-CHO                                                                      287 3-CHO                                                                      288 4-CHO                                                                      289 2-CO--CH.sub.3                                                             290 3-CO--CH.sub.3                                                             291 4-CO--CH.sub.3                                                             292 2-CO--CH.sub.2 --CH.sub.3                                                  293 3-CO--CH.sub.2 --CH.sub.3                                                  294 4-CO--CH.sub.2 --CH.sub.3                                                  295 2-CO--CH.sub.2 --CH.sub.2 --CH.sub.3                                       296 3-CO--CH.sub.2 --CH.sub.2 --CH.sub.3                                       297 4-CO--CH.sub.2 --CH.sub.2 --CH.sub.3                                       298 2-CO--CH(CH.sub.3)--CH.sub.3                                               299 3-CO--CH(CH.sub.3)--CH.sub.3                                               300 4-CO--CH(CH.sub.3)--CH.sub.3                                               301 2-Me-4-CHO                                                                 302 2-Me-4-CO--CH.sub.3                                                        303 2-Me-4-CH.sub.3 --CH.sub.2 --CO                                            304 2-Me-4-CO--CH.sub.2 --CH.sub.2 --CH.sub.3                                  305 2-Me-4-CO--CH(CH.sub.3).sub.2                                              306 2,5-Me.sub.2 -4-CHO                                                        307 2,5-Me.sub.2 -4-CO--CH.sub.3                                               308 2,5-Me.sub.2 -4-CO--CH.sub.2 --CH.sub.3                                    309 2,5-Me.sub.2 -4-CH.sub.2 --CH.sub.2 --CO--CH.sub.3                         310 2,5-Me.sub.2 -4-CO--CH(CH.sub.3).sub.2                                     311 2-Cl-4-CHO                                                                 312 2-Cl-4-CO--CH.sub.3                                                        313 2-Cl-4-CO--CH.sub.2 --CH.sub.3                                             314 2-Cl-4-CO--CH(CH.sub.3).sub.2                                              315 2,5-Cl.sub.2 -4-CHO                                                        316 2,5-Cl.sub.2 -4-CO--CH.sub.3                                               317 2,5-Cl.sub.2 -4-CO--CH.sub.2 --CH.sub.3                                    318 2,5-Cl.sub.2 -4-CO--CH.sub.2 --CH.sub.2 --CH.sub.3                         319 2,5-Cl.sub.2 -4-CO--CH(CH.sub.3).sub.2                                     320 2-C(═NOCH.sub.3)--CH.sub.3                                             321 3-C(═NOCH.sub.3)--CH.sub.3                                             322 4-C(═NCCH.sub.3)--CH.sub.3                                             323 2-C(═NOC.sub.2 H.sub.5)--CH.sub.3                                      324 3-C(═NOC.sub.2 H.sub.5)--CH.sub.3                                      325 4-C(═NOC.sub.2 H.sub.5)--CH.sub.3                                      326 2-C(═NO-n-C.sub.3 H.sub.7)--CH.sub.3                                   327 3-C(═NO-n-C.sub.3 H.sub.7)--CH.sub.3                                   328 4-C(═NO-n-C.sub.3 H.sub.7)--CH.sub.3                                   329 2-C(═NO-i-C.sub.3 H.sub.7)--CH.sub.3                                   330 3-C(═NO-i-C.sub.3 H.sub.7)--CH.sub.3                                   331 4-C(═NO-i-C.sub.3 H.sub.7)--CH.sub.3                                   332 2-C(═NO-Allyl)-CH.sub.3                                                333 3-C(═NO-Allyl)-CH.sub.3                                                334 4-C(═NO-Allyl)-CH.sub.3                                                335 2-C(═NO-trans-Chloroallyl)-CH.sub.3                                    336 3-C(═NO-trans-Chloroallyl)-CH.sub.3                                    337 4-C(═NO-trans-Chloroallyl)-CH.sub.3                                    338 2-C(═NO-Propargyl)-CH.sub.3                                            339 3-C(═NO-Propargyl)-CH.sub.3                                            340 4-C(═NO-Propargyl)-CH.sub.3                                            341 2-C(═NO-n-C.sub.4 H.sub.9)--CH.sub.3                                   342 3-C(═NO-n-C.sub.4 H.sub.9)--CH.sub.3                                   343 4-C(═NO-n-C.sub.4 H.sub.9)--CH.sub.3                                   344 2-C(═NO--CH.sub.2 --C.sub.6 H.sub.5)--CH.sub.3                         345 3-C(═NO--CH.sub.2 --C.sub.6 H.sub.5)--CH.sub.3                         346 4-C(═NO--CH.sub.2 --C.sub.6 H.sub.5)--CH.sub.3                         347 2-CH.sub.3 -4-CH═NOCH.sub.3                                            348 2-CH.sub.3 -4-CH═NOC.sub.2 H.sub.5                                     349 2-CH.sub.3 -4-CH═NO-n-C.sub.3 H.sub.7                                  350 2-CH.sub.3 -4-CH═NO-i-C.sub.3 H.sub.7                                  351 2-CH.sub.3 -4-CH═NO-Allyl                                              352 2-CH.sub.3 -4-CH═NO-(trans-Chloroallyl)                                353 2-CH.sub.3 -4-CH═NO-Propargyl                                          354 2-CH.sub.3 -4-CH═NO-n-C.sub.4 H.sub.9                                  355 2-CH.sub.3 -4-CH═NO--CH.sub.2 --C.sub.6 H.sub.5                        356 2-CH.sub.3 -4-(CH.sub.3 --C═NOCH.sub.3)                                357 2-CH.sub.3 -4-(CH.sub.3 --C═NOC.sub.2 H.sub.5)                         358 2-CH.sub.3 -4-(CH.sub.3 --C═NO-n-C.sub.3 H.sub.7)                      359 2-CH.sub.3 -4-(CH.sub.3 --C═NO-i-C.sub.3 H.sub.7)                      360 2-CH.sub.3 -4-(CH.sub.3 --C═NO-Allyl)                                  361 2-CH.sub.3 -4-(CH.sub.3 --C═NO-trans-Chloroallyl)                      362 2-CH.sub.3 -4-(CH.sub.3 --C═NO-Propargyl)                              363 2-CH.sub.3 -4-(CH.sub.3 --C═NO-n-C.sub.4 H.sub.9)                      364 2-CH.sub.3 -4-(CH.sub.3 --C═NO--CH.sub.2 --C.sub.6 H.sub.5)                   365 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C═NO--CH.sub.3)                       366 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C═NO--C.sub.2 H.sub.5)                367 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C═NO-n-C.sub.3 H.sub.7)        368 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C═NO-i-C.sub.3 H.sub.7                       369 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C═NO-Allyl)                    370 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C═NO-trans-Chloroallyl)                      371 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C═NO-Propargyl)                       372 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C═NO-n-C.sub.4 H.sub.9)        373 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C═NO--CH.sub.2 --C.sub.6                    H.sub.5)                                                                 374 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C═NOCH.sub.3)                      375 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C═NOC.sub.2 H.sub.5)                      376 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C═NO-n-C.sub.3                    H.sub.7)                                                                 377 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C═NO-i-C.sub.3 H.sub.7)                   378 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C═NO-Allyl)                 379 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C═NO-trans-Chloroallyl)                   380 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C═NO-Propargyl)                    381 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C═NO-n-C.sub.4                    H.sub.9)                                                                 382 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C═NO--CH.sub.2 --C.sub.6                 H.sub.5)                                                                 383 2-C.sub.6 H.sub.5                                                          384 3-C.sub.6 H.sub.5                                                          385 4-C.sub.6 H.sub.5                                                          386 2-(2'-F--C.sub.6 H.sub.4)                                                  387 2-(3'-F--C.sub.6 H.sub.4)                                                  388 2-(4'-F--C.sub.6 H.sub.4)                                                  389 3-(2'-F--C.sub.6 H.sub.4)                                                  390 3-(3'-F--C.sub.6 H.sub.4)                                                  391 3-(4'-F--C.sub.6 H.sub.4)                                                  392 4-(2'-F--C.sub.6 H.sub.4)                                                  393 4-(3'-F--C.sub.6 H.sub.4)                                                  394 4-(4'-F--C.sub.6 H.sub.4)                                                  395 2-(2'-Cl--C.sub.6 H.sub.4)                                                 396 2-(3'-Cl--C.sub.6 H.sub.4)                                                 397 2-(4'-Cl--C.sub.6 H.sub.4)                                                 398 3-(2'-Cl--C.sub.6 H.sub.4)                                                 399 3-(3'-Cl--C.sub.6 H.sub.4)                                                 400 3-(4'-Cl--C.sub.6 H.sub.4)                                                 401 4-(2'-Cl--C.sub.6 H.sub.4)                                                 402 4-(3'-Cl--C.sub.6 H.sub.4)                                                 403 4-(4'-Cl--C.sub.6 H.sub.4)                                                 405 2-(2'-CH.sub.3 --C.sub.6 H.sub.4)                                          406 2-(3'-CH.sub.3 --C.sub.6 H.sub.4)                                          407 2-(4'-CH.sub.3 --C.sub.6 H.sub.4)                                          408 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)                                          409 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)                                          410 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)                                          411 4-(2'-CH.sub.3 --C.sub.6 H.sub.4)                                          412 4-(3'-CH.sub.3 --C.sub.6 H.sub.4)                                          413 4-(4'-CH.sub.3 --C.sub.6 H.sub.4)                                          414 2-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                      415 2-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                      416 2-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                      417 3-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                      418 3-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                      419 3-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                      420 4-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                      421 4-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                      422 4-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                      423 2-(2'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                       424 2-(3'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                       425 2-(4'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                       426 3-(2'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                       427 3-(3'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                       428 3-(4'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                       429 4-(2'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                       430 4-(3'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                       431 4-(4'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                       432 2-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                                 433 2-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                                 434 2-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                                 435 3-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                                 436 3-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                                 437 3-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                                 438 4-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                                 439 4-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                                 440 4-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                                 441 2-(2'-CH.sub.3 O--C.sub.6 H.sub.4)                                         442 2-(3'-CH.sub.3 O--C.sub.6 H.sub.4)                                         443 2-(4'-CH.sub.3 O--C.sub.6 H.sub.4)                                         444 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)                                         445 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)                                         446 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)                                         447 4-(2'-CH.sub.3 O--C.sub.6 H.sub.4)                                         448 4-(3'-CH.sub.3 O--C.sub.6 H.sub.4)                                         449 4-(4'-CH.sub.3 O--C.sub.6 H.sub.4)                                         450 2-(2'-O.sub.2 N--C.sub.6 H.sub.4)                                          451 2-(3'-O.sub.2 N--C.sub.6 H.sub.4)                                          452 2-(4'-O.sub.2 N--C.sub.6 H.sub.4)                                          453 3-(2'-O.sub.2 N--C.sub.6 H.sub.4)                                          454 3-(3'-O.sub.2 N--C.sub.6 H.sub.4)                                          455 3-(4'-O.sub.2 N--C.sub.6 H.sub.4)                                          456 4-(2'-O.sub.2 N--C.sub.6 H.sub.4)                                          457 4-(3'-O.sub.2 N--C.sub.6 H.sub.4)                                          458 4-(4'-O.sub.2 N--C.sub.6 H.sub.4)                                          459 2-(2'-NC--C.sub.6 H.sub.4)                                                 460 2-(3'-NC--C.sub.6 H.sub.4)                                                 461 2-(4'-NC--C.sub.6 H.sub.4)                                                 462 3-(2'-NC--C.sub.6 H.sub.4)                                                 463 3-(3'-NC--C.sub.6 H.sub.4)                                                 464 3-(4'-NC--C.sub.6 H.sub.4)                                                 465 4-(2'-NC--C.sub.6 H.sub.4)                                                 466 4-(3'-NC--C.sub.6 H.sub.4)                                                 467 4-(4'-NC--C.sub.6 H.sub.4)                                                 468 2-(2'-CF.sub.3 --C.sub.6 H.sub.4)                                          469 2-(3'-CF.sub.3 --C.sub.6 H.sub.4)                                          470 2-(4'-CF.sub.3 --C.sub.6 H.sub.4)                                          471 3-(2'-CF.sub.3 --C.sub.6 H.sub.4)                                          472 3-(3'-CF.sub.3 --C.sub.6 H.sub.4)                                          473 3-(4'-CF.sub.3 --C.sub.6 H.sub.4)                                          474 4-(2'-CF.sub.3 --C.sub.6 H.sub.4)                                          475 4-(3'-CF.sub.3 --C.sub.6 H.sub.4)                                          476 4-(4'-CF.sub.3 --C.sub.6 H.sub.4)                                          477 2-O--C.sub.6 H.sub.5                                                       475 3-O--C.sub.6 H.sub.5                                                       476 4-O--C.sub.6 H.sub.5                                                       478 2-O-(2'-F--C.sub.6 H.sub.4)                                                479 2-O-(3'-F--C.sub.6 H.sub.4)                                                480 2-O-(4'-F--C.sub.6 H.sub.4)                                                481 3-O-(2'-F--C.sub.6 H.sub.4)                                                482 3-O-(3'-F--C.sub.6 H.sub.4)                                                483 3-O-(4'-F--C.sub.6 H.sub.4)                                                484 4-O-(2'-F--C.sub.6 H.sub.4)                                                485 4-O-(3'-F--C.sub.6 H.sub.4)                                                486 4-O-(4'-F--C.sub.6 H.sub.4)                                                487 2-O-(2'-Cl--C.sub.6 H.sub.4)                                               488 2-O-(3'-Cl--C.sub.6 H.sub.4)                                               489 2-O-(4'-Cl--C.sub.6 H.sub.4)                                               490 3-O-(2'-Cl--C.sub.6 H.sub.4)                                               491 3-O-(3'-Cl--C.sub.6 H.sub.4)                                               492 3-O-(4'-Cl--C.sub.6 H.sub.4)                                               493 3-O-(4'-Cl--C.sub.6 H.sub.4)                                               494 4-O-(2'-Cl--C.sub.6 H.sub.4)                                               495 4-O-(3'-Cl--C.sub.6 H.sub.4)                                               496 4-O-(4'-Cl--C.sub.6 H.sub.4)                                               497 2-O-(2'-CH.sub.3 --C.sub.6 H.sub.4)                                        498 2-O-(3'-CH.sub.3 --C.sub.6 H.sub.4)                                        499 2-O-(4'-CH.sub.3 --C.sub.6 H.sub.4)                                        500 3-O-(2'-CH.sub.3 --C.sub.6 H.sub.4)                                        501 3-O-(3'-CH.sub.3 --C.sub.6 H.sub.4)                                        502 3-O-(4'-CH.sub.3 --C.sub.6 H.sub.4)                                        503 4-O-(2'-CH.sub.3 --C.sub.6 H.sub.4)                                        504 4-O-(3'-CH.sub.3 --C.sub.6 H.sub.4)                                        505 4-O-(4'-CH.sub.3 --C.sub.6 H.sub.4)                                        506 2-O-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                    507 2-O-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                    508 2-O-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                    509 3-O-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                    510 3-O-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                    511 3-O-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                    512 4-O-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                    513 4-O-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                    514 4-O-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                    515 2-O-(2'-(CH.sub.3 --C(═NOAllyl))-C.sub.6 H.sub.4)                      516 2-O-(3'-(CH.sub.3 --C(═NOAllyl))-C.sub.6 H.sub.4)                      517 2-O-(4'-(CH.sub.3 --C(═NOAllyl))-C.sub.6 H.sub.4)                      518 3-O-(2'-(CH.sub.3 --C(═NOAllyl))-C.sub.6 H.sub.4)                      519 3-O-(3'-(CH.sub.3 --C(═NOAllyl))-C.sub.6 H.sub.4)                      520 3-O-(4'-(CH.sub.3 --C(═NOAllyl))-C.sub.6 H.sub.4)                      521 4-O-(2'-(CH.sub.3 --C(═NOAllyl))-C.sub.6 H.sub.4)                      522 4-O-(3'-(CH.sub.3 --C(═NOAllyl))-C.sub.6 H.sub.4)                      523 4-O-(4'-(CH.sub.3 --C(═NOAllyl))-C.sub.6 H.sub.4)                      524 2-O-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                               525 2-O-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                               526 2-O-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                               527 3-O-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                               528 3-O-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                               529 3-O-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                               530 4-O-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                               531 4-O-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                               532 4-O-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                               533 2-O-(2'-CH.sub.3 O--C.sub.6 H.sub.4)                                       534 2-O-(3'-CH.sub.3 O--C.sub.6 H.sub.4)                                       535 2-O-(4'-CH.sub.3 O--C.sub.6 H.sub.4)                                       536 3-O-(2'-CH.sub.3 O--C.sub.6 H.sub.4)                                       537 3-O-(3'-CH.sub.3 O--C.sub.6 H.sub.4)                                       538 3-O-(4'-CH.sub.3 O--C.sub.6 H.sub.4)                                       539 4-O-(2'-CH.sub.3 O--C.sub.6 H.sub.4)                                       540 4-O-(3'-CH.sub.3 O--C.sub.6 H.sub.4)                                       541 4-O-(4'-CH.sub.3 O--C.sub.6 H.sub.4)                                       542 2-O-(2'-O.sub.2 N--C.sub.6 H.sub.4)                                        543 2-O-(3'-O.sub.2 N--C.sub.6 H.sub.4)                                        544 2-O-(4'-O.sub.2 N--C.sub.6 H.sub.4)                                        545 3-O-(2'-O.sub.2 N--C.sub.6 H.sub.4)                                        546 3-O-(3'-O.sub.2 N--C.sub.6 H.sub.4)                                        547 3-O-(4'-O.sub.2 N--C.sub.6 H.sub.4)                                        548 4-O-(2'-O.sub.2 N--C.sub.6 H.sub.4)                                        549 4-O-(3'-O.sub.2 N--C.sub.6 H.sub.4)                                        550 4-O-(4'-O.sub.2 N--C.sub.6 H.sub.4)                                        551 2-O-(2'-NC--C.sub.6 H.sub.4)                                               552 2-O-(3'-NC--C.sub.6 H.sub.4)                                               553 2-O-(4'-NC--C.sub.6 H.sub.4)                                               554 3-O-(2'-NC--C.sub.6 H.sub.4)                                               555 3-O-(3'-NC--C.sub.6 H.sub.4)                                               556 3-O-(4'-NC--C.sub.6 H.sub.4)                                               557 4-O-(2'-NC--C.sub.6 H.sub.4)                                               558 4-O-(3'-NC--C.sub.6 H.sub.4)                                               559 4-O-(4'-NC--C.sub.6 H.sub.4)                                               560 2-O-(2'-CF.sub.3 --C.sub.6 H.sub.4)                                        561 2-O-(3'-CF.sub.3 --C.sub.6 H.sub.4)                                        562 2-O-(4'-CF.sub.3 --C.sub.6 H.sub.4)                                        563 3-O-(2'-CF.sub.3 --C.sub.6 H.sub.4)                                        564 3-O-(3'-CF.sub.3 --C.sub.6 H.sub.4)                                        565 3-O-(4'-CF.sub.3 --C.sub.6 H.sub.4)                                        566 4-O-(2'-CF.sub.3 --C.sub.6 H.sub.4)                                        567 4-O-(3'-CF.sub.3 --C.sub.6 H.sub.4)                                        568 4-O-(4'-CF.sub.3 --C.sub.6 H.sub.4)                                        569 2-Pyridinyl-2'                                                             570 2-Pyridinyl-3'                                                             571 2-Pyridinyl-4'                                                             572 3-Pyridinyl-2'                                                             573 3-Pyridinyl-3'                                                             574 3-Pyridinyl-4'                                                             575 4-Pyridinyl-2'                                                             576 4-Pyridinyl-3'                                                             577 4-Pyridinyl-4'                                                             578 2-Pyrimidinyl-2'                                                           579 2-Pyrimidinyl-3'                                                           580 2-Pyrimidinyl-4'                                                           581 3-Pyrimidinyl-2'                                                           582 3-Pyrimidinyl-3'                                                           583 3-Pyrimidinyl-4'                                                           584 4-Pyrimidinyl-2'                                                           585 4-Pyrimidinyl-3'                                                           586 4-Pyrimidinyl-4'                                                           587 2-Pyrazolyl-1'                                                             588 2-Pyrazolyl-3'                                                             589 2-Pyrazolyl-4'                                                             590 3-Pyrazolyl-1'                                                             591 3-Pyrazolyl-3'                                                             592 3-Pyrazolyl-4'                                                             593 4-Pyrazolyl-1'                                                             594 4-Pyrazolyl-3'                                                             595 4-Pyrazolyl-4'                                                             596 2-Isoxazolyl-3'                                                            597 2-Isoxazolyl-4'                                                            598 2-Isoxazolyl-5'                                                            599 3-Isoxazolyl-3'                                                            600 3-Isoxazoiyl-4'                                                            601 3-Isoxazolyl-5'                                                            602 4-Isoxazolyl-3'                                                            603 4-Isoxazolyl-4'                                                            604 4-Isoxazolyl-5'                                                            605 2-Isothiazolyl-3'                                                          606 2-Isothiazolyl-4'                                                          607 2-Isothiazolyl-5'                                                          608 3-Isothiazolyl-3'                                                          609 3-Isothiazolyl-4'                                                          610 3-Isothiazolyl-5'                                                          611 4-Isothiazolyl-3'                                                          612 4-Isothiazolyl-4'                                                          613 4-Isothiazolyl-5'                                                          614 2-Imidazolyl-1'                                                            615 2-Imidazolyl-2'                                                            616 2-Imidazolyl-4'                                                            617 3-Imidazolyl-1'                                                            618 3-Imidazolyl-2'                                                            619 3-Imidazolyl-4'                                                            620 4-Imidazolyl-1'                                                            621 4-Imidazolyl-2                                                             622 4-Imidazolyl-4'                                                            623 2-Oxazolyl-2'                                                              624 2-Oxazolyl-4'                                                              625 2-Oxazolyl-5'                                                              626 3-Oxazolyl-2'                                                              627 3-Oxazolyl-4'                                                              628 3-Oxazolyl-5'                                                              629 4-Oxazolyl-2'                                                              630 4-Oxazolyl-4'                                                              631 4-Oxazolyl-5'                                                              632 2-Thiazolyl-2'                                                             633 2-Thiazolyl-4'                                                             634 2-Thiazolyl-5'                                                             635 3-Thiazolyl-2'                                                             636 3-Thiazolyl-4'                                                             637 3-Thiazolyl-5'                                                             638 4-Thiazolyl-2'                                                             639 4-Thiazolyl-4'                                                             640 4-Thiazolyl-5'                                                             641 2-CH.sub.3 -4-(CH.sub.3 --C═N--O--CH.sub.2 --CH.sub.2 --OCH.sub.             3)                                                                       642 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C═N--O--CH.sub.2 --CH.sub.2                 --OCH.sub.3)                                                             643 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C═N--O--CH.sub.2 --CH.sub.2              --OCH.sub.3)                                                             644 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C═N--OCH.sub.3)                     645 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C═N--OC.sub.2 H.sub.5)                     646 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C═N--O-n-C.sub.3                   H.sub.7)                                                                 647 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C═N--O-i-C.sub.3 H.sub.7)                  648 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C═N--O-Allyl)                       649 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C═N--O-trans-Chloroall             yl)                                                                      650 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C═N--O-Propargyl)                   651 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C═N--O-n-C.sub.4 H.sub.9)                  652 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C═N--O--CH.sub.2                   --C.sub.6 H.sub.5)                                                       653 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C═N--OCH.sub.3)                     654 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C═N--OC.sub.2 H.sub.5)                     655 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C═N--O-n-C.sub.3                   H.sub.7)                                                                 656 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C═N--O-i-C.sub.3 H.sub.7)                  657 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C═N--O-Allyl)                       658 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C═N--O-trans-Chloroall             yl)                                                                      659 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C═N--O-Propargyl)                   660 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C═N--O-n-C.sub.4 H.sub.9)                  661 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C═N--O--CH.sub.2                   --C.sub.6 H.sub.5)                                                       662 2-O-n-C.sub.4 H.sub.9                                                      663 2-O-i-C.sub.4 H.sub.9                                                      664 2-O-s-C.sub.4 H.sub.9                                                      665 2-O-t-C.sub.4 H.sub.9                                                      666 2-Neopentyloxy                                                             667 3-O-n-C.sub.4 H.sub.9                                                      668 3-O-i-C.sub.4 H.sub.9                                                      669 3-O-s-C.sub.4 H.sub.9                                                      670 3-C-t-C.sub.4 H.sub.9                                                      671 3-Neopentyloxy                                                             672 4-O-n-C.sub.4 H.sub.9                                                      673 4-O-i-C.sub.4 H.sub.9                                                      674 4-O-s-C.sub.4 H.sub.9                                                      675 4-O-t-C.sub.4 H.sub.9                                                      676 4-Neopentyloxy                                                             677 3-CH.sub.3 -4-OCH.sub.3                                                    678 3-CH.sub.3 -4-OC.sub.2 H.sub.5                                             679 3-CH.sub.3 -4-O-n-C.sub.3 H.sub.7                                          680 3-CH.sub.3 -4-O-n-C.sub.4 H.sub.9                                          681 3-CH.sub.3 -4-O-i-C.sub.4 H.sub.9                                          682 3-CH.sub.3 -4-O-s-C.sub.4 H.sub.9                                          683 3-CH.sub.3 -4-O-t-C.sub.4 H.sub.9                                          684 3-CH.sub.3 -4-Neopentyloxy                                                 685 2-CH.sub.3 -3-OCH.sub.3                                                    686 2-CH.sub.3 -4-OCH.sub.3                                                    687 2-CH.sub.3 -5-OCH.sub.3                                                    688 2-CH.sub.3 -6-OCH.sub.3                                                    689 3-CH.sub.3 -4-CCH.sub.3                                                    690 3-CH.sub.3 -5-OCH.sub.3                                                    691 3-CH.sub.3 -6-OCH.sub.3                                                    692 4-CH.sub.3 -5-OCH.sub.3                                                    693 4-CH.sub.3 -6-OCH.sub.3                                                    694 4-CH.sub.3 -6-OCH.sub.3                                                    695 2-CH.sub.3 -3-O-i-C.sub.3 H.sub.7                                          696 2-CH.sub.3 -4-O-i-C.sub.3 H.sub.7                                          697 2-CH.sub.3 -5-O-i-C.sub.3 H.sub.7                                          698 2-CH.sub.3 -6-O-i-C.sub.3 H.sub.7                                          699 3-CH.sub.3 -4-O-i-C.sub.3 H.sub.7                                          700 3-CH.sub.3 -5-O-i-C.sub.3 H.sub.7                                          701 3-CH.sub.3 -6-O-i-C.sub.3 H.sub.7                                          702 4-CH.sub.3 -5-O-i-C.sub.3 H.sub.7                                          703 4-CH.sub.3 -6-O-i-C.sub.3 H.sub.7                                          704 5-CH.sub.3 -6-O-i-C.sub.3 H.sub.7                                          705 2-Cl-3-OCH.sub.3                                                           706 2-Cl-4-OCH.sub.3                                                           707 2-Cl-5-OCH.sub.3                                                           708 2-Cl-6-OCH.sub.3                                                           709 3-Cl-4-OCH.sub.3                                                           710 3-Cl-5-OCH.sub.3                                                           711 3-Cl-6-OCH.sub.3                                                           712 4-Cl-5-OCH.sub.3                                                           713 4-Cl-6-OCH.sub.3                                                           714 5-Cl-6-OCH.sub.3                                                         ______________________________________                                    

                  TABLE 33                                                         ______________________________________                                         1  STR253##                                                                      I: R.sup.1 = H, Z = C.sub.2 H.sub.5                                                               IX: R.sup.1 = CH.sub.3, Z = NH(CH.sub.3)                    II: R.sup.1 = CH.sub.3, Z = C.sub.2 H.sub.5 X: R.sup.1 = C.sub.2                                  H.sub.5, Z = NH(CH.sub.3)                                   III: R.sup.1 = C.sub.2 H.sub.5, Z = C.sub.2 H.sub.5 XI: R.sup.1 =                                 Allyl, Z = NH(CH.sub.3)                                     IV: R.sup.1 = Allyl, Z = C.sub.2 H.sub.5 XII: R.sup.1 = Propargyl, Z =                            NH(CH.sub.3)                                                V: R.sup.1 = Propargyl, Z = C.sub.2 H.sub.5 XIII: R.sup.1 = CH.sub.2                              --OCH.sub.3,                                                VI: R.sup.1 = CH.sub.2 --OCH.sub.3, Z = C.sub.2 H.sub.5 Z = NH(CH.sub.3)       VII: R.sup.1 = CO--C.sub.2 H.sub.5, Z = C.sub.2 H.sub.5 XIV: R.sup.1 =                            CO--C.sub.2 H.sub.5, Z = NH(CH.sub.3)                       VIII: R.sup.1 = H, Z = NH(CH.sub.3)                                             -                                                                           No.     X.sub.m                                                                ______________________________________                                          1      H                                                                         2 2-F                                                                          3 3-F                                                                          4 4-F                                                                          5 2,4-F.sub.2                                                                  6 2,4,6-F.sub.3                                                                7 2,3,4,5,6-F.sub.5                                                            8 2,3-F.sub.2                                                                  9 2-Cl                                                                         10 3-Cl                                                                        11 4-Cl                                                                        12 2,3-Cl.sub.2                                                                13 2,4-Cl.sub.2                                                                14 2,5-Cl.sub.2                                                                15 2,6-Cl.sub.2                                                                16 3,4-Cl.sub.2                                                                17 3,5-Cl.sub.2                                                                18 2,3,4-Cl.sub.3                                                              19 2,3,5-Cl.sub.3                                                              20 2,3,6-Cl.sub.3                                                              21 2,4,5-Cl.sub.3                                                              22 2,4,6-Cl.sub.3                                                              23 3,4,5-Cl.sub.3                                                              24 2,3,4,6-Cl.sub.4                                                            25 2,3,5,6-Cl.sub.4                                                            26 2,3,4,5,6-Cl.sub.5                                                          27 2-Br                                                                        28 3-Br                                                                        29 4-Br                                                                        30 2,4-Br.sub.2                                                                31 2,5-Br.sub.2                                                                32 2,6-Br.sub.2                                                                33 2,4,6-Br.sub.3                                                              34 2,3,4,5,6-Br.sub.5                                                          35 2-I                                                                         36 3-I                                                                         37 4-I                                                                         38 2,4-I.sub.2                                                                 39 2-Cl, 3-F                                                                   40 2-Cl, 4-F                                                                   41 2-Cl, 5-F                                                                   42 2-Cl, 6-F                                                                   43 2-Cl, 3-Br                                                                  44 2-Cl, 4-Br                                                                  45 2-Cl, 5-Br                                                                  46 2-Cl, 6-Br                                                                  47 2-Br, 3-Cl                                                                  48 2-Br, 4-Cl                                                                  49 2-Br, 5-Cl                                                                  50 2-Br, 3-F                                                                   51 2-Br, 4-F                                                                   52 2-Br, 5-F                                                                   53 2-Br, 6-F                                                                   54 2-F, 3-Cl                                                                   55 2-F, 4-Cl                                                                   56 2-F, 5-Cl                                                                   57 3-Cl, 4-F                                                                   58 3-Cl, 5-F                                                                   59 3-Cl, 4-Br                                                                  60 3-Cl, 5-Br                                                                  61 3-F, 4-Cl                                                                   62 3-F, 4-Br                                                                   63 3-Br, 4-Cl                                                                  64 3-Br, 4-F                                                                   65 2,6-Cl.sub.2, 4-Br                                                          66 2-CH.sub.3                                                                  67 3-CH.sub.3                                                                  68 4-CH.sub.3                                                                  69 2,3-(CH.sub.3).sub.2                                                        70 2,4-(CH.sub.3).sub.2                                                        71 2,5-(CH.sub.3).sub.2                                                        72 2,6-(CH.sub.3).sub.2                                                        73 3,4-(CH.sub.3).sub.2                                                        74 3,5-(CH.sub.3).sub.2                                                        75 2,3,5-(CH.sub.3).sub.3                                                      76 2,3,4-(CH.sub.3).sub.3                                                      77 2,3,6-(CH.sub.3).sub.3                                                      78 2,4,5-(CH.sub.3).sub.3                                                      79 2,4,6-(CH.sub.3).sub.3                                                      80 3,4,5-(CH.sub.3).sub.3                                                      81 2,3,4,6-(CH.sub.3).sub.4                                                    82 2,3,5,6-(CH.sub.3).sub.4                                                    83 2,3,4,5,6-(CH.sub.3).sub.5                                                  84 2-C.sub.2 H.sub.5                                                           85 3-C.sub.2 H.sub.5                                                           86 4-C.sub.2 H.sub.5                                                           87 2,4-(C.sub.2 H.sub.5).sub.2                                                 88 2,6-(C.sub.2 H.sub.5).sub.2                                                 89 3,5-(C.sub.2 H.sub.5).sub.2                                                 90 2,4,6-(C.sub.2 H.sub.5).sub.3                                               91 2-n-C.sub.3 H.sub.7                                                         92 3-n-C.sub.3 H.sub.7                                                         93 4-n-C.sub.3 H.sub.7                                                         94 2-i-C.sub.3 H.sub.7                                                         95 3-i-C.sub.3 H.sub.7                                                         96 4-i-C.sub.3 H.sub.7                                                         97 2,4-(i-C.sub.3 H.sub.7).sub.2                                               98 2,6-(i-C.sub.3 H.sub.7).sub.2                                               99 3,5-(i-C.sub.3 H.sub.7).sub.2                                              100 2,4,6-(i-C.sub.3 H.sub.7).sub.3                                            101 2-s-C.sub.4 H.sub.9                                                        102 3-s-C.sub.4 H.sub.9                                                        103 4-s-C.sub.4 H.sub.9                                                        104 2-t-C.sub.4 H.sub.9                                                        105 3-t-C.sub.4 H.sub.9                                                        106 4-t-C.sub.4 H.sub.9                                                        107 2,3-(t-C.sub.4 H.sub.9).sub.2                                              108 2,4-(t-C.sub.4 H.sub.9).sub.2                                              109 2,5-(t-C.sub.4 H.sub.9).sub.2                                              110 2,6-(t-C.sub.4 H.sub.9).sub.2                                              111 3,4-(t-C.sub.4 H.sub.9).sub.2                                              112 2,4,6-(t-C.sub.4 H.sub.9).sub.3                                            113 4-n-C.sub.9 H.sub.19                                                       114 4-n-C.sub.12 H.sub.25                                                      115 4-n-C.sub.15 H.sub.31                                                      116 4-(1,1,3,3-Tetramethylbutyl)                                               117 4-(2,4,4-Trimethylpropyl)                                                  118 2-t-C.sub.4 H.sub.9, 4-CH.sub.3                                            119 2-t-C.sub.4 H.sub.9, 5-CH.sub.3                                            120 2,6-(t-C.sub.4 H.sub.9).sub.2, 4-CH.sub.3                                  121 2-CH.sub.3, 4-t-C.sub.4 H.sub.9                                            122 2-CH.sub.3, 6-t-C.sub.4 H.sub.9                                            123 2-CH.sub.3, 4-i-C.sub.3 H.sub.7                                            124 2-CH.sub.3, 5-i-C.sub.3 H.sub.7                                            125 3-CH.sub.3, 4-i-C.sub.3 H.sub.7                                            126 2-i-C.sub.3 H.sub.7, 5-CH.sub.3                                            127 2,4-(t-C.sub.4 H.sub.9).sub.2, 6-i-C.sub.3 H.sub.7                         128 2-Allyl                                                                    129 3-Allyl                                                                    130 4-Allyl                                                                    131 2-Allyl, 6-CH.sub.3                                                        132 2-cyclo-C.sub.6 H.sub.11                                                   133 3-cyclo-C.sub.6 H.sub.11                                                   134 4-cyclo-C.sub.6 H.sub.11                                                   135 2,4-(cyclo-C.sub.6 H.sub.11).sub.2, 6-CH.sub.3                             136 2-CH.sub.3, 4-cyclo-C.sub.6 H.sub.11                                       137 2-CH.sub.2 --C.sub.6 H.sub.5                                               138 3-CH.sub.2 --C.sub.6 H.sub.5                                               139 4-CH.sub.2 --C.sub.6 H.sub.5                                               140 2-CH.sub.2 --C.sub.6 H.sub.5, 4-CH.sub.3                                   141 2-CH.sub.3, 4-CH.sub.2 --C.sub.6 H.sub.5                                   142 2-C.sub.6 H.sub.5                                                          143 3-C.sub.6 H.sub.5                                                          144 4-C.sub.6 H.sub.5                                                          145 4-(2-i-C.sub.3 H.sub.7 --C.sub.6 H.sub.4)                                  146 4-C.sub.6 H.sub.5, 2,6-(CH.sub.3).sub.2                                    147 2-Cl, 4-C.sub.6 H.sub.5                                                    148 2-Br, 4-C.sub.6 H.sub.5                                                    149 2-C.sub.6 H.sub.5, 4-Cl                                                    150 2-C.sub.6 H.sub.5, 4-Br                                                    151 2-CH.sub.2 C.sub.6 H.sub.5, 4-Cl                                           152 2-CH.sub.2 C.sub.6 H.sub.5, 4-Br                                           153 2-Cl, 4-CH.sub.2 C.sub.6 H.sub.5                                           154 2-Br, 4-CH.sub.2 C.sub.6 H.sub.5                                           155 2-cyclo-C.sub.6 H.sub.11, 4-Cl                                             156 2-cyclo-C.sub.6 H.sub.11, 4-Br                                             157 2-Cl, 4-cyclo-C.sub.6 H.sub.11                                             158 2-Br, 4-cyclo-C.sub.6 H.sub.11                                             159 2-OCH.sub.3                                                                160 3-OCH.sub.3                                                                161 4-OCH.sub.3                                                                162 2-OC.sub.2 H.sub.5                                                         163 3-O--C.sub.2 H.sub.5                                                       164 4-O--C.sub.2 H.sub.5                                                       165 2-O-n-C.sub.3 H.sub.7                                                      166 3-O-n-C.sub.3 H.sub.7                                                      167 4-O-n-C.sub.3 H.sub.7                                                      168 2-O-i-C.sub.3 H.sub.7                                                      169 3-O-i-C.sub.3 H.sub.7                                                      170 4-O-i-C.sub.3 H.sub.7                                                      171 2-O-n-C.sub.6 H.sub.13                                                     172 3-O-n-C.sub.6 H.sub.13                                                     173 4-O-n-C.sub.6 H.sub.13                                                     174 2-O-n-C.sub.8 H.sub.17                                                     175 3-O-n-C.sub.8 H.sub.17                                                     176 4-O-n-C.sub.8 H.sub.17                                                     177 2-O--CH.sub.2 C.sub.6 H.sub.5                                              178 3-O--CH.sub.2 C.sub.6 H.sub.5                                              179 4-O--CH.sub.2 C.sub.6 H.sub.5                                              180 2-O--(CH.sub.2).sub.3 C.sub.6 H.sub.5                                      181 3-O--(CH.sub.2).sub.3 C.sub.6 H.sub.5                                      182 4-O--(CH.sub.2).sub.3 C.sub.6 H.sub.5                                      183 2,4-(OCH.sub.3).sub.2                                                      184 2-CF.sub.3                                                                 185 3-CF.sub.3                                                                 186 4-CF.sub.3                                                                 187 2-OCF.sub.3                                                                188 3-OCF.sub.3                                                                189 4-OCF.sub.3                                                                190 3-OCH.sub.2 CHF.sub.2                                                      191 2-NO.sub.2                                                                 192 3-NO.sub.2                                                                 193 4-NO.sub.2                                                                 194 2-CN                                                                       195 3-CN                                                                       196 4-CN                                                                       197 2-CH.sub.3, 3-Cl                                                           198 2-CH.sub.3, 4-Cl                                                           199 2-CH.sub.3, 5-Cl                                                           200 2-CH.sub.3, 6-Cl                                                           201 2-CH.sub.3, 3-F                                                            202 2-CH.sub.3, 4-F                                                            203 2-CH.sub.3, 5-F                                                            204 2-CH.sub.3, 6-F                                                            205 2-CH.sub.3, 3-Br                                                           206 2-CH.sub.3, 4-Br                                                           207 2-CH.sub.3, 5-Br                                                           208 2-CH.sub.3, 6-Br                                                           209 2-Cl, 3-CH.sub.3                                                           210 2-Cl, 4-CH.sub.3                                                           211 2-Cl, 5-CH.sub.3                                                           212 2-F, 3-CH.sub.3                                                            213 2-F, 4-CH.sub.3                                                            214 2-F, 5-CH.sub.3                                                            215 2-Br, 3-CH.sub.3                                                           216 2-Br, 4-CH.sub.3                                                           217 2-Br, 5-CH.sub.3                                                           218 3-CH.sub.3, 4-Cl                                                           219 3-CH.sub.3, 5-Cl                                                           220 3-CH.sub.3, 4-F                                                            221 3-CH.sub.3, 5-F                                                            222 3-CH.sub.3, 4-Br                                                           223 3-CH.sub.3, 5-Br                                                           224 3-F, 4-CH.sub.3                                                            225 3-Cl, 4-CH.sub.3                                                           226 3-Br, 4-CH.sub.3                                                           227 2-Cl, 4,5-(CH.sub.3).sub.2                                                 228 2-Br, 4,5-(CH.sub.3).sub.2                                                 229 2-Cl, 3,5-(CH.sub.3).sub.2                                                 230 2-Br, 3,5-(CH.sub.3).sub.2                                                 231 2,6-Cl.sub.2, 4-CH.sub.3                                                   232 2,6-F.sub.2, 4-CH.sub.3                                                    233 2,6-Br.sub.2, 4-CH.sub.3                                                   234 2,4-Br.sub.2, 6-CH.sub.3                                                   235 2,4-F.sub.2, 6-CH.sub.3                                                    236 2,4-Br.sub.2, 6-CH.sub.3                                                   237 2,6-(CH.sub.3).sub.2, 4-F                                                  238 2,6-(CH.sub.3).sub.2, 4-Cl                                                 239 2,6-(CH.sub.3).sub.2, 4-Br                                                 240 3,5-(CH.sub.3).sub.2, 4-F                                                  241 3,5-(CH.sub.3).sub.2, 4-Cl                                                 242 3,5-(CH.sub.3).sub.2, 4-Br                                                 243 2,3,6-(CH.sub.3).sub.3, 4-F                                                244 2,3,6-(CH.sub.3).sub.3, 4-Cl                                               245 2,3,6-(CH.sub.3).sub.3, 4-Br                                               246 2,4-(CH.sub.3).sub.2, 6-F                                                  247 2,4-(CH.sub.3).sub.2, 6-Cl                                                 248 2,4-(CH.sub.3).sub.2, 6-Br                                                 249 2-i-C.sub.3 H.sub.7, 4-Cl, 5-CH.sub.3                                      250 2-Cl, 4-NO.sub.2                                                           251 2-NO.sub.2, 4-Cl                                                           252 2-OCH.sub.3, 5-NO.sub.2                                                    253 2,4-Cl.sub.2, 5-NO.sub.2                                                   254 2,4-Cl.sub.2, 6-NO.sub.2                                                   255 2,6-Cl.sub.2, 4-NO.sub.2                                                   256 2,6-Br.sub.2, 4-NO.sub.2                                                   257 2,6-I.sub.2, 4-NO.sub.2                                                    258 2-CH.sub.3, 5-i-C.sub.3 H.sub.7, 4-Cl                                      259 2-CO.sub.2 CH.sub.3                                                        260 3-CO.sub.2 CH.sub.3                                                        261 4-CO.sub.2 CH.sub.3                                                        262 2-CO.sub.2 (C.sub.2 H.sub.5)                                               263 3-CO.sub.2 (C.sub.2 H.sub.5)                                               264 4-CO.sub.2 (C.sub.2 H.sub.5)                                               265 2-CO.sub.2 (n-C.sub.3 H.sub.7)                                             266 3-CO.sub.2 (n-C.sub.3 H.sub.7)                                             267 4-CO.sub.2 (n-C.sub.3 H.sub.7)                                             268 2-CO.sub.2 (i-C.sub.3 H.sub.7)                                             269 3-CO.sub.2 (i-C.sub.3 H.sub.7)                                             270 4-CO.sub.2 (i-C.sub.3 H.sub.7)                                             271 2-CO.sub.2 (n-C.sub.6 H.sub.13)                                            272 3-CO.sub.2 (n-C.sub.6 H.sub.13)                                            273 4-CO.sub.2 (n-C.sub.6 H.sub.13)                                            274 2-CH.sub.2 --OCH.sub.3                                                     275 3-CH.sub.2 --OCH.sub.3                                                     276 4-CH.sub.2 --OCH.sub.3                                                     277 2-CH.sub.2 O(C.sub.2 H.sub.5)                                              278 3-CH.sub.2 O(C.sub.2 H.sub.5)                                              279 4-CH.sub.2 O(C.sub.2 H.sub.5)                                              280 2-CH.sub.2 O(n-C.sub.3 H.sub.7)                                            281 3-CH.sub.2 O(n-C.sub.3 H.sub.7)                                            282 4-CH.sub.2 O(n-C.sub.3 H.sub.7)                                            283 2-CH.sub.2 O(i-C.sub.3 H.sub.7)                                            284 3-CH.sub.2 O(i-C.sub.3 H.sub.7)                                            285 4-CH.sub.2 O(i-C.sub.3 H.sub.7)                                            286 2-CHO                                                                      287 3-CHO                                                                      288 4-CHO                                                                      289 2-CO--CH.sub.3                                                             290 3-CO--CH.sub.3                                                             291 4-CO--CH.sub.3                                                             292 2-CO--CH.sub.2 --CH.sub.3                                                  293 3-CO--CH.sub.2 --CH.sub.3                                                  294 4-CO--CH.sub.2 --CH.sub.3                                                  295 2-CO--CH.sub.2 --CH.sub.2 --CH.sub.3                                       296 3-CO--CH.sub.2 --CH.sub.2 --CH.sub.3                                       297 4-CO--CH.sub.2 --CH.sub.2 --CH.sub.3                                       298 2-CO--CH(CH.sub.3)--CH.sub.3                                               299 3-CO--CH(CH.sub.3)--CH.sub.3                                               300 4-CO--CH(CH.sub.3)--CH.sub.3                                               301 2-Me-4-CHO                                                                 302 2-Me-4-CO--CH.sub.3                                                        303 2-Me-4-CO--CH.sub.2 --CH.sub.3                                             304 2-Me-4-CO--CH.sub.2 --CH.sub.2 --CH.sub.3                                  305 2-Me-4-CO--CH(CH.sub.3).sub.2                                              306 2,5-Me.sub.2 -4-CHO                                                        307 2, 5-Me.sub.2 -4-CO--CH.sub.3                                              308 2, 5-Me.sub.2 -4-CO--CH.sub.2 --CH.sub.3                                   309 2, 5-Me.sub.2 -4-CH.sub.2 --CH.sub.2 --CO--CH.sub.3                        310 2, 5-Me.sub.2 -4-CO--CH(CH.sub.3).sub.2                                    311 2-Cl-4-CHO                                                                 312 2-Cl-4-CO--CH.sub.3                                                        313 2-Cl-4-CO--CH.sub.2 --CH.sub.3                                             314 2-Cl-4-CO--CH(CH.sub.3).sub.2                                              315 2,5-Cl.sub.2 -4-CHO                                                        316 2,5-Cl.sub.2 -4-CO--CH.sub.3                                               317 2,5-Cl.sub.2 -4-CO--CH.sub.2 --CH.sub.3                                    318 2,5-Cl.sub.2 -4-CO--CH.sub.2 --CH.sub.2 --CH.sub.3                         319 2,5-Cl.sub.2 -4-CO--CH(CH.sub.3).sub.2                                     320 2-C(═NOCH.sub.3)--CH.sub.3                                             321 3-C(═NOCH.sub.3)--CH.sub.3                                             322 4-C(═NOCH.sub.3)--CH.sub.3                                             323 2-C(═NOC.sub.2 H.sub.5)--CH.sub.3                                      324 3-C(═NOC.sub.2 H.sub.5)--CH.sub.3                                      325 4-C(═NOC.sub.2 H.sub.5)--CH.sub.3                                      326 2-C(═NO-n-C.sub.3 H.sub.7)--CH.sub.3                                   327 3-C(═NO-n-C.sub.3 H.sub.7)--CH.sub.3                                   328 4-C(═NO-n-C.sub.3 H.sub.7)--CH.sub.3                                   329 2-C(═NO-i-C.sub.3 H.sub.7)--CH.sub.3                                   330 3-C(═NO-i-C.sub.3 H.sub.7)--CH.sub.3                                   331 4-C(═NO-i-C.sub.3 H.sub.7)--CH.sub.3                                   332 2-C(═NO-Allyl)--CH.sub.3                                               333 3-C(═NO-Allyl)--CH.sub.3                                               334 4-C(═NO-Allyl)--CH.sub.3                                               335 2-C(═NO-trans-Chloroallyl)--CH.sub.3                                   336 3-C(═NO-trans-Chloroallyl)--CH.sub.3                                   337 4-C(═NO-trans-Chloroallyl)--CH.sub.3                                   338 2-C(═NO-Propargyl)--CH.sub.3                                           339 3-C(═NO-Propargyl)--CH.sub.3                                           340 4-C(═NO-Propargyl)--CH.sub.3                                           341 2-C(═NO-n-C.sub.4 H.sub.9)--CH.sub.3                                   342 3-C(═NO-n-C.sub.4 H.sub.9)--CH.sub.3                                   343 4-C(═NO-n-C.sub.4 H.sub.9)--CH.sub.3                                   344 2-C(═NO--CH.sub.2 --C.sub.6 H.sub.5)--CH.sub.3                         345 3-C(═NO--CH.sub.2 --C.sub.6 H.sub.5)--CH.sub.3                         346 4-C(═NO--CH.sub.2 --C.sub.6 H.sub.5)--CH.sub.3                         347 2-CH.sub.3 -4-CH═NOCH.sub.3                                            348 2-CH.sub.3 -4-CH═NOC.sub.2 H.sub.5                                     349 2-CH.sub.3 -4-CH═NO-n-C.sub.3 H.sub.7                                  350 2-CH.sub.3 -4-CH═NO-i-C.sub.3 H.sub.7                                  351 2-CH.sub.3 -4-CH═NO-Allyl                                              352 2-CH.sub.3 -4-CH═NO-(trans-Chloroallyl)                                353 2-CH.sub.3 -4-CH═NO-Propargyl                                          354 2-CH.sub.3 -4-CH═NO-n-C.sub.4 H.sub.9                                  355 2-CH.sub.3 -4-CH═NO-CH.sub.2 --C.sub.6 H.sub.5                         356 2-CH.sub.3 -4-(CH.sub.3 --C═NOCH.sub.3)                                357 2-CH.sub.3 -4-(CH.sub.3 --C═NOC.sub.2 H.sub.5)                         358 2-CH.sub.3 -4-(CH.sub.3 --C═NO-n-C.sub.3 H.sub.7)                      359 2-CH.sub.3 -4-(CH.sub.3 --C═NO-i-C.sub.3 H.sub.7)                      360 2-CH.sub.3 -4-(CH.sub.3 --C═NO-Allyl)                                  361 2-CH.sub.3 -4-(CH.sub.3 --C═NO-trans-Chloroallyl)                      362 2-CH.sub.3 -4-(CH.sub.3 --C═NO-Propargyl)                              363 2-CH.sub.3 -4-(CH.sub.3 --C═NO-n-C.sub.4 H.sub.9)                      364 2-CH.sub.3 -4-(CH.sub.3 --C═NO--CH.sub.2 --C.sub.6 H.sub.5)                   365 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C═NO--CH.sub.3)                       366 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C═NO--C.sub.2 H.sub.5)                367 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C═NO-n-C.sub.3 H.sub.7)        368 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C═NO-i-C.sub.3 H.sub.7                       369 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C═NO-Allyl)                    370 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C═NO-trans-Chloroallyl)                      371 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C═NO-Propargyl)                       372 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C═NO-n-C.sub.4 H.sub.9)        373 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C═NO--CH.sub.2 --C.sub.6                    H.sub.5)                                                                 374 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C═NOCH.sub.3)                      375 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C═NOC.sub.2 H.sub.5)                      376 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C═NO-n-C.sub.3                    H.sub.7)                                                                 377 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C═NO-i-C.sub.3 H.sub.7)                   378 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C═NO-Allyl)                 379 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C═NO-trans-Chloroallyl)                   380 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C═NO-Proparyl)                     381 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C═NO-n-C.sub.4                    H.sub.9)                                                                 382 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C═NO--CH.sub.2 --C.sub.6                 H.sub.5)                                                                 383 2-C.sub.6 H.sub.5                                                          384 3-C.sub.6 H.sub.5                                                          385 4-C.sub.6 H.sub.5                                                          386 2-(2'-F--C.sub.6 H.sub.4)                                                  387 2-(3'-F--C.sub.6 H.sub.4)                                                  388 2-(4'-F--C.sub.6 H.sub.4)                                                  389 3-(2'-F--C.sub.6 H.sub.4)                                                  390 3-(3'-F--C.sub.6 H.sub.4)                                                  391 3-(4'-F--C.sub.6 H.sub.4)                                                  392 4-(2'-F--C.sub.6 H.sub.4)                                                  393 4-(3'-F--C.sub.6 H.sub.4)                                                  394 4-(4'-F--C.sub.6 H.sub.4)                                                  395 2-(2'-Cl--C.sub.6 H.sub.4)                                                 396 2-(3'-Cl--C.sub.6 H.sub.4)                                                 397 2-(4'-Cl--C.sub.6 H.sub.4)                                                 398 3-(2'-Cl--C.sub.6 H.sub.4)                                                 399 3-(3'-Cl--C.sub.6 H.sub.4)                                                 400 3-(4'-Cl--C.sub.6 H.sub.4)                                                 401 4-(2'-Cl--C.sub.6 H.sub.4)                                                 402 4-(3'-Cl--C.sub.6 H.sub.4)                                                 403 4-(4'-Cl--C.sub.6 H.sub.4)                                                 405 2-(2'-CH.sub.3 --C.sub.6 H.sub.4)                                          406 2-(3'-CH.sub.3 --C.sub.6 H.sub.4)                                          407 2-(4'-CH.sub.3 --C.sub.6 H.sub.4)                                          408 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)                                          409 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)                                          410 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)                                          411 4-(2'-CH.sub.3 --C.sub.6 H.sub.4)                                          412 4-(3'-CH.sub.3 --C.sub.6 H.sub.4)                                          413 4-(4'-CH.sub.3 --C.sub.6 H.sub.4)                                          414 2-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                      415 2-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                      416 2-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                      417 3-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                      418 3-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                      419 3-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                      420 4-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                      421 4-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                      422 4-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                      423 2-(2'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                       424 2-(3'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                       425 2-(4'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                       426 3-(2'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                       427 3-(3'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                       428 3-(4'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                       429 4-(2'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                       430 4-(3'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                       431 4-(4'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                       432 2-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                                 433 2-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                                 434 2-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                                 435 3-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                                 436 3-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                                 437 3-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                                 438 4-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                                 439 4-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                                 440 4-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                                 441 2-(2'-CH.sub.3 O--C.sub.6 H.sub.4)                                         442 2-(3'-CH.sub.3 O--C.sub.6 H.sub.4)                                         443 2-(4'-CH.sub.3 O--C.sub.6 H.sub.4)                                         444 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)                                         445 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)                                         446 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)                                         447 4-(2'-CH.sub.3 O--C.sub.6 H.sub.4)                                         448 4-(3'-CH.sub.3 O--C.sub.6 H.sub.4)                                         449 4-(4'-CH.sub.3 O--C.sub.6 H.sub.4)                                         450 2-(2'-O.sub.2 N--C.sub.6 H.sub.4)                                          451 2-(3'-O.sub.2 N--C.sub.6 H.sub.4)                                          452 2-(4'-O.sub.2 N--C.sub.6 H.sub.4)                                          453 3-(2'-O.sub.2 N--C.sub.6 H.sub.4)                                          454 3-(3'-O.sub.2 N--C.sub.6 H.sub.4)                                          455 3-(4'-O.sub.2 N--C.sub.6 H.sub.4)                                          456 4-(2'-O.sub.2 N--C.sub.6 H.sub.4)                                          457 4-(3'-O.sub.2 N--C.sub.6 H.sub.4)                                          458 4-(4'-O.sub.2 N--C.sub.6 H.sub.4)                                          459 2-(2'-NC--C.sub.6 H.sub.4)                                                 460 2-(3'-NC--C.sub.6 H.sub.4)                                                 461 2-(4'-NC--C.sub.6 H.sub.4)                                                 462 3-(2'-NC--C.sub.6 H.sub.4)                                                 463 3-(3'-NC--C.sub.6 H.sub.4)                                                 464 3-(4'-NC--C.sub.6 H.sub.4)                                                 465 4-(2'-NC--C.sub.6 H.sub.4)                                                 466 4-(3'-NC--C.sub.6 H.sub.4)                                                 467 4-(4'-NC--C.sub.6 H.sub.4)                                                 468 2-(2'-CF.sub.3 --C.sub.6 H.sub.4)                                          469 2-(3'-CF.sub.3 --C.sub.6 H.sub.4)                                          470 2-(4'-CF.sub.3 --C.sub.6 H.sub.4)                                          471 3-(2'-CF.sub.3 --C.sub.6 H.sub.4)                                          472 3-(3'-CF.sub.3 --C.sub.6 H.sub.4)                                          473 3-(4'-CF.sub.3 --C.sub.6 H.sub.4)                                          474 4-(2'-CF.sub.3 --C.sub.6 H.sub.4)                                          475 4-(3'-CF.sub.3 --C.sub.6 H.sub.4)                                          476 4-(4'-CF.sub.3 --C.sub.6 H.sub.4)                                          477 2-O--C.sub.6 H.sub.5                                                       475 3-O--C.sub.6 H.sub.5                                                       476 4-O--C.sub.6 H.sub.5                                                       478 2-O--(2'-F--C.sub.6 H.sub.4)                                               479 2-O--(3'-F--C.sub.6 H.sub.4)                                               480 2-O--(4'-F--C.sub.6 H.sub.4)                                               481 3-O--(2'-F--C.sub.6 H.sub.4)                                               482 3-O--(3'-F--C.sub.6 H.sub.4)                                               483 3-O--(4'-F--C.sub.6 H.sub.4)                                               484 4-O--(2'-F--C.sub.6 H.sub.4)                                               485 4-O--(3'-F--C.sub.6 H.sub.4)                                               486 4-O--(4'-F--C.sub.6 H.sub.4)                                               487 2-O--(2'-Cl--C.sub.6 H.sub.4)                                              488 2-O--(3'-Cl--C.sub.6 H.sub.4)                                              489 2-O--(4'-Cl--C.sub.6 H.sub.4)                                              490 3-O--(2'-Cl--C.sub.6 H.sub.4)                                              491 3-O--(3'-Cl--C.sub.6 H.sub.4)                                              492 3-O--(4'-Cl--C.sub.6 H.sub.4)                                              493 3-O--(4'-Cl--C.sub.6 H.sub.4)                                              494 4-O--(2'-Cl--C.sub.6 H.sub.4)                                              495 4-O--(3'-Cl--C.sub.6 H.sub.4)                                              496 4-O--(4'-Cl--C.sub.6 H.sub.4)                                              497 2-O--(2'-CH.sub.3 --C.sub.6 H.sub.4)                                       498 2-O--(3'-CH.sub.3 --C.sub.6 H.sub.4)                                       499 2-O--(4'-CH.sub.3 --C.sub.6 H.sub.4)                                       500 3-O--(2'-CH.sub.3 --C.sub.6 H.sub.4)                                       501 3-O--(3'-CH.sub.3 --C.sub.6 H.sub.4)                                       502 3-O--(4'-CH.sub.3 --C.sub.6 H.sub.4)                                       503 4-O--(2'-CH.sub.3 --C.sub.6 H.sub.4)                                       504 4-O--(3'-CH.sub.3 --C.sub.6 H.sub.4)                                       505 4-O--(4'-CH.sub.3 --C.sub.6 H.sub.4)                                       506 2-O--(2'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                   507 2-O--(3'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                   508 2-O--(4'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                   509 3-O--(2'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                   510 3-O--(3'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                   511 3-O--(4'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                   512 4-O--(2'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                   513 4-O--(3'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                   514 4-O--(4'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                   515 2-O--(2'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                    516 2-O--(3'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                    517 2-O--(4'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                    518 3-O--(2'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                    519 3-O--(3'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                    520 3-O--(4'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                    521 4-O--(2'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                    522 4-O--(3'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                    523 4-O--(4'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                    524 2-O--(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                              525 2-O--(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                              526 2-O--(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                              527 3-O--(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                              528 3-O--(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                              529 3-O--(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                              530 4-O--(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                              531 4-O--(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                              532 4-O--(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                              533 2-O--(2'-CH.sub.3 O--C.sub.6 H.sub.4)                                      534 2-O--(3'-CH.sub.3 O--C.sub.6 H.sub.4)                                      535 2-O--(4'-CH.sub.3 O--C.sub.6 H.sub.4)                                      536 3-O--(2'-CH.sub.3 O--C.sub.6 H.sub.4)                                      537 3-O--(3'-CH.sub.3 O--C.sub.6 H.sub.4)                                      538 3-O--(4'-CH.sub.3 O--C.sub.6 H.sub.4)                                      539 4-O--(2'-CH.sub.3 O--C.sub.6 H.sub.4)                                      540 4-O--(3'-CH.sub.3 O--C.sub.6 H.sub.4)                                      541 4-O--(4'-CH.sub.3 O--C.sub.6 H.sub.4)                                      542 2-O--(2'-O.sub.2 N--C.sub.6 H.sub.4)                                       543 2-O--(3'-O.sub.2 N--C.sub.6 H.sub.4)                                       544 2-O--(4'-O.sub.2 N--C.sub.6 H.sub.4)                                       545 3-O--(2'-O.sub.2 N--C.sub.6 H.sub.4)                                       546 3-O--(3'-O.sub.2 N--C.sub.6 H.sub.4)                                       547 3-O--(4'-O.sub.2 N--C.sub.6 H.sub.4)                                       548 4-O--(2'-O.sub.2 N--C.sub.6 H.sub.4)                                       549 4-O--(3'-O.sub.2 N--C.sub.6 H.sub.4)                                       550 4-O--(4'-O.sub.2 N--C.sub.6 H.sub.4)                                       551 2-O--(2'-NC--C.sub.6 H.sub.4)                                              552 2-O--(3'-NC--C.sub.6 H.sub.4)                                              553 2-O--(4'-NC--C.sub.6 H.sub.4)                                              554 3-O--(2'-NC--C.sub.6 H.sub.4)                                              555 3-O--(3'-NC--C.sub.6 H.sub.4)                                              556 3-O--(4'-NC--C.sub.6 H.sub.4)                                              557 4-O--(2'-NC--C.sub.6 H.sub.4)                                              558 4-O--(3'-NC--C.sub.6 H.sub.4)                                              559 4-O--(4'-NC--C.sub.6 H.sub.4)                                              560 2-O--(2'-CF.sub.3 --C.sub.6 H.sub.4)                                       561 2-O--(3'-CF.sub.3 --C.sub.6 H.sub.4)                                       562 2-O--(4'-CF.sub.3 --C.sub.6 H.sub.4)                                       563 3-O--(2'-CF.sub.3 --C.sub.6 H.sub.4)                                       564 3-O--(3'-CF.sub.3 --C.sub.6 H.sub.4)                                       565 3-O--(4'-CF.sub.3 --C.sub.6 H.sub.4)                                       566 4-O--(2'-CF.sub.3 --C.sub.6 H.sub.4)                                       567 4-O--(3'-CF.sub.3 --C.sub.6 H.sub.4)                                       568 4-O--(4'-CF.sub.3 --C.sub.6 H.sub.4)                                       569 2-Pyridinyl-2'                                                             570 2-Pyridinyl-3'                                                             571 2-Pyridinyl-4'                                                             572 3-Pyridinyl-2'                                                             573 3-Pyridinyl-3'                                                             574 3-Pyridinyl-4'                                                             575 4-Pyridinyl-2'                                                             576 4-Pyridinyl-3'                                                             577 4-Pyridinyl-4'                                                             578 2-Pyrimidinyl-2'                                                           579 2-Pyrimidinyl-3'                                                           580 2-Pyrimidinyl-4'                                                           581 3-Pyrimidinyl-2'                                                           582 3-Pyrimidinyl-3'                                                           583 3-Pyrimidinyl-4'                                                           584 4-Pyrimidinyl-2'                                                           585 4-Pyrimidinyl-3'                                                           586 4-Pyrimidinyl-4'                                                           587 2-Pyrazolyl-1'                                                             588 2-Pyrazolyl-3'                                                             589 2-Pyrazolyl-4'                                                             590 3-Pyrazolyl-1'                                                             591 3-Pyrazolyl-3'                                                             592 3-Pyrazolyl-4'                                                             593 4-Pyrazolyl-1'                                                             594 4-Pyrazolyl-3'                                                             595 4-Pyrazolyl-4'                                                             596 2-Isoxazolyl-3'                                                            597 2-Isoxazolyl-4'                                                            598 2-Isoxazolyl-5'                                                            599 3-Isoxazolyl-3'                                                            600 3-Isoxazolyl-4'                                                            601 3-Isoxazolyl-5'                                                            602 4-Isoxazolyl-3'                                                            603 4-Isoxazolyl-4'                                                            604 4-Isoxazolyl-5'                                                            605 2-Isothiazolyl-3'                                                          606 2-Isothiazolyl-4'                                                          607 2-Isothiazolyl-5'                                                          608 3-Isothiazolyl-3'                                                          609 3-Isothiazolyl-4'                                                          610 3-Isothiazolyl-5'                                                          611 4-Isothiazolyl-3'                                                          612 4-Isothiazolyl-4'                                                          613 4-Isothiazolyl-5'                                                          614 2-Imidazolyl-1'                                                            615 2-Imidazolyl-2'                                                            616 2-Imidazolyl-4'                                                            617 3-Imidazolyl-1'                                                            618 3-Imidazolyl-2'                                                            619 3-Imidazolyl-4'                                                            620 4-Imidazolyl-1'                                                            621 4-Imidazolyl-2'                                                            622 4-Imidazolyl-4'                                                            623 2-Oxazolyl-2'                                                              624 2-Oxazolyl-4'                                                              625 2-Oxazolyl-5'                                                              626 3-Oxazolyl-2'                                                              627 3-Oxazolyl-4'                                                              628 3-Oxazolyl-5'                                                              629 4-Oxazolyl-2'                                                              630 4-Oxazolyl-4'                                                              631 4-Oxazolyl-5'                                                              632 2-Thiazolyl-2'                                                             633 2-Thiazolyl-4'                                                             634 2-Thiazolyl-5'                                                             635 3-Thiazolyl-2'                                                             636 3-Thiazolyl-4'                                                             637 3-Thiazolyl-5'                                                             638 4-Thiazolyl-2'                                                             639 4-Thiazolyl-4'                                                             640 4-Thiazolyl-5'                                                             641 2-CH.sub.3 -4-(CH.sub.3 --C═N--O--CH.sub.2 --CH.sub.2 --OCH.sub.             3)                                                                       642 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C═N--O--CH.sub.2 --CH.sub.2                 --OCH.sub.3)                                                             643 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C═N--O--CH.sub.2 --CH.sub.2              --OCH.sub.3)                                                             644 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C═N--OCH.sub.3)                     645 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C═N--OC.sub.2 H.sub.5)                     646 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C═N--O-n-C.sub.3                   H.sub.7)                                                                 647 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C═N--O-i-C.sub.3 H.sub.7)                  648 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C═N--O-Allyl)                       649 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C═N--O-trans-Chloroall             yl)                                                                      650 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C═N--O-Propargyl)                   651 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C═N--O-n-C.sub.4 H.sub.9)                  652 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C═N--O--CH.sub.2                   --C.sub.6 H.sub.5)                                                       653 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C═N--OCH.sub.3)                     654 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C═N--OC.sub.2 H.sub.5)                     655 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C═N--O-n-C.sub.3                   H.sub.7)                                                                 656 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C═N--O-i-C.sub.3 H.sub.7)                  657 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C═N--O-Allyl)                       658 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C═N--O-trans-Chloroall             yl)                                                                      659 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C═N--O-Propargyl)                   660 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C═N--O-n-C.sub.4 H.sub.9)                  661 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C═N--O--CH.sub.2                   --C.sub.6 H.sub.5)                                                       662 2-O-n-C.sub.4 H.sub.9                                                      663 2-O-i-C.sub.4 H.sub.9                                                      664 2-O-s-C.sub.4 H.sub.9                                                      665 2-O-t-C.sub.4 H.sub.9                                                      666 2-Neopentyloxy                                                             667 3-O-n-C.sub.4 H.sub.9                                                      668 3-O-i-C.sub.4 H.sub.9                                                      669 3-O-s-C.sub.4 H.sub.9                                                      670 3-O-t-C.sub.4 H.sub.9                                                      671 3-Neopentyloxy                                                             672 4-O-n-C.sub.4 H.sub.9                                                      673 4-O-i-C.sub.4 H.sub.9                                                      674 4-O-s-C.sub.4 H.sub.9                                                      675 4-O-t-C.sub.4 H.sub.9                                                      676 4-Neopentyloxy                                                             677 3-CH.sub.3 -4-OCH.sub.3                                                    678 3-CH.sub.3 -4-OC.sub.2 H.sub.5                                             679 3-CH.sub.3 -4-O-n-C.sub.3 H.sub.7                                          680 3-CH.sub.3 -4-O-n-C.sub.4 H.sub.9                                          681 3-CH.sub.3 -4-O-i-C.sub.4 H.sub.9                                          682 3-CH.sub.3 -4-O-s-C.sub.4 H.sub.9                                          683 3-CH.sub.3 -4-O-t-C.sub.4 H.sub.9                                          684 3-CH.sub.3 -4-Neopentyloxy                                                 685 2-CH.sub.3 -3-OCH.sub.3                                                    686 2-CH.sub.3 -4-OCH.sub.3                                                    687 2-CH.sub.3 -5-OCH.sub.3                                                    688 2-CH.sub.3 -6-OCH.sub.3                                                    689 3-CH.sub.3 -4-OCH.sub.3                                                    690 3-CH.sub.3 -5-OCH.sub.3                                                    691 3-CH.sub.3 -6-OCH.sub.3                                                    692 4-CH.sub.3 -5-O--CH.sub.3                                                  693 4-CH.sub.3 -6-O--CH.sub.3                                                  694 4-CH.sub.3 -6-OCH.sub.3                                                    695 2-CH.sub.3 -3-O-i-C.sub.3 H.sub.7                                          696 2-CH.sub.3 -4-O-i-C.sub.3 H.sub.7                                          697 2-CH.sub.3 -5-O-i-C.sub.3 H.sub.7                                          698 2-CH.sub.3 -6-O-i-C.sub.3 H.sub.7                                          699 3-CH.sub.3 -4-O-i-C.sub.3 H.sub.7                                          700 3-CH.sub.3 -5-O-i-C.sub.3 H.sub.7                                          701 3-CH.sub.3 -6-O-i-C.sub.3 H.sub.7                                          702 4-CH.sub.3 -5-O-i-C.sub.3 H.sub.7                                          703 4-CH.sub.3 -6-O-i-C.sub.3 H.sub.7                                          704 5-CH.sub.3 -6-O-i-C.sub.3 H.sub.7                                          705 2-Cl-3-OCH.sub.3                                                           706 2-Cl-4-OCH.sub.3                                                           707 2-Cl-5-OCH.sub.3                                                           708 2-Cl-6-OCH.sub.3                                                           709 3-Cl-4-OCH.sub.3                                                           710 3-Cl-5-OCH.sub.3                                                           711 3-Cl-6-OCH.sub.3                                                           712 4-Cl-5-OCH.sub.3                                                           713 4-Cl-6-OCH.sub.3                                                           714 5-Cl-6-OCH.sub.3                                                         ______________________________________                                    

                  TABLE 34                                                         ______________________________________                                         1  STR254##                                                                      I: R.sup.1 = H, Z = C.sub.2 H.sub.5                                                              VIII: R.sup.1 = H, Z = NH(CH.sub.3)                          II: R.sup.1 = CH.sub.3, Z = C.sub.2 H.sub.5 IX: R.sup.1 = CH.sub.3, Z =                          NH(CH.sub.3)                                                 III: R.sup.1 = C.sub.2 H.sub.5, Z = C.sub.2 H.sub.5 X: R.sup.1 =                                 C.sub.2 H.sub.5, Z = NH(CH.sub.3)                            IV: R.sup.1 = Allyl, Z = C.sub.2 H.sub.5 XI: R.sup.1 = Allyl, Z =                                NH(CH.sub.3)                                                 V: R.sup.1 = Propargyl, Z = C.sub.2 H.sub.5 XII: R.sup.1 = Propargyl, Z                          = NH(CH.sub.3)                                               VI: R.sup.1 = CH.sub.2 --OCH.sub.3, XIII: R.sup.1 = CH.sub.2 --OCH.sub.3                         , Z = NH(CH.sub.3)                                           Z = C.sub.2 H.sub.5 XIV: R.sup.1 = CO--C.sub.2 H.sub.5, Z = NH(CH.sub.3)       VII: R.sup.1 = CO--C.sub.2 H.sub.5, Z = C.sub.2 H.sub.5                         -                                                                           No.       X.sub.m                                                              ______________________________________                                         1         H                                                                      2 2-F                                                                          3 3-F                                                                          4 4-F                                                                          5 2,4-F.sub.2                                                                  6 2,4,6-F.sub.3                                                                7 2,3,4,5,6-F.sub.5                                                            8 2,3-F.sub.2                                                                  9 2-Cl                                                                         10 3-Cl                                                                        11 4-Cl                                                                        12 2,3-Cl.sub.2                                                                13 2,4-Cl.sub.2                                                                14 2,5-Cl.sub.2                                                                15 2,6-Cl.sub.2                                                                16 3,4-Cl.sub.2                                                                17 3,5-Cl.sub.2                                                                18 2,3,4-Cl.sub.3                                                              19 2,3,5-Cl.sub.3                                                              20 2,3,6-Cl.sub.3                                                              21 2,4,5-Cl.sub.3                                                              22 2,4,6-Cl.sub.3                                                              23 3,4,5-Cl.sub.3                                                              24 2,3,4,6-Cl.sub.4                                                            25 2,3,5,6-Cl.sub.4                                                            26 2,3,4,5,6-Cl.sub.5                                                          27 2-Br                                                                        28 3-Br                                                                        29 4-Br                                                                        30 2,4-Br.sub.2                                                                31 2,5-Br.sub.2                                                                32 2,6-Br.sub.2                                                                33 2,4,6-Br.sub.3                                                              34 2,3,4,5,6-Br.sub.5                                                          35 2-I                                                                         36 3-I                                                                         37 4-I                                                                         38 2,4-I.sub.2                                                                 39 2-Cl, 3-F                                                                   40 2-Cl, 4-F                                                                   41 2-Cl, 5-F                                                                   42 2-Cl, 6-F                                                                   43 2-Cl, 3-Br                                                                  44 2-Cl, 4-Br                                                                  45 2-Cl, 5-Br                                                                  46 2-Cl, 6-Br                                                                  47 2-Br, 3-Cl                                                                  48 2-Br, 4-Cl                                                                  49 2-Br, 5-Cl                                                                  50 2-Br, 3-F                                                                   51 2-Br, 4-F                                                                   52 2-Br, 5-F                                                                   53 2-Br, 6-F                                                                   54 2-F, 3-Cl                                                                   55 2-F, 4-Cl                                                                   56 2-F, 5-Cl                                                                   57 3-Cl, 4-F                                                                   58 3-Cl, 5-F                                                                   59 3-Cl, 4-Br                                                                  60 3-Cl, 5-Br                                                                  61 3-F, 4-Cl                                                                   62 3-F, 4-Br                                                                   63 3-Br, 4-Cl                                                                  64 3-Br, 4-F                                                                   65 2,6-Cl.sub.2, 4-Br                                                          66 2-CH.sub.3                                                                  67 3-CH.sub.3                                                                  68 4-CH.sub.3                                                                  69 2,3-(CH.sub.3).sub.2                                                        70 2,4-(CH.sub.3).sub.2                                                        71 2,5-(CH.sub.3).sub.2                                                        72 2,6-(CH.sub.3).sub.2                                                        73 3,4-(CH.sub.3).sub.2                                                        74 3,5-(CH.sub.3).sub.2                                                        75 2,3,5-(CH.sub.3).sub.3                                                      76 2,3,4-(CH.sub.3).sub.3                                                      77 2,3,6-(CH.sub.3).sub.3                                                      78 2,4,5-(CH.sub.3).sub.3                                                      79 2,4,6-(CH.sub.3).sub.3                                                      80 3,4,5-(CH.sub.3).sub.3                                                      81 2,3,4,6-(CH.sub.3).sub.4                                                    82 2,3,5,6-(CH.sub.3).sub.4                                                    83 2,3,4,5,6-(CH.sub.3).sub.5                                                  84 2-C.sub.2 H.sub.5                                                           85 3-C.sub.2 H.sub.5                                                           86 4-C.sub.2 H.sub.5                                                           87 2,4-(C.sub.2 H.sub.5).sub.2                                                 88 2,6-(C.sub.2 H.sub.5).sub.2                                                 89 3,5-(C.sub.2 H.sub.5).sub.2                                                 90 2,4,6-(C.sub.2 H.sub.5).sub.3                                               91 2-n-C.sub.3 H.sub.7                                                         92 3-n-C.sub.3 H.sub.7                                                         93 4-n-C.sub.3 H.sub.7                                                         94 2-i-C.sub.3 H.sub.7                                                         95 3-i-C.sub.3 H.sub.7                                                         96 4-i-C.sub.3 H.sub.7                                                         97 2,4-(i-C.sub.3 H.sub.7).sub.2                                               98 2,6-(i-C.sub.3 H.sub.7).sub.2                                               99 3,5-(i-C.sub.3 H.sub.7).sub.2                                               100 2,4,6-(i-C.sub.3 H.sub.7).sub.3                                            101 2-s-C.sub.4 H.sub.9                                                        102 3-s-C.sub.4 H.sub.9                                                        103 4-s-C.sub.4 H.sub.9                                                        104 2-t-C.sub.4 H.sub.9                                                        105 3-t-C.sub.4 H.sub.9                                                        106 4-t-C.sub.4 H.sub.9                                                        107 2,3-(t-C.sub.4 H.sub.9).sub.2                                              108 2,4-(t-C.sub.4 H.sub.9).sub.2                                              109 2,5-(t-C.sub.4 H.sub.9).sub.2                                              110 2,6-(t-C.sub.4 H.sub.9).sub.2                                              111 3,4-(t-C.sub.4 H.sub.9).sub.2                                              112 2,4,6-(t-C.sub.4 H.sub.9).sub.3                                            113 4-n-C.sub.9 H.sub.19                                                       114 4-n-C.sub.12 H.sub.25                                                      115 4-n-C.sub.15 H.sub.31                                                      116 4-(1,1,3,3-Tetramethylbutyl)                                               117 4-(2,4,4-Trimethylpropyl)                                                  118 2-t-C.sub.4 H.sub.9, 4-CH.sub.3                                            119 2-t-C.sub.4 H.sub.9, 5-CH.sub.3                                            120 2,6-(t-C.sub.4 H.sub.9).sub.2, 4-CH.sub.3                                  121 2-CH.sub.3, 4-t-C.sub.4 H.sub.9                                            122 2-CH.sub.3, 6-t-C.sub.4 H.sub.9                                            123 2-CH.sub.3, 4-i-C.sub.3 H.sub.7                                            124 2-CH.sub.3, 5-i-C.sub.3 H.sub.7                                            125 3-CH.sub.3, 4-i-C.sub.3 H.sub.7                                            126 2-i-C.sub.3 H.sub.7, 5-CH.sub.3                                            127 2,4-(t-C.sub.4 H.sub.9).sub.2, 6-i-C.sub.3 H.sub.7                         128 2-Allyl                                                                    129 3-Allyl                                                                    130 4-Allyl                                                                    131 2-Allyl, 6-CH.sub.3                                                        132 2-cyclo-C.sub.6 H.sub.11                                                   133 3-cyclo-C.sub.6 H.sub.11                                                   134 4-cyclo-C.sub.6 H.sub.11                                                   135 2,4-(cyclo-C.sub.6 H.sub.11).sub.2, 6-CH.sub.3                             136 2-CH.sub.3, 4-cyclo-C.sub.6 H.sub.11                                       137 2-CH.sub.2 --C.sub.6 H.sub.5                                               138 3-CH.sub.2 --C.sub.6 H.sub.5                                               139 4-CH.sub.2 --C.sub.6 H.sub.5                                               140 2-CH.sub.2 --C.sub.6 H.sub.5, 4-CH.sub.3                                   141 2-CH.sub.3, 4-CH.sub.2 --C.sub.6 H.sub.5                                   142 2-C.sub.6 H.sub.5                                                          143 3-C.sub.6 H.sub.5                                                          144 4-C.sub.6 H.sub.5                                                          145 4-(2-i-C.sub.3 H.sub.7 --C.sub.6 H.sub.4)                                  146 4-C.sub.6 H.sub.5, 2,6-(CH.sub.3).sub.2                                    147 2-Cl, 4-C.sub.6 H.sub.5                                                    148 2-Br, 4-C.sub.6 H.sub.5                                                    149 2-C.sub.6 H.sub.5, 4-Cl                                                    150 2-C.sub.6 H.sub.5, 4-Br                                                    151 2-CH.sub.2 C.sub.6 H.sub.5, 4-Cl                                           152 2-CH.sub.2 C.sub.6 H.sub.5, 4-Br                                           153 2-Cl, 4-CH.sub.2 C.sub.6 H.sub.5                                           154 2-Br, 4-CH.sub.2 C.sub.6 H.sub.5                                           155 2-cyclo-C.sub.6 H.sub.11, 4-Cl                                             156 2-cyclo-C.sub.6 H.sub.11, 4-Br                                             157 2-Cl, 4-cyclo-C.sub.6 H.sub.11                                             158 2-Br, 4-cyclo-C.sub.6 H.sub.11                                             159 2-OCH.sub.3                                                                160 3-OCH.sub.3                                                                161 4-OCH.sub.3                                                                162 2-OC.sub.2 H.sub.5                                                         163 3-O--C.sub.2 H.sub.5                                                       164 4-O--C.sub.2 H.sub.5                                                       165 2-O-n-C.sub.3 H.sub.7                                                      166 3-O-n-C.sub.3 H.sub.7                                                      167 4-O-n-C.sub.3 H.sub.7                                                      168 2-O-i-C.sub.3 H.sub.7                                                      169 3-O-i-C.sub.3 H.sub.7                                                      170 4-O-i-C.sub.3 H.sub.7                                                      171 2-O-n-C.sub.6 H.sub.13                                                     172 3-O-n-C.sub.6 H.sub.13                                                     173 4-O-n-C.sub.6 H.sub.13                                                     174 2-O-n-C.sub.8 H.sub.17                                                     175 3-O-n-C.sub.8 H.sub.17                                                     176 4-O-n-C.sub.8 H.sub.17                                                     177 2-O--CH.sub.2 C.sub.6 H.sub.5                                              178 3-O--CH.sub.2 C.sub.6 H.sub.5                                              179 4-O--CH.sub.2 C.sub.6 H.sub.5                                              180 2-O--(CH.sub.2).sub.3 C.sub.6 H.sub.5                                      181 3-O--(CH.sub.2).sub.3 C.sub.6 H.sub.5                                      182 4-O--(CH.sub.2).sub.3 C.sub.6 H.sub.5                                      183 2,4-(OCH.sub.3).sub.2                                                      184 2-CF.sub.3                                                                 185 3-CF.sub.3                                                                 186 4-CF.sub.3                                                                 187 2-OCF.sub.3                                                                188 3-OCF.sub.3                                                                189 4-OCF.sub.3                                                                190 3-OCH.sub.2 CHF.sub.2                                                      191 2-NO.sub.2                                                                 192 3-NO.sub.2                                                                 193 4-NO.sub.2                                                                 194 2-CN                                                                       195 3-CN                                                                       196 4-CN                                                                       197 2-CH.sub.3, 3-Cl                                                           198 2-CH.sub.3, 4-Cl                                                           199 2-CH.sub.3, 5-Cl                                                           200 2-CH.sub.3, 6-Cl                                                           201 2-CH.sub.3, 3-F                                                            202 2-CH.sub.3, 4-F                                                            203 2-CH.sub.3, 5-F                                                            204 2-CH.sub.3, 6-F                                                            205 2-CH.sub.3, 3-Br                                                           206 2-CH.sub.3, 4-Br                                                           207 2-CH.sub.3, 5-Br                                                           208 2-CH.sub.3, 6-Br                                                           209 2-Cl, 3-CH.sub.3                                                           210 2-Cl, 4-CH.sub.3                                                           211 2-Cl, 5-CH.sub.3                                                           212 2-F, 3-CH.sub.3                                                            213 2-F, 4-CH.sub.3                                                            214 2-F, 5-CH.sub.3                                                            215 2-Br, 3-CH.sub.3                                                           216 2-Br, 4-CH.sub.3                                                           217 2-Br, 5-CH.sub.3                                                           218 3-CH.sub.3, 4-Cl                                                           219 3-CH.sub.3, 5-Cl                                                           220 3-CH.sub.3, 4-F                                                            221 3-CH.sub.3, 5-F                                                            222 3-CH.sub.3, 4-Br                                                           223 3-CH.sub.3, 5-Br                                                           224 3-F, 4-CH.sub.3                                                            225 3-Cl, 4-CH.sub.3                                                           226 3-Br, 4-CH.sub.3                                                           227 2-Cl, 4,5-(CH.sub.3).sub.2                                                 228 2-Br, 4,5-(CH.sub.3).sub.2                                                 229 2-Cl, 3,5-(CH.sub.3).sub.2                                                 230 2-Br, 3,5-(CH.sub.3).sub.2                                                 231 2,6-Cl.sub.2, 4-CH.sub.3                                                   232 2,6-F.sub.2, 4-CH.sub.3                                                    233 2,6-Br.sub.2, 4-CH.sub.3                                                   234 2,4-Br.sub.2, 6-CH.sub.3                                                   235 2,4-F.sub.2, 6-CH.sub.3                                                    236 2,4-Br.sub.2, 6-CH.sub.3                                                   237 2,6-(CH.sub.3).sub.2, 4-F                                                  238 2,6-(CH.sub.3).sub.2, 4-Cl                                                 239 2,6-(CH.sub.3).sub.2, 4-Br                                                 240 3,5-(CH.sub.3).sub.2, 4-F                                                  241 3,5-(CH.sub.3).sub.2, 4-Cl                                                 242 3,5-(CH.sub.3).sub.2, 4-Br                                                 243 2,3,6-(CH.sub.3).sub.3, 4-F                                                244 2,3,6-(CH.sub.3).sub.3, 4-Cl                                               245 2,3,6-(CH.sub.3).sub.3, 4-Br                                               246 2,4-(CH.sub.3).sub.2, 6-F                                                  247 2,4-(CH.sub.3).sub.2, 6-Cl                                                 248 2,4-(CH.sub.3).sub.2, 6-Br                                                 249 2-i-C.sub.3 H.sub.7, 4-Cl, 5-CH.sub.3                                      250 2-Cl, 4-NO.sub.2                                                           251 2-NO.sub.2, 4-Cl                                                           252 2-OCH.sub.3, 5-NO.sub.2                                                    253 2,4-Cl.sub.2, 5-NO.sub.2                                                   254 2,4-Cl.sub.2, 6-NO.sub.2                                                   255 2,6-Cl.sub.2, 4-NO.sub.2                                                   256 2,6-Br.sub.2, 4-NO.sub.2                                                   257 2,6-I.sub.2, 4-NO.sub.2                                                    258 2-CH.sub.3, 5-i-C.sub.3 H.sub.7, 4-Cl                                      259 2-CO.sub.2 CH.sub.3                                                        260 3-CO.sub.2 CH.sub.3                                                        261 4-CO.sub.2 CH.sub.3                                                        262 2-CO.sub.2 (C.sub.2 H.sub.5)                                               263 3-CO.sub.2 (C.sub.2 H.sub.5)                                               264 4-CO.sub.2 (C.sub.2 H.sub.5)                                               265 2-CO.sub.2 (n-C.sub.3 H.sub.7)                                             266 3-CO.sub.2 (n-C.sub.3 H.sub.7)                                             267 4-CO.sub.2 (n-C.sub.3 H.sub.7)                                             268 2-CO.sub.2 (i-C.sub.3 H.sub.7)                                             269 3-CO.sub.2 (i-C.sub.3 H.sub.7)                                             270 4-CO.sub.2 (i-C.sub.3 H.sub.7)                                             271 2-CO.sub.2 (n-C.sub.6 H.sub.13)                                            272 3-CO.sub.2 (n-C.sub.6 H.sub.13)                                            273 4-CO.sub.2 (n-C.sub.6 H.sub.13)                                            274 2-CH.sub.2 --OCH.sub.3                                                     275 3-CH.sub.2 --OCH.sub.3                                                     276 4-CH.sub.2 --OCH.sub.3                                                     277 2-CH.sub.2 O(C.sub.2 H.sub.5)                                              278 3-CH.sub.2 O(C.sub.2 H.sub.5)                                              279 4-CH.sub.2 O(C.sub.2 H.sub.5)                                              280 2-CH.sub.2 O(n-C.sub.3 H.sub.7)                                            281 3-CH.sub.2 O(n-C.sub.3 H.sub.7)                                            282 4-CH.sub.2 O(n-C.sub.3 H.sub.7)                                            283 2-CH.sub.2 O(i-C.sub.3 H.sub.7)                                            284 3-CH.sub.2 O(i-C.sub.3 H.sub.7)                                            285 4-CH.sub.2 O(i-C.sub.3 H.sub.7)                                            286 2-CHO                                                                      287 3-CHO                                                                      288 4-CHO                                                                      289 2-CO--CH.sub.3                                                             290 3-CO--CH.sub.3                                                             291 4-CO--CH.sub.3                                                             292 2-CO--CH.sub.2 --CH.sub.3                                                  293 3-CO--CH.sub.2 --CH.sub.3                                                  294 4-CO--CH.sub.2 --CH.sub.3                                                  295 2-CO--CH.sub.2 --CH.sub.2 --CH.sub.3                                       296 3-CO--CH.sub.2 --CH.sub.2 --CH.sub.3                                       297 4-CO--CH.sub.2 --CH.sub.2 --CH.sub.3                                       298 2-CO--CH(CH.sub.3)--CH.sub.3                                               299 3-CO--CH(CH.sub.3)--CH.sub.3                                               300 4-CO--CH(CH.sub.3)--CH.sub.3                                               301 2-Me-4-CHO                                                                 302 2-Me-4-CO--CH.sub.3                                                        303 2-Me-4-CO--CH.sub.2 --CH.sub.3                                             304 2-Me-4-CO--CH.sub.2 --CH.sub.2 --CH.sub.3                                  305 2-Me-4-CO--CH(CH.sub.3).sub.2                                              306 2,5-Me.sub.2 -4-CHO                                                        307 2,5-Me.sub.2 -4-CO--CH.sub.3                                               308 2,5-Me.sub.2 -4-CO--CH.sub.2 --CH.sub.3                                    309 2,5-Me.sub.2 -4-CH.sub.2 --CH.sub.2 --CO--CH.sub.3                         310 2,5-Me.sub.2 -4-CO--CH(CH.sub.3).sub.2                                     311 2-Cl-4-CHO                                                                 312 2-Cl-4-CO--CH.sub.3                                                        313 2-Cl-4-CO--CH.sub.2 --CH.sub.3                                             314 2-Cl-4-CO--CH(CH.sub.3).sub.2                                              315 2,5-Cl.sub.2 -4-CHO                                                        316 2,5-Cl.sub.2 -4-CO--CH.sub.3                                               317 2,5-Cl.sub.2 -4-CO--CH.sub.2 --CH.sub.3                                    318 2,5-Cl.sub.2 -4-CO--CH.sub.2 --CH.sub.2 --CH.sub.3                         319 2,5-Cl.sub.2 -4-CO--CH(CH.sub.3).sub.2                                     320 2-C(═NOCH.sub.3)--CH.sub.3                                             321 3-C(═NOCH.sub.3)--CH.sub.3                                             322 4-C(═NOCH.sub.3)--CH.sub.3                                             323 2-C(═NOC.sub.2 H.sub.5)--CH.sub.3                                      324 3-C(═NOC.sub.2 H.sub.5)--CH.sub.3                                      325 4-C(═NOC.sub.2 H.sub.5)--CH.sub.3                                      326 2-C(═NO-n-C.sub.3 H.sub.7)--CH.sub.3                                   327 3-C(═NO-n-C.sub.3 H.sub.7)--CH.sub.3                                   328 4-C(═NO-n-C.sub.3 H.sub.7)--CH.sub.3                                   329 2-C(═NO-i-C.sub.3 H.sub.7)--CH.sub.3                                   330 3-C(═NO-i-C.sub.3 H.sub.7)--CH.sub.3                                   331 4-C(═NO-i-C.sub.3 H.sub.7)--CH.sub.3                                   332 2-C(═NO-Allyl)--CH.sub.3                                               333 3-C(═NO-Allyl)--CH.sub.3                                               334 4-C(═NO-Allyl)--CH.sub.3                                               335 2-C(═NO-trans-Chloroallyl)--CH.sub.3                                   336 3-C(═NO-trans-Chloroallyl)--CH.sub.3                                   337 4-C(═NO-trans-Chloroallyl)--CH.sub.3                                   338 2-C(═NO-Propargyl)--CH.sub.3                                           339 3-C(═NO-Propargyl)--CH.sub.3                                           340 4-C(═NO-Propargyl)--CH.sub.3                                           341 2-C(═NO-n-C.sub.4 H.sub.9)--CH.sub.3                                   342 3-C(═NO-n-C.sub.4 H.sub.9)--CH.sub.3                                   343 4-C(═NO-n-C.sub.4 H.sub.9)--CH.sub.3                                   344 2-C(═NO--CH.sub.2 --C.sub.6 H.sub.5)--CH.sub.3                         345 3-C(═NO--CH.sub.2 --C.sub.6 H.sub.5)--CH.sub.3                         346 4-C(═NO--CH.sub.2 --C.sub.6 H.sub.5)--CH.sub.3                         347 2-CH.sub.3 -4-CH═NOCH.sub.3                                            348 2-CH.sub.3 -4-CH═NOC.sub.2 H.sub.5                                     349 2-CH.sub.3 -4-CH═NO-n-C.sub.3 H.sub.7                                  350 2-CH.sub.3 -4-CH═NO-i-C.sub.3 H.sub.7                                  351 2-CH.sub.3 -4-CH═NO-Allyl                                              352 2-CH.sub.3 -4-CH═NO-(trans-Chloroallyl)                                353 2-CH.sub.3 -4-CH═NO-Propargyl                                          354 2-CH.sub.3 -4-CH═NO-n-C.sub.4 H.sub.9                                  355 2-CH.sub.3 -4-CH═NO--CH.sub.2 --C.sub.6 H.sub.5                        356 2-CH.sub.3 -4-(CH.sub.3 --C═NOCH.sub.3)                                357 2-CH.sub.3 -4-(CH.sub.3 --C═NOC.sub.2 H.sub.5)                         358 2-CH.sub.3 -4-(CH.sub.3 --C═NO-n-C.sub.3 H.sub.7)                      359 2-CH.sub.3 -4-(CH.sub.3 --C═NO-i-C.sub.3 H.sub.7)                      360 2-CH.sub.3 -4-(CH.sub.3 --C═NO-Allyl)                                  361 2-CH.sub.3 -4-(CH.sub.3 --C═NO-trans-Chloroallyl)                      362 2-CH.sub.3 -4-(CH.sub.3 --C═NO-Propargyl)                              363 2-CH.sub.3 -4-(CH.sub.3 --C═NO-n-C.sub.4 H.sub.9)                      364 2-CH.sub.3 -4-(CH.sub.3 --C═NO--CH.sub.2 --C.sub.6 H.sub.5)                     365 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C═NO--CH.sub.3)                       366 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C═NO--C.sub.2                        H.sub.5)                                                               367 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C═NO-n-C.sub.3 H.sub.7)                        368 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C═NO-i-C.sub.3                       H.sub.7)                                                               369 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C═NO-Allyl)                           370 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C═NO-trans-Chloroallyl)                        371 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C═NO-Propargyl)                       372 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C═NO-n-C.sub.4                       H.sub.9)                                                               373 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C═NO--CH.sub.2 --C.sub.6                      H.sub.5)                                                               374 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C═NOCH.sub.3)                      375 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C═NOC.sub.2 H.sub.5)                        376 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C═NO-n-C.sub.3                    H.sub.7)                                                               377 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C═NO-i-C.sub.3 H.sub.7)                     378 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C═NO-Allyl)                        379 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C═NO-trans-Chloroal               lyl)                                                                   380 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C═NO-Proparyl)                     381 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C═NO-n-C.sub.4 H.sub.9)                     382 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C═NO--CH.sub.2                    --C.sub.6 H.sub.5)                                                     383 2-C.sub.6 H.sub.5                                                          384 3-C.sub.6 H.sub.5                                                          385 4-C.sub.6 H.sub.5                                                          386 2-(2'-F--C.sub.6 H.sub.4)                                                  387 2-(3'-F--C.sub.6 H.sub.4)                                                  388 2-(4'-F--C.sub.6 H.sub.4)                                                  389 3-(2'-F--C.sub.6 H.sub.4)                                                  390 3-(3'-F--C.sub.6 H.sub.4)                                                  391 3-(4'-F--C.sub.6 H.sub.4)                                                  392 4-(2'-F--C.sub.6 H.sub.4)                                                  393 4-(3'-F--C.sub.6 H.sub.4)                                                  394 4-(4'-F--C.sub.6 H.sub.4)                                                  395 2-(2'-Cl--C.sub.6 H.sub.4)                                                 396 2-(3'-Cl--C.sub.6 H.sub.4)                                                 397 2-(4'-Cl--C.sub.6 H.sub.4)                                                 398 3-(2'-Cl--C.sub.6 H.sub.4)                                                 399 3-(3'-Cl--C.sub.6 H.sub.4)                                                 400 3-(4'-Cl--C.sub.6 H.sub.4)                                                 401 4-(2'-Cl--C.sub.6 H.sub.4)                                                 402 4-(3'-Cl--C.sub.6 H.sub.4)                                                 403 4-(4'-Cl--C.sub.6 H.sub.4)                                                 405 2-(2'-CH.sub.3 --C.sub.6 H.sub.4)                                          406 2-(3'-CH.sub.3 --C.sub.6 H.sub.4)                                          407 2-(4'-CH.sub.3 --C.sub.6 H.sub.4)                                          408 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)                                          409 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)                                          410 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)                                          411 4-(2'-CH.sub.3 --C.sub.6 H.sub.4)                                          412 4-(3'-CH.sub.3 --C.sub.6 H.sub.4)                                          413 4-(4'-CH.sub.3 --C.sub.6 H.sub.4)                                          414 2-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                      415 2-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                      416 2-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                      417 3-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                      418 3-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                      419 3-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                      420 4-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                      421 4-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                      422 4-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                      423 2-(2'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                       424 2-(3'-(CH.sub.3 --C(═NOAllyl))--C6H.sub.4)                             425 2-(4'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                       426 3-(2'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                       427 3-(3'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                       428 3-(4'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                       429 4-(2'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                       430 4-(3'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                       431 4-(4'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                       432 2-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                                 433 2-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                                 434 2-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                                 435 3-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                                 436 3-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                                 437 3-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                                 438 4-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                                 439 4-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                                 440 4-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                                 441 2-(2'-CH.sub.3 O--C.sub.6 H.sub.4)                                         442 2-(3'-CH.sub.3 O--C.sub.6 H.sub.4)                                         443 2-(4'-CH.sub.3 O--C.sub.6 H.sub.4)                                         444 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)                                         445 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)                                         446 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)                                         447 4-(2'-CH.sub.3 O--C.sub.6 H.sub.4)                                         448 4-(3'-CH.sub.3 O--C.sub.6 H.sub.4)                                         449 4-(4'-CH.sub.3 O--C.sub.6 H.sub.4)                                         450 2-(2'-O.sub.2 N--C.sub.6 H.sub.4)                                          451 2-(3'-O.sub.2 N--C.sub.6 H.sub.4)                                          452 2-(4'-O.sub.2 N--C.sub.6 H.sub.4)                                          453 3-(2'-O.sub.2 N--C.sub.6 H.sub.4)                                          454 3-(3'-O.sub.2 N--C.sub.6 H.sub.4)                                          455 3-(4'-O.sub.2 N--C.sub.6 H.sub.4)                                          456 4-(2'-O.sub.2 N--C.sub.6 H.sub.4)                                          457 4-(3'-O.sub.2 N--C.sub.6 H.sub.4)                                          458 4-(4'-O.sub.2 N--C.sub.6 H.sub.4)                                          459 2-(2'-NC--C.sub.6 H.sub.4)                                                 460 2-(3'-NC--C.sub.6 H.sub.4)                                                 461 2-(4'-NC--C.sub.6 H.sub.4)                                                 462 3-(2'-NC--C.sub.6 H.sub.4)                                                 463 3-(3'-NC--C.sub.6 H.sub.4)                                                 464 3-(4'-NC--C.sub.6 H.sub.4)                                                 465 4-(2'-NC--C.sub.6 H.sub.4)                                                 466 4-(3'-NC--C.sub.6 H.sub.4)                                                 467 4-(4'-NC--C.sub.6 H.sub.4)                                                 468 2-(2'-CF.sub.3 --C.sub.6 H.sub.4)                                          469 2-(3'-CF.sub.3 --C.sub.6 H.sub.4)                                          470 2-(4'-CF.sub.3 --C.sub.6 H.sub.4)                                          471 3-(2'-CF.sub.3 --C.sub.6 H.sub.4)                                          472 3-(3'-CF.sub.3 --C.sub.6 H.sub.4)                                          473 3-(4'-CF.sub.3 --C.sub.6 H.sub.4)                                          474 4-(2'-CF.sub.3 --C.sub.6 H.sub.4)                                          475 4-(3'-CF.sub.3 --C.sub.6 H.sub.4)                                          476 4-(4'-CF.sub.3 --C.sub.6 H.sub.4)                                          477 2-O--C.sub.6 H.sub.5                                                       475 3-O--C.sub.6 H.sub.5                                                       476 4-O--C.sub.6 H.sub.5                                                       478 2-O-(2'-F--C.sub.6 H.sub.4)                                                479 2-O-(3'-F--C.sub.6 H.sub.4)                                                480 2-O-(4'-F--C.sub.6 H.sub.4)                                                481 3-O-(2'-F--C.sub.6 H.sub.4)                                                482 3-O-(3'-F--C.sub.6 H.sub.4)                                                483 3-O-(4'-F--C.sub.6 H.sub.4)                                                484 4-O-(2'-F--C.sub.6 H.sub.4)                                                485 4-O-(3'-F--C.sub.6 H.sub.4)                                                486 4-O-(4'-F--C.sub.6 H.sub.4)                                                487 2-O-(2'-Cl--C.sub.6 H.sub.4)                                               488 2-O-(3'-Cl--C.sub.6 H.sub.4)                                               489 2-O-(4'-Cl--C.sub.6 H.sub.4)                                               490 3-O-(2'-Cl--C.sub.6 H.sub.4)                                               491 3-O-(3'-Cl--C.sub.6 H.sub.4)                                               492 3-O-(4'-Cl--C.sub.6 H.sub.4)                                               493 3-O-(4'-Cl--C.sub.6 H.sub.4)                                               494 4-O-(2'-Cl--C.sub.6 H.sub.4)                                               495 4-O-(3'-Cl--C.sub.6 H.sub.4)                                               496 4-O-(4'-Cl--C.sub.6 H.sub.4)                                               497 2-O-(2'-CH.sub.3 --C.sub.6 H.sub.4)                                        498 2-O-(3'-CH.sub.3 --C.sub.6 H.sub.4)                                        499 2-O-(4'-CH.sub.3 --C.sub.6 H.sub.4)                                        500 3-O-(2'-CH.sub.3 --C.sub.6 H.sub.4)                                        501 3-O-(3'-CH.sub.3 --C.sub.6 H.sub.4)                                        502 3-O-(4'-CH.sub.3 --C.sub.6 H.sub.4)                                        503 4-O-(2'-CH.sub.3 --C.sub.6 H.sub.4)                                        504 4-O-(3'-CH.sub.3 --C.sub.6 H.sub.4)                                        505 4-O-(4'-CH.sub.3 --C.sub.6 H.sub.4)                                        506 2-O-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                    507 2-O-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                    508 2-O-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                    509 3-O-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                    510 3-O-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                    511 3-O-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                    512 4-O-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                    513 4-O-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                    514 4-O-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                    515 2-O-(2'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                     516 2-O-(3'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                     517 2-O-(4'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                     518 3-O-(2'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                     519 3-O-(3'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                     520 3-O-(4'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                     521 4-O-(2'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                     522 4-O-(3'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                     523 4-O-(4'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                     524 2-O-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                               525 2-O-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                               526 2-O-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                               527 3-O-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                               528 3-O-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                               529 3-O-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                               530 4-O-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                               531 4-O-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                               532 4-O-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                               533 2-O-(2'-CH.sub.3 O--C.sub.6 H.sub.4)                                       534 2-O-(3'-CH.sub.3 O--C.sub.6 H.sub.4)                                       535 2-O-(4'-CH.sub.3 O--C.sub.6 H.sub.4)                                       536 3-O-(2'-CH.sub.3 O--C.sub.6 H.sub.4)                                       537 3-O-(3'-CH.sub.3 O--C.sub.6 H.sub.4)                                       538 3-O-(4'-CH.sub.3 O--C.sub.6 H.sub.4)                                       539 4-O-(2'-CH.sub.3 O--C.sub.6 H.sub.4)                                       540 4-O-(3'-CH.sub.3 O--C.sub.6 H.sub.4)                                       541 4-O-(4'-CH.sub.3 O--C.sub.6 H.sub.4)                                       542 2-O-(2'-O.sub.2 N--C.sub.6 H.sub.4)                                        543 2-O-(3'-O.sub.2 N--C.sub.6 H.sub.4)                                        544 2-O-(4'-O.sub.2 N--C.sub.6 H.sub.4)                                        545 3-O-(2'-O.sub.2 N--C.sub.6 H.sub.4)                                        546 3-O-(3'-O.sub.2 N--C.sub.6 H.sub.4)                                        547 3-O-(4'-O.sub.2 N--C.sub.6 H.sub.4)                                        548 4-O-(2'-O.sub.2 N--C.sub.6 H.sub.4)                                        549 4-O-(3'-O.sub.2 N--C.sub.6 H.sub.4)                                        550 4-O-(4'-O.sub.2 N--C.sub.6 H.sub.4)                                        551 2-O-(2'-NC--C.sub.6 H.sub.4)                                               552 2-O-(3'-NC--C.sub.6 H.sub.4)                                               553 2-O-(4'-NC--C.sub.6 H.sub.4)                                               554 3-O-(2'-NC--C.sub.6 H.sub.4)                                               555 3-O-(3'-NC--C.sub.6 H.sub.4)                                               556 3-O-(4'-NC--C.sub.6 H.sub.4)                                               557 4-O-(2'-NC--C.sub.6 H.sub.4)                                               558 4-O-(3'-NC--C.sub.6 H.sub.4)                                               559 4-O-(4'-NC--C.sub.6 H.sub.4)                                               560 2-O-(2'-CF.sub.3 --C.sub.6 H.sub.4)                                        561 2-O-(3'-CF.sub.3 --C.sub.6 H.sub.4)                                        562 2-O-(4'-CF.sub.3 --C.sub.6 H.sub.4)                                        563 3-O-(2'-CF.sub.3 --C.sub.6 H.sub.4)                                        564 3-O-(3'-CF.sub.3 --C.sub.6 H.sub.4)                                        565 3-O-(4'-CF.sub.3 --C.sub.6 H.sub.4)                                        566 4-O-(2'-CF.sub.3 --C.sub.6 H.sub.4)                                        567 4-O-(3'-CF.sub.3 --C.sub.6 H.sub.4)                                        568 4-O-(4'-CF.sub.3 --C.sub.6 H.sub.4)                                        569 2-Pyridinyl-2'                                                             570 2-Pyridinyl-3'                                                             571 2-Pyridinyl-4'                                                             572 3-Pyridinyl-2'                                                             573 3-Pyridinyl-3'                                                             574 3-Pyridinyl-4'                                                             575 4-Pyridinyl-2'                                                             576 4-Pyridinyl-3'                                                             577 4-Pyridinyl-4'                                                             578 2-Pyrimidinyl-2'                                                           579 2-Pyrimidinyl-3'                                                           580 2-Pyrimidinyl-4'                                                           581 3-Pyrimidinyl-2'                                                           582 3-Pyrimidinyl-3'                                                           583 3-Pyrimidinyl-4'                                                           584 4-Pyrimidinyl-2'                                                           585 4-Pyrimidinyl-3'                                                           586 4-Pyrimidinyl-4'                                                           587 2-Pyrazolyl-1'                                                             588 2-Pyrazolyl-3'                                                             589 2-Pyrazolyl-4'                                                             590 3-Pyrazolyl-1'                                                             591 3-Pyrazolyl-3'                                                             592 3-Pyrazolyl-4'                                                             593 4-Pyrazolyl-1'                                                             594 4-Pyrazolyl-3'                                                             595 4-Pyrazolyl-4'                                                             596 2-Isoxazolyl-3'                                                            597 2-Isoxazolyl-4'                                                            598 2-Isoxazolyl-5'                                                            599 3-Isoxazolyl-3'                                                            600 3-Isoxazolyl-4'                                                            601 3-Isoxazolyl-5'                                                            602 4-Isoxazolyl-3'                                                            603 4-Isoxazolyl-4'                                                            604 4-Isoxazolyl-5'                                                            605 2-Isothiazolyl-3'                                                          606 2-Isothiazolyl-4'                                                          607 2-Isothiazolyl-5'                                                          608 3-Isothiazolyl-3'                                                          609 3-Isothiazolyl-4'                                                          610 3-Isothiazolyl-5'                                                          611 4-Isothiazolyl-3'                                                          612 4-Isothiazolyl-4'                                                          613 4-Isothiazolyl-5'                                                          614 2-Imidazolyl-1'                                                            615 2-Imidazolyl-2'                                                            616 2-Imidazolyl-4'                                                            617 3-Imidazolyl-1'                                                            618 3-Imidazolyl-2'                                                            619 3-Imidazolyl-4'                                                            620 4-Imidazolyl-1'                                                            621 4-Imidazolyl-2'                                                            622 4-Imidazolyl-4'                                                            623 2-Oxazolyl-2'                                                              624 2-Oxazolyl-4'                                                              625 2-Oxazolyl-5'                                                              626 3-Oxazolyl-2'                                                              627 3-Oxazolyl-4'                                                              628 3-Oxazolyl-5'                                                              629 4-Oxazolyl-2'                                                              630 4-Oxazolyl-4'                                                              631 4-Oxazolyl-5'                                                              632 2-Thiazolyl-2'                                                             633 2-Thiazolyl-4'                                                             634 2-Thiazolyl-5'                                                             635 3-Thiazolyl-2'                                                             636 3-Thiazolyl-4'                                                             637 3-Thiazolyl-5'                                                             638 4-Thiazolyl-2'                                                             639 4-Thiazolyl-4'                                                             640 4-Thiazolyl-5'                                                             641 2-CH.sub.3 -4-(CH.sub.3 --C═N--O--CH.sub.2 --CH.sub.2 --OCH.sub.               3)                                                                     642 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C═N--O--CH.sub.2 --CH.sub.2                   --OCH.sub.3)                                                           643 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C═N--O--CH.sub.2 --CH.sub.2                --OCH.sub.3)                                                           644 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C═N--OCH.sub.3)                     645 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C═N--OC.sub.2 H.sub.5)                       646 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C═N--O-n-C.sub.3                   H.sub.7)                                                               647 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C═N--O-i-C.sub.3 H.sub.7)                    648 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C═N--O-Allyl)                       649 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C═N--O-trans-Chloroa               llyl)                                                                  650 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C═N--O-Propargyl)                   651 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C═N--O-n-C.sub.4 H.sub.9)                    652 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C═N--O--CH.sub.2                   --C.sub.6 H.sub.5)                                                     653 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C═N--OCH.sub.3)                     654 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C═N--OC.sub.2 H.sub.5)                       655 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C═N--O-n-C.sub.3                   H.sub.7)                                                               656 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C═N--O-i-C.sub.3 H.sub.7)                    657 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C═N--O-Allyl)                       658 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C═N--O-trans-Chloroa               llyl)                                                                  659 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C═N--O-Propargyl)                   660 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C═N--O-n-C.sub.4 H.sub.9)                    661 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C═N--O--CH.sub.2                   --C.sub.6 H.sub.5)                                                     662 2-O-n-C.sub.4 H.sub.9                                                      663 2-O-i-C.sub.4 H.sub.9                                                      664 2-O-s-C.sub.4 H.sub.9                                                      665 2-O-t-C.sub.4 H.sub.9                                                      666 2-Neopentyloxy                                                             667 3-O-n-C.sub.4 H.sub.9                                                      668 3-O-i-C.sub.4 H.sub.9                                                      669 3-O-s-C.sub.4 H.sub.9                                                      670 3-O-t-C.sub.4 H.sub.9                                                      671 3-Neopentyloxy                                                             672 4-O-n-C.sub.4 H.sub.9                                                      673 4-O-i-C.sub.4 H.sub.9                                                      674 4-O-s-C.sub.4 H.sub.9                                                      675 4-O-t-C.sub.4 H.sub.9                                                      676 4-Neopentyloxy                                                             677 3-CH.sub.3 -4-OCH.sub.3                                                    678 3-CH.sub.3 -4-OC.sub.2 H.sub.5                                             679 3-CH.sub.3 -4-O-n-C.sub.3 H.sub.7                                          680 3-CH.sub.3 -4-O-n-C.sub.4 H.sub.9                                          681 3-CH.sub.3 -4-O-i-C.sub.4 H.sub.9                                          682 3-CH.sub.3 -4-O-s-C.sub.4 H.sub.9                                          683 3-CH.sub.3 -4-O-t-C.sub.4 H.sub.9                                          684 3-CH.sub.3 -4-Neopentyloxy                                                 685 2-CH.sub.3 -3-OCH.sub.3                                                    686 2-CH.sub.3 -4-OCH.sub.3                                                    687 2-CH.sub.3 -5-OCH.sub.3                                                    688 2-CH.sub.3 -6-OCH.sub.3                                                    689 3-CH.sub.3 -4-OCH.sub.3                                                    690 3-CH.sub.3 -5-OCH.sub.3                                                    691 3-CH.sub.3 -6-OCH.sub.3                                                    692 4-CH.sub.3 -5-O--CH.sub.3                                                  693 4-CH.sub.3 -6-O--CH.sub.3                                                  694 4-CH.sub.3 -6-OCH.sub.3                                                    695 2-CH.sub.3 -3-O-i-C.sub.3 H.sub.7                                          696 2-CH.sub.3 -4-O-i-C.sub.3 H.sub.7                                          697 2-CH.sub.3 -5-O-i-C.sub.3 H.sub.7                                          698 2-CH.sub.3 -6-O-i-C.sub.3 H.sub.7                                          699 3-CH.sub.3 -4-O-i-C.sub.3 H.sub.7                                          700 3-CH.sub.3 -5-O-i-C.sub.3 H.sub.7                                          701 3-CH.sub.3 -6-O-i-C.sub.3 H.sub.7                                          702 4-CH.sub.3 -5-O-i-C.sub.3 H.sub.7                                          703 4-CH.sub.3 -6-O-i-C.sub.3 H.sub.7                                          704 5-CH.sub.3 -6-O-i-C.sub.3 H.sub.7                                          705 2-Cl-3-OCH.sub.3                                                           706 2-Cl-4-OCH.sub.3                                                           707 2-Cl-5-OCH.sub.3                                                           708 2-Cl-6-OCH.sub.3                                                           709 3-Cl-4-OCH.sub.3                                                           710 3-Cl-5-OCH.sub.3                                                           711 3-Cl-6-OCH.sub.3                                                           712 4-Cl-5-OCH.sub.3                                                           713 4-Cl-6-OCH.sub.3                                                           714 5-Cl-6-OCH.sub.3                                                         ______________________________________                                    

                  TABLE 35                                                         ______________________________________                                         1  STR255##                                                                      I: R.sup.1 = H, Z = C.sub.2 H.sub.5                                                              VIII: R.sup.1 = H, Z = NH(CH.sub.3)                          II: R.sup.1 = CH.sub.3, Z = C.sub.2 H.sub.5 IX: R.sup.1 = CH.sub.3, Z =                          NH(CH.sub.3)                                                 III: R.sup.1 = C.sub.2 H.sub.5, Z = C.sub.2 H.sub.5 X: R.sup.1 =                                 C.sub.2 H.sub.5, Z = NH(CH.sub.3)                            IV: R.sup.1 = Allyl, Z = C.sub.2 H.sub.5 XI: R.sup.1 = Allyl, Z =                                NH(CH.sub.3)                                                 V: R.sup.1 = Propargyl, Z = C.sub.2 H.sub.5 XII: R.sup.1 = Propargyl, Z                          = NH(CH.sub.3)                                               VI: R.sup.1 = CH.sub.2 --OCH.sub.3, XIII: R.sup.1 = CH.sub.2 --OCH.sub.3                         , Z = NH(CH.sub.3)                                           Z = C.sub.2 H.sub.5 XIV: R.sup.1 = CO--C.sub.2 H.sub.5, Z = NH(CH.sub.3)       VII: R.sup.1 = CO--C.sub.2 H.sub.5, Z = C.sub.2 H.sub.5                         -                                                                           No.       X.sub.m                                                              ______________________________________                                         1         H                                                                      2 2-F                                                                          3 3-F                                                                          4 4-F                                                                          5 2,4-F.sub.2                                                                  6 2,4,6-F.sub.3                                                                7 2,3,4,5,6-F.sub.5                                                            8 2,3-F.sub.2                                                                  9 2-Cl                                                                         10 3-Cl                                                                        11 4-Cl                                                                        12 2,3-Cl.sub.2                                                                13 2,4-Cl.sub.2                                                                14 2,5-Cl.sub.2                                                                15 2,6-Cl.sub.2                                                                16 3,4-Cl.sub.2                                                                17 3,5-Cl.sub.2                                                                18 2,3,4-Cl.sub.3                                                              19 2,3,5-Cl.sub.3                                                              20 2,3,6-Cl.sub.3                                                              21 2,4,5-Cl.sub.3                                                              22 2,4,6-Cl.sub.3                                                              23 3,4,5-Cl.sub.3                                                              24 2,3,4,6-Cl.sub.4                                                            25 2,3,5,6-Cl.sub.4                                                            26 2,3,4,5,6-Cl.sub.5                                                          27 2-Br                                                                        28 3-Br                                                                        29 4-Br                                                                        30 2,4-Br.sub.2                                                                31 2,5-Br.sub.2                                                                32 2,6-Br.sub.2                                                                33 2,4,6-Br.sub.3                                                              34 2,3,4,5,6-Br.sub.5                                                          35 2-I                                                                         36 3-I                                                                         37 4-I                                                                         38 2,4-I.sub.2                                                                 39 2-Cl, 3-F                                                                   40 2-Cl, 4-F                                                                   41 2-Cl, 5-F                                                                   42 2-Cl, 6-F                                                                   43 2-Cl, 3-Br                                                                  44 2-Cl, 4-Br                                                                  45 2-Cl, 5-Br                                                                  46 2-Cl, 6-Br                                                                  47 2-Br, 3-Cl                                                                  48 2-Br, 4-Cl                                                                  49 2-Br, 5-Cl                                                                  50 2-Br, 3-F                                                                   51 2-Br, 4-F                                                                   52 2-Br, 5-F                                                                   53 2-Br, 6-F                                                                   54 2-F, 3-Cl                                                                   55 2-F, 4-Cl                                                                   56 2-F, 5-Cl                                                                   57 3-Cl, 4-F                                                                   58 3-Cl, 5-F                                                                   59 3-Cl, 4-Br                                                                  60 3-Cl, 5-Br                                                                  61 3-F, 4-Cl                                                                   62 3-F, 4-Br                                                                   63 3-Br, 4-Cl                                                                  64 3-Br, 4-F                                                                   65 2,6-Cl.sub.2, 4-Br                                                          66 2-CH.sub.3                                                                  67 3-CH.sub.3                                                                  68 4-CH.sub.3                                                                  69 2,3-(CH.sub.3).sub.2                                                        70 2,4-(CH.sub.3).sub.2                                                        71 2,5-(CH.sub.3).sub.2                                                        72 2,6-(CH.sub.3).sub.2                                                        73 3,4-(CH.sub.3).sub.2                                                        74 3,5-(CH.sub.3).sub.2                                                        75 2,3,5-(CH.sub.3).sub.3                                                      76 2,3,4-(CH.sub.3).sub.3                                                      77 2,3,6-(CH.sub.3).sub.3                                                      78 2,4,5-(CH.sub.3).sub.3                                                      79 2,4,6-(CH.sub.3).sub.3                                                      80 3,4,5-(CH.sub.3).sub.3                                                      81 2,3,4,6-(CH.sub.3).sub.4                                                    82 2,3,5,6-(CH.sub.3).sub.4                                                    83 2,3,4,5,6-(CH.sub.3).sub.5                                                  84 2-C.sub.2 H.sub.5                                                           85 3-C.sub.2 H.sub.5                                                           86 4-C.sub.2 H.sub.5                                                           87 2,4-(C.sub.2 H.sub.5).sub.2                                                 88 2,6-(C.sub.2 H.sub.5).sub.2                                                 89 3,5-(C.sub.2 H.sub.5).sub.2                                                 90 2,4,6-(C.sub.2 H.sub.5).sub.3                                               91 2-n-C.sub.3 H.sub.7                                                         92 3-n-C.sub.3 H.sub.7                                                         93 4-n-C.sub.3 H.sub.7                                                         94 2-i-C.sub.3 H.sub.7                                                         95 3-i-C.sub.3 H.sub.7                                                         96 4-i-C.sub.3 H.sub.7                                                         97 2,4-(i-C.sub.3 H.sub.7).sub.2                                               98 2,6-(i-C.sub.3 H.sub.7).sub.2                                               99 3,5-(i-C.sub.3 H.sub.7).sub.2                                               100 2,4,6-(i-C.sub.3 H.sub.7).sub.3                                            101 2-s-C.sub.4 H.sub.9                                                        102 3-s-C.sub.4 H.sub.9                                                        103 4-s-C.sub.4 H.sub.9                                                        104 2-t-C.sub.4 H.sub.9                                                        105 3-t-C.sub.4 H.sub.9                                                        106 4-t-C.sub.4 H.sub.9                                                        107 2,3-(t-C.sub.4 H.sub.9).sub.2                                              108 2,4-(t-C.sub.4 H.sub.9).sub.2                                              109 2,5-(t-C.sub.4 H.sub.9).sub.2                                              110 2,6-(t-C.sub.4 H.sub.9).sub.2                                              111 3,4-(t-C.sub.4 H.sub.9).sub.2                                              112 2,4,6-(t-C.sub.4 H.sub.9).sub.3                                            113 4-n-C.sub.9 H.sub.19                                                       114 4-n-C.sub.12 H.sub.25                                                      115 4-n-C.sub.15 H.sub.31                                                      116 4-(1,1,3,3-Tetramethylbutyl)                                               117 4-(2,4,4-Trimethylpropyl)                                                  118 2-t-C.sub.4 H.sub.9, 4-CH.sub.3                                            119 2-t-C.sub.4 H.sub.9, 5-CH.sub.3                                            120 2,6-(t-C.sub.4 H.sub.9).sub.2, 4-CH.sub.3                                  121 2-CH.sub.3, 4-t-C.sub.4 H.sub.9                                            122 2-CH.sub.3, 6-t-C.sub.4 H.sub.9                                            123 2-CH.sub.3, 4-i-C.sub.3 H.sub.7                                            124 2-CH.sub.3, 5-i-C.sub.3 H.sub.7                                            125 3-CH.sub.3, 4-i-C.sub.3 H.sub.7                                            126 2-i-C.sub.3 H.sub.7, 5-CH.sub.3                                            127 2,4-(t-C.sub.4 H.sub.9).sub.2, 6-i-C.sub.3 H.sub.7                         128 2-Allyl                                                                    129 3-Allyl                                                                    130 4-Allyl                                                                    131 2-Allyl, 6-CH.sub.3                                                        132 2-cyclo-C.sub.6 H.sub.11                                                   133 3-cyclo-C.sub.6 H.sub.11                                                   134 4-cyclo-C.sub.6 H.sub.11                                                   135 2,4-(cyclo-C.sub.6 H.sub.11).sub.2, 6-CH.sub.3                             136 2-CH.sub.3, 4-cyclo-C.sub.6 H.sub.11                                       137 2-CH.sub.2 --C.sub.6 H.sub.5                                               138 3-CH.sub.2 --C.sub.6 H.sub.5                                               139 4-CH.sub.2 --C.sub.6 H.sub.5                                               140 2-CH.sub.2 --C.sub.6 H.sub.5, 4-CH.sub.3                                   141 2-CH.sub.3, 4-CH.sub.2 --C.sub.6 H.sub.5                                   142 2-C.sub.6 H.sub.5                                                          143 3-C.sub.6 H.sub.5                                                          144 4-C.sub.6 H.sub.5                                                          145 4-(2-i-C.sub.3 H.sub.7 --C.sub.6 H.sub.4)                                  146 4-C.sub.6 H.sub.5, 2,6-(CH.sub.3).sub.2                                    147 2-Cl, 4-C.sub.6 H.sub.5                                                    148 2-Br, 4-C.sub.6 H.sub.5                                                    149 2-C.sub.6 H.sub.5, 4-Cl                                                    150 2-C.sub.6 H.sub.5, 4-Br                                                    151 2-CH.sub.2 C.sub.6 H.sub.5, 4-Cl                                           152 2-CH.sub.2 C.sub.6 H.sub.5, 4-Br                                           153 2-Cl, 4-CH.sub.2 C.sub.6 H.sub.5                                           154 2-Br, 4-CH.sub.2 C.sub.6 H.sub.5                                           155 2-cyclo-C.sub.6 H.sub.11, 4-Cl                                             156 2-cyclo-C.sub.6 H.sub.11, 4-Br                                             157 2-Cl, 4-cyclo-C.sub.6 H.sub.11                                             158 2-Br, 4-cyclo-C.sub.6 H.sub.11                                             159 2-OCH.sub.3                                                                160 3-OCH.sub.3                                                                161 4-OCH.sub.3                                                                162 2-OC.sub.2 H.sub.5                                                         163 3-O--C.sub.2 H.sub.5                                                       164 4-O--C.sub.2 H.sub.5                                                       165 2-O-n-C.sub.3 H.sub.7                                                      166 3-O-n-C.sub.3 H.sub.7                                                      167 4-O-n-C.sub.3 H.sub.7                                                      168 2-O-i-C.sub.3 H.sub.7                                                      169 3-O-i-C.sub.3 H.sub.7                                                      170 4-O-i-C.sub.3 H.sub.7                                                      171 2-O-n-C.sub.6 H.sub.13                                                     172 3-O-n-C.sub.6 H.sub.13                                                     173 4-O-n-C.sub.6 H.sub.13                                                     174 2-O-n-C.sub.8 H.sub.17                                                     175 3-O-n-C.sub.8 H.sub.17                                                     176 4-O-n-C.sub.8 H.sub.17                                                     177 2-O--CH.sub.2 C.sub.6 H.sub.5                                              178 3-O--CH.sub.2 C.sub.6 H.sub.5                                              179 4-O--CH.sub.2 C.sub.6 H.sub.5                                              180 2-O--(CH.sub.2).sub.3 C.sub.6 H.sub.5                                      181 3-O--(CH.sub.2).sub.3 C.sub.6 H.sub.5                                      182 4-O--(CH.sub.2).sub.3 C.sub.6 H.sub.5                                      183 2,4-(OCH.sub.3).sub.2                                                      184 2-CF.sub.3                                                                 185 3-CF.sub.3                                                                 186 4-CF.sub.3                                                                 187 2-OCF.sub.3                                                                188 3-OCF.sub.3                                                                189 4-OCF.sub.3                                                                190 3-OCH.sub.2 CHF.sub.2                                                      191 2-NO.sub.2                                                                 192 3-NO.sub.2                                                                 193 4-NO.sub.2                                                                 194 2-CN                                                                       195 3-CN                                                                       196 4-CN                                                                       197 2-CH.sub.3, 3-Cl                                                           198 2-CH.sub.3, 4-Cl                                                           199 2-CH.sub.3, 5-Cl                                                           200 2-CH.sub.3, 6-Cl                                                           201 2-CH.sub.3, 3-F                                                            202 2-CH.sub.3, 4-F                                                            203 2-CH.sub.3, 5-F                                                            204 2-CH.sub.3, 6-F                                                            205 2-CH.sub.3, 3-Br                                                           206 2-CH.sub.3, 4-Br                                                           207 2-CH.sub.3, 5-Br                                                           208 2-CH.sub.3, 6-Br                                                           209 2-Cl, 3-CH.sub.3                                                           210 2-Cl, 4-CH.sub.3                                                           211 2-Cl, 5-CH.sub.3                                                           212 2-F, 3-CH.sub.3                                                            213 2-F, 4-CH.sub.3                                                            214 2-F, 5-CH.sub.3                                                            215 2-Br, 3-CH.sub.3                                                           216 2-Br, 4-CH.sub.3                                                           217 2-Br, 5-CH.sub.3                                                           218 3-CH.sub.3, 4-Cl                                                           219 3-CH.sub.3, 5-Cl                                                           220 3-CH.sub.3, 4-F                                                            221 3-CH.sub.3, 5-F                                                            222 3-CH.sub.3, 4-Br                                                           223 3-CH.sub.3, 5-Br                                                           224 3-F, 4-CH.sub.3                                                            225 3-Cl, 4-CH.sub.3                                                           226 3-Br, 4-CH.sub.3                                                           227 2-Cl, 4,5-(CH.sub.3).sub.2                                                 228 2-Br, 4,5-(CH.sub.3).sub.2                                                 229 2-Cl, 3,5-(CH.sub.3).sub.2                                                 230 2-Br, 3,5-(CH.sub.3).sub.2                                                 231 2,6-Cl.sub.2, 4-CH.sub.3                                                   232 2,6-F.sub.2, 4-CH.sub.3                                                    233 2,6-Br.sub.2, 4-CH.sub.3                                                   234 2,4-Br.sub.2, 6-CH.sub.3                                                   235 2,4-F.sub.2, 6-CH.sub.3                                                    236 2,4-Br.sub.2, 6-CH.sub.3                                                   237 2,6-(CH.sub.3).sub.2, 4-F                                                  238 2,6-(CH.sub.3).sub.2, 4-Cl                                                 239 2,6-(CH.sub.3).sub.2, 4-Br                                                 240 3,5-(CH.sub.3).sub.2, 4-F                                                  241 3,5-(CH.sub.3).sub.2, 4-Cl                                                 242 3,5-(CH.sub.3).sub.2, 4-Br                                                 243 2,3,6-(CH.sub.3).sub.3, 4-F                                                244 2,3,6-(CH.sub.3).sub.3, 4-Cl                                               245 2,3,6-(CH.sub.3).sub.3, 4-Br                                               246 2,4-(CH.sub.3).sub.2, 6-F                                                  247 2,4-(CH.sub.3).sub.2, 6-Cl                                                 248 2,4-(CH.sub.3).sub.2, 6-Br                                                 249 2-i-C.sub.3 H.sub.7, 4-Cl, 5-CH.sub.3                                      250 2-Cl, 4-NO.sub.2                                                           251 2-NO.sub.2, 4-Cl                                                           252 2-OCH.sub.3, 5-NO.sub.2                                                    253 2,4-Cl.sub.2, 5-NO.sub.2                                                   254 2,4-Cl.sub.2, 6-NO.sub.2                                                   255 2,6-Cl.sub.2, 4-NO.sub.2                                                   256 2,6-Br.sub.2, 4-NO.sub.2                                                   257 2,6-I.sub.2, 4-NO.sub.2                                                    258 2-CH.sub.3, 5-i-C.sub.3 H.sub.7, 4-Cl                                      259 2-CO.sub.2 CH.sub.3                                                        260 3-CO.sub.2 CH.sub.3                                                        261 4-CO.sub.2 CH.sub.3                                                        262 2-CO.sub.2 (C.sub.2 H.sub.5)                                               263 3-CO.sub.2 (C.sub.2 H.sub.5)                                               264 4-CO.sub.2 (C.sub.2 H.sub.5)                                               265 2-CO.sub.2 (n-C.sub.3 H.sub.7)                                             266 3-CO.sub.2 (n-C.sub.3 H.sub.7)                                             267 4-CO.sub.2 (n-C.sub.3 H.sub.7)                                             268 2-CO.sub.2 (i-C.sub.3 H.sub.7)                                             269 3-CO.sub.2 (i-C.sub.3 H.sub.7)                                             270 4-CO.sub.2 (i-C.sub.3 H.sub.7)                                             271 2-CO.sub.2 (n-C.sub.6 H.sub.13)                                            272 3-CO.sub.2 (n-C.sub.6 H.sub.13)                                            273 4-CO.sub.2 (n-C.sub.6 H.sub.13)                                            274 2-CH.sub.2 --OCH.sub.3                                                     275 3-CH.sub.2 --OCH.sub.3                                                     276 4-CH.sub.2 --OCH.sub.3                                                     277 2-CH.sub.2 O(C.sub.2 H.sub.5)                                              278 3-CH.sub.2 O(C.sub.2 H.sub.5)                                              279 4-CH.sub.2 O(C.sub.2 H.sub.5)                                              280 2-CH.sub.2 O(n-C.sub.3 H.sub.7)                                            281 3-CH.sub.2 O(n-C.sub.3 H.sub.7)                                            282 4-CH.sub.2 O(n-C.sub.3 H.sub.7)                                            283 2-CH.sub.2 O(i-C.sub.3 H.sub.7)                                            284 3-CH.sub.2 O(i-C.sub.3 H.sub.7)                                            285 4-CH.sub.2 O(i-C.sub.3 H.sub.7)                                            286 2-CHO                                                                      287 3-CHO                                                                      288 4-CHO                                                                      289 2-CO--CH.sub.3                                                             290 3-CO--CH.sub.3                                                             291 4-CO--CH.sub.3                                                             292 2-CO--CH.sub.2 --CH.sub.3                                                  293 3-CO--CH.sub.2 --CH.sub.3                                                  294 4-CO--CH.sub.2 --CH.sub.3                                                  295 2-CO--CH.sub.2 --CH.sub.2 --CH.sub.3                                       296 3-CO--CH.sub.2 --CH.sub.2 --CH.sub.3                                       297 4-CO--CH.sub.2 --CH.sub.2 --CH.sub.3                                       298 2-CO--CH(CH.sub.3)--CH.sub.3                                               299 3-CO--CH(CH.sub.3)--CH.sub.3                                               300 4-CO--CH(CH.sub.3)--CH.sub.3                                               301 2-Me-4-CHO                                                                 302 2-Me-4-CH.sub.3 --CO                                                       303 2-Me-4-CO--CH.sub.2 --CH.sub.3                                             304 2-Me-4-CO--CH.sub.2 --CH.sub.2 --CH.sub.3                                  305 2-Me-4-CO--CH(CH.sub.3).sub.2                                              306 2,5-Me.sub.2 -4-CHO                                                        307 2,5-Me.sub.2 -4-CO--CH.sub.3                                               308 2,5-Me.sub.2 -4-CO--CH.sub.2 --CH.sub.3                                    309 2,5-Me.sub.2 -4-CH.sub.2 --CH.sub.2 --CO--CH.sub.3                         310 2,5-Me.sub.2 -4-CO--CH(CH.sub.3).sub.2                                     311 2-Cl-4-CHO                                                                 312 2-Cl-4-CO--CH.sub.3                                                        313 2-Cl-4-CO--CH.sub.2 --CH.sub.3                                             314 2-Cl-4-CO--CH(CH.sub.3).sub.2                                              315 2,5-Cl.sub.2 -4-CHO                                                        316 2,5-Cl.sub.2 -4-CO--CH.sub.3                                               317 2,5-Cl.sub.2 -4-CO--CH.sub.2 --CH.sub.3                                    318 2,5-Cl.sub.2 -4-CO--CH.sub.2 --CH.sub.2 --CH.sub.3                         319 2,5-Cl.sub.2 -4-CO--CH(CH.sub.3).sub.2                                     320 2-C(═NOCH.sub.3)--CH.sub.3                                             321 3-C(═NOCH.sub.3)--CH.sub.3                                             322 4-C(═NOCH.sub.3)--CH.sub.3                                             323 2-C(═NOC.sub.2 H.sub.5)--CH.sub.3                                      324 3-C(═NOC.sub.2 H.sub.5)--CH.sub.3                                      325 4-C(═NOC.sub.2 H.sub.5)--CH.sub.3                                      326 2-C(═NO-n-C.sub.3 H.sub.7)--CH.sub.3                                   327 3-C(═NO-n-C.sub.3 H.sub.7)--CH.sub.3                                   328 4-C(═NO-n-C.sub.3 H.sub.7)--CH.sub.3                                   329 2-C(═NO-i-C.sub.3 H.sub.7)--CH.sub.3                                   330 3-C(═NO-i-C.sub.3 H.sub.7)--CH.sub.3                                   331 4-C(═NO-i-C.sub.3 H.sub.7)--CH.sub.3                                   332 2-C(═NO-Allyl)--CH.sub.3                                               333 3-C(═NO-Allyl)--CH.sub.3                                               334 4-C(═NO-Allyl)--CH.sub.3                                               335 2-C(═NO-trans-Chloroallyl)--CH.sub.3                                   336 3-C(═NO-trans-Chloroallyl)--CH.sub.3                                   337 4-C(═NO-trans-Chloroallyl)--CH.sub.3                                   338 2-C(═NO-Propargyl)--CH.sub.3                                           339 3-C(═NO-Propargyl)--CH.sub.3                                           340 4-C(═NO-Propargyl)--CH.sub.3                                           341 2-C(═NO-n-C.sub.4 H.sub.9)--CH.sub.3                                   342 3-C(═NO-n-C.sub.4 H.sub.9)--CH.sub.3                                   343 4-C(═NO-n-C.sub.4 H.sub.9)--CH.sub.3                                   344 2-C(═NO--CH.sub.2 --C.sub.6 H.sub.5)--CH.sub.3                         345 3-C(═NO--CH.sub.2 --C.sub.6 H.sub.5)--CH.sub.3                         346 4-C(═NO--CH.sub.2 --C.sub.6 H.sub.5)--CH.sub.3                         347 2-CH.sub.3 -4-CH═NOCH.sub.3                                            348 2-CH.sub.3 -4-CH═NOC.sub.2 H.sub.5                                     349 2-CH.sub.3 -4-CH═NO-n-C.sub.3 H.sub.7                                  350 2-CH.sub.3 -4-CH═NO-i-C.sub.3 H.sub.7                                  351 2-CH.sub.3 -4-CH═NO-Allyl                                              352 2-CH.sub.3 -4-CH═NO-(trans-Chloroallyl)                                353 2-CH.sub.3 -4-CH═NO-Propargyl                                          354 2-CH.sub.3 -4-CH═NO-n-C.sub.4 H.sub.9                                  355 2-CH.sub.3 -4-CH═NO--CH.sub.2 --C.sub.6 H.sub.5                        356 2-CH.sub.3 -4-(CH.sub.3 --C═NOCH.sub.3)                                357 2-CH.sub.3 -4-(CH.sub.3 --C═NOC.sub.2 H.sub.5)                         358 2-CH.sub.3 -4-(CH.sub.3 --C═NO-n-C.sub.3 H.sub.7)                      359 2-CH.sub.3 -4-(CH.sub.3 --C═NO-i-C.sub.3 H.sub.7)                      360 2-CH.sub.3 -4-(CH.sub.3 --C═NO-Allyl)                                  361 2-CH.sub.3 -4-(CH.sub.3 --C═NO-trans-Chloroallyl)                      362 2-CH.sub.3 -4-(CH.sub.3 --C═NO-Propargyl)                              363 2-CH.sub.3 -4-(CH.sub.3 --C═NO-n-C.sub.4 H.sub.9)                      364 2-CH.sub.3 -4-(CH.sub.3 --C═NO--CH.sub.2 --C.sub.6 H.sub.5)                     365 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C═NO--CH.sub.3)                       366 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C═NO--C.sub.2                        H.sub.5)                                                               367 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C═NO-n-C.sub.3 H.sub.7)                        368 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C═NO-i-C.sub.3                       H.sub.7)                                                               369 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C═NO-Allyl)                           370 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C═NO-trans-Chloroallyl)                        371 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C═NO-Propargyl)                       372 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C═NO-n-C.sub.4                       H.sub.9)                                                               373 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C═NO--CH.sub.2 --C.sub.6                      H.sub.5)                                                               374 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C═NOCH.sub.3)                      375 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C═NOC.sub.2 H.sub.5)                        376 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C═NO-n-C.sub.3                    H.sub.7)                                                               377 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C═NO-i-C.sub.3 H.sub.7)                     378 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C═NO-Allyl)                        379 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C═NO-trans-Chloroal               lyl)                                                                   380 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C═NO-Proparyl)                     381 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C═NO-n-C.sub.4 H.sub.9)                     382 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C═NO--CH.sub.2                    --C.sub.6 H.sub.5)                                                     383 2-C.sub.6 H.sub.5                                                          384 3-C.sub.6 H.sub.5                                                          385 4-C.sub.6 H.sub.5                                                          386 2-(2'-F--C.sub.6 H.sub.4)                                                  387 2-(3'-F--C.sub.6 H.sub.4)                                                  388 2-(4'-F--C.sub.6 H.sub.4)                                                  389 3-(2'-F--C.sub.6 H.sub.4)                                                  390 3-(3'-F--C.sub.6 H.sub.4)                                                  391 3-(4'-F--C.sub.6 H.sub.4)                                                  392 4-(2'-F--C.sub.6 H.sub.4)                                                  393 4-(3'-F--C.sub.6 H.sub.4)                                                  394 4-(4'-F--C.sub.6 H.sub.4)                                                  395 2-(2'-Cl--C.sub.6 H.sub.4)                                                 396 2-(3'-Cl--C.sub.6 H.sub.4)                                                 397 2-(4'-Cl--C.sub.6 H.sub.4)                                                 398 3-(2'-Cl--C.sub.6 H.sub.4)                                                 399 3-(3'-Cl--C.sub.6 H.sub.4)                                                 400 3-(4'-Cl--C.sub.6 H.sub.4)                                                 401 4-(2'-Cl--C.sub.6 H.sub.4)                                                 402 4-(3'-Cl--C.sub.6 H.sub.4)                                                 403 4-(4'-Cl--C.sub.6 H.sub.4)                                                 405 2-(2'-CH.sub.3 --C.sub.6 H.sub.4)                                          406 2-(3'-CH.sub.3 --C.sub.6 H.sub.4)                                          407 2-(4'-CH.sub.3 --C.sub.6 H.sub.4)                                          408 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)                                          409 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)                                          410 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)                                          411 4-(2'-CH.sub.3 --C.sub.6 H.sub.4)                                          412 4-(3'-CH.sub.3 --C.sub.6 H.sub.4)                                          413 4-(4'-CH.sub.3 --C.sub.6 H.sub.4)                                          414 2-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                      415 2-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                      416 2-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                      417 3-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                      418 3-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                      419 3-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                      420 4-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                      421 4-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                      422 4-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                      423 2-(2'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                       424 2-(3'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                       425 2-(4'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                       426 3-(2'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                       427 3-(3'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                       428 3-(4'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                       429 4-(2'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                       430 4-(3'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                       431 4-(4'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                       432 2-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                                 433 2-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                                 434 2-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                                 435 3-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                                 436 3-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                                 437 3-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                                 438 4-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                                 439 4-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                                 440 4-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                                 441 2-(2'-CH.sub.3 O--C.sub.6 H.sub.4)                                         442 2-(3'-CH.sub.3 O--C.sub.6 H.sub.4)                                         443 2-(4'-CH.sub.3 O--C.sub.6 H.sub.4)                                         444 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)                                         445 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)                                         446 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)                                         447 4-(2'-CH.sub.3 O--C.sub.6 H.sub.4)                                         448 4-(3'-CH.sub.3 O--C.sub.6 H.sub.4)                                         449 4-(4'-CH.sub.3 O--C.sub.6 H.sub.4)                                         450 2-(2'-O.sub.2 N--C.sub.6 H.sub.4)                                          451 2-(3'-O.sub.2 N--C.sub.6 H.sub.4)                                          452 2-(4'-O.sub.2 N--C.sub.6 H.sub.4)                                          453 3-(2'-O.sub.2 N--C.sub.6 H.sub.4)                                          454 3-(3'-O.sub.2 N--C.sub.6 H.sub.4)                                          455 3-(4'-O.sub.2 N--C.sub.6 H.sub.4)                                          456 4-(2'-O.sub.2 N--C.sub.6 H.sub.4)                                          457 4-(3'-O.sub.2 N--C.sub.6 H.sub.4)                                          458 4-(4'-O.sub.2 N--C.sub.6 H.sub.4)                                          459 2-(2'-NC--C.sub.6 H.sub.4)                                                 460 2-(3'-NC--C.sub.6 H.sub.4)                                                 461 2-(4'-NC--C.sub.6 H.sub.4)                                                 462 3-(2'-NC--C.sub.6 H.sub.4)                                                 463 3-(3'-NC--C.sub.6 H.sub.4)                                                 464 3-(4'-NC--C.sub.6 H.sub.4)                                                 465 4-(2'-NC--C.sub.6 H.sub.4)                                                 466 4-(3'-NC--C.sub.6 H.sub.4)                                                 467 4-(4'-NC--C.sub.6 H.sub.4)                                                 468 2-(2'-CF.sub.3 --C.sub.6 H.sub.4)                                          469 2-(3'-CF.sub.3 --C.sub.6 H.sub.4)                                          470 2-(4'-CF.sub.3 --C.sub.6 H.sub.4)                                          471 3-(2'-CF.sub.3 --C.sub.6 H.sub.4)                                          472 3-(3'-CF.sub.3 --C.sub.6 H.sub.4)                                          473 3-(4'-CF.sub.3 --C.sub.6 H.sub.4)                                          474 4-(2'-CF.sub.3 --C.sub.6 H.sub.4)                                          475 4-(3'-CF.sub.3 --C.sub.6 H.sub.4)                                          476 4-(4'-CF.sub.3 --C.sub.6 H.sub.4)                                          477 2-O--C.sub.6 H.sub.5                                                       475 3-O--C.sub.6 H.sub.5                                                       476 4-O--C.sub.6 H.sub.5                                                       478 2-O-(2'-F--C.sub.6 H.sub.4)                                                479 2-O-(3'-F--C.sub.6 H.sub.4)                                                480 2-O-(4'-F--C.sub.6 H.sub.4)                                                481 3-O-(2'-F--C.sub.6 H.sub.4)                                                482 3-O-(3'-F--C.sub.6 H.sub.4)                                                483 3-O-(4'-F--C.sub.6 H.sub.4)                                                484 4-O-(2'-F--C.sub.6 H.sub.4)                                                485 4-O-(3'-F--C.sub.6 H.sub.4)                                                486 4-O-(4'-F--C.sub.6 H.sub.4)                                                487 2-O-(2'-Cl--C.sub.6 H.sub.4)                                               488 2-O-(3'-Cl--C.sub.6 H.sub.4)                                               489 2-O-(4'-Cl--C.sub.6 H.sub.4)                                               490 3-O-(2'-Cl--C.sub.6 H.sub.4)                                               491 3-O-(3'-Cl--C.sub.6 H.sub.4)                                               492 3-O-(4'-Cl--C.sub.6 H.sub.4)                                               493 3-O-(4'-Cl--C.sub.6 H.sub.4)                                               494 4-O-(2'-Cl--C.sub.6 H.sub.4)                                               495 4-O-(3'-Cl--C.sub.6 H.sub.4)                                               496 4-O-(4'-Cl--C.sub.6 H.sub.4)                                               497 2-O-(2'-CH.sub.3 --C.sub.6 H.sub.4)                                        498 2-O-(3'-CH.sub.3 --C.sub.6 H.sub.4)                                        499 2-O-(4'-CH.sub.3 --C.sub.6 H.sub.4)                                        500 3-O-(2'-CH.sub.3 --C.sub.6 H.sub.4)                                        501 3-O-(3'-CH.sub.3 --C.sub.6 H.sub.4)                                        502 3-O-(4'-CH.sub.3 --C.sub.6 H.sub.4)                                        503 4-O-(2'-CH.sub.3 --C.sub.6 H.sub.4)                                        504 4-O-(3'-CH.sub.3 --C.sub.6 H.sub.4)                                        505 4-O-(4'-CH.sub.3 --C.sub.6 H.sub.4)                                        506 2-O-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                    507 2-O-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                    508 2-O-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                    509 3-O-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                    510 3-O-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                    511 3-O-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                    512 4-O-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                    513 4-O-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                    514 4-O-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                    515 2-O-(2'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                     516 2-O-(3'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                     517 2-O-(4'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                     518 3-O-(2'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                     519 3-O-(3'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                     520 3-O-(4'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                     521 4-O-(2'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                     522 4-O-(3'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                     523 4-O-(4'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                     524 2-O-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                               525 2-O-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                               526 2-O-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                               527 3-O-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                               528 3-O-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                               529 3-O-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                               530 4-O-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                               531 4-O-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                               532 4-O-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                               533 2-O-(2'-CH.sub.3 O--C.sub.6 H.sub.4)                                       534 2-O-(3'-CH.sub.3 O--C.sub.6 H.sub.4)                                       535 2-O-(4'-CH.sub.3 O--C.sub.6 H.sub.4)                                       536 3-O-(2'-CH.sub.3 O--C.sub.6 H.sub.4)                                       537 3-O-(3'-CH.sub.3 O--C.sub.6 H.sub.4)                                       538 3-O-(4'-CH.sub.3 O--C.sub.6 H.sub.4)                                       539 4-O-(2'-CH.sub.3 O--C.sub.6 H.sub.4)                                       540 4-O-(3'-CH.sub.3 O--C.sub.6 H.sub.4)                                       541 4-O-(4'-CH.sub.3 O--C.sub.6 H.sub.4)                                       542 2-O-(2'-O.sub.2 N--C.sub.6 H.sub.4)                                        543 2-O-(3'-O.sub.2 N--C.sub.6 H.sub.4)                                        544 2-O-(4'-O.sub.2 N--C.sub.6 H.sub.4)                                        545 3-O-(2'-O.sub.2 N--C.sub.6 H.sub.4)                                        546 3-O-(3'-O.sub.2 N--C.sub.6 H.sub.4)                                        547 3-O-(4'-O.sub.2 N--C.sub.6 H.sub.4)                                        548 4-O-(2'-O.sub.2 N--C.sub.6 H.sub.4)                                        549 4-O-(3'-O.sub.2 N--C.sub.6 H.sub.4)                                        550 4-O-(4'-O.sub.2 N--C.sub.6 H.sub.4)                                        551 2-O-(2'-NC--C.sub.6 H.sub.4)                                               552 2-O-(3'-NC--C.sub.6 H.sub.4)                                               553 2-O-(4'-NC--C.sub.6 H.sub.4)                                               554 3-O-(2'-NC--C.sub.6 H.sub.4)                                               555 3-O-(3'-NC--C.sub.6 H.sub.4)                                               556 3-O-(4'-NC--C.sub.6 H.sub.4)                                               557 4-O-(2'-NC--C.sub.6 H.sub.4)                                               558 4-O-(3'-NC--C.sub.6 H.sub.4)                                               559 4-O-(4'-NC--C.sub.6 H.sub.4)                                               560 2-O-(2'-CF.sub.3 --C.sub.6 H.sub.4)                                        561 2-O-(3'-CF.sub.3 --C.sub.6 H.sub.4)                                        562 2-O-(4'-CF.sub.3 --C.sub.6 H.sub.4)                                        563 3-O-(2'-CF.sub.3 --C.sub.6 H.sub.4)                                        564 3-O-(3'-CF.sub.3 --C.sub.6 H.sub.4)                                        565 3-O-(4'-CF.sub.3 --C.sub.6 H.sub.4)                                        566 4-O-(2'-CF.sub.3 --C.sub.6 H.sub.4)                                        567 4-O-(3'-CF.sub.3 --C.sub.6 H.sub.4)                                        568 4-O-(4'-CF.sub.3 --C.sub.6 H.sub.4)                                        569 2-Pyridinyl-2'                                                             570 2-Pyridinyl-3'                                                             571 2-Pyridinyl-4'                                                             572 3-Pyridinyl-2'                                                             573 3-Pyridinyl-3'                                                             574 3-Pyridinyl-4'                                                             575 4-Pyridinyl-2'                                                             576 4-Pyridinyl-3'                                                             577 4-Pyridinyl-4'                                                             578 2-Pyrimidinyl-2'                                                           579 2-Pyrimidinyl-3'                                                           580 2-Pyrimidinyl-4'                                                           581 3-Pyrimidinyl-2'                                                           582 3-Pyrimidinyl-3'                                                           583 3-Pyrimidinyl-4'                                                           584 4-Pyrimidinyl-2'                                                           585 4-Pyrimidinyl-3'                                                           586 4-Pyrimidinyl-4'                                                           587 2-Pyrazolyl-1'                                                             588 2-Pyrazolyl-3'                                                             589 2-Pyrazolyl-4'                                                             590 3-Pyrazolyl-1'                                                             591 3-Pyrazolyl-3'                                                             592 3-Pyrazolyl-4'                                                             593 4-Pyrazolyl-1'                                                             594 4-Pyrazolyl-3'                                                             595 4-Pyrazolyl-4'                                                             596 2-Isoxazolyl-3'                                                            597 2-Isoxazolyl-4'                                                            598 2-Isoxazolyl-5'                                                            599 3-Isoxazolyl-3'                                                            600 3-Isoxazolyl-4'                                                            601 3-Isoxazolyl-5'                                                            602 4-Isoxazolyl-3'                                                            603 4-Isoxazolyl-4'                                                            604 4-Isoxazolyl-5'                                                            605 2-Isothiazolyl-3'                                                          606 2-Isothiazolyl-4'                                                          607 2-Isothiazolyl-5'                                                          608 3-Isothiazolyl-3'                                                          609 3-Isothiazolyl-4'                                                          610 3-Isothiazolyl-5'                                                          611 4-Isothiazolyl-3'                                                          612 4-Isothiazolyl-4'                                                          613 4-Isothiazolyl-5'                                                          614 2-Imidazolyl-1'                                                            615 2-Imidazolyl-2'                                                            616 2-Imidazolyl-4'                                                            617 3-Imidazolyl-1'                                                            618 3-Imidazolyl-2'                                                            619 3-Imidazolyl-4'                                                            620 4-Imidazolyl-1'                                                            621 4-Imidazolyl-2'                                                            622 4-Imidazolyl-4'                                                            623 2-Oxazolyl-2'                                                              624 2-Oxazolyl-4'                                                              625 2-Oxazolyl-5'                                                              626 3-Oxazolyl-2'                                                              627 3-Oxazolyl-4'                                                              628 3-Oxazolyl-5'                                                              629 4-Oxazolyl-2'                                                              630 4-Oxazolyl-4'                                                              631 4-Oxazolyl-5'                                                              632 2-Thiazolyl-2'                                                             633 2-Thiazolyl-4'                                                             634 2-Thiazolyl-5'                                                             635 3-Thiazolyl-2'                                                             636 3-Thiazolyl-4'                                                             637 3-Thiazolyl-5'                                                             638 4-Thiazolyl-2'                                                             639 4-Thiazolyl-4'                                                             640 4-Thiazolyl-5'                                                             641 2-CH.sub.3 -4-(CH.sub.3 --C═N--O--CH.sub.2 --CH.sub.2 --OCH.sub.               3)                                                                     642 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C═N--O--CH.sub.2 --CH.sub.2                   --OCH.sub.3)                                                           643 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C═N--O--CH.sub.2 --CH.sub.2                --OCH.sub.3)                                                           644 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C═N--OCH.sub.3)                     645 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C═N--OC.sub.2 H.sub.5)                       646 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C═N--O-n-C.sub.3                   H.sub.7)                                                               647 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C═N--O-i-C.sub.3 H.sub.7)                    648 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C═N--O-Allyl)                       649 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C═N--O-trans-Chloroa               llyl)                                                                  650 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C═N--O-Propargyl)                   651 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C═N--O-n-C.sub.4 H.sub.9)                    652 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C═N--O--CH.sub.2                   --C.sub.6 H.sub.5)                                                     653 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C═N--OCH.sub.3)                     654 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C═N--OC.sub.2 H.sub.5)                       655 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C═N--O-n-C.sub.3                   H.sub.7)                                                               656 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C═N--O-i-C.sub.3 H.sub.7)                    657 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C═N--O-Allyl)                       658 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C═N--O-trans-Chloroa               llyl)                                                                  659 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C═N--O-Propargyl)                   660 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C═N--O-n-C.sub.4 H.sub.9)                    661 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C═N--O--CH.sub.2                   --C.sub.6 H.sub.5)                                                     662 2-O-n-C.sub.4 H.sub.9                                                      663 2-O-i-C.sub.4 H.sub.9                                                      664 2-O-s-C.sub.4 H.sub.9                                                      665 2-O-t-C.sub.4 H.sub.9                                                      666 2-Neopentyloxy                                                             667 3-O-n-C.sub.4 H.sub.9                                                      668 3-O-i-C.sub.4 H.sub.9                                                      669 3-O-s-C.sub.4 H.sub.9                                                      670 3-O-t-C.sub.4 H.sub.9                                                      671 3-Neopentyloxy                                                             672 4-O-n-C.sub.4 H.sub.9                                                      673 4-O-i-C.sub.4 H.sub.9                                                      674 4-O-s-C.sub.4 H.sub.9                                                      675 4-O-t-C.sub.4 H.sub.9                                                      676 4-Neopentyloxy                                                             677 3-CH.sub.3 -4-OCH.sub.3                                                    678 3-CH.sub.3 -4-OC.sub.2 H.sub.5                                             679 3-CH.sub.3 -4-O-n-C.sub.3 H.sub.7                                          680 3-CH.sub.3 -4-O-n-C.sub.4 H.sub.9                                          681 3-CH.sub.3 -4-O-i-C.sub.4 H.sub.9                                          682 3-CH.sub.3 -4-O-s-C.sub.4 H.sub.9                                          683 3-CH.sub.3 -4-O-t-C.sub.4 H.sub.9                                          684 3-CH.sub.3 -4-Neopentyloxy                                                 685 2-CH.sub.3 -3-OCH.sub.3                                                    686 2-CH.sub.3 -4-OCH.sub.3                                                    687 2-CH.sub.3 -5-OCH.sub.3                                                    688 2-CH.sub.3 -6-OCH.sub.3                                                    689 3-CH.sub.3 -4-OCH.sub.3                                                    690 3-CH.sub.3 -5-OCH.sub.3                                                    691 3-CH.sub.3 -6-OCH.sub.3                                                    692 4-CH.sub.3 -5-O--CH.sub.3                                                  693 4-CH.sub.3 -6-O--CH.sub.3                                                  694 4-CH.sub.3 -6-OCH.sub.3                                                    695 2-CH.sub.3 -3-O-i-C.sub.3 H.sub.7                                          696 2-CH.sub.3 -4-O-i-C.sub.3 H.sub.7                                          697 2-CH.sub.3 -5-O-i-C.sub.3 H.sub.7                                          698 2-CH.sub.3 -6-O-i-C.sub.3 H.sub.7                                          699 3-CH.sub.3 -4-O-i-C.sub.3 H.sub.7                                          700 3-CH.sub.3 -5-O-i-C.sub.3 H.sub.7                                          701 3-CH.sub.3 -6-O-i-C.sub.3 H.sub.7                                          702 4-CH.sub.3 -5-O-i-C.sub.3 H.sub.7                                          703 4-CH.sub.3 -6-O-i-C.sub.3 H.sub.7                                          704 5-CH.sub.3 -6-O-i-C.sub.3 H.sub.7                                          705 2-Cl-3-OCH.sub.3                                                           706 2-Cl-4-OCH.sub.3                                                           707 2-Cl-5-OCH.sub.3                                                           708 2-Cl-6-OCH.sub.3                                                           709 3-Cl-4-OCH.sub.3                                                           710 3-Cl-5-OCH.sub.3                                                           711 3-Cl-6-OCH.sub.3                                                           712 4-Cl-5-OCH.sub.3                                                           713 4-Cl-6-OCH.sub.3                                                           714 5-Cl-6-OCH.sub.3                                                         ______________________________________                                    

                  TABLE 36                                                         ______________________________________                                         1  STR256##                                                                      I: R.sup.1 = H, Z = C.sub.2 H.sub.5                                                              VIII: R.sup.1 = H, Z = NH(CH.sub.3)                          II: R.sup.1 = CH.sub.3, Z = C.sub.2 H.sub.5 IX: R.sup.1 = CH.sub.3, Z =                          NH(CH.sub.3)                                                 III: R.sup.1 = C.sub.2 H.sub.5, Z = C.sub.2 H.sub.5 X: R.sup.1 =                                 C.sub.2 H.sub.5, Z = NH(CH.sub.3)                            IV: R.sup.1 = Allyl, Z = C.sub.2 H.sub.5 XI: R.sup.1 = Allyl, Z =                                NH(CH.sub.3)                                                 V: R.sup.1 = Propargyl, Z = C.sub.2 H.sub.5 XII: R.sup.1 = Propargyl, Z                          = NH(CH.sub.3)                                               VI: R.sup.1 = CH.sub.2 --OCH.sub.3, XIII: R.sup.1 = CH.sub.2 --OCH.sub.3                         , Z = NH(CH.sub.3)                                           Z = C.sub.2 H.sub.5 XIV: R.sup.1 = CO--C.sub.2 H.sub.5, Z = NH(CH.sub.3)       VII: R.sup.1 = CO--C.sub.2 H.sub.5, Z = C.sub.2 H.sub.5                         -                                                                           No.       X.sub.m                                                              ______________________________________                                         1         H                                                                      2 2-F                                                                          3 3-F                                                                          4 4-F                                                                          5 2,4-F.sub.2                                                                  6 2,4,6-F.sub.3                                                                7 2,3,4,5,6-F.sub.5                                                            8 2,3-F.sub.2                                                                  9 2-Cl                                                                         10 3-Cl                                                                        11 4-Cl                                                                        12 2,3-Cl.sub.2                                                                13 2,4-Cl.sub.2                                                                14 2,5-Cl.sub.2                                                                15 2,6-Cl.sub.2                                                                16 3,4-Cl.sub.2                                                                17 3,5-Cl.sub.2                                                                18 2,3,4-Cl.sub.3                                                              19 2,3,5-Cl.sub.3                                                              20 2,3,6-Cl.sub.3                                                              21 2,4,5-Cl.sub.3                                                              22 2,4,6-Cl.sub.3                                                              23 3,4,5-Cl.sub.3                                                              24 2,3,4,6-Cl.sub.4                                                            25 2,3,5,6-Cl.sub.4                                                            26 2,3,4,5,6-Cl.sub.5                                                          27 2-Br                                                                        28 3-Br                                                                        29 4-Br                                                                        30 2,4-Br.sub.2                                                                31 2,5-Br.sub.2                                                                32 2,6-Br.sub.2                                                                33 2,4,6-Br.sub.3                                                              34 2,3,4,5,6-Br.sub.5                                                          35 2-I                                                                         36 3-I                                                                         37 4-I                                                                         38 2,4-I.sub.2                                                                 39 2-Cl, 3-F                                                                   40 2-Cl, 4-F                                                                   41 2-Cl, 5-F                                                                   42 2-Cl, 6-F                                                                   43 2-Cl, 3-Br                                                                  44 2-Cl, 4-Br                                                                  45 2-Cl, 5-Br                                                                  46 2-Cl, 6-Br                                                                  47 2-Br, 3-Cl                                                                  48 2-Br, 4-Cl                                                                  49 2-Br, 5-Cl                                                                  50 2-Br, 3-F                                                                   51 2-Br, 4-F                                                                   52 2-Br, 5-F                                                                   53 2-Br, 6-F                                                                   54 2-F, 3-Cl                                                                   55 2-F, 4-Cl                                                                   56 2-F, 5-Cl                                                                   57 3-Cl, 4-F                                                                   58 3-Cl, 5-F                                                                   59 3-Cl, 4-Br                                                                  60 3-Cl, 5-Br                                                                  61 3-F, 4-Cl                                                                   62 3-F, 4-Br                                                                   63 3-Br, 4-Cl                                                                  64 3-Br, 4-F                                                                   65 2,6-Cl.sub.2, 4-Br                                                          66 2-CH.sub.3                                                                  67 3-CH.sub.3                                                                  68 4-CH.sub.3                                                                  69 2,3-(CH.sub.3).sub.2                                                        70 2,4-(CH.sub.3).sub.2                                                        71 2,5-(CH.sub.3).sub.2                                                        72 2,6-(CH.sub.3).sub.2                                                        73 3,4-(CH.sub.3).sub.2                                                        74 3,5-(CH.sub.3).sub.2                                                        75 2,3,5-(CH.sub.3).sub.3                                                      76 2,3,4-(CH.sub.3).sub.3                                                      77 2,3,6-(CH.sub.3).sub.3                                                      78 2,4,5-(CH.sub.3).sub.3                                                      79 2,4,6-(CH.sub.3).sub.3                                                      80 3,4,5-(CH.sub.3).sub.3                                                      81 2,3,4,6-(CH.sub.3).sub.4                                                    82 2,3,5,6-(CH.sub.3).sub.4                                                    83 2,3,4,5,6-(CH.sub.3).sub.5                                                  84 2-C.sub.2 H.sub.5                                                           85 3-C.sub.2 H.sub.5                                                           86 4-C.sub.2 H.sub.5                                                           87 2,4-(C.sub.2 H.sub.5).sub.2                                                 88 2,6-(C.sub.2 H.sub.5).sub.2                                                 89 3,5-(C.sub.2 H.sub.5).sub.2                                                 90 2,4,6-(C.sub.2 H.sub.5).sub.3                                               91 2-n-C.sub.3 H.sub.7                                                         92 3-n-C.sub.3 H.sub.7                                                         93 4-n-C.sub.3 H.sub.7                                                         94 2-i-C.sub.3 H.sub.7                                                         95 3-i-C.sub.3 H.sub.7                                                         96 4-i-C.sub.3 H.sub.7                                                         97 2,4-(i-C.sub.3 H.sub.7).sub.2                                               98 2,6-(i-C.sub.3 H.sub.7).sub.2                                               99 3,5-(i-C.sub.3 H.sub.7).sub.2                                               100 2,4,6-(i-C.sub.3 H.sub.7).sub.3                                            101 2-s-C.sub.4 H.sub.9                                                        102 3-s-C.sub.4 H.sub.9                                                        103 4-s-C.sub.4 H.sub.9                                                        104 2-t-C.sub.4 H.sub.9                                                        105 3-t-C.sub.4 H.sub.9                                                        106 4-t-C.sub.4 H.sub.9                                                        107 2,3-(t-C.sub.4 H.sub.9).sub.2                                              108 2,4-(t-C.sub.4 H.sub.9).sub.2                                              109 2,5-(t-C.sub.4 H.sub.9).sub.2                                              110 2,6-(t-C.sub.4 H.sub.9).sub.2                                              111 3,4-(t-C.sub.4 H.sub.9).sub.2                                              112 2,4,6-(t-C.sub.4 H.sub.9).sub.3                                            113 4-n-C.sub.9 H.sub.19                                                       114 4-n-C.sub.12 H.sub.25                                                      115 4-n-C.sub.15 H.sub.31                                                      116 4-(1,1,3,3-Tetramethylbutyl)                                               117 4-(2,4,4-Trimethylpropyl)                                                  118 2-t-C.sub.4 H.sub.9, 4-CH.sub.3                                            119 2-t-C.sub.4 H.sub.9, 5-CH.sub.3                                            120 2,6-(t-C.sub.4 H.sub.9).sub.2, 4-CH.sub.3                                  121 2-CH.sub.3, 4-t-C.sub.4 H.sub.9                                            122 2-CH.sub.3, 6-t-C.sub.4 H.sub.9                                            123 2-CH.sub.3, 4-i-C.sub.3 H.sub.7                                            124 2-CH.sub.3, 5-i-C.sub.3 H.sub.7                                            125 3-CH.sub.3, 4-i-C.sub.3 H.sub.7                                            126 2-i-C.sub.3 H.sub.7, 5-CH.sub.3                                            127 2,4-(t-C.sub.4 H.sub.9).sub.2, 6-i-C.sub.3 H.sub.7                         128 2-Allyl                                                                    129 3-Allyl                                                                    130 4-Allyl                                                                    131 2-Allyl, 6-CH.sub.3                                                        132 2-cyclo-C.sub.6 H.sub.11                                                   133 3-cyclo-C.sub.6 H.sub.11                                                   134 4-cyclo-C.sub.6 H.sub.11                                                   135 2,4-(cyclo-C.sub.6 H.sub.11).sub.2, 6-CH.sub.3                             136 2-CH.sub.3, 4-cyclo-C.sub.6 H.sub.11                                       137 2-CH.sub.2 --C.sub.6 H.sub.5                                               138 3-CH.sub.2 --C.sub.6 H.sub.5                                               139 4-CH.sub.2 --C.sub.6 H.sub.5                                               140 2-CH.sub.2 --C.sub.6 H.sub.5, 4-CH.sub.3                                   141 2-CH.sub.3, 4-CH.sub.2 --C.sub.6 H.sub.5                                   142 2-C.sub.6 H.sub.5                                                          143 3-C.sub.6 H.sub.5                                                          144 4-C.sub.6 H.sub.5                                                          145 4-(2-i-C.sub.3 H.sub.7 --C.sub.6 H.sub.4)                                  146 4-C.sub.6 H.sub.5, 2,6-(CH.sub.3).sub.2                                    147 2-Cl, 4-C.sub.6 H.sub.5                                                    148 2-Br, 4-C.sub.6 H.sub.5                                                    149 2-C.sub.6 H.sub.5, 4-Cl                                                    150 2-C.sub.6 H.sub.5, 4-Br                                                    151 2-CH.sub.2 C.sub.6 H.sub.5, 4-Cl                                           152 2-CH.sub.2 C.sub.6 H.sub.5, 4-Br                                           153 2-Cl, 4-CH.sub.2 C.sub.6 H.sub.5                                           154 2-Br, 4-CH.sub.2 C.sub.6 H.sub.5                                           155 2-cyclo-C.sub.6 H.sub.11, 4-Cl                                             156 2-cyclo-C.sub.6 H.sub.11, 4-Br                                             157 2-Cl, 4-cyclo-C.sub.6 H.sub.11                                             158 2-Br, 4-cyclo-C.sub.6 H.sub.11                                             159 2-OCH.sub.3                                                                160 3-OCH.sub.3                                                                161 4-OCH.sub.3                                                                162 2-OC.sub.2 H.sub.5                                                         163 3-O--C.sub.2 H.sub.5                                                       164 4-O--C.sub.2 H.sub.5                                                       165 2-O-n-C.sub.3 H.sub.7                                                      166 3-O-n-C.sub.3 H.sub.7                                                      167 4-O-n-C.sub.3 H.sub.7                                                      168 2-O-i-C.sub.3 H.sub.7                                                      169 3-O-i-C.sub.3 H.sub.7                                                      170 4-O-i-C.sub.3 H.sub.7                                                      171 2-O-n-C.sub.6 H.sub.13                                                     172 3-O-n-C.sub.6 H.sub.13                                                     173 4-O-n-C.sub.6 H.sub.13                                                     174 2-O-n-C.sub.8 H.sub.17                                                     175 3-O-n-C.sub.8 H.sub.17                                                     176 4-O-n-C.sub.8 H.sub.17                                                     177 2-O--CH.sub.2 C.sub.6 H.sub.5                                              178 3-O--CH.sub.2 C.sub.6 H.sub.5                                              179 4-O--CH.sub.2 C.sub.6 H.sub.5                                              180 2-O--(CH.sub.2).sub.3 C.sub.6 H.sub.5                                      181 3-O--(CH.sub.2).sub.3 C.sub.6 H.sub.5                                      182 4-O--(CH.sub.2).sub.3 C.sub.6 H.sub.5                                      183 2,4-(OCH.sub.3).sub.2                                                      184 2-CF.sub.3                                                                 185 3-CF.sub.3                                                                 186 4-CF.sub.3                                                                 187 2-OCF.sub.3                                                                188 3-OCF.sub.3                                                                189 4-OCF.sub.3                                                                190 3-OCH.sub.2 CHF.sub.2                                                      191 2-NO.sub.2                                                                 192 3-NO.sub.2                                                                 193 4-NO.sub.2                                                                 194 2-CN                                                                       195 3-CN                                                                       196 4-CN                                                                       197 2-CH.sub.3, 3-Cl                                                           198 2-CH.sub.3, 4-Cl                                                           199 2-CH.sub.3, 5-Cl                                                           200 2-CH.sub.3, 6-Cl                                                           201 2-CH.sub.3, 3-F                                                            202 2-CH.sub.3, 4-F                                                            203 2-CH.sub.3, 5-F                                                            204 2-CH.sub.3, 6-F                                                            205 2-CH.sub.3, 3-Br                                                           206 2-CH.sub.3, 4-Br                                                           207 2-CH.sub.3, 5-Br                                                           208 2-CH.sub.3, 6-Br                                                           209 2-Cl, 3-CH.sub.3                                                           210 2-Cl, 4-CH.sub.3                                                           211 2-Cl, 5-CH.sub.3                                                           212 2-F, 3-CH.sub.3                                                            213 2-F, 4-CH.sub.3                                                            214 2-F, 5-CH.sub.3                                                            215 2-Br, 3-CH.sub.3                                                           216 2-Br, 4-CH.sub.3                                                           217 2-Br, 5-CH.sub.3                                                           218 3-CH.sub.3, 4-Cl                                                           219 3-CH.sub.3, 5-Cl                                                           220 3-CH.sub.3, 4-F                                                            221 3-CH.sub.3, 5-F                                                            222 3-CH.sub.3, 4-Br                                                           223 3-CH.sub.3, 5-Br                                                           224 3-F, 4-CH.sub.3                                                            225 3-Cl, 4-CH.sub.3                                                           226 3-Br, 4-CH.sub.3                                                           227 2-Cl, 4,5-(CH.sub.3).sub.2                                                 228 2-Br, 4,5-(CH.sub.3).sub.2                                                 229 2-Cl, 3,5-(CH.sub.3).sub.2                                                 230 2-Br, 3,5-(CH.sub.3).sub.2                                                 231 2,6-Cl.sub.2, 4-CH.sub.3                                                   232 2,6-F.sub.2, 4-CH.sub.3                                                    233 2,6-Br.sub.2, 4-CH.sub.3                                                   234 2,4-Br.sub.2, 6-CH.sub.3                                                   235 2,4-F.sub.2, 6-CH.sub.3                                                    236 2,4-Br.sub.2, 6-CH.sub.3                                                   237 2,6-(CH.sub.3).sub.2, 4-F                                                  238 2,6-(CH.sub.3).sub.2, 4-Cl                                                 239 2,6-(CH.sub.3).sub.2, 4-Br                                                 240 3,5-(CH.sub.3).sub.2, 4-F                                                  241 3,5-(CH.sub.3).sub.2, 4-Cl                                                 242 3,5-(CH.sub.3).sub.2, 4-Br                                                 243 2,3,6-(CH.sub.3).sub.3, 4-F                                                244 2,3,6-(CH.sub.3).sub.3, 4-Cl                                               245 2,3,6-(CH.sub.3).sub.3, 4-Br                                               246 2,4-(CH.sub.3).sub.2, 6-F                                                  247 2,4-(CH.sub.3).sub.2, 6-Cl                                                 248 2,4-(CH.sub.3).sub.2, 6-Br                                                 249 2-i-C.sub.3 H.sub.7, 4-Cl, 5-CH.sub.3                                      250 2-Cl, 4-NO.sub.2                                                           251 2-NO.sub.2, 4-Cl                                                           252 2-OCH.sub.3, 5-NO.sub.2                                                    253 2,4-Cl.sub.2, 5-NO.sub.2                                                   254 2,4-Cl.sub.2, 6-NO.sub.2                                                   255 2,6-Cl.sub.2, 4-NO.sub.2                                                   256 2,6-Br.sub.2, 4-NO.sub.2                                                   257 2,6-I.sub.2, 4-NO.sub.2                                                    258 2-CH.sub.3, 5-i-C.sub.3 H.sub.7, 4-Cl                                      259 2-CO.sub.2 CH.sub.3                                                        260 3-CO.sub.2 CH.sub.3                                                        261 4-CO.sub.2 CH.sub.3                                                        262 2-CO.sub.2 (C.sub.2 H.sub.5)                                               263 3-CO.sub.2 (C.sub.2 H.sub.5)                                               264 4-CO.sub.2 (C.sub.2 H.sub.5)                                               265 2-CO.sub.2 (n-C.sub.3 H.sub.7)                                             266 3-CO.sub.2 (n-C.sub.3 H.sub.7)                                             267 4-CO.sub.2 (n-C.sub.3 H.sub.7)                                             268 2-CO.sub.2 (i-C.sub.3 H.sub.7)                                             269 3-CO.sub.2 (i-C.sub.3 H.sub.7)                                             270 4-CO.sub.2 (i-C.sub.3 H.sub.7)                                             271 2-CO.sub.2 (n-C.sub.6 H.sub.13)                                            272 3-CO.sub.2 (n-C.sub.6 H.sub.13)                                            273 4-CO.sub.2 (n-C.sub.6 H.sub.13)                                            274 2-CH.sub.2 --OCH.sub.3                                                     275 3-CH.sub.2 --OCH.sub.3                                                     276 4-CH.sub.2 --OCH.sub.3                                                     277 2-CH.sub.2 O(C.sub.2 H.sub.5)                                              278 3-CH.sub.2 O(C.sub.2 H.sub.5)                                              279 4-CH.sub.2 O(C.sub.2 H.sub.5)                                              280 2-CH.sub.2 O(n-C.sub.3 H.sub.7)                                            281 3-CH.sub.2 O(n-C.sub.3 H.sub.7)                                            282 4-CH.sub.2 O(n-C.sub.3 H.sub.7)                                            283 2-CH.sub.2 O(i-C.sub.3 H.sub.7)                                            284 3-CH.sub.2 O(i-C.sub.3 H.sub.7)                                            285 4-CH.sub.2 O(i-C.sub.3 H.sub.7)                                            286 2-CHO                                                                      287 3-CHO                                                                      288 4-CHO                                                                      289 2-CO--CH.sub.3                                                             290 3-CO--CH.sub.3                                                             291 4-CO--CH.sub.3                                                             292 2-CO--CH.sub.2 --CH.sub.3                                                  293 3-CO--CH.sub.2 --CH.sub.3                                                  294 4-CO--CH.sub.2 --CH.sub.3                                                  295 2-CO--CH.sub.2 --CH.sub.2 --CH.sub.3                                       296 3-CO--CH.sub.2 --CH.sub.2 --CH.sub.3                                       297 4-CO--CH.sub.2 --CH.sub.2 --CH.sub.3                                       298 2-CO--CH(CH.sub.3)--CH.sub.3                                               299 3-CO--CH(CH.sub.3)--CH.sub.3                                               300 4-CO--CH(CH.sub.3)--CH.sub.3                                               301 2-Me-4-CHO                                                                 302 2-Me-4-CH.sub.3 --CO                                                       303 2-Me-4-CO--CH.sub.2 --CH.sub.3                                             304 2-Me-4-CO--CH.sub.2 --CH.sub.2 --CH.sub.3                                  305 2-Me-4-CO--CH(CH.sub.3).sub.2                                              306 2,5-Me.sub.2 -4-CHO                                                        307 2,5-Me.sub.2 -4-CO--CH.sub.3                                               308 2,5-Me.sub.2 -4-CO--CH.sub.2 --CH.sub.3                                    309 2,5-Me.sub.2 -4-CH.sub.2 --CH.sub.2 --CO--CH.sub.3                         310 2,5-Me.sub.2 -4-CO--CH(CH.sub.3).sub.2                                     311 2-Cl-4-CHO                                                                 312 2-Cl-4-CO--CH.sub.3                                                        313 2-Cl-4-CO--CH.sub.2 --CH.sub.3                                             314 2-Cl-4-CO--CH(CH.sub.3).sub.2                                              315 2,5-Cl.sub.2 -4-CHO                                                        316 2,5-Cl.sub.2 -4-CO--CH.sub.3                                               317 2,5-Cl.sub.2 -4-CO--CH.sub.2 --CH.sub.3                                    318 2,5-Cl.sub.2 -4-CO--CH.sub.2 --CH.sub.2 --CH.sub.3                         319 2,5-Cl.sub.2 -4-CO--CH(CH.sub.3).sub.2                                     320 2-C(═NOCH.sub.3)--CH.sub.3                                             321 3-C(═NOCH.sub.3)--CH.sub.3                                             322 4-C(═NOCH.sub.3)--CH.sub.3                                             323 2-C(═NOC.sub.2 H.sub.5)--CH.sub.3                                      324 3-C(═NOC.sub.2 H.sub.5)--CH.sub.3                                      325 4-C(═NOC.sub.2 H.sub.5)--CH.sub.3                                      326 2-C(═NO-n-C.sub.3 H.sub.7)--CH.sub.3                                   327 3-C(═NO-n-C.sub.3 H.sub.7)--CH.sub.3                                   328 4-C(═NO-n-C.sub.3 H.sub.7)--CH.sub.3                                   329 2-C(═NO-i-C.sub.3 H.sub.7)--CH.sub.3                                   330 3-C(═NO-i-C.sub.3 H.sub.7)--CH.sub.3                                   331 4-C(═NO-i-C.sub.3 H.sub.7)--CH.sub.3                                   332 2-C(═NO-Allyl)--CH.sub.3                                               333 3-C(═NO-Allyl)--CH.sub.3                                               334 4-C(═NO-Allyl)--CH.sub.3                                               335 2-C(═NO-trans-Chloroallyl)--CH.sub.3                                   336 3-C(═NO-trans-Chloroallyl)--CH.sub.3                                   337 4-C(═NO-trans-Chloroallyl)--CH.sub.3                                   338 2-C(═NO-Propargyl)--CH.sub.3                                           339 3-C(═NO-Propargyl)--CH.sub.3                                           340 4-C(═NO-Propargyl)--CH.sub.3                                           341 2-C(═NO-n-C.sub.4 H.sub.9)--CH.sub.3                                   342 3-C(═NO-n-C.sub.4 H.sub.9)--CH.sub.3                                   343 4-C(═NO-n-C.sub.4 H.sub.9)--CH.sub.3                                   344 2-C(═NO--CH.sub.2 --C.sub.6 H.sub.5)--CH.sub.3                         345 3-C(═NO--CH.sub.2 --C.sub.6 H.sub.5)--CH.sub.3                         346 4-C(═NO--CH.sub.2 --C.sub.6 H.sub.5)--CH.sub.3                         347 2-CH.sub.3 -4-CH═NOCH.sub.3                                            348 2-CH.sub.3 -4-CH═NOC.sub.2 H.sub.5                                     349 2-CH.sub.3 -4-CH═NO-n-C.sub.3 H.sub.7                                  350 2-CH.sub.3 -4-CH═NO-i-C.sub.3 H.sub.7                                  351 2-CH.sub.3 -4-CH═NO-Allyl                                              352 2-CH.sub.3 -4-CH═NO-(trans-Chloroallyl)                                353 2-CH.sub.3 -4-CH═NO-Propargyl                                          354 2-CH.sub.3 -4-CH═NO-n-C.sub.4 H.sub.9                                  355 2-CH.sub.3 -4-CH═NO--CH.sub.2 --C.sub.6 H.sub.5                        356 2-CH.sub.3 -4-(CH.sub.3 --C═NOCH.sub.3)                                357 2-CH.sub.3 -4-(CH.sub.3 --C═NOC.sub.2 H.sub.5)                         358 2-CH.sub.3 -4-(CH.sub.3 --C═NO-n-C.sub.3 H.sub.7)                      359 2-CH.sub.3 -4-(CH.sub.3 --C═NO-i-C.sub.3 H.sub.7)                      360 2-CH.sub.3 -4-(CH.sub.3 --C═NO-Allyl)                                  361 2-CH.sub.3 -4-(CH.sub.3 --C═NO-trans-Chloroallyl)                      362 2-CH.sub.3 -4-(CH.sub.3 --C═NO-Propargyl)                              363 2-CH.sub.3 -4-(CH.sub.3 --C═NO-n-C.sub.4 H.sub.9)                      364 2-CH.sub.3 -4-(CH.sub.3 --C═NO--CH.sub.2 --C.sub.6 H.sub.5)                     365 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C═NO--CH.sub.3)                       366 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C═NO--C.sub.2                        H.sub.5)                                                               367 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C═NO-n-C.sub.3 H.sub.7)                        368 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C═NO-i-C.sub.3                       H.sub.7                                                                369 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C═NO-Allyl)                           370 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C═NO-trans-Chloroallyl)                        371 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C═NO-Propargyl)                       372 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C═NO-n-C.sub.4                       H.sub.9)                                                               373 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C═NO--CH.sub.2 --C.sub.6                      H.sub.5)                                                               374 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C═NOCH.sub.3)                      375 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C═NOC.sub.2 H.sub.5)                        376 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C═NO-n-C.sub.3                    H.sub.7)                                                               377 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C═NO-i-C.sub.3 H.sub.7)                     378 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C═NO-Allyl)                        379 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C═NO-trans-Chloroal               lyl)                                                                   380 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C═NO-Proparyl)                     381 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C═NO-n-C.sub.4 H.sub.9)                     382 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C═NO--CH.sub.2                    --C.sub.6 H.sub.5)                                                     383 2-C.sub.6 H.sub.5                                                          384 3-C.sub.6 H.sub.5                                                          385 4-C.sub.6 H.sub.5                                                          386 2-(2'-F--C.sub.6 H.sub.4)                                                  387 2-(3'-F--C.sub.6 H.sub.4)                                                  388 2-(4'-F--C.sub.6 H.sub.4)                                                  389 3-(2'-F--C.sub.6 H.sub.4)                                                  390 3-(3'-F--C.sub.6 H.sub.4)                                                  391 3-(4'-F--C.sub.6 H.sub.4)                                                  392 4-(2'-F--C.sub.6 H.sub.4)                                                  393 4-(3'-F--C.sub.6 H.sub.4)                                                  394 4-(4'-F--C.sub.6 H.sub.4)                                                  395 2-(2'-Cl--C.sub.6 H.sub.4)                                                 396 2-(3'-Cl--C.sub.6 H.sub.4)                                                 397 2-(4'-Cl--C.sub.6 H.sub.4)                                                 398 3-(2'-Cl--C.sub.6 H.sub.4)                                                 399 3-(3'-Cl--C.sub.6 H.sub.4)                                                 400 3-(4'-Cl--C.sub.6 H.sub.4)                                                 401 4-(2'-Cl--C.sub.6 H.sub.4)                                                 402 4-(3'-Cl--C.sub.6 H.sub.4)                                                 403 4-(4'-Cl--C.sub.6 H.sub.4)                                                 405 2-(2'-CH.sub.3 --C.sub.6 H.sub.4)                                          406 2-(3'-CH.sub.3 --C.sub.6 H.sub.4)                                          407 2-(4'-CH.sub.3 --C.sub.6 H.sub.4)                                          408 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)                                          409 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)                                          410 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)                                          411 4-(2'-CH.sub.3 --C.sub.6 H.sub.4)                                          412 4-(3'-CH.sub.3 --C.sub.6 H.sub.4)                                          413 4-(4'-CH.sub.3 --C.sub.6 H.sub.4)                                          414 2-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                      415 2-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                      416 2-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                      417 3-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                      418 3-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                      419 3-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                      420 4-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                      421 4-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                      422 4-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                      423 2-(2'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                       424 2-(3'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                       425 2-(4'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                       426 3-(2'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                       427 3-(3'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                       428 3-(4'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                       429 4-(2'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                       430 4-(3'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                       431 4-(4'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                       432 2-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                                 433 2-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                                 434 2-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                                 435 3-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                                 436 3-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                                 437 3-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                                 438 4-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                                 439 4-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                                 440 4-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                                 441 2-(2'-CH.sub.3 O--C.sub.6 H.sub.4)                                         442 2-(3'-CH.sub.3 O--C.sub.6 H.sub.4)                                         443 2-(4'-CH.sub.3 O--C.sub.6 H.sub.4)                                         444 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)                                         445 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)                                         446 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)                                         447 4-(2'-CH.sub.3 O--C.sub.6 H.sub.4)                                         448 4-(3'-CH.sub.3 O--C.sub.6 H.sub.4)                                         449 4-(4'-CH.sub.3 O--C.sub.6 H.sub.4)                                         450 2-(2'-O.sub.2 N--C.sub.6 H.sub.4)                                          451 2-(3'-O.sub.2 N--C.sub.6 H.sub.4)                                          452 2-(4'-O.sub.2 N--C.sub.6 H.sub.4)                                          453 3-(2'-O.sub.2 N--C.sub.6 H.sub.4)                                          454 3-(3'-O.sub.2 N--C.sub.6 H.sub.4)                                          455 3-(4'-O.sub.2 N--C.sub.6 H.sub.4)                                          456 4-(2'-O.sub.2 N--C.sub.6 H.sub.4)                                          457 4-(3'-O.sub.2 N--C.sub.6 H.sub.4)                                          458 4-(4'-O.sub.2 N--C.sub.6 H.sub.4)                                          459 2-(2'-NC--C.sub.6 H.sub.4)                                                 460 2-(3'-NC--C.sub.6 H.sub.4)                                                 461 2-(4'-NC--C.sub.6 H.sub.4)                                                 462 3-(2'-NC--C.sub.6 H.sub.4)                                                 463 3-(3'-NC--C.sub.6 H.sub.4)                                                 464 3-(4'-NC--C.sub.6 H.sub.4)                                                 465 4-(2'-NC--C.sub.6 H.sub.4)                                                 466 4-(3'-NC--C.sub.6 H.sub.4)                                                 467 4-(4'-NC--C.sub.6 H.sub.4)                                                 468 2-(2'-CF.sub.3 --C.sub.6 H.sub.4)                                          469 2-(3'-CF.sub.3 --C.sub.6 H.sub.4)                                          470 2-(4'-CF.sub.3 --C.sub.6 H.sub.4)                                          471 3-(2'-CF.sub.3 --C.sub.6 H.sub.4)                                          472 3-(3'-CF.sub.3 --C.sub.6 H.sub.4)                                          473 3-(4'-CF.sub.3 --C.sub.6 H.sub.4)                                          474 4-(2'-CF.sub.3 --C.sub.6 H.sub.4)                                          475 4-(3'-CF.sub.3 --C.sub.6 H.sub.4)                                          476 4-(4'-CF.sub.3 --C.sub.6 H.sub.4)                                          477 2-O--C.sub.6 H.sub.5                                                       475 3-O--C.sub.6 H.sub.5                                                       476 4-O--C.sub.6 H.sub.5                                                       478 2-O-(2'-F--C.sub.6 H.sub.4)                                                479 2-O-(3'-F--C.sub.6 H.sub.4)                                                480 2-O-(4'-F--C.sub.6 H.sub.4)                                                481 3-O-(2'-F--C.sub.6 H.sub.4)                                                482 3-O-(3'-F--C.sub.6 H.sub.4)                                                483 3-O-(4'-F--C.sub.6 H.sub.4)                                                484 4-O-(2'-F--C.sub.6 H.sub.4)                                                485 4-O-(3'-F--C.sub.6 H.sub.4)                                                486 4-O-(4'-F--C.sub.6 H.sub.4)                                                487 2-O-(2'-Cl--C.sub.6 H.sub.4)                                               488 2-O-(3'-Cl--C.sub.6 H.sub.4)                                               489 2-O-(4'-Cl--C.sub.6 H.sub.4)                                               490 3-O-(2'-Cl--C.sub.6 H.sub.4)                                               491 3-O-(3'-Cl--C.sub.6 H.sub.4)                                               492 3-O-(4'-Cl--C.sub.6 H.sub.4)                                               493 3-O-(4'-Cl--C.sub.6 H.sub.4)                                               494 4-O-(2'-Cl--C.sub.6 H.sub.4)                                               495 4-O-(3'-Cl--C.sub.6 H.sub.4)                                               496 4-O-(4'-Cl--C.sub.6 H.sub.4)                                               497 2-O-(2'-CH.sub.3 --C.sub.6 H.sub.4)                                        498 2-O-(3'-CH.sub.3 --C.sub.6 H.sub.4)                                        499 2-O-(4'-CH.sub.3 --C.sub.6 H.sub.4)                                        500 3-O-(2'-CH.sub.3 --C.sub.6 H.sub.4)                                        501 3-O-(3'-CH.sub.3 --C.sub.6 H.sub.4)                                        502 3-O-(4'-CH.sub.3 --C.sub.6 H.sub.4)                                        503 4-O-(2'-CH.sub.3 --C.sub.6 H.sub.4)                                        504 4-O-(3'-CH.sub.3 --C.sub.6 H.sub.4)                                        505 4-O-(4'-CH.sub.3 --C.sub.6 H.sub.4)                                        506 2-O-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                    507 2-O-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                    508 2-O-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                    509 3-O-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                    510 3-O-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                    511 3-O-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                    512 4-O-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                    513 4-O-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                    514 4-O-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                    515 2-O-(2'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                     516 2-O-(3'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                     517 2-O-(4'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                     518 3-O-(2'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                     519 3-O-(3'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                     520 3-O-(4'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                     521 4-O-(2'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                     522 4-O-(3'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                     523 4-O-(4'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                     524 2-O-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                               525 2-O-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                               526 2-O-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                               527 3-O-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                               528 3-O-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                               529 3-O-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                               530 4-O-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                               531 4-O-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                               532 4-O-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                               533 2-O-(2'-CH.sub.3 O--C.sub.6 H.sub.4)                                       534 2-O-(3'-CH.sub.3 O--C.sub.6 H.sub.4)                                       535 2-O-(4'-CH.sub.3 O--C.sub.6 H.sub.4)                                       536 3-O-(2'-CH.sub.3 O--C.sub.6 H.sub.4)                                       537 3-O-(3'-CH.sub.3 O--C.sub.6 H.sub.4)                                       538 3-O-(4'-CH.sub.3 O--C.sub.6 H.sub.4)                                       539 4-O-(2'-CH.sub.3 O--C.sub.6 H.sub.4)                                       540 4-O-(3'-CH.sub.3 O--C.sub.6 H.sub.4)                                       541 4-O-(4'-CH.sub.3 O--C.sub.6 H.sub.4)                                       542 2-O-(2'-O.sub.2 N--C.sub.6 H.sub.4)                                        543 2-O-(3'-O.sub.2 N--C.sub.6 H.sub.4)                                        544 2-O-(4'-O.sub.2 N--C.sub.6 H.sub.4)                                        545 3-O-(2'-O.sub.2 N--C.sub.6 H.sub.4)                                        546 3-O-(3'-O.sub.2 N--C.sub.6 H.sub.4)                                        547 3-O-(4'-O.sub.2 N--C.sub.6 H.sub.4)                                        548 4-O-(2'-O.sub.2 N--C.sub.6 H.sub.4)                                        549 4-O-(3'-O.sub.2 N--C.sub.6 H.sub.4)                                        550 4-O-(4'-O.sub.2 N--C.sub.6 H.sub.4)                                        551 2-O-(2'-NC--C.sub.6 H.sub.4)                                               552 2-O-(3'-NC--C.sub.6 H.sub.4)                                               553 2-O-(4'-NC--C.sub.6 H.sub.4)                                               554 3-O-(2'-NC--C.sub.6 H.sub.4)                                               555 3-O-(3'-NC--C.sub.6 H.sub.4)                                               556 3-O-(4'-NC--C.sub.6 H.sub.4)                                               557 4-O-(2'-NC--C.sub.6 H.sub.4)                                               558 4-O-(3'-NC--C.sub.6 H.sub.4)                                               559 4-O-(4'-NC--C.sub.6 H.sub.4)                                               560 2-O-(2'-CF.sub.3 --C.sub.6 H.sub.4)                                        561 2-O-(3'-CF.sub.3 --C.sub.6 H.sub.4)                                        562 2-O-(4'-CF.sub.3 --C.sub.6 H.sub.4)                                        563 3-O-(2'-CF.sub.3 --C.sub.6 H.sub.4)                                        564 3-O-(3'-CF.sub.3 --C.sub.6 H.sub.4)                                        565 3-O-(4'-CF.sub.3 --C.sub.6 H.sub.4)                                        566 4-O-(2'-CF.sub.3 --C.sub.6 H.sub.4)                                        567 4-O-(3'-CF.sub.3 --C.sub.6 H.sub.4)                                        568 4-O-(4'-CF.sub.3 --C.sub.6 H.sub.4)                                        569 2-Pyridinyl-2'                                                             570 2-Pyridinyl-3'                                                             571 2-Pyridinyl-4'                                                             572 3-Pyridinyl-2'                                                             573 3-Pyridinyl-3'                                                             574 3-Pyridinyl-4'                                                             575 4-Pyridinyl-2'                                                             576 4-Pyridinyl-3'                                                             577 4-Pyridinyl-4'                                                             578 2-Pyrimidinyl-2'                                                           579 2-Pyrimidinyl-3'                                                           580 2-Pyrimidinyl-4'                                                           581 3-Pyrimidinyl-2'                                                           582 3-Pyrimidinyl-3'                                                           583 3-Pyrimidinyl-4'                                                           584 4-Pyrimidinyl-2'                                                           585 4-Pyrimidinyl-3'                                                           586 4-Pyrimidinyl-4'                                                           587 2-Pyrazolyl-1'                                                             588 2-Pyrazolyl-3'                                                             589 2-Pyrazolyl-4'                                                             590 3-Pyrazolyl-1'                                                             591 3-Pyrazolyl-3'                                                             592 3-Pyrazolyl-4'                                                             593 4-Pyrazolyl-1'                                                             594 4-Pyrazolyl-3'                                                             595 4-Pyrazolyl-4'                                                             596 2-Isoxazolyl-3'                                                            597 2-Isoxazolyl-4'                                                            598 2-Isoxazolyl-5'                                                            599 3-Isoxazolyl-3'                                                            600 3-Isoxazolyl-4'                                                            601 3-Isoxazolyl-5'                                                            602 4-Isoxazolyl-3'                                                            603 4-Isoxazolyl-4'                                                            604 4-Isoxazolyl-5'                                                            605 2-Isothiazolyl-3'                                                          606 2-Isothiazolyl-4'                                                          607 2-Isothiazolyl-5'                                                          608 3-Isothiazolyl-3'                                                          609 3-Isothiazolyl-4'                                                          610 3-Isothiazolyl-5'                                                          611 4-Isothiazolyl-3'                                                          612 4-Isothiazolyl-4'                                                          613 4-Isothiazolyl-5'                                                          614 2-Imidazolyl-1'                                                            615 2-Imidazolyl-2'                                                            616 2-Imidazolyl-4'                                                            617 3-Imidazolyl-1'                                                            618 3-Imidazolyl-2'                                                            619 3-Imidazolyl-4'                                                            620 4-Imidazolyl-1'                                                            621 4-Imidazolyl-2'                                                            622 4-Imidazolyl-4'                                                            623 2-Oxazolyl-2'                                                              624 2-Oxazolyl-4'                                                              625 2-Oxazolyl-5'                                                              626 3-Oxazolyl-2'                                                              627 3-Oxazolyl-4'                                                              628 3-Oxazolyl-5'                                                              629 4-Oxazolyl-2'                                                              630 4-Oxazolyl-4'                                                              631 4-Oxazolyl-5'                                                              632 2-Thiazolyl-2'                                                             633 2-Thiazolyl-4'                                                             634 2-Thiazolyl-5'                                                             635 3-Thiazolyl-2'                                                             636 3-Thiazolyl-4'                                                             637 3-Thiazolyl-5'                                                             638 4-Thiazolyl-2'                                                             639 4-Thiazolyl-4'                                                             640 4-Thiazolyl-5'                                                           ______________________________________                                    

                  TABLE 37                                                         ______________________________________                                         1  STR257##                                                                      I: R.sup.1 = H, Z = C.sub.2 H.sub.5                                                               IX: R.sup.1 = CH.sub.3, Z = NH(CH.sub.3)                    II: R.sup.1 = CH.sub.3, Z = C.sub.2 H.sub.5 X: R.sup.1 = C.sub.2                                  H.sub.5, Z = NH(CH.sub.3)                                   III: R.sup.1 = C.sub.2 H.sub.5, Z = C.sub.2 H.sub.5 XI: R.sup.1 =                                 Allyl, Z = NH(CH.sub.3)                                     IV: R.sup.1 = Allyl, Z = C.sub.2 H.sub.5 XII: R.sup.1 = Propargyl, Z =                            NH(CH.sub.3)                                                V: R.sup.1 = Propargyl, Z = C.sub.2 H.sub.5 XIII: R.sup.1 = CH.sub.2                              --OCH.sub.3,                                                VI: R.sup.1 = CH.sub.2 --OCH.sub.3, Z = C.sub.2 H.sub.5 Z = NH(CH.sub.3)       VII: R.sup.1 = CO--C.sub.2 H.sub.5, Z = C.sub.2 H.sub.5 XIV: R.sup.1 =                            CO--C.sub.2 H.sub.5, Z = NH(CH.sub.3)                       VIII: R.sup.1 = H, Z = NH(CH.sub.3)                                             -                                                                           No.       B                                                                    ______________________________________                                          1        Pyrrolyl-3                                                              2 N--CH.sub.3 -Pyrrolyl-3                                                      3 N--C.sub.6 H.sub.5 -Pyrrolyl-3                                               4 N--(4'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrrolyl-3                                5 N--(3'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrrolyl-3                                6 N--(2'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrrolyl-3                                7 N--(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrrolyl-3                               8 N--(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrrolyl-3                               9 N--(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrrolyl-3                               10 N--(4'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrrolyl-3                               11 N--(3'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrrolyl-3                               12 N--(2'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrrolyl-3                               13 N--(4'-CN--C.sub.6 H.sub.4)-Pyrrolyl-3                                      14 N--(3'-CN--C.sub.6 H.sub.4)-Pyrrolyl-3                                      15 N--(2'-CN--C.sub.6 H.sub.4)-Pyrrolyl-3                                      16 N--(4'-Cl--C.sub.6 H.sub.4)-Pyrrolyl-3                                      17 N--(3'-Cl--C.sub.6 H.sub.4)-Pyrrolyl-3                                      18 N--(2'-Cl--C.sub.6 H.sub.4)-Pyrrolyl-3                                      19 Pyrrolyl-2                                                                  20 N--CH.sub.3 -Pyrrolyl-2                                                     21 N--C.sub.6 H.sub.5 -Pyrrolyl-2                                              22 N--(4'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrrolyl-2                               23 N--(3'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrrolyl-2                               24 N--(2'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrrolyl-2                               25 N--(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrrolyl-2                              26 N--(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrrolyl-2                              27 N--(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrrolyl-2                              28 N--(4'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrrolyl-2                               29 N--(3'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrrolyl-2                               30 N--(2'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrrolyl-2                               31 N--(4'-CN--C.sub.6 H.sub.4)-Pyrrolyl-2                                      32 N--(3'-CN--C.sub.6 H.sub.4)-Pyrrolyl-2                                      33 N--(2'-CN--C.sub.6 H.sub.4)-Pyrrolyl-2                                      34 N--(4 -Cl--C.sub.6 H.sub.4)-Pyrrolyl-2                                      35 N--(3'-Cl--C.sub.6 H.sub.4)-Pyrrolyl-2                                      36 N--(2'-Cl--C.sub.6 H.sub.4)-Pyrrolyl-2                                      37 Furyl-2                                                                     38 5-CH.sub.3 -Furyl-2                                                         39 5-C.sub.6 H.sub.5 -Furyl-2                                                  40 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Furyl-2                                   41 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Furyl-2                                   42 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Furyl-2                                   43 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Furyl-2                                  44 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Furyl-2                                  45 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Furyl-2                                  46 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Furyl-2                                   47 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Furyl-2                                   48 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Furyl-2                                   49 5-(4'-CN--C.sub.6 H.sub.4)-Furyl-2                                          50 5-(3'-CN--C.sub.6 H.sub.4)-Furyl-2                                          51 5-(2'-CN--C.sub.6 H.sub.4)-Furyl-2                                          52 5-(4'-Cl--C.sub.6 H.sub.4)-Furyl-2                                          53 5-(3'-Cl--C.sub.6 H.sub.4)-Furyl-2                                          54 5-(2'-Cl--C.sub.6 H.sub.4)-Furyl-2                                          55 4-CH.sub.3 -Furyl-2                                                         56 4-C.sub.6 H.sub.5 -Furyl-2                                                  57 4-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Furyl-2                                   58 4-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Furyl-2                                   59 4-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Furyl-2                                   60 4-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Furyl-2                                  61 4-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Furyl-2                                  62 4-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Furyl-2                                  63 4-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Furyl-2                                   64 4-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Furyl-2                                   65 4-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Furyl-2                                   66 4-(4'-CN--C.sub.6 H.sub.4)-Furyl-2                                          67 4-(3'-CN--C.sub.6 H.sub.4)-Furyl-2                                          68 4-(2'-CN--C.sub.6 H.sub.4)-Furyl-2                                          69 4-(4'-Cl--C.sub.6 H.sub.4)-Furyl-2                                          70 4-(3'-Cl--C.sub.6 H.sub.4)-Furyl-2                                          71 4-(2'-Cl--C.sub.6 H.sub.4)-Furyl-2                                          72 Thienyl-2                                                                   73 5-CH.sub.3 -Thienyl-2                                                       74 5-C.sub.6 H.sub.5 -Thienyl-2                                                75 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-2                                 76 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-2                                 77 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-2                                 78 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-2                                79 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-2                                80 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-2                                81 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-2                                 82 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-2                                 83 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-2                                 84 5-(4'-CN--C.sub.6 H.sub.4)-Thienyl-2                                        85 5-(3'-CN--C.sub.6 H.sub.4)-Thienyl-2                                        86 5-(2'-CN--C.sub.6 H.sub.4)-Thienyl-2                                        87 5-(4'-Cl--C.sub.6 H.sub.4)-Thienyl-2                                        88 5-(3'-Cl--C.sub.6 H.sub.4)-Thienyl-2                                        89 5-(2'-Cl--C.sub.6 H.sub.4)-Thienyl-2                                        90 4-CH.sub.3 -Thienyl-2                                                       91 4-C.sub.6 H.sub.5 -Thienyl-2                                                92 4-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-2                                 93 4-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-2                                 94 4-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-2                                 95 4-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-2                                96 4-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-2                                97 4-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-2                                98 4-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-2                                 99 4-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-2                                100 4-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-2                                101 4-(4'-CN--C.sub.6 H.sub.4)-Thienyl-2                                       102 4-(3'-CN--C.sub.6 H.sub.4)-Thienyl-2                                       103 4-(2 1-CN--C.sub.6 H.sub.4)-Thienyl-2                                      104 4-(4'-Cl--C.sub.6 H.sub.4)-Thienyl-2                                       105 4-(3'-Cl--C.sub.6 H.sub.4)-Thienyl-2                                       106 4-(2'-Cl--C.sub.6 H.sub.4)-Thienyl-2                                       107 Thienyl-3                                                                  108 5-CH.sub.3 -Thienyl-3                                                      109 5-C.sub.6 H.sub.5 -Thienyl-3                                               110 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-3                                111 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-3                                112 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-3                                113 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-3                               114 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-3                               115 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-3                               116 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-3                                117 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-3                                118 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-3                                119 5-(4'-CN--C.sub.6 H.sub.4)-Thienyl-3                                       120 5-(3'-CN--C.sub.6 H.sub.4)-Thienyl-3                                       121 5-(2'-CN--C.sub.6 H.sub.4)-Thienyl-3                                       122 5-(4'-Cl--C.sub.6 H.sub.4)-Thienyl-3                                       123 5-(3'-Cl--C.sub.6 H.sub.4)-Thienyl-3                                       124 5-(2'-Cl--C.sub.6 H.sub.4)-Thienyl-3                                       125 Pyrazolyl-4                                                                126 N--CH.sub.3 -Pyrazolyl-4                                                   127 N--C.sub.6 H.sub.5 -Pyrazolyl-4                                            128 N--(4'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrazolyl-4                             129 N--(3'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrazolyl-4                             130 N--(2'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrazolyl-4                             131 N--(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrazolyl-4                            132 N--(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrazolyl-4                            133 N--(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrazolyl-4                            134 N--(4'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrazolyl-4                             135 N--(3'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrazolyl-4                             136 N--(2'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrazolyl-4                             137 N--(4'-CN--C.sub.6 H.sub.4)-Pyrazolyl-4                                    138 N--(3'-CN--C.sub.6 H.sub.4)-Pyrazolyl-4                                    139 N--(2'-CN--C.sub.6 H.sub.4)-Pyrazolyl-4                                    140 N--(4'-Cl--C.sub.6 H.sub.4)-Pyrazolyl-4                                    141 N--(3'-Cl--C.sub.6 H.sub.4)-Pyrazolyl-4                                    142 N--(2'-Cl--C.sub.6 H.sub.4)-Pyrazolyl-4                                    143 3-CH.sub.3 --N-Methylpyrazolyl-4                                           144 3-C.sub.6 H.sub.5 --N-Methylpyrazolyl-4                                    145 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)--N-Methylpyrazolyl-4                     146 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)--N-Methylpyrazolyl-4                     147 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)--N-Methylpyrazolyl-4                     148 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)--N-Methylpyrazolyl-4                    149 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)--N-Methylpyrazolyl-4                    150 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)--N-Methylpyrazolyl-4                    151 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)--N-Methylpyrazolyl-4                     152 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)--N-Methylpyrazolyl-4                     153 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)--N-Methylpyrazolyl-4                     154 3-(4'-CN--C.sub.6 H.sub.4)--N-Methylpyrazolyl-4                            155 3-(3'-CN--C.sub.6 H.sub.4)--N-Methylpyrazolyl-4                            156 3-(2'-CN--C.sub.6 H.sub.4)--N-Methylpyrazolyl-4                            157 3-(4'-Cl--C.sub.6 H.sub.4)--N-Methylpyrazolyl-4                            158 3-(3'-Cl--C.sub.6 H.sub.4)--N-Methylpyrazolyl-4                            159 3-(2'-Cl--C.sub.6 H.sub.4)--N-Methylpyrazolyl-4                            160 Isoxazolyl-5                                                               161 3-CH.sub.3 -Isoxazolyl-5                                                   162 3-C.sub.6 H.sub.5 -Isoxazolyl-5                                            163 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Isoxazolyl-5                             164 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Isoxazolyl-5                             165 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Isoxazolyl-5                             166 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Isoxazolyl-5                            167 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Isoxazolyl-5                            168 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Isoxazolyl-5                            169 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Isoxazolyl-5                             170 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Isoxazolyl-5                             171 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Isoxazolyl-5                             172 3-(4'-CN--C.sub.6 H.sub.4)-Isoxazolyl-5                                    173 3-(3'-CN--C.sub.6 H.sub.4)-Isoxazolyl-5                                    174 3-(2'-CN--C.sub.6 H.sub.4)-Isoxazolyl-5                                    175 3-(4'-Cl--C.sub.6 H.sub.4)-Isoxazolyl-5                                    176 3-(3'-Cl--C.sub.6 H.sub.4)-Isoxazolyl-5                                    177 3-(2'-Cl--C.sub.6 H.sub.4)-Isoxazolyl-5                                    178 4-Chloroisoxazolyl-5                                                       179 3-CH.sub.3 -4-Chloroisoxazolyl-5                                           180 3-C.sub.6 H.sub.5 -4-Chloroisoxazolyl-5                                    181 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                     182 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                     183 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                     184 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                    185 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                    186 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                    187 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                     188 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                     189 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                     190 3-(4'-CN--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                            191 3-(3'-CN--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                            192 3-(2'-CN--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                            193 3-(4'-Cl--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                            194 3-(3'-Cl--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                            195 3-(2'-Cl--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                            196 Isoxazolyl-3                                                               197 5-CH.sub.3 -Isoxazolyl-3                                                   198 5-C.sub.6 H.sub.5 -Isoxazolyl-3                                            199 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Isoxazolyl-3                             200 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Isoxazolyl-3                             201 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Isoxazolyl-3                             202 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Isoxazolyl-3                            203 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Isoxazolyl-3                            204 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Isoxazolyl-3                            205 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Isoxazolyl-3                             206 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Isoxazolyl-3                             207 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Isoxazolyl-3                             208 5-(4'-CN--C.sub.6 H.sub.4)-Isoxazolyl-3                                    209 5-(3'-CN--C.sub.6 H.sub.4)-Isoxazolyl-3                                    210 5-(2'-CN--C.sub.6 H.sub.4)-Isoxazolyl-3                                    211 5-(4'-Cl--C.sub.6 H.sub.4)-Isoxazolyl-3                                    212 5-(3'-Cl--C.sub.6 H.sub.4)-Isoxazolyl-3                                    213 5-(2'-Cl--C.sub.6 H.sub.4)-Isoxazolyl-3                                    214 Isothiazolyl-5                                                             215 3-CH.sub.3 -Isothiazolyl-5                                                 216 3-C.sub.6 H.sub.5 -Isothiazolyl-5                                          217 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Isothiazolyl-5                           218 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Isothiazolyl-5                           219 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Isothiazolyl-5                           220 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Isothiazolyl-5                          221 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Isothiazolyl-5                          222 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Isothiazolyl-5                          223 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Isothiazolyl-5                           224 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Isothiazolyl-5                           225 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Isothiazolyl-5                           226 3-(4'-CN--C.sub.6 H.sub.4)-Isothiazolyl-5                                  227 3-(3'-CN--C.sub.6 H.sub.4)-Isothiazolyl-5                                  228 3-(2'-CN--C.sub.6 H.sub.4)-Isothiazolyl-5                                  229 3-(4'-Cl--C.sub.6 H.sub.4)-Isothiazolyl-5                                  230 3-(3'-Cl--C.sub.6 H.sub.4)-Isothiazolyl-5                                  231 3-(2'-Cl--C.sub.6 H.sub.4)-Isothiazolyl-5                                  232 Oxazolyl-4                                                                 233 3-CH.sub.3 -Oxazolyl-4                                                     234 3-C.sub.6 H.sub.5 -Oxazolyl-4                                              235 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Oxazolyl-4                               236 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Oxazolyl-4                               237 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Oxazolyl-4                               238 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Oxazolyl-4                              239 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Oxazolyl-4                              240 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Oxazolyl-4                              241 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Oxazolyl-4                               242 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Oxazolyl-4                               243 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Oxazolyl-4                               244 3-(4'-CN--C.sub.6 H.sub.4)-Oxazolyl-4                                      245 3-(3'-CN--C.sub.6 H.sub.4)-Oxazolyl-4                                      246 3-(2'-CN--C.sub.6 H.sub.4)-Oxazolyl-4                                      247 3-(4'-Cl--C.sub.6 H.sub.4)-Oxazolyl-4                                      248 3-(3'-Cl--C.sub.6 H.sub.4)-Oxazolyl-4                                      249 3-(2'-Cl--C.sub.6 H.sub.4)-Oxazolyl-4                                      250 Thiazolyl-4                                                                251 2-CH.sub.3 -Thiazolyl-4                                                    252 2-C.sub.6 H.sub.5 -Thiazolyl-4                                             253 2-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Thiazolyl-4                              254 2-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Thiazolyl-4                              255 2-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Thiazolyl-4                              256 2-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Thiazolyl-4                             267 2-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Thiazolyl-4                             258 2-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Thiazolyl-4                             259 2-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Thiazolyl-4                              260 2-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Thiazolyl-4                              261 2-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Thiazolyl-4                              262 2-(4'-CN--C.sub.6 H.sub.4)-Thiazolyl-4                                     263 2-(3'-CN--C.sub.6 H.sub.4)-Thiazolyl-4                                     264 2-(2'-CN--C.sub.6 H.sub.4)-Thiazolyl-4                                     265 2-(4'-Cl--C.sub.6 H.sub.4)-Thiazolyl-4                                     266 2-(3'-Cl--C.sub.6 H.sub.4)-Thiazolyl-4                                     267 2-(2'-Cl--C.sub.6 H.sub.4)-Thiazolyl-4                                     268 N--CH.sub.3 -1,2,4-Triazolyl-5                                             269 3-CH.sub.3 --N--CH.sub.3 -1,2,4-Triazolyl-5                                270 3-C.sub.6 H.sub.5 --N--CH.sub.3 -1,2,4-Triazolyl-5                         271 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5                   272 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triaz               olyl-5                                                                 273 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5                   274 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Tria               zolyl-5                                                                275 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5                  276 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Tria               zolyl-5                                                                277 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5                   278 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triaz               olyl-5                                                                 279 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5                   280 3-(4'-CN--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5        281 3-(3'-CN--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5                 282 3-(2'-CN--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5                 283 3-(4'-Cl--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5                 284 3-(3'-Cl--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5                 285 3-(2'-Cl--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5                 286 1,3,4-Oxadiazolyl-2                                                        287 5-CH.sub.3 -1,3,4-Oxadiazolyl-2                                            288 5-C.sub.6 H.sub.5 -1,3,4-Oxadiazolyl-2                                     289 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                      290 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                      291 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                      292 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                     293 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                     294 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                     295 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                      296 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                      297 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                      298 5-(4'-CN--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                             299 5-(3'-CN--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                             300 5-(2'-CN--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                             301 5-(4'-Cl--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                             302 5-(3'-Cl--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                             303 5-(2'-Cl--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                             304 1,2,4-Oxadiazolyl-3                                                        305 5-CH.sub.3 -1,2,4-Oxadiazolyl-3                                            306 5-C.sub.6 H.sub.5 -1,2,4-Oxadiazolyl-3                                     307 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                      308 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                      309 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                      310 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                     311 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                     312 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                     313 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                      314 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                      315 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                      316 5-(4'-CN--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                             317 5-(3'-CN--C.sub.6 H.sub.4)-1,2, 4-Oxadiazolyl-3                            318 5-(2'-CN--C.sub.6 H.sub.4)-1,2, 4-Oxadiazolyl-3                            319 5-(4'-Cl--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                             320 5-(3'-Cl--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                             321 5-(2'-Cl--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                             322 1,2,4-Oxadiazolyl-5                                                        323 3-CH.sub.3 -1,2,4-Oxadiazolyl-5                                            324 3-C.sub.6 H.sub.5 -1,2,4-Oxadiazolyl-5                                     325 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                      326 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                      327 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                      328 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                     329 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                     330 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                     331 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                      332 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                      333 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                      334 3-(4'-CN--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                             335 3-(3'-CN--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                             336 3-(2'-CN--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                             337 3-(4'-Cl--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                             338 3-(3'-Cl--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                             339 3-(2'-Cl--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                             340 1,2,4-Thiadiazolyl-3                                                       341 5-CH.sub.3 -1,2,4-Thiadiazolyl-3                                           342 5-C.sub.6 H.sub.5 -1,2,4-Thiadiazolyl-3                                    343 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                     344 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                     345 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                     346 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                    347 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                    348 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                    349 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                     350 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                     351 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                     352 5-(4'-CN--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                            353 5-(3'-CN--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                            354 5-(2'-CN--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                            355 5-(4'-Cl--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                            356 5-(3'-Cl--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                            357 5-(2'-Cl--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                            358 1,3,4-Thiadiazolyl-2                                                       359 5-CH.sub.3 -1,3,4-Thiadiazolyl-2                                           360 5-C.sub.6 H.sub.5 -1,3,4-Thiadiazolyl-2                                    361 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                     362 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                     363 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                     364 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                    365 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                    366 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                    367 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                     368 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                     369 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                     370 5-(4'-CN--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                            371 5-(3'-CN--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                            372 5-(2'-CN--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                            373 5-(4,-Cl--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                            374 5-(3'-Cl--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                            375 5-(2'-Cl--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                            376 Pyridinyl-2                                                                377 Pyridinyl-4                                                                378 Pyridazinyl-3                                                              379 Pyridazinyl-4                                                              380 pyridazinyl-2                                                              381 Pyrimidinyl-4                                                              382 Pyrimidinyl-5                                                              383 Pyrimidinyl-2                                                            ______________________________________                                    

                                      TABLE 38                                     __________________________________________________________________________     Selected physical data of some compounds                                                                IR (cm.sup.-1)                                            or .sup.1 H-NMR                                                              No. Compound (ppm) mp (° C.)                                          __________________________________________________________________________       1                                                                                                            2   128 8##                                       - 2                                                                                                         3   144 9##                                       - 3                                                                                                         4  STR260##                                       - 4                                                                                                         5  STR261##                                       - 5                                                                                                         6    80 2##                                       - 6                                                                                                         5    75 3##                                       - 7                                                                                                         7   188 4##                                       - 8                                                                                                         8   115 5##                                       - 9                                                                                                         9    76 6##                                       - 10                                                                                                        0    96 7##                                       - 11                                                                                                        1  3.3(s, 3H); 2.25(2, 3H)                     __________________________________________________________________________

                  TABLE 58                                                         ______________________________________                                         Selected physical data of some compounds                                       2  STR269##                                                                       -                                IR                                              (cm.sup.-1)                                                                    or .sup.1 H-                                                                   NMR mp                                                                      No. X.sub.m R.sup.1 (ppm) (° C.)                                      ______________________________________                                          1  2-CH.sub.3          H             120                                         2 2-CH.sub.3 CH.sub.3 oil                                                      3 2-CH.sub.3 C.sub.2 H.sub.5 oil                                               4 2-CH.sub.3 Allyl oil                                                         5 2-CH.sub.3 Propargyl oil                                                     6 2-CH.sub.3 CH.sub.2 --OCH.sub.3 oil                                          7 2,5-(CH.sub.3).sub.2 H 170                                                   8 2,5-(CH.sub.3).sub.2 CH.sub.3 oil                                            9 2,5-(CH.sub.3).sub.2 C.sub.2 H.sub.5 oil                                    10 2,5-(CH.sub.3).sub.2 Allyl oil                                              11 2,5-(CH.sub.3).sub.2 Propargyl oil                                          12 2,5-(CH.sub.3).sub.2 CH.sub.2 --OCH.sub.3 oil                               13 2-CH.sub.3 -4-C(CH.sub.3)═N--OCH.sub.3 H 125                            14 2-CH.sub.3 -4-C(CH.sub.3)═N--OCH.sub.3 CH.sub.3 oil                     15 2-CH.sub.3 -4-C(CH.sub.3)═N--OCH.sub.3 C.sub.2 H.sub.5 oil                                                   16 2-CH.sub.3 -4-C(CH.sub.3)═N-                                           -OCH.sub.3 Allyl  87                       17 2-CH.sub.3 -4-C(CH.sub.3)═N--OCH.sub.3 Propargyl oil                    18 2-CH.sub.3 -4-C(CH.sub.3)═N--OCH.sub.3 CH.sub.2 --OCH.sub.3 oil                                              19 2,5-(CH.sub.3).sub.2 -4-C(CH.sub                                           .3)═N--O-Allyl H  85                   20 2,5-(CH.sub.3).sub.2 -4-C(CH.sub.3)═N--O-Allyl CH.sub.3 oil                                                  21 2,5-(CH.sub.3).sub.2 -4-C(CH.sub                                           .3)═N--O-Allyl C.sub.2 H.sub.5                                             oil                                        22 2,5-(CH.sub.3).sub.2 -4-C(CH.sub.3)═N--O-Allyl Allyl  87                                                     23 2,5-(CH.sub.3).sub.2 -4-C(CH.sub                                           .3)═N--O-Allyl Propargyl oil                                                24 2,5-(CH.sub.3).sub.2 -4-C(CH.sub                                           .3)═N--O-Allyl CH.sub.2                                                    --OCH.sub.3 oil                          ______________________________________                                    

                  TABLE 59                                                         ______________________________________                                         Selected physical data of some compounds                                       3  STR270##                                                                       -                          IR (cm.sup.-1)                                        or .sup.1 H-NMR                                                             No. X.sub.m R.sup.1 (ppm) mp (° C.)                                   ______________________________________                                         1       4-CH.sub.3                                                                              H                118                                            2 4-CH.sub.3 CH.sub.3 oil                                                      3 4-CH.sub.3 C.sub.2 H.sub.5 oil                                               4 4-CH.sub.3 Allyl oil                                                         5 4-CH.sub.3 Propargyl oil                                                     6 4-CH.sub.3 CH.sub.2 --OCH.sub.3 oil                                          7 3,5-Cl.sub.2 H 160                                                           8 3,5-Cl.sub.2 CH.sub.3 oil                                                    9 3,5-Cl.sub.2 C.sub.2 H.sub.5 oil                                             10  3,5-Cl.sub.2 Allyl  85                                                     11  3,5-Cl.sub.2 Propargyl oil                                                 12  3,5-Cl.sub.2 CH.sub.2 --OCH.sub.3 oil                                    ______________________________________                                    

                  TABLE 39                                                         ______________________________________                                         4  STR271##                                                                      No.     X      R.sup.1 Z      A                                              ______________________________________                                          1    H      H         CH.sub.3                                                                              --CH.sub.2 O--                                      2 H H CH.sub.3 --CH.sub.2 O--N═C(CH.sub.3)--                               3 H H CH.sub.3 --CH═CH--                                                   4 H H NH.sub.2 --CH.sub.2 O--                                                  5 H H NH.sub.2 --CH.sub.2 O--N═C(CH.sub.3)--                               6 H H NH.sub.2 --CH═CH--                                                   7 H H N(CH.sub.3).sub.2 --CH.sub.2 O--                                         8 H H N(CH.sub.3).sub.2 --CH.sub.2 O--N═C(CH.sub.3)--                      9 H H N(CH.sub.3).sub.2 --CH═CH--                                         10 H H CCl.sub.3 --CH.sub.2 O--                                                11 H H CCl.sub.3 --CH.sub.2 O--N═C(CH.sub.3)--                             12 H H CCl.sub.3 --CH═CH--                                                 13 H H CF.sub.3 --CH.sub.2 O--                                                 14 H H CF.sub.3 --CH.sub.2 O--N═C(CH.sub.3)--                              15 H H CF.sub.3 --CH═CH--                                                  16 H Propargyl CH.sub.3 --CH.sub.2 O--                                         17 H Propargyl CH.sub.3 --CH.sub.2 O--N═C(CH.sub.3)--                      18 H Propargyl CH.sub.3 --CH═CH--                                          19 H Propargyl NH.sub.2 --CH.sub.2 O--                                         20 H Propargyl NH.sub.2 --CH.sub.2 O--N═C(CH.sub.3)--                      21 H Propargyl NH.sub.2 --CH═CH--                                          22 H Propargyl N(CH.sub.3).sub.2 --CH.sub.2 O--                                23 H Propargyl N(CH.sub.3).sub.2 --CH.sub.2 O--N--═C(CH.sub.3)--                                        24 H Propargyl N(CH.sub.3).sub.2 --CH═C                                   H--                                                25 H Propargyl CCl.sub.3 --CH.sub.2 O--                                        26 H Propargyl CCl.sub.3 --CH.sub.2 O--N═C(CH.sub.3)--                     27 H Propargyl CCl.sub.3 --CH═CH--                                         28 H Propargyl CF.sub.3 --CH.sub.2 O--                                         29 H Propargyl CF.sub.3 --CH.sub.2 O--N═C(CH.sub.3)--                      30 H Propargyl CF.sub.3 --CH═CH--                                          31 CH.sub.3 H CH.sub.3 --CH.sub.2 O--                                          32 CH.sub.3 H CH.sub.3 --CH.sub.2 O--N═C(CH.sub.3)--                       33 CH.sub.3 H CH.sub.3 --CH═CH--                                           34 CH.sub.3 H NH.sub.2 --CH.sub.2 O--                                          35 CH.sub.3 H NH.sub.2 --CH.sub.2 O--N═C(CH.sub.3)--                       36 CH.sub.3 H NH.sub.2 --CH═CH--                                           37 CH.sub.3 H N(CH.sub.3).sub.2 --CH.sub.2 O--                                 38 CH.sub.3 H N(CH.sub.3).sub.2 --CH.sub.2 O--N═C(CH.sub.3)--                                           39 CH.sub.3 H N(CH.sub.3).sub.2 --CH═CH                                   --                                                 40 CH.sub.3 H CCl.sub.3 --CH.sub.2 O--                                         41 CH.sub.3 H CCl.sub.3 --CH.sub.2 O--N═C(CH.sub.3)--                      42 CH.sub.3 H CCl.sub.3 --CH═CH--                                          43 CH.sub.3 H CF.sub.3 --CH.sub.2 O--                                          44 CH.sub.3 H CF.sub.3 --CH.sub.2 O--N═C(CH.sub.3)--                       45 CH.sub.3 H CF.sub.3 --CH═CH--                                           46 CH.sub.3 Propargyl CH.sub.3 --CH.sub.2 O--                                  47 CH.sub.3 Propargyl CH.sub.3 --CH.sub.2 O--N═C(CH.sub.3)--                                            48 CH.sub.3 Propargyl CH.sub.3 --CH═CH-                                   -                                                  49 CH.sub.3 Propargyl NH.sub.2 --CH.sub.2 O--                                  50 CH.sub.3 Propargyl NH.sub.2 --CH.sub.2 O--N═C(CH.sub.3)--                                            51 CH.sub.3 Propargyl NH.sub.2 --CH═CH-                                   -                                                  52 CH.sub.3 Propargyl N(CH.sub.3).sub.2 --CH.sub.2 O--                         53 CH.sub.3 Propargyl N(CH.sub.3).sub.2 --CH.sub.2 O--N═C(CH.sub.3)-                                   -                                                  54 CH.sub.3 Propargyl N(CH.sub.3).sub.2 --CH═CH--                          55 CH.sub.3 Propargyl CCl.sub.3 --CH.sub.2 O--                                 56 CH.sub.3 Propargyl CCl.sub.3 --CH.sub.2 O--N═C(CH.sub.3)--                                           57 CH.sub.3 Propargyl CCl.sub.3 --CH═CH                                   --                                                 58 CH.sub.3 Propargyl CF.sub.3 --CH.sub.2 O--                                  59 CH.sub.3 Propargyl CF.sub.3 --CH.sub.2 O--N═C(CH.sub.3)--                                            60 CH.sub.3 Propargyl CF.sub.3 --CH═CH-                                   -                                                  61 Cl H CH.sub.3 --CH.sub.2 O--                                                62 Cl H CH.sub.3 --CH.sub.2 O--N═C(CH.sub.3)--                             63 Cl H CH.sub.3 --CH═CH--                                                 64 Cl H NH.sub.2 --CH.sub.2 O--                                                65 Cl H NH.sub.2 --CH.sub.2 O--N═C(CH.sub.3)--                             66 Cl H NH.sub.2 --CH═CH--                                                 67 Cl H N(CH.sub.3).sub.2 --CH.sub.2 O--                                       68 Cl H N(CH.sub.3).sub.2 --CH.sub.2 O--N═C(CH.sub.3)--                    69 Cl H N(CH.sub.3).sub.2 --CH═CH--                                        70 Cl H CCl.sub.3 --CH.sub.2 O--                                               71 Cl H CCl.sub.3 --CH.sub.2 O--N═C(CH.sub.3)--                            72 Cl H CCl.sub.3 --CH═CH--                                                73 Cl H CF.sub.3 --CH.sub.2 O--                                                74 Cl H CF.sub.3 --CH.sub.2 O--N═C(CH.sub.3)--                             75 Cl H CF.sub.3 --CH═CH--                                                 76 Cl Propargyl CH.sub.3 --CH.sub.2 O--                                        77 Cl Propargyl CH.sub.3 --CH.sub.2 O--N═C(CH.sub.3)--                     78 Cl Propargyl CH.sub.3 --CH═CH--                                         79 Cl Propargyl NH.sub.2 --CH.sub.2 O--                                        80 Cl Propargyl NH.sub.2 --CH.sub.2 O--N═C(CH.sub.3)--                     81 Cl Propargyl NH.sub.2 --CH═CH--                                         82 Cl Propargyl N(CH.sub.3).sub.2 --CH.sub.2 O--                               83 Cl Propargyl N(CH.sub.3).sub.2 --CH.sub.2 O--N═C(CH.sub.3)--                                         84 Cl Propargyl N(CH.sub.3).sub.2 --CH═                                   CH--                                               85 Cl Propargyl CCl.sub.3 --CH.sub.2 O--                                       86 Cl Propargyl CCl.sub.3 --CH.sub.2 O--N═C(CH.sub.3)--                    87 Cl Propargyl CCl.sub.3 --CH═CH--                                        88 Cl Propargyl CF.sub.3 --CH.sub.2 O--                                        89 Cl Propargyl CF.sub.3 --CH.sub.2 O--N═C(CH.sub.3)--                     90 Cl Propargyl CF.sub.3 --CH═CH--                                       ______________________________________                                    

                  TABLE 40                                                         ______________________________________                                         5  STR272##                                                                      I: R.sup.1 = H, Z = C.sub.2 H.sub.5                                                               VIII: R.sup.1 = H, Z = NH(CH.sub.3)                         II: R.sup.1 = CH.sub.3, Z = C.sub.2 H.sub.5 IX: R.sup.1 = CH.sub.3, Z =                           NH(CH.sub.3)                                                III: R.sup.1 = C.sub.2 H.sub.5, Z = C.sub.2 H.sub.5 X: R.sup.1 =                                  C.sub.2 H.sub.5, Z = NH(CH.sub.3)                           IV: R.sup.1 = Allyl, Z = C.sub.2 H.sub.5 XI: R.sup.1 = Allyl, Z =                                 NH(CH.sub.3)                                                V: R.sup.1 = Propargyl, Z = C.sub.2 H.sub.5 XII: R.sup.1 = Propargyl, Z                           = NH(CH.sub.3)                                              VI: R.sup.1 = CH.sub.2 --OCH.sub.3, Z = C.sub.2 H.sub.5 XIII: R.sup.1 =                           CH.sub.2 --OCH.sub.3,                                       VII: R.sup.1 = CO--C.sub.2 H.sub.5, Z = C.sub.2 H.sub.5 Z = NH(CH.sub.3)        XIV: R.sup.1 = CO--C.sub.2 H.sub.5, Z = NH(CH.sub.3)                           -                                                                           No.         B                                                                  ______________________________________                                         1           2-Pyridyl                                                            2 3-Trifluoromethyl-2-pyridyl                                                  3 5-Trifluoromethyl-2-pyridyl                                                  4 3,5-Bis-(trifluoromethyl)-2-pyridyl                                          5 3,5-Dichloro-2-pyridyl                                                       6 3-Chloroo-5-trifluoromethyl-2-pyridyl                                        7 3,5-Dichloro-2-pyridyl                                                       8 2-Chloroo-4-trifluoromethylphenyl                                            9 2-Benzothiazolyl                                                             10  5-Chloroo-1-methyl-2-benzimidazolyl                                        11  2-Benzoxazolyl                                                             12  1-Methyl-5-trifluoromethylimidazo-                                          [5,4-a]-pyridin-2-yl                                                          13  5-Chloroo-2-pyrimidinyl                                                    14  4-Methyl-5-phenyl-2-thiazolin-2-yl                                         15  4-Methyl-5-phenyl-2-oxazolin-2-yl                                          16  7-Trifluoromethyl-4-quinolinyl                                           ______________________________________                                    

Example 16

Methyl N-[2-(3",4"-dichlorophenyl-1-'1-methyliminooxymethyl-4')-6-methylphenyl]-carbamate (Table 47, No. 2)

a) 2-(Methanesulfonyloxymethyl)-6-methyl-nitrobenzene

At 10-15° C., 27 g (0.23 mol) of methanesulfonyl chloride dissolved in 20 ml of CH₂ Cl₂ is dripped into a mixture of 34 g (0.2 mol) of 3-methyl-2-nitrobenzyl alcohol and 27 g (0.27 mol) of triethylamine in 100 ml of CH₂ Cl₂. The reaction mixture is stirred for 1 hour at room temperature and is then extracted with water. The organic phase is dried over MgSO₄ and evaporated down. There is obtained as residue 48 g of the title compound as a yellow oil, containing about 10% of the corresponding benzyl chloride as impurity. The crude product is used for the next reaction without any further purification.

¹ H-NMR(COCl₃ ; δ in ppm): 7.3-7.6 (m, 3H, phenyl); 5.3 (S, 2H, OCH₂); 3.0 (S, 3H, CH₃ --SO3); 2.4 (S, 3H, CH₃)

b) 2-(3",4"-Dichlorophenyl-1'-1-methyl-iminooxymethyl-4')-6-methyl-nitrobenzene

At room temperature, 1.8 g (75 mmol) of sodium hydride is added in portions to a solution of 13 g (64 mmol) of 3,4-dichloroacetophenonoxime in 100 ml of dimethylformamide. Upon conclusion of gas evolution, a solution of 16 g (65 mmol) of the mesylate from Example 1a in 30 ml of dimethylformamide is dripped in at 25-30° C., and the mixture is then stirred for 1 hour at room temperature. The reaction mixture is diluted with water and the aqueous phase is then extracted three times with methyl tert-butyl ether. The combined organic phases are washed with water, dried over MGSO₄ and evaporated down. The residue crystallizes and is stirred with methanol. The mother liquor is purified by column chromatography with mixtures of cyclohexane and ethyl acetate. There is obtained a total of 20.4 g (58 mmol=90%) of the title compound as pale yellow crystals.

¹ H-NMR(CDCl₃ ; δ in ppm): 7.7 (S, broad, 1H, phenyl); 7.2-7.6 (m, 5H, phenyl); 5.3 (S, 2H, OCH₂); 2.4 (S, 3H, CH₃); 2.2 (S, 3H, CH₃)

c) 2-(3',4'-Dichlorophenyl-1'-methyl-iminooxymethyl-4')-6-methyl-aniline

At 20-30° C., 53 g of 21.8% strength Na₂ [Fe(CO)₄ ] solution (1 kg of the solution contains 633 g of water, 218 g of Na₂ [Fe(CO)₄ ], 108 g of Na₂ CO₃ and 41 g of NaOH) is added dropwise to 19 g (52.8 mmol) of the nitrobenzene from Example 16b in 150 ml of methanol. The brown suspension is stirred for 2 hours at room temperature, and the reaction mixture is then diluted with methylene chloride and the mixture is suction filtered using kieselguhr. The residue is again washed with CH₂ Cl₂ and the combined extracts are extracted with water, dried over MgSO₄ and evaporated down. The brown residue is purified by column chromatography with mixtures of cyclohexane and ethyl acetate. There is obtained 14.3 g (44.3 mmol=82%) of the title compound as a beige solid.

¹ H-NMR(CDCl₃ ; δ in ppm): 7.7 (S, 1H, phenyl); 7.5 (m, 2H, phenyl); 7.1 (t, broad, 2H, phenyl); 6.7 (t, 1H, I=8 Hz, phenyl); 5.2 (S, 2H, OCH₂); 4.15 (S, 2H, NH₂ ; 2.2 (S, 3H, CH₃)

d) Methyl N-[2-(3",4"-dichlorophenyl-1'-methyl-iminooxymethyl-4'-6-methylphenyl]-carbamate (Table 47, No. 2)

At 20-30° C., 4.8 g (50 mmol) of methyl chloroformate and subsequently 4.8 g (60 mmol) of pyridine are dripped into a solution of 14.3 g (44 mmol) of the aniline from Example 1c in 150 ml of CH₂ Cl₂. The mixture is stirred overnight at room temperature and is then extracted with dilute hydrochloric acid and water. The reaction mixture is suction filtered using silica gel, dried over MgSO₄ and evaporated down. The residue crystallizes and is stirred with cyclohexane. There is obtained 13.8 g (36 mmol=82%) of the title compound as a colorless solid (mp=109° C.).

¹ H-NMR(CDCl₃ ; δ in ppm): 7.8 (S, 1H, phenyl); 7.6 (S, broad, 1H, NH); 7.4 (S, 2H, phenyl); 7.2 (m, 3H, phenyl); 5.2 (S, 2H, OCH₂); 3.8 (S, 3H, OCH₃); 2.3 (S, 3H, CH₃); 2.2 (S, 3H, CH₃)

Example 17

Methyl N-[2-(3",4"-dichlorophenyl-1'-methyl-iminooxymethyl-4')-6-methylphenyl]-N-propargyl-carbamate (Table 47, No. 13)

At 25-30° C., 0.15 g (6.3 mmol) of sodium hydride is added in portions to a solution of 1.9 g (5 mmol) of the carbamate from Example 16d in 20 ml of dimethylformamide. When no more gas evolves, 0.75 g (6.3 mmol) of propargyl bromide is added and the whole is stirred overnight at room temperature. The reaction mixture is diluted with water and the aqueous phase is extracted three times with methyl tert-butyl ether. The combined organic phases are extracted with water, dried over MgSO₄ and evaporated down. There is obtained 1.4 g (3.3 mmol=67%) of the title compound as a yellow oil.

¹ H-NMR (CDCl₃ ; δ in ppm): 7.75 (S, broad, 1H, phenyl); 7.2-7.6 (m, 5H, phenyl); 5.2 (dd, 2H, I=12 Hz, OCH₂); 4.4 (dd, broad, I=16 Hz, NCH₂); (S, 3H, OCH₃); 2.3 (S, 3H, CH₃); 2.25 (S, broad, 1H, C.tbd.CH); 2.2 (S, 3H, CH₃); the ¹ H-NMR spectrum also contains signals of about 20% of the amide rotamer.

The compounds described in the following tables may be prepared analogously.

                  TABLE 41                                                         ______________________________________                                         1  STR273##                                                                      I: R.sup.1 = H, X = CH.sub.3                                                                      VIII: R.sup.1 = H, X = Cl                                   II: R.sup.1 = CH.sub.3, X = CH.sub.3 IX: R.sup.1 = CH.sub.3, X = Cl                                III: R.sup.1 = C.sub.2 H.sub.5, X = CH.sub.3 X:                               R.sup.1 = C.sub.2 H.sub.5, X = Cl                           IV: R.sup.1 = Allyl, X = CH.sub.3 XI: R.sup.1 = Allyl, X = Cl                  V: R.sup.1 = Propargyl, X = CH.sub.3 XII: R.sup.1 = Propargyl, X = Cl                              VI: R.sup.1 = CH.sub.2 --OCH.sub.3, X = CH.sub.3                              XIII: R.sup.1 = CH.sub.2 --OCH.sub.3, X = Cl                                    VII: R.sup.1 = CO.sub.2 CH.sub.3, X = CH.sub.3 XIV:                           R.sup.1 = CO.sub.2 CH.sub.3, X = Cl                          -                                                                           Compound I from Table 41 has for instance the following                          structural formula:                                                             -                                                                           2  STR274##                                                                      No.         T.sub.m                                                          ______________________________________                                         1         H                                                                      2 2-F                                                                          3 3-F                                                                          4 4-F                                                                          5 2,4-F.sub.2                                                                  6 2,4,6-F.sub.3                                                                7 2,3,4,5,6-F.sub.5                                                            8 2,3-F.sub.2                                                                  9 2-Cl                                                                         10 3-Cl                                                                        11 4-Cl                                                                        12 2,3-Cl.sub.2                                                                13 2,4-Cl.sub.2                                                                14 2,5-Cl.sub.2                                                                15 2,6-Cl.sub.2                                                                16 3,4-Cl.sub.2                                                                17 3,5-Cl.sub.2                                                                18 2,3,4-Cl.sub.3                                                              19 2,3,5-Cl.sub.3                                                              20 2,3,6-Cl.sub.3                                                              21 2,4,5-Cl.sub.3                                                              22 2,4,6-Cl.sub.3                                                              23 3,4,5-Cl.sub.3                                                              24 2,3,4,6-Cl.sub.4                                                            25 2,3,5,6-Cl.sub.4                                                            26 2,3,4,5,6-Cl.sub.5                                                          27 2-Br                                                                        28 3-Br                                                                        29 4-Br                                                                        30 2,4-Br.sub.2                                                                31 2,5-Br.sub.2                                                                32 2,6-Br.sub.2                                                                33 2,4,6-Br.sub.3                                                              34 2,3,4,5,6-Br.sub.5                                                          35 2-I                                                                         36 3-I                                                                         37 4-I                                                                         38 2,4-I.sub.2                                                                 39 2-Cl, 3-F                                                                   40 2-Cl, 4-F                                                                   41 2-Cl, 5-F                                                                   42 2-Cl, 6-F                                                                   43 2-Cl, 3-Br                                                                  44 2-Cl, 4-Br                                                                  45 2-Cl, 5-Br                                                                  46 2-Cl, 6-Br                                                                  47 2-Br, 3-Cl                                                                  48 2-Br, 4-Cl                                                                  49 2-Br, 5-Cl                                                                  50 2-Br, 3-F                                                                   51 2-Br, 4-F                                                                   52 2-Br, 5-F                                                                   53 2-Br, 6-F                                                                   54 2-F, 3-Cl                                                                   55 2-F, 4-Cl                                                                   56 2-F, 5-Cl                                                                   57 3-Cl, 4-F                                                                   58 3-Cl, 5-F                                                                   59 3-Cl, 4-Br                                                                  60 3-Cl, 5-Br                                                                  61 3-F, 4-Cl                                                                   62 3-F, 4-Br                                                                   63 3-Br, 4-Cl                                                                  64 3-Br, 4-F                                                                   65 2,6-Cl.sub.2, 4-Br                                                          66 2-CH.sub.3                                                                  67 3-CH.sub.3                                                                  68 4-CH.sub.3                                                                  69 2,3-(CH.sub.3).sub.2                                                        70 2,4-(CH.sub.3).sub.2                                                        71 2,5-(CH.sub.3).sub.2                                                        72 2,6-(CH.sub.3).sub.2                                                        73 3,4-(CH.sub.3).sub.2                                                        74 3,5-(CH.sub.3).sub.2                                                        75 2,3,5-(CH.sub.3).sub.3                                                      76 2,3,4-(CH.sub.3).sub.3                                                      77 2,3,6-(CH.sub.3).sub.3                                                      78 2,4,5-(CH.sub.3).sub.3                                                      79 2,4,6-(CH.sub.3).sub.3                                                      80 3,4,5-(CH.sub.3).sub.3                                                      81 2,3,4,6-(CH.sub.3).sub.4                                                    82 2,3,5,6-(CH.sub.3).sub.4                                                    83 2,3,4,5,6-(CH.sub.3).sub.5                                                  84 2-C.sub.2 H.sub.5                                                           85 3-C.sub.2 H.sub.5                                                           86 4-C.sub.2 H.sub.5                                                           87 2,4-(C.sub.2 H.sub.5).sub.2                                                 88 2,6-(C.sub.2 H.sub.5).sub.2                                                 89 3,5-(C.sub.2 H.sub.5).sub.2                                                 90 2,4,6-(C.sub.2 H.sub.5).sub.3                                               91 2-n-C.sub.3 H.sub.7                                                         92 3-n-C.sub.3 H.sub.7                                                         93 4-n-C.sub.3 H.sub.7                                                         94 2-i-C.sub.3 H.sub.7                                                         95 3-i-C.sub.3 H.sub.7                                                         96 4-i-C.sub.3 H.sub.7                                                         97 2,4-(i-C.sub.3 H.sub.7).sub.2                                               98 2,6-(i-C.sub.3 H.sub.7).sub.2                                               99 3,5-(i-C.sub.3 H.sub.7).sub.2                                               100 2,4,6-(i-C.sub.3 H.sub.7).sub.3                                            101 2-s-C.sub.4 H.sub.9                                                        102 3-s-C.sub.4 H.sub.9                                                        103 4-s-C.sub.4 H.sub.9                                                        104 2-t-C.sub.4 H.sub.9                                                        105 3-t-C.sub.4 H.sub.9                                                        106 4-t-C.sub.4 H.sub.9                                                        107 2,3-(t-C.sub.4 H.sub.9).sub.2                                              108 2,4-(t-C.sub.4 H.sub.9).sub.2                                              109 2,5-(t-C.sub.4 H.sub.9).sub.2                                              110 2,6-(t-C.sub.4 H.sub.9).sub.2                                              111 3,4-(t-C.sub.4 H.sub.9).sub.2                                              112 2,4,6-(t-C.sub.4 H.sub.9).sub.3                                            113 4-n-C.sub.9 H.sub.19                                                       114 4-n-C.sub.12 H.sub.25                                                      115 4-n-C.sub.15 H.sub.31                                                      116 4-(1,1,3,3-Tetramethylbutyl)                                               117 4-(2,4,4-Trimethylpropyl)                                                  118 2-t-C.sub.4 H.sub.9, 4-CH.sub.3                                            119 2-t-C.sub.4 H.sub.9, 5-CH.sub.3                                            120 2,6-(t-C.sub.4 H.sub.9).sub.2, 4-CH.sub.3                                  121 2-CH.sub.3, 4-t-C.sub.4 H.sub.9                                            122 2-CH.sub.3, 6-t-C.sub.4 H.sub.9                                            123 2-CH.sub.3, 4-i-C.sub.3 H.sub.7                                            124 2-CH.sub.3, 5-i-C.sub.3 H.sub.7                                            125 3-CH.sub.3, 4-i-C.sub.3 H.sub.7                                            126 2-i-C.sub.3 H.sub.7, 5-CH.sub.3                                            127 2,4-(t-C.sub.4 H.sub.9).sub.2, 6-i-C.sub.3 H.sub.7                         128 2-Allyl                                                                    129 3-Allyl                                                                    130 4-Allyl                                                                    131 2-Allyl, 6-CH.sub.3                                                        132 2-cyclo-C.sub.6 H.sub.11                                                   133 3-cyclo-C.sub.6 H.sub.11                                                   134 4-cyclo-C.sub.6 H.sub.11                                                   135 2,4-(cyclo-C.sub.6 H.sub.11).sub.2, 6-CH.sub.3                             136 2-CH.sub.3, 4-cyclo-C.sub.6 H.sub.11                                       137 2-CH.sub.2 --C.sub.6 H.sub.5                                               138 3-CH.sub.2 --C.sub.6 H.sub.5                                               139 4-CH.sub.2 --C.sub.6 H.sub.5                                               140 2-CH.sub.2 --C.sub.6 H.sub.5, 4-CH.sub.3                                   141 2-CH.sub.3, 4-CH.sub.2 --C.sub.6 H.sub.5                                   142 2-C.sub.6 H.sub.5                                                          143 3-C.sub.6 H.sub.5                                                          144 4-C.sub.6 H.sub.5                                                          145 4-(2-i-C.sub.3 H.sub.7 --C.sub.6 H.sub.4)                                  146 4-C.sub.6 H.sub.5, 2,6-(CH.sub.3).sub.2                                    147 2-Cl, 4-C.sub.6 H.sub.5                                                    148 2-Br, 4-C.sub.6 H.sub.5                                                    149 2-C.sub.6 H.sub.5, 4-Cl                                                    150 2-C.sub.6 H.sub.5, 4-Br                                                    151 2-CH.sub.2 C.sub.6 H.sub.5, 4-Cl                                           152 2-CH.sub.2 C.sub.6 H.sub.5, 4-Br                                           153 2-Cl, 4-CH.sub.2 C.sub.6 H.sub.5                                           154 2-Br, 4-CH.sub.2 C.sub.6 H.sub.5                                           155 2-cyclo-C.sub.6 H.sub.11, 4-Cl                                             156 2-cyclo-C.sub.6 H.sub.11, 4-Br                                             157 2-Cl, 4-cyclo-C.sub.6 H.sub.11                                             158 2-Br, 4-cyclo-C.sub.6 H.sub.11                                             159 2-OCH.sub.3                                                                160 3-OCH.sub.3                                                                161 4-OCH.sub.3                                                                162 2-OC.sub.2 H.sub.5                                                         163 3-O--C.sub.2 H.sub.5                                                       164 4-O--C.sub.2 H.sub.5                                                       165 2-O-n-C.sub.3 H.sub.7                                                      166 3-O-n-C.sub.3 H.sub.7                                                      167 4-O-n-C.sub.3 H.sub.7                                                      168 2-O-i-C.sub.3 H.sub.7                                                      169 3-O-i-C.sub.3 H.sub.7                                                      170 4-O-i-C.sub.3 H.sub.7                                                      171 2-O-n-C.sub.6 H.sub.13                                                     172 3-O-n-C.sub.6 H.sub.13                                                     173 4-O-n-C.sub.6 H.sub.13                                                     174 2-O-n-C.sub.8 H.sub.17                                                     175 3-O-n-C.sub.8 H.sub.17                                                     176 4-O-n-C.sub.8 H.sub.17                                                     177 2-O--CH.sub.2 C.sub.6 H.sub.5                                              178 3-O--CH.sub.2 C.sub.6 H.sub.5                                              179 4-O--CH.sub.2 C.sub.6 H.sub.5                                              180 2-O--(CH.sub.2).sub.3 C.sub.6 H.sub.5                                      181 3-O--(CH.sub.2).sub.3 C.sub.6 H.sub.5                                      182 4-O--(CH.sub.2).sub.3 C.sub.6 H.sub.5                                      183 2,4-(OCH.sub.3).sub.2                                                      184 2-CF.sub.3                                                                 185 3-CF.sub.3                                                                 186 4-CF.sub.3                                                                 187 2-OCF.sub.3                                                                188 3-OCF.sub.3                                                                189 4-OCF.sub.3                                                                190 3-OCH.sub.2 CHF.sub.2                                                      191 2-NO.sub.2                                                                 192 3-NO.sub.2                                                                 193 4-NO.sub.2                                                                 194 2-CN                                                                       195 3-CN                                                                       196 4-CN                                                                       197 2-CH.sub.3, 3-Cl                                                           198 2-CH.sub.3, 4-Cl                                                           199 2-CH.sub.3, 5-Cl                                                           200 2-CH.sub.3, 6-Cl                                                           201 2-CH.sub.3, 3-F                                                            202 2-CH.sub.3, 4-F                                                            203 2-CH.sub.3, 5-F                                                            204 2-CH.sub.3, 6-F                                                            205 2-CH.sub.3, 3-Br                                                           206 2-CH.sub.3, 4-Br                                                           207 2-CH.sub.3, 5-Br                                                           208 2-CH.sub.3, 6-Br                                                           209 2-Cl, 3-CH.sub.3                                                           210 2-Cl, 4-CH.sub.3                                                           211 2-Cl, 5-CH.sub.3                                                           212 2-F, 3-CH.sub.3                                                            213 2-F, 4-CH.sub.3                                                            214 2-F, 5-CH.sub.3                                                            215 2-Br, 3-CH.sub.3                                                           216 2-Br, 4-CH.sub.3                                                           217 2-Br, 5-CH.sub.3                                                           218 3-CH.sub.3, 4-Cl                                                           219 3-CH.sub.3, 5-Cl                                                           220 3-CH.sub.3, 4-F                                                            221 3-CH.sub.3, 5-F                                                            222 3-CH.sub.3, 4-Br                                                           223 3-CH.sub.3, 5-Br                                                           224 3-F, 4-CH.sub.3                                                            225 3-Cl, 4-CH.sub.3                                                           226 3-Br, 4-CH.sub.3                                                           227 2-Cl, 4,5-(CH.sub.3).sub.2                                                 228 2-Br, 4,5-(CH.sub.3).sub.2                                                 229 2-Cl, 3,5-(CH.sub.3).sub.2                                                 230 2-Br, 3,5-(CH.sub.3).sub.2                                                 231 2,6-Cl.sub.2, 4-CH.sub.3                                                   232 2,6-F.sub.2, 4-CH.sub.3                                                    233 2,6-Br.sub.2, 4-CH.sub.3                                                   234 2,4-Br.sub.2, 6-CH.sub.3                                                   235 2,4-F.sub.2, 6-CH.sub.3                                                    236 2,4-Br.sub.2, 6-CH.sub.3                                                   237 2,6-(CH.sub.3).sub.2, 4-F                                                  238 2,6-(CH.sub.3).sub.2, 4-Cl                                                 239 2,6-(CH.sub.3).sub.2, 4-Br                                                 240 3,5-(CH.sub.3).sub.2, 4-F                                                  241 3,5-(CH.sub.3).sub.2, 4-Cl                                                 242 3,5-(CH.sub.3).sub.2, 4-Br                                                 243 2,3,6-(CH.sub.3).sub.3, 4-F                                                244 2,3,6-(CH.sub.3).sub.3, 4-Cl                                               245 2,3,6-(CH.sub.3).sub.3, 4-Br                                               246 2,4-(CH.sub.3).sub.2, 6-F                                                  247 2,4-(CH.sub.3).sub.2, 6-Cl                                                 248 2,4-(CH.sub.3).sub.2, 6-Br                                                 249 2-i-C.sub.3 H.sub.7, 4-Cl, 5-CH.sub.3                                      250 2-Cl, 4-NO.sub.2                                                           251 2-NO.sub.2, 4-Cl                                                           252 2-OCH.sub.3, 5-NO.sub.2                                                    253 2,4-Cl.sub.2, 5-NO.sub.2                                                   254 2,4-Cl.sub.2, 6-NO.sub.2                                                   255 2,6-Cl.sub.2, 4-NO.sub.2                                                   256 2,6-Br.sub.2, 4-NO.sub.2                                                   257 2,6-I.sub.2, 4-NO.sub.2                                                    258 2-CH.sub.3, 5-i-C.sub.3 H.sub.7, 4-Cl                                      259 2-CO.sub.2 CH.sub.3                                                        260 3-CO.sub.2 CH.sub.3                                                        261 4-CO.sub.2 CH.sub.3                                                        262 2-CO.sub.2 (C.sub.2 H.sub.5)                                               263 3-CO.sub.2 (C.sub.2 H.sub.5)                                               264 4-CO.sub.2 (C.sub.2 H.sub.5)                                               265 2-CO.sub.2 (n-C.sub.3 H.sub.7)                                             266 3-CO.sub.2 (n-C.sub.3 H.sub.7)                                             267 4-CO.sub.2 (n-C.sub.3 H.sub.7)                                             268 2-CO.sub.2 (i-C.sub.3 H.sub.7)                                             269 3-CO.sub.2 (i-C.sub.3 H.sub.7)                                             270 4-CO.sub.2 (i-C.sub.3 H.sub.7)                                             271 2-CO.sub.2 (n-C.sub.6 H.sub.13)                                            272 3-CO.sub.2 (n-C.sub.6 H.sub.13)                                            273 4-CO.sub.2 (n-C.sub.6 H.sub.13)                                            274 2-CH.sub.2 --OCH.sub.3                                                     275 3-CH.sub.2 --OCH.sub.3                                                     276 4-CH.sub.2 --OCH.sub.3                                                     277 2-CH.sub.2 O(C.sub.2 H.sub.5)                                              278 3-CH.sub.2 O(C.sub.2 H.sub.5)                                              279 4-CH.sub.2 O(C.sub.2 H.sub.5)                                              280 2-CH.sub.2 O(n-C.sub.3 H.sub.7)                                            281 3-CH.sub.2 O(n-C.sub.3 H.sub.7)                                            282 4-CH.sub.2 O(n-C.sub.3 H.sub.7)                                            283 2-CH.sub.2 O(i-C.sub.3 H.sub.7)                                            284 3-CH.sub.2 O(i-C.sub.3 H.sub.7)                                            285 4-CH.sub.2 O(i-C.sub.3 H.sub.7)                                            286 2-CHO                                                                      287 3-CHO                                                                      288 4-CHO                                                                      289 2-CO--CH.sub.3                                                             290 3-CO--CH.sub.3                                                             291 4-CO--CH.sub.3                                                             292 2-CO--CH.sub.2 --CH.sub.3                                                  293 3-CO--CH.sub.2 --CH.sub.3                                                  294 4-CO--CH.sub.2 --CH.sub.3                                                  295 2-CO--CH.sub.2 --CH.sub.2 --CH.sub.3                                       296 3-CO--CH.sub.2 --CH.sub.2 --CH.sub.3                                       297 4-CO--CH.sub.2 --CH.sub.2 --CH.sub.3                                       298 2-CO--CH(CH.sub.3)--CH.sub.3                                               299 3-CO--CH(CH.sub.3)--CH.sub.3                                               300 4-CO--CH(CH.sub.3)--CH.sub.3                                               301 2-Me-4-CHO                                                                 302 2-Me-4-CH.sub.3 --CO                                                       303 2-Me-4-CH.sub.3 --CH.sub.2 --CO                                            304 2-Me-4-CH.sub.3 --CH.sub.2 --CH.sub.2 --CO                                 305 2-Me-4-CH.sub.3 --CH(CH.sub.3)--CO                                         306 2,5-Me.sub.2 -4-CHO                                                        307 2,5-Me.sub.2 -4-CH.sub.3 --CO                                              308 2,5-Me.sub.2 -4-CH.sub.3 --CH.sub.2 --CO                                   309 2,5-Me.sub.2 -4-CH.sub.3 --CH.sub.2 --CH.sub.2 --CO                        310 2,5-Me.sub.2 -4-CH.sub.3 --CH(CH.sub.3)--CO                                311 2-Cl-4-CHO                                                                 312 2-Cl-4-CH.sub.3 --CO                                                       313 2-Cl-4-CH.sub.3 --CH.sub.2 --CO                                            314 2-Cl-4-CH.sub.3 --CH(CH.sub.3)--CO                                         315 2,5-Cl.sub.2 -4-CHO                                                        316 2,5-Cl.sub.2 -4-CH.sub.3 --CO                                              317 2,5-Cl.sub.2 -4-CH.sub.3 --CH.sub.2 --CO                                   318 2,5-Cl.sub.2 -4-CH.sub.3 --CH.sub.2 --CH.sub.2 --CO                        319 2,5-Cl.sub.2 -4-CH.sub.3 --CH(CH.sub.3)--CO                                320 2-C(═NOCH.sub.3)--CH.sub.3                                             321 3-C(═NOCH.sub.3)--CH.sub.3                                             322 4-C(═NOCH.sub.3)--CH.sub.3                                             323 2-C(═NOC.sub.2 H.sub.5)--CH.sub.3                                      324 3-C(═NOC.sub.2 H.sub.5)--CH.sub.3                                      325 4-C(═NOC.sub.2 H.sub.5)--CH.sub.3                                      326 2-C(═NO-n-C.sub.3 H.sub.7)--CH.sub.3                                   327 3-C(═NO-n-C.sub.3 H.sub.7)--CH.sub.3                                   328 4-C(═NO-n-C.sub.3 H.sub.7)--CH.sub.3                                   329 2-C(═NO-i-C.sub.3 H.sub.7)--CH.sub.3                                   330 3-C(═NO-i-C.sub.3 H.sub.7)--CH.sub.3                                   331 4-C(═NO-i-C.sub.3 H.sub.7)--CH.sub.3                                   332 2-C(═NO-Allyl)--CH.sub.3                                               333 3-C(═NO-Allyl)--CH.sub.3                                               334 4-C(═NO-Allyl)--CH.sub.3                                               335 2-C(═NO-trans-Chloroallyl)--CH.sub.3                                   336 3-C(═NO-trans-Chloroallyl)--CH.sub.3                                   337 4-C(═NO-trans-Chloroallyl)--CH.sub.3                                   338 2-C(═NO-Propargyl)--CH.sub.3                                           339 3-C(═NO-Propargyl)--CH.sub.3                                           340 4-C(═NO-Propargyl)--CH.sub.3                                           341 2-C(═NO-n-C.sub.4 H.sub.9)--CH.sub.3                                   342 3-C(═NO-n-C.sub.4 H.sub.9)--CH.sub.3                                   343 4-C(═NO-n-C.sub.4 H.sub.9)--CH.sub.3                                   344 2-C(═NO--CH.sub.2 --C.sub.6 H.sub.5)--CH.sub.3                         345 3-C(═NO--CH.sub.2 --C.sub.6 H.sub.5)--CH.sub.3                         346 4-C(═NO--CH.sub.2 --C.sub.6 H.sub.5)--CH.sub.3                         347 2-CH.sub.3 -4-CH═NOCH.sub.3                                            348 2-CH.sub.3 -4-CH═NOC.sub.2 H.sub.5                                     349 2-CH.sub.3 -4-CH═NO-n-C.sub.3 H.sub.7                                  350 2-CH.sub.3 -4-CH═NO-i-C.sub.3 H.sub.7                                  351 2-CH.sub.3 -4-CH═NO-Allyl                                              352 2-CH.sub.3 -4-CH═NO-(trans-Chloroallyl)                                353 2-CH.sub.3 -4-CH═NO-Propargyl                                          354 2-CH.sub.3 -4-CH═NO-n-C.sub.4 H.sub.9                                  355 2-CH.sub.3 -4-CH═NO--CH.sub.2 --C.sub.6 H.sub.5                        356 2-CH.sub.3 -4-(CH.sub.3 --C═NOCH.sub.3)                                357 2-CH.sub.3 -4-(CH.sub.3 --C═NOC.sub.2 H.sub.5)                         358 2-CH.sub.3 -4-(CH.sub.3 --C═NO-n-C.sub.3 H.sub.7)                      359 2-CH.sub.3 -4-(CH.sub.3 --C═NO-i-C.sub.3 H.sub.7)                      360 2-CH.sub.3 -4-(CH.sub.3 --C═NO-Allyl)                                  361 2-CH.sub.3 -4-(CH.sub.3 --C═NO-trans-Chloroallyl)                      362 2-CH.sub.3 -4-(CH.sub.3 --C═NO-Propargyl)                              363 2-CH.sub.3 -4-(CH.sub.3 --C═NO-n-C.sub.4 H.sub.9)                      364 2-CH.sub.3 -4-(CH.sub.3 --C═NO--CH.sub.2 --C.sub.6 H.sub.5)                     365 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C═NO--CH.sub.3)                       366 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C═NO--C.sub.2                        H.sub.5)                                                               367 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C═NO-n-C.sub.3 H.sub.7)                        368 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C═NO-i-C.sub.3                       H.sub.7                                                                369 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C═NO-Allyl)                           370 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C═NO-trans-Chloroallyl)                        371 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C═NO-Propargyl)                       372 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C═NO-n-C.sub.4                       H.sub.9)                                                               373 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C═NO--CH.sub.2 --C.sub.6                      H.sub.5)                                                               374 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C═NOCH.sub.3)                      375 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C═NOC.sub.2 H.sub.5)                        376 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C═NO-n-C.sub.3                    H.sub.7)                                                               377 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C═NO-i-C.sub.3 H.sub.7)                     378 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C═NO-Allyl)                        379 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C═NO-trans-Chloroal               lyl)                                                                   380 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C═NO-Proparyl)                     381 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C═NO-n-C.sub.4 H.sub.9)                     382 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C═NO--CH.sub.2                    --C.sub.6 H.sub.5)                                                     383 2-C.sub.6 H.sub.5                                                          384 3-C.sub.6 H.sub.5                                                          385 4-C.sub.6 H.sub.5                                                          386 2-(2'-F--C.sub.6 H.sub.4)                                                  387 2-(3'-F--C.sub.6 H.sub.4)                                                  388 2-(4'-F--C.sub.6 H.sub.4)                                                  389 3-(2'-F--C.sub.6 H.sub.4)                                                  390 3-(3'-F--C.sub.6 H.sub.4)                                                  391 3-(4'-F--C.sub.6 H.sub.4)                                                  392 4-(2'-F--C.sub.6 H.sub.4)                                                  393 4-(3'-F--C.sub.6 H.sub.4)                                                  394 4-(4'-F--C.sub.6 H.sub.4)                                                  395 2-(2'-Cl--C.sub.6 H.sub.4)                                                 396 2-(3'-Cl--C.sub.6 H.sub.4)                                                 397 2-(4'-Cl--C.sub.6 H.sub.4)                                                 398 3-(2'-Cl--C.sub.6 H.sub.4)                                                 399 3-(3'-Cl--C.sub.6 H.sub.4)                                                 400 3-(4'-Cl--C.sub.6 H.sub.4)                                                 401 4-(2'-Cl--C.sub.6 H.sub.4)                                                 402 4-(3'-Cl--C.sub.6 H.sub.4)                                                 403 4-(4'-Cl--C.sub.6 H.sub.4)                                                 405 2-(2'-CH.sub.3 --C.sub.6 H.sub.4)                                          406 2-(3'-CH.sub.3 --C.sub.6 H.sub.4)                                          407 2-(4'-CH.sub.3 --C.sub.6 H.sub.4)                                          408 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)                                          409 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)                                          410 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)                                          411 4-(2'-CH.sub.3 --C.sub.6 H.sub.4)                                          412 4-(3'-CH.sub.3 --C.sub.6 H.sub.4)                                          413 4-(4'-CH.sub.3 --C.sub.6 H.sub.4)                                          414 2-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                      415 2-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                      416 2-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                      417 3-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                      418 3-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                      419 3-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                      420 4-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                      421 4-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                      422 4-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                      423 2-(2'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                       424 2-(3'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                       425 2-(4'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                       426 3-(2'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                       427 3-(3'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                       428 3-(4'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                       429 4-(2'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                       430 4-(3'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                       431 4-(4'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                       432 2-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                                 433 2-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                                 434 2-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                                 435 3-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                                 436 3-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                                 437 3-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                                 438 4-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                                 439 4-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                                 440 4-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                                 441 2-(2'-CH.sub.3 O--C.sub.6 H.sub.4)                                         442 2-(3'-CH.sub.3 O--C.sub.6 H.sub.4)                                         443 2-(4'-CH.sub.3 O--C.sub.6 H.sub.4)                                         444 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)                                         445 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)                                         446 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)                                         447 4-(2'-CH.sub.3 O--C.sub.6 H.sub.4)                                         448 4-(3'-CH.sub.3 O--C.sub.6 H.sub.4)                                         449 4-(4'-CH.sub.3 O--C.sub.6 H.sub.4)                                         450 2-(2'-O.sub.2 N--C.sub.6 H.sub.4)                                          451 2-(3'-O.sub.2 N--C.sub.6 H.sub.4)                                          452 2-(4'-O.sub.2 N--C.sub.6 H.sub.4)                                          453 3-(2'-O.sub.2 N--C.sub.6 H.sub.4)                                          454 3-(3'-O.sub.2 N--C.sub.6 H.sub.4)                                          455 3-(4'-O.sub.2 N--C.sub.6 H.sub.4)                                          456 4-(2'-O.sub.2 N--C.sub.6 H.sub.4)                                          457 4-(3'-O.sub.2 N--C.sub.6 H.sub.4)                                          458 4-(4'-O.sub.2 N--C.sub.6 H.sub.4)                                          459 2-(2'-NC--C.sub.6 H.sub.4)                                                 460 2-(3'-NC--C.sub.6 H.sub.4)                                                 461 2-(4'-NC--C.sub.6 H.sub.4)                                                 462 3-(2'-NC--C.sub.6 H.sub.4)                                                 463 3-(3'-NC--C.sub.6 H.sub.4)                                                 464 3-(4'-NC--C.sub.6 H.sub.4)                                                 465 4-(2'-NC--C.sub.6 H.sub.4)                                                 466 4-(3'-NC--C.sub.6 H.sub.4)                                                 467 4-(4'-NC--C.sub.6 H.sub.4)                                                 468 2-(2'-CF.sub.3 --C.sub.6 H.sub.4)                                          469 2-(3'-CF.sub.3 --C.sub.6 H.sub.4)                                          470 2-(4'-CF.sub.3 --C.sub.6 H.sub.4)                                          471 3-(2'-CF.sub.3 --C.sub.6 H.sub.4)                                          472 3-(3'-CF.sub.3 --C.sub.6 H.sub.4)                                          473 3-(4'-CF.sub.3 --C.sub.6 H.sub.4)                                          474 4-(2'-CF.sub.3 --C.sub.6 H.sub.4)                                          475 4-(3'-CF.sub.3 --C.sub.6 H.sub.4)                                          476 4-(4'-CF.sub.3 --C.sub.6 H.sub.4)                                          477 2-O--C.sub.6 H.sub.5                                                       475 3-O--C.sub.6 H.sub.5                                                       476 4-O--C.sub.6 H.sub.5                                                       478 2-O-(2'-F--C.sub.6 H.sub.4)                                                479 2-O-(3'-F--C.sub.6 H.sub.4)                                                480 2-O-(4'-F--C.sub.6 H.sub.4)                                                481 3-O-(2'-F--C.sub.6 H.sub.4)                                                482 3-O-(3'-F--C.sub.6 H.sub.4)                                                483 3-O-(4'-F--C.sub.6 H.sub.4)                                                484 4-O-(2'-F--C.sub.6 H.sub.4)                                                485 4-O-(3'-F--C.sub.6 H.sub.4)                                                486 4-O-(4'-F--C.sub.6 H.sub.4)                                                487 2-O-(2'-Cl--C.sub.6 H.sub.4)                                               488 2-O-(3'-Cl--C.sub.6 H.sub.4)                                               489 2-O-(4'-Cl--C.sub.6 H.sub.4)                                               490 3-O-(2'-Cl--C.sub.6 H.sub.4)                                               491 3-O-(3'-Cl--C.sub.6 H.sub.4)                                               492 3-O-(4'-Cl--C.sub.6 H.sub.4)                                               493 3-O-(4'-Cl--C.sub.6 H.sub.4)                                               494 4-O-(2'-Cl--C.sub.6 H.sub.4)                                               495 4-O-(3'-Cl--C.sub.6 H.sub.4)                                               496 4-O-(4'-Cl--C.sub.6 H.sub.4)                                               497 2-O-(2'-CH.sub.3 --C.sub.6 H.sub.4)                                        498 2-O-(3'-CH.sub.3 --C.sub.6 H.sub.4)                                        499 2-O-(4'-CH.sub.3 --C.sub.6 H.sub.4)                                        500 3-O-(2'-CH.sub.3 --C.sub.6 H.sub.4)                                        501 3-O-(3'-CH.sub.3 --C.sub.6 H.sub.4)                                        502 3-O-(4'-CH.sub.3 --C.sub.6 H.sub.4)                                        503 4-O-(2'-CH.sub.3 --C.sub.6 H.sub.4)                                        504 4-O-(3'-CH.sub.3 --C.sub.6 H.sub.4)                                        505 4-O-(4'-CH.sub.3 --C.sub.6 H.sub.4)                                        506 2-O-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                    507 2-O-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                    508 2-O-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                    509 3-O-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                    510 3-O-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                    511 3-O-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                    512 4-O-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                    513 4-O-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                    514 4-O-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                    515 2-O-(2'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                     516 2-O-(3'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                     517 2-O-(4'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                     518 3-O-(2'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                     519 3-O-(3'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                     520 3-O-(4'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                     521 4-O-(2'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                     522 4-O-(3'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                     523 4-O-(4'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                     524 2-O-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                               525 2-O-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                               526 2-O-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                               527 3-O-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                               528 3-O-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                               529 3-O-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                               530 4-O-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                               531 4-O-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                               532 4-O-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                               533 2-O-(2'-CH.sub.3 O--C.sub.6 H.sub.4)                                       534 2-O-(3'-CH.sub.3 O--C.sub.6 H.sub.4)                                       535 2-O-(4'-CH.sub.3 O--C.sub.6 H.sub.4)                                       536 3-O-(2'-CH.sub.3 O--C.sub.6 H.sub.4)                                       537 3-O-(3'-CH.sub.3 O--C.sub.6 H.sub.4)                                       538 3-O-(4'-CH.sub.3 O--C.sub.6 H.sub.4)                                       539 4-O-(2'-CH.sub.3 O--C.sub.6 H.sub.4)                                       540 4-O-(3'-CH.sub.3 O--C.sub.6 H.sub.4)                                       541 4-O-(4'-CH.sub.3 O--C.sub.6 H.sub.4)                                       542 2-O-(2'-O.sub.2 N--C.sub.6 H.sub.4)                                        543 2-O-(3'-O.sub.2 N--C.sub.6 H.sub.4)                                        544 2-O-(4'-O.sub.2 N--C.sub.6 H.sub.4)                                        545 3-O-(2'-O.sub.2 N--C.sub.6 H.sub.4)                                        546 3-O-(3'-O.sub.2 N--C.sub.6 H.sub.4)                                        547 3-O-(4'-O.sub.2 N--C.sub.6 H.sub.4)                                        548 4-O-(2'-O.sub.2 N--C.sub.6 H.sub.4)                                        549 4-O-(3'-O.sub.2 N--C.sub.6 H.sub.4)                                        550 4-O-(4'-O.sub.2 N--C.sub.6 H.sub.4)                                        551 2-O-(2'-NC--C.sub.6 H.sub.4)                                               552 2-O-(3'-NC--C.sub.6 H.sub.4)                                               553 2-O-(4'-NC--C.sub.6 H.sub.4)                                               554 3-O-(2'-NC--C.sub.6 H.sub.4)                                               555 3-O-(3'-NC--C.sub.6 H.sub.4)                                               556 3-O-(4'-NC--C.sub.6 H.sub.4)                                               557 4-O-(2'-NC--C.sub.6 H.sub.4)                                               558 4-O-(3'-NC--C.sub.6 H.sub.4)                                               559 4-O-(4'-NC--C.sub.6 H.sub.4)                                               560 2-O-(2'-CF.sub.3 --C.sub.6 H.sub.4)                                        561 2-O-(3'-CF.sub.3 --C.sub.6 H.sub.4)                                        562 2-O-(4'-CF.sub.3 --C.sub.6 H.sub.4)                                        563 3-O-(2'-CF.sub.3 --C.sub.6 H.sub.4)                                        564 3-O-(3'-CF.sub.3 --C.sub.6 H.sub.4)                                        565 3-O-(4'-CF.sub.3 --C.sub.6 H.sub.4)                                        566 4-O-(2'-CF.sub.3 --C.sub.6 H.sub.4)                                        567 4-O-(3'-CF.sub.3 --C.sub.6 H.sub.4)                                        568 4-O-(4'-CF.sub.3 --C.sub.6 H.sub.4)                                        569 2-Pyridinyl-2'                                                             570 2-Pyridinyl-3'                                                             571 2-Pyridinyl-4'                                                             572 3-Pyridinyl-2'                                                             573 3-Pyridinyl-3'                                                             574 3-Pyridinyl-4'                                                             575 4-Pyridinyl-2'                                                             576 4-Pyridinyl-3'                                                             577 4-Pyridinyl-4'                                                             578 2-Pyrimidinyl-2'                                                           579 2-Pyrimidinyl-3'                                                           580 2-Pyrimidinyl-4'                                                           581 3-Pyrimidinyl-2'                                                           582 3-Pyrimidinyl-3'                                                           583 3-Pyrimidinyl-4'                                                           584 4-Pyrimidinyl-2'                                                           585 4-Pyrimidinyl-3'                                                           586 4-Pyrimidinyl-4'                                                           587 2-Pyrazolyl-1'                                                             588 2-Pyrazolyl-3'                                                             589 2-Pyrazolyl-4'                                                             590 3-Pyrazolyl-1'                                                             591 3-Pyrazolyl-3'                                                             592 3-Pyrazolyl-4'                                                             593 4-Pyrazolyl-1'                                                             594 4-Pyrazolyl-3'                                                             595 4-Pyrazolyl-4'                                                             596 2-Isoxazolyl-3'                                                            597 2-Isoxazolyl-4'                                                            598 2-Isoxazolyl-5'                                                            599 3-Isoxazolyl-3'                                                            600 3-Isoxazolyl-4'                                                            601 3-Isoxazolyl-5'                                                            602 4-Isoxazolyl-3'                                                            603 4-Isoxazolyl-4'                                                            604 4-Isoxazolyl-5'                                                            605 2-Isothiazolyl-3'                                                          606 2-Isothiazolyl-4'                                                          607 2-Isothiazolyl-5'                                                          608 3-Isothiazolyl-3'                                                          609 3-Isothiazolyl-4'                                                          610 3-Isothiazolyl-5'                                                          611 4-Isothiazolyl-3'                                                          612 4-Isothiazolyl-4'                                                          613 4-Isothiazolyl-5'                                                          614 2-Imidazolyl-1'                                                            615 2-Imidazolyl-2'                                                            616 2-Imidazolyl-4'                                                            617 3-Imidazolyl-1'                                                            618 3-Imidazolyl-2'                                                            619 3-Imidazolyl-4'                                                            620 4-Imidazolyl-1'                                                            621 4-Imidazolyl-2'                                                            622 4-Imidazolyl-4'                                                            623 2-Oxazolyl-2'                                                              624 2-Oxazolyl-4'                                                              625 2-Oxazolyl-5'                                                              626 3-Oxazolyl-2'                                                              627 3-Oxazolyl-4'                                                              628 3-Oxazolyl-5'                                                              629 4-Oxazolyl-2'                                                              630 4-Oxazolyl-4'                                                              631 4-Oxazolyl-5'                                                              632 2-Thiazolyl-2'                                                             633 2-Thiazolyl-4'                                                             634 2-Thiazolyl-5'                                                             635 3-Thiazolyl-2'                                                             636 3-Thiazolyl-4'                                                             637 3-Thiazolyl-5'                                                             638 4-Thiazolyl-2'                                                             639 4-Thiazolyl-4'                                                             640 4-Thiazolyl-5'                                                             641 2-CH.sub.3 -4-(CH.sub.3 --C═N--O--CH.sub.2 --CH.sub.2 --OCH.sub.               3)                                                                     642 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C═N--O--CH.sub.2 --CH.sub.2                   --OCH.sub.3)                                                           643 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C═N--O--CH.sub.2 --CH.sub.2                --OCH.sub.3)                                                           644 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C═N--OCH.sub.3)                     645 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C═N--OC.sub.2 H.sub.5)                       646 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C═N--O-n-C.sub.3                   H.sub.7)                                                               647 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C═N--O-i-C.sub.3 H.sub.7)                    648 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C═N--O-Allyl)                       649 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C═N--O-trans-Chloroa               llyl)                                                                  650 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C═N--O-Propargyl)                   651 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C═N--O-n-C.sub.4 H.sub.9)                    652 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C═N--O--CH.sub.2                   --C.sub.6 H.sub.5)                                                     653 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C═N--OCH.sub.3)                     654 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C═N--OC.sub.2 H.sub.5)                       655 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C═N--O-n-C.sub.3                   H.sub.7)                                                               656 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C═N--O-i-C.sub.3 H.sub.7)                    657 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C═N--O-Allyl)                       658 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C═N--O-trans-Chloroa               llyl)                                                                  659 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C═N--O-Propargyl)                   660 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C═N--O-n-C.sub.4 H.sub.9)                    661 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C═N--O--CH.sub.2                   --C.sub.6 H.sub.5)                                                     662 2-O-n-C.sub.4 H.sub.9                                                      663 2-O-i-C.sub.4 H.sub.9                                                      664 2-O-s-C.sub.4 H.sub.9                                                      665 2-O-t-C.sub.4 H.sub.9                                                      666 2-Neopentyloxy                                                             667 3-O-n-C.sub.4 H.sub.9                                                      668 3-O-i-C.sub.4 H.sub.9                                                      669 3-O-s-C.sub.4 H.sub.9                                                      670 3-O-t-C.sub.4 H.sub.9                                                      671 3-Neopentyloxy                                                             672 4-O-n-C.sub.4 H.sub.9                                                      673 4-O-i-C.sub.4 H.sub.9                                                      674 4-O-s-C.sub.4 H.sub.9                                                      675 4-O-t-C.sub.4 H.sub.9                                                      676 4-Neopentyloxy                                                             677 3-CH.sub.3 -4-OCH.sub.3                                                    678 3-CH.sub.3 -4-OC.sub.2 H.sub.5                                             679 3-CH.sub.3 -4-O-n-C.sub.3 H.sub.7                                          680 3-CH.sub.3 -4-O-n-C.sub.4 H.sub.9                                          681 3-CH.sub.3 -4-O-i-C.sub.4 H.sub.9                                          682 3-CH.sub.3 -4-O-s-C.sub.4 H.sub.9                                          683 3-CH.sub.3 -4-O-t-C.sub.4 H.sub.9                                          684 3-CH.sub.3 -4-Neopentyloxy                                                 685 2-CH.sub.3 -3-OCH.sub.3                                                    686 2-CH.sub.3 -4-OCH.sub.3                                                    687 2-CH.sub.3 -5-OCH.sub.3                                                    688 2-CH.sub.3 -6-OCH.sub.3                                                    689 3-CH.sub.3 -4-OCH.sub.3                                                    690 3-CH.sub.3 -5-OCH.sub.3                                                    691 3-CH.sub.3 -6-OCH.sub.3                                                    692 4-CH.sub.3 -5-O--CH.sub.3                                                  693 4-CH.sub.3 -6-O--CH.sub.3                                                  694 4-CH.sub.3 -6-OCH.sub.3                                                    695 2-CH.sub.3 -3-O-i-C.sub.3 H.sub.7                                          696 2-CH.sub.3 -4-O-i-C.sub.3 H.sub.7                                          697 2-CH.sub.3 -5-O-i-C.sub.3 H.sub.7                                          698 2-CH.sub.3 -6-O-i-C.sub.3 H.sub.7                                          699 3-CH.sub.3 -4-O-i-C.sub.3 H.sub.7                                          700 3-CH.sub.3 -5-O-i-C.sub.3 H.sub.7                                          701 3-CH.sub.3 -6-O-i-C.sub.3 H.sub.7                                          702 4-CH.sub.3 -5-O-i-C.sub.3 H.sub.7                                          703 4-CH.sub.3 -6-O-i-C.sub.3 H.sub.7                                          704 5-CH.sub.3 -6-O-i-C.sub.3 H.sub.7                                          705 2-Cl-3-OCH.sub.3                                                           706 2-Cl-4-OCH.sub.3                                                           707 2-Cl-5-OCH.sub.3                                                           708 2-Cl-6-OCH.sub.3                                                           709 3-Cl-4-OCH.sub.3                                                           710 3-Cl-5-OCH.sub.3                                                           711 3-Cl-6-OCH.sub.3                                                           712 4-Cl-5-OCH.sub.3                                                           713 4-Cl-6-OCH.sub.3                                                           714 5-Cl-6-OCH.sub.3                                                         ______________________________________                                    

                  TABLE 42                                                         ______________________________________                                         2  STR275##                                                                       -                                                                               I: R.sup.1 = H, X = CH.sub.3                                                                     VIII: R.sup.1 = H, X = Cl                                  II: R.sup.1 = CH.sub.3, X = CH.sub.3 IX: R.sup.1 = CH.sub.3, X = Cl                                 III: R.sup.1 = C.sub.2 H.sub.5, X = CH.sub.3 X:                               R.sup.1 = C.sub.2 H.sub.5, X = Cl                          IV: R.sup.1 = Allyl, X = CH.sub.3 XI: R.sup.1 = Allyl, X = Cl                  V: R.sup.1 = Propargyl, X = CH.sub.3 XII: R.sup.1 = Propargyl, X = Cl                               VI: R.sup.1 = CH.sub.2 --OCH.sub.3, X = CH.sub.3                              XIII: R.sup.1 = CH.sub.2 --OCH.sub.3, X = Cl                                    VII: R.sup.1 = CO.sub.2 CH.sub.3, X = CH.sub.3                                XIV: R.sup.1 = CO.sub.2 CH.sub.3, X = Cl                 No.       B                                                                    ______________________________________                                          1        Pyrrolyl-3                                                              2 N--CH.sub.3 -Pyrrolyl-3                                                      3 N--C.sub.6 H.sub.5 -Pyrrolyl-3                                               4 N-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrrolyl-3                                 5 N-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrrolyl-3                                 6 N-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrrolyl-3                                 7 N-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrrolyl-3                                8 N-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrrolyl-3                                9 N-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrrolyl-3                                10 N-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrrolyl-3                                11 N-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrrolyl-3                                12 N-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrrolyl-3                                13 N-(4'-CN--C.sub.6 H.sub.4)-Pyrrolyl-3                                       14 N-(3'-CN--C.sub.6 H.sub.4)-Pyrrolyl-3                                       15 N-(2'-CN--C.sub.6 H.sub.4)-Pyrrolyl-3                                       16 N-(4'-Cl--C.sub.6 H.sub.4)-Pyrrolyl-3                                       17 N-(3'-Cl--C.sub.6 H.sub.4)-Pyrrolyl-3                                       18 N-(2'-Cl--C.sub.6 H.sub.4)-Pyrrolyl-3                                       19 Pyrrolyl-2                                                                  20 N--CH.sub.3 -Pyrrolyl-2                                                     21 N--C.sub.6 H.sub.5 -Pyrrolyl-2                                              22 N-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrrolyl-2                                23 N-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrrolyl-2                                24 N-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrrolyl-2                                25 N-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrrolyl-2                               26 N-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrrolyl-2                               27 N-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrrolyl-2                               28 N-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrrolyl-2                                29 N-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrrolyl-2                                30 N-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrrolyl-2                                31 N-(4'-CN--C.sub.6 H.sub.4)-Pyrrolyl-2                                       32 N-(3'-CN--C.sub.6 H.sub.4)-Pyrrolyl-2                                       33 N-(2'-CN--C.sub.6 H.sub.4)-Pyrrolyl-2                                       34 N-(4'-Cl--C.sub.6 H.sub.4)-Pyrrolyl-2                                       35 N-(3'-Cl--C.sub.6 H.sub.4)-Pyrrolyl-2                                       36 N-(2'-Cl--C.sub.6 H.sub.4)-Pyrrolyl-2                                       37 Furyl-2                                                                     38 5-CH.sub.3 -Furyl-2                                                         39 5-C.sub.6 H.sub.5 -Furyl-2                                                  40 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Furyl-2                                   41 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Furyl-2                                   42 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Furyl-2                                   43 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Furyl-2                                  44 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Furyl-2                                  45 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Furyl-2                                  46 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Furyl-2                                   47 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Furyl-2                                   48 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Furyl-2                                   49 5-(4'-CN--C.sub.6 H.sub.4)-Furyl-2                                          50 5-(3'-CN--C.sub.6 H.sub.4)-Furyl-2                                          51 5-(2'-CN--C.sub.6 H.sub.4)-Furyl-2                                          52 5-(4'-Cl--C.sub.6 H.sub.4)-Furyl-2                                          53 5-(3'-Cl--C.sub.6 H.sub.4)-Furyl-2                                          54 5-(2'-Cl--C.sub.6 H.sub.4)-Furyl-2                                          55 4-CH.sub.3 -Furyl-2                                                         56 4-C.sub.6 H.sub.5 -Furyl-2                                                  57 4-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Furyl-2                                   58 4-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Furyl-2                                   59 4-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Furyl-2                                   60 4-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Furyl-2                                  61 4-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Furyl-2                                  62 4-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Furyl-2                                  63 4-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Furyl-2                                   64 4-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Furyl-2                                   65 4-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Furyl-2                                   66 4-(4'-CN--C.sub.6 H.sub.4)-Furyl-2                                          67 4-(3'-CN--C.sub.6 H.sub.4)-Furyl-2                                          68 4-(2'-CN--C.sub.6 H.sub.4)-Furyl-2                                          69 4-(4'-Cl--C.sub.6 H.sub.4)-Furyl-2                                          70 4-(3'-Cl--C.sub.6 H.sub.4)-Furyl-2                                          71 4-(2'-Cl--C.sub.6 H.sub.4)-Furyl-2                                          72 Thienyl-2                                                                   73 5-CH.sub.3 -Thienyl-2                                                       74 5-C.sub.6 H.sub.5 -Thienyl-2                                                75 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-2                                 76 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-2                                 77 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-2                                 78 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-2                                79 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-2                                80 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-2                                81 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-2                                 82 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-2                                 83 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-2                                 84 5-(4'-CN--C.sub.6 H.sub.4)-Thienyl-2                                        85 5-(3'-CN--C.sub.6 H.sub.4)-Thienyl-2                                        86 5-(2'-CN--C.sub.6 H.sub.4)-Thienyl-2                                        87 5-(4'-Cl--C.sub.6 H.sub.4)-Thienyl-2                                        88 5-(3'-Cl--C.sub.6 H.sub.4)-Thienyl-2                                        89 5-(2'-Cl--C.sub.6 H.sub.4)-Thienyl-2                                        90 4-CH.sub.3 -Thienyl-2                                                       91 4-C.sub.6 H.sub.5 -Thienyl-2                                                92 4-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-2                                 93 4-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-2                                 94 4-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-2                                 95 4-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-2                                96 4-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-2                                97 4-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-2                                98 4-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-2                                 99 4-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-2                                100 4-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-2                                101 4-(4'-CN--C.sub.6 H.sub.4)-Thienyl-2                                       102 4-(3'-CN--C.sub.6 H.sub.4)-Thienyl-2                                       103 4-(2'-CN--C.sub.6 H.sub.4)-Thienyl-2                                       104 4-(4'-Cl--C.sub.6 H.sub.4)-Thienyl-2                                       105 4-(3'-Cl--C.sub.6 H.sub.4)-Thienyl-2                                       106 4-(2'-Cl--C.sub.6 H.sub.4)-Thienyl-2                                       107 Thienyl-3                                                                  108 5-CH.sub.3 -Thienyl-3                                                      109 5-C.sub.6 H.sub.5 -Thienyl-3                                               110 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-3                                111 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-3                                112 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-3                                113 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-3                               114 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-3                               115 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-3                               116 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-3                                117 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-3                                118 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-3                                119 5-(4'-CN--C.sub.6 H.sub.4)-Thienyl-3                                       120 5-(3'-CN--C.sub.6 H.sub.4)-Thienyl-3                                       121 5-(2'-CN--C.sub.6 H.sub.4)-Thienyl-3                                       122 5-(4'-Cl--C.sub.6 H.sub.4)-Thienyl-3                                       123 5-(3'-Cl--C.sub.6 H.sub.4)-Thienyl-3                                       124 5-(2'-Cl--C.sub.6 H.sub.4)-Thienyl-3                                       125 Pyrazolyl-4                                                                126 N--CH.sub.3 -Pyrazolyl-4                                                   127 N--C.sub.6 H.sub.5 -Pyrazolyl-4                                            128 N-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrazolyl-4                              129 N-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrazolyl-4                              130 N-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrazolyl-4                              131 N-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrazolyl-4                             132 N-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrazolyl-4                             133 N-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrazolyl-4                             134 N-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrazolyl-4                              135 N-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrazolyl-4                              136 N-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrazolyl-4                              137 N-(4'-CN--C.sub.6 H.sub.4)-Pyrazolyl-4                                     138 N-(3'-CN--C.sub.6 H.sub.4)-Pyrazolyl-4                                     139 N-(2'-CN--C.sub.6 H.sub.4)-Pyrazolyl-4                                     140 N-(4'-Cl--C.sub.6 H.sub.4)-Pyrazolyl-4                                     141 N-(3'-Cl--C.sub.6 H.sub.4)-Pyrazolyl-4                                     142 N-(2'-Cl--C.sub.6 H.sub.4)-Pyrazolyl-4                                     143 3-CH.sub.3 --N-Methylpyrazolyl-4                                           144 3-C.sub.6 H.sub.4 --N-Methylpyrazolyl-4                                    145 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)--N-Methylpyrazolyl-4                     146 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)--N-Methylpyrazolyl-4                     147 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)--N-Methylpyrazolyl-4                     148 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)--N-Methylpyrazolyl-4                    149 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)--N-Methylpyrazolyl-4                    150 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)--N-Methylpyrazolyl-4                    151 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)--N-Methylpyrazolyl-4                     152 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)--N-Methylpyrazolyl-4                     153 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)--N-Methylpyrazolyl-4                     154 3-(4'-CN--C.sub.6 H.sub.4)--N-Methylpyrazolyl-4                            155 3-(3'-CN--C.sub.6 H.sub.4)--N-Methylpyrazolyl-4                            156 3-(2'-CN--C.sub.6 H.sub.4)--N-Methylpyrazolyl-4                            157 3-(4'-Cl--C.sub.6 H.sub.4)--N-Methylpyrazolyl-4                            158 3-(3'-Cl--C.sub.6 H.sub.4)--N-Methylpyrazolyl-4                            159 3-(2'-Cl--C.sub.6 H.sub.4)--N-Methylpyrazolyl-4                            160 Isoxazolyl-5                                                               161 3-CH.sub.3 -Isoxazolyl-5                                                   162 3-C.sub.6 H.sub.5 -Isoxazolyl-5                                            163 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Isoxazolyl-5                             164 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Isoxazolyl-5                             165 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Isoxazolyl-5                             166 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Isoxazolyl-5                            167 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Isoxazolyl-5                            168 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Isoxazolyl-5                            169 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Isoxazolyl-5                             170 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Isoxazolyl-5                             171 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Isoxazolyl-5                             172 3-(4'-CN--C.sub.6 H.sub.4)-Isoxazolyl-5                                    173 3-(3'-CN--C.sub.6 H.sub.4)-Isoxazolyl-5                                    174 3-(2'-CN--C.sub.6 H.sub.4)-Isoxazolyl-5                                    175 3-(4'-Cl--C.sub.6 H.sub.4)-Isoxazolyl-5                                    176 3-(3'-Cl--C.sub.6 H.sub.4)-Isoxazolyl-5                                    177 3-(2'-Cl--C.sub.6 H.sub.4)-Isoxazolyl-5                                    178 4-Chloroisoxazolyl-5                                                       179 3-CH.sub.3 -4-Chloroisoxazolyl-5                                           180 3-C.sub.6 H.sub.5 -4-Chloroisoxazolyl-5                                    181 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                     182 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                     183 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                     184 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                    185 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                    186 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                    187 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                     188 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                     189 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                     190 3-(4'-CN--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                            191 3-(3'-CN--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                            192 3-(2'-CN--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                            193 3-(4'-Cl--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                            194 3-(3'-Cl--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                            195 3-(2'-Cl--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                            196 Isoxazolyl-3                                                               197 5-CH.sub.3 -Isoxazolyl-3                                                   198 5-C.sub.6 H.sub.5 -Isoxazolyl-3                                            199 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Isoxazolyl-3                             200 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Isoxazolyl-3                             201 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Isoxazolyl-3                             202 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Isoxazolyl-3                            203 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Isoxazolyl-3                            204 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Isoxazolyl-3                            205 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Isoxazolyl-3                             206 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Isoxazolyl-3                             207 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Isoxazolyl-3                             208 5-(4'-CN--C.sub.6 H.sub.4)-Isoxazolyl-3                                    209 5-(3'-CN--C.sub.6 H.sub.4)-Isoxazolyl-3                                    210 5-(2'-CN--C.sub.6 H.sub.4)-Isoxazolyl-3                                    211 5-(4'-Cl--C.sub.6 H.sub.4)-Isoxazolyl-3                                    212 5-(3'-Cl--C.sub.6 H.sub.4)-Isoxazolyl-3                                    213 5-(2'-Cl--C.sub.6 H.sub.4)-Isoxazolyl-3                                    214 Isothiazolyl-5                                                             215 3-CH.sub.3 -Isothiazolyl-5                                                 216 3-C.sub.6 H.sub.5 -Isothiazolyl-5                                          217 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Isothiazolyl-5                           218 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Isothiazolyl-5                           219 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Isothiazolyl-5                           220 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Isothiazolyl-5                          221 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Isothiazolyl-5                          222 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Isothiazolyl-5                          223 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Isothiazolyl-5                           224 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Isothiazolyl-5                           225 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Isothiazolyl-5                           226 3-(4'-CN--C.sub.6 H.sub.4)-Isothiazolyl-5                                  227 3-(3'-CN--C.sub.6 H.sub.4)-Isothiazolyl-5                                  228 3-(2'-CN--C.sub.6 H.sub.4)-Isothiazolyl-5                                  229 3-(4'-Cl--C.sub.6 H.sub.4)-Isothiazolyl-5                                  230 3-(3'-Cl--C.sub.6 H.sub.4)-Isothiazolyl-5                                  231 3-(2'-Cl--C.sub.6 H.sub.4)-Isothiazolyl-5                                  232 Oxazolyl-4                                                                 233 3-CH.sub.3 -Oxazolyl-4                                                     234 3-C.sub.6 H.sub.5 -Oxazolyl-4                                              235 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Oxazolyl-4                               236 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Oxazolyl-4                               237 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Oxazolyl-4                               238 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Oxazolyl-4                              239 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Oxazolyl-4                              240 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Oxazolyl-4                              241 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Oxazolyl-4                               242 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Oxazolyl-4                               243 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Oxazolyl-4                               244 3-(4'-CN--C.sub.6 H.sub.4)-Oxazolyl-4                                      245 3-(3'-CN--C.sub.6 H.sub.4)-Oxazolyl-4                                      246 3-(2'-CN--C.sub.6 H.sub.4)-Oxazolyl-4                                      247 3-(4'-Cl--C.sub.6 H.sub.4)-Oxazolyl-4                                      248 3-(3'-Cl--C.sub.6 H.sub.4)-Oxazolyl-4                                      249 3-(2'-Cl--C.sub.6 H.sub.4)-Oxazolyl-4                                      250 Thiazolyl-4                                                                251 2-CH.sub.3 -Thiazolyl-4                                                    252 2-C.sub.6 H.sub.5 -Thiazolyl-4                                             253 2-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Thiazolyl-4                              254 2-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Thiazolyl-4                              255 2-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Thiazolyl-4                              256 2-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Thiazolyl-4                             267 2-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Thiazolyl-4                             258 2-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Thiazolyl-4                             259 2-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Thiazolyl-4                              260 2-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Thiazolyl-4                              261 2-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Thiazolyl-4                              262 2-(4'-CN--C.sub.6 H.sub.4)-Thiazolyl-4                                     263 2-(3'-CN--C.sub.6 H.sub.4)-Thiazolyl-4                                     264 2-(2'-CN--C.sub.6 H.sub.4)-Thiazolyl-4                                     265 2-(4'-Cl--C.sub.6 H.sub.4)-Thiazolyl-4                                     266 2-(3'-Cl--C.sub.6 H.sub.4)-Thiazolyl-4                                     267 2-(2'-Cl--C.sub.6 H.sub.4)-Thiazolyl-4                                     268 N--CH.sub.3 -1,2,4-Triazolyl-5                                             269 3-CH.sub.3 --N--CH.sub.3 -1,2,4-Triazolyl-5                                270 3-C.sub.6 H.sub.5 --N--CH.sub.3 -1,2,4-Triazolyl-5                         271 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5                   272 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triaz               olyl-5                                                                 273 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5                   274 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Tria               zolyl-5                                                                275 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5                  276 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Tria               zolyl-5                                                                277 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5                   278 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triaz               olyl-5                                                                 279 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5                   280 3-(4'-CN--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5        281 3-(3'-CN--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5                 282 3-(2'-CN--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5                 283 3-(4'-Cl--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5                 284 3-(3'-Cl--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5                 285 3-(2'-Cl--C.sub.6 H.sub.4)--N--CH.sub.3 -1,2,4-Triazolyl-5                 286 1,3,4-Oxadiazolyl-2                                                        287 5-CH.sub.3 -1,3,4-Oxadiazolyl-2                                            288 5-C.sub.6 H.sub.5 -1,3,4-Oxadiazolyl-2                                     289 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                      290 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                      291 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                      292 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                     293 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                     294 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                     295 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                      296 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                      297 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                      298 5-(4'-CN--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                             299 5-(3'-CN--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                             300 5-(2'-CN--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                             301 5-(4'-Cl--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                             302 5-(3'-Cl--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                             303 5-(2'-Cl--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                             304 1,2,4-Oxadiazolyl-3                                                        305 5-CH.sub.3 -1,2,4-Oxadiazolyl-3                                            306 5-C.sub.6 H.sub.5 -1,2,4-Oxadiazolyl-3                                     307 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                      308 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                      309 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                      310 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                     311 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                     312 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                     313 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                      314 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                      315 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                      316 5-(4'-CN--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                             317 5-(3'-CN--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                             318 5-(2'-CN--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                             319 5-(4'-Cl--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                             320 5-(3'-Cl--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                             321 5-(2'-Cl--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                             322 1,2,4-Oxadiazolyl-5                                                        323 3-CH.sub.3 -1,2,4-Oxadiazolyl-5                                            324 3-C.sub.6 H.sub.5 -1,2,4-Oxadiazolyl-5                                     325 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                      326 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                      327 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                      328 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                     329 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                     330 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                     331 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                      332 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                      333 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                      334 3-(4'-CN--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                             335 3-(3'-CN--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                             336 3-(2'-CN--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                             337 3-(4'-Cl--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                             338 3-(3'-Cl--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                             339 3-(2'-Cl--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                             340 1,2,4-Thiadiazolyl-3                                                       341 5-CH.sub.3 -1,2,4-Thiadiazolyl-3                                           342 5-C.sub.6 H.sub.5 -1,2,4-Thiadiazolyl-3                                    343 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                     344 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                     345 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                     346 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                    347 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                    348 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                    349 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                     350 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                     351 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                     352 5-(4'-CN--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                            353 5-(3'-CN--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                            354 5-(2'-CN--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                            355 5-(4'-Cl--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                            356 5-(3'-Cl--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                            357 5-(2'-Cl--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                            358 1,3,4-Thiadiazolyl-2                                                       359 5-CH.sub.3 -1,3,4-Thiadiazolyl-2                                           360 5-C.sub.6 H.sub.5 -1,3,4-Thiadiazolyl-2                                    361 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                     362 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                     363 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                     364 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                    365 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                    366 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                    367 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                     368 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                     369 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                     370 5-(4'-CN--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                            371 5-(3'-CN--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                            372 5-(2'-CN--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                            373 5-(4'-Cl--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                            374 5-(3'-Cl--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                            375 5-(2'-Cl--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                            376 Pyridinyl-2                                                                377 Pyridinyl-4                                                                378 Pyridazinyl-3                                                              379 Pyridazinyl-4                                                              380 Pyridazinyl-2                                                              381 Pyrimidinyl-4                                                              382 Pyrimidinyl-5                                                              383 Pyrimidinyl-2                                                              384 1-Naphthyl                                                                 385 2-Naphthyl                                                               ______________________________________                                    

                  TABLE 43                                                         ______________________________________                                         1  STR276##                                                                      I: R.sup.1 = H, X = CH.sub.3                                                                      VIII: R.sup.1 = H, X = Cl                                   II: R.sup.1 = CH.sub.3, X = CH.sub.3 IX: R.sup.1 = CH.sub.3, X = Cl                                III: R.sup.1 = C.sub.2 H.sub.5, X = CH.sub.3 X:                               R.sup.1 = C.sub.2 H.sub.5, X = Cl                           IV: R.sup.1 = Allyl, X = CH.sub.3 XI: R.sup.1 = Allyl, X = Cl                  V: R.sup.1 = Propargyl, X = CH.sub.3 XII: R.sup.1 = Propargyl, X = Cl                              VI: R.sup.1 = CH.sub.2 --OCH.sub.3, X = CH.sub.3                              XIII: R.sup.1 = CH.sub.2 --OCH.sub.3, X = Cl                                    VII: R.sup.1 = CO.sub.2 CH.sub.3, X = CH.sub.3 XIV:                           R.sup.1 = CO.sub.2 CH.sub.3, X = Cl                          -                                                                           No.       T.sub.m                                                              ______________________________________                                         1         H                                                                      2 2-F                                                                          3 3-F                                                                          4 4-F                                                                          5 2,4-F.sub.2                                                                  6 2,4,6-F.sub.3                                                                7 2,3,4,5,6-F.sub.5                                                            8 2,3-F.sub.2                                                                  9 2-Cl                                                                         10 3-Cl                                                                        11 4-Cl                                                                        12 2,3-Cl.sub.2                                                                13 2,4-Cl.sub.2                                                                14 2,5-Cl.sub.2                                                                15 2,6-Cl.sub.2                                                                16 3,4-Cl.sub.2                                                                17 3,5-Cl.sub.2                                                                18 2,3,4-Cl.sub.3                                                              19 2,3,5-Cl.sub.3                                                              20 2,3,6-Cl.sub.3                                                              21 2,4,5-Cl.sub.3                                                              22 2,4,6-Cl.sub.3                                                              23 3,4,5-Cl.sub.3                                                              24 2,3,4,6-Cl.sub.4                                                            25 2,3,5,6-Cl.sub.4                                                            26 2,3,4,5,6-Cl.sub.5                                                          27 2-Br                                                                        28 3-Br                                                                        29 4-Br                                                                        30 2,4-Br.sub.2                                                                31 2,5-Br.sub.2                                                                32 2,6-Br.sub.2                                                                33 2,4,6-Br.sub.3                                                              34 2,3,4,5,6-Br.sub.5                                                          35 2-I                                                                         36 3-I                                                                         37 4-I                                                                         38 2,4-I.sub.2                                                                 39 2-Cl, 3-F                                                                   40 2-Cl, 4-F                                                                   41 2-Cl, 5-F                                                                   42 2-Cl, 6-F                                                                   43 2-Cl, 3-Br                                                                  44 2-Cl, 4-Br                                                                  45 2-Cl, 5-Br                                                                  46 2-Cl, 6-Br                                                                  47 2-Br, 3-Cl                                                                  48 2-Br, 4-Cl                                                                  49 2-Br, 5-Cl                                                                  50 2-Br, 3-F                                                                   51 2-Br, 4-F                                                                   52 2-Br, 5-F                                                                   53 2-Br, 6-F                                                                   54 2-F, 3-Cl                                                                   55 2-F, 4-Cl                                                                   56 2-F, 5-Cl                                                                   57 3-Cl, 4-F                                                                   58 3-Cl, 5-F                                                                   59 3-Cl, 4-Br                                                                  60 3-Cl, 5-Br                                                                  61 3-F, 4-Cl                                                                   62 3-F, 4-Br                                                                   63 3-Br, 4-Cl                                                                  64 3-Br, 4-F                                                                   65 2,6-Cl.sub.2, 4-Br                                                          66 2-CH.sub.3                                                                  67 3-CH.sub.3                                                                  68 4-CH.sub.3                                                                  69 2,3-(CH.sub.3).sub.2                                                        70 2,4-(CH.sub.3).sub.2                                                        71 2,5-(CH.sub.3).sub.2                                                        72 2,6-(CH.sub.3).sub.2                                                        73 3,4-(CH.sub.3).sub.2                                                        74 3,5-(CH.sub.3).sub.2                                                        75 2,3,5-(CH.sub.3).sub.3                                                      76 2,3,4-(CH.sub.3).sub.3                                                      77 2,3,6-(CH.sub.3).sub.3                                                      78 2,4,5-(CH.sub.3).sub.3                                                      79 2,4,6-(CH.sub.3).sub.3                                                      80 3,4,5-(CH.sub.3).sub.3                                                      81 2,3,4,6-(CH.sub.3).sub.4                                                    82 2,3,5,6-(CH.sub.3).sub.4                                                    83 2,3,4,5,6-(CH.sub.3).sub.5                                                  84 2-C.sub.2 H.sub.5                                                           85 3-C.sub.2 H.sub.5                                                           86 4-C.sub.2 H.sub.5                                                           87 2,4-(C.sub.2 H.sub.5).sub.2                                                 88 2,6-(C.sub.2 H.sub.5).sub.2                                                 89 3,5-(C.sub.2 H.sub.5).sub.2                                                 90 2,4,6-(C.sub.2 H.sub.5).sub.3                                               91 2-n-C.sub.3 H.sub.7                                                         92 3-n-C.sub.3 H.sub.7                                                         93 4-n-C.sub.3 H.sub.7                                                         94 2-i-C.sub.3 H.sub.7                                                         95 3-i-C.sub.3 H.sub.7                                                         96 4-i-C.sub.3 H.sub.7                                                         97 2,4-(i-C.sub.3 H.sub.7).sub.2                                               98 2,6-(i-C.sub.3 H.sub.7).sub.2                                               99 3,5-(i-C.sub.3 H.sub.7).sub.2                                               100 2,4,6-(i-C.sub.3 H.sub.7).sub.3                                            101 2-s-C.sub.4 H.sub.9                                                        102 3-s-C.sub.4 H.sub.9                                                        103 4-s-C.sub.4 H.sub.9                                                        104 2-t-C.sub.4 H.sub.9                                                        105 3-t-C.sub.4 H.sub.9                                                        106 4-t-C.sub.4 H.sub.9                                                        107 2,3-(t-C.sub.4 H.sub.9).sub.2                                              108 2,4-(t-C.sub.4 H.sub.9).sub.2                                              109 2,5-(t-C.sub.4 H.sub.9).sub.2                                              110 2,6-(t-C.sub.4 H.sub.9).sub.2                                              111 3,4-(t-C.sub.4 H.sub.9).sub.2                                              112 2,4,6-(t-C.sub.4 H.sub.9).sub.3                                            113 4-n-C.sub.9 H.sub.19                                                       114 4-n-C.sub.12 H.sub.25                                                      115 4-n-C.sub.15 H.sub.31                                                      116 4-(1,1,3,3-Tetramethylbutyl)                                               117 4-(2,4,4-Trimethylpropyl)                                                  118 2-t-C.sub.4 H.sub.9, 4-CH.sub.3                                            119 2-t-C.sub.4 H.sub.9, 5-CH.sub.3                                            120 2,6-(t-C.sub.4 H.sub.9).sub.2, 4-CH.sub.3                                  121 2-CH.sub.3, 4-t-C.sub.4 H.sub.9                                            122 2-CH.sub.3, 6-t-C.sub.4 H.sub.9                                            123 2-CH.sub.3, 4-i-C.sub.3 H.sub.7                                            124 2-CH.sub.3, 5-i-C.sub.3 H.sub.7                                            125 3-CH.sub.3, 4-i-C.sub.3 H.sub.7                                            126 2-i-C.sub.3 H.sub.7, 5-CH.sub.3                                            127 2,4-(t-C.sub.4 H.sub.9).sub.2, 6-i-C.sub.3 H.sub.7                         128 2-Allyl                                                                    129 3-Allyl                                                                    130 4-Allyl                                                                    131 2-Allyl, 6-CH.sub.3                                                        132 2-cyclo-C.sub.6 H.sub.11                                                   133 3-cyclo-C.sub.6 H.sub.11                                                   134 4-cyclo-C.sub.6 H.sub.11                                                   135 2,4-(cyclo-C.sub.6 H.sub.11).sub.2, 6-CH.sub.3                             136 2-CH.sub.3, 4-cyclo-C.sub.6 H.sub.11                                       137 2-CH.sub.2 --C.sub.6 H.sub.5                                               138 3-CH.sub.2 --C.sub.6 H.sub.5                                               139 4-CH.sub.2 --C.sub.6 H.sub.5                                               140 2-CH.sub.2 --C.sub.6 H.sub.5, 4-CH.sub.3                                   141 2-CH.sub.3, 4-CH.sub.2 --C.sub.6 H.sub.5                                   142 2-C.sub.6 H.sub.5                                                          143 3-C.sub.6 H.sub.5                                                          144 4-C.sub.6 H.sub.5                                                          145 4-(2-i-C.sub.3 H.sub.7 --C.sub.6 H.sub.4)                                  146 4-C.sub.6 H.sub.5, 2,6-(CH.sub.3).sub.2                                    147 2-Cl, 4-C.sub.6 H.sub.5                                                    148 2-Br, 4-C.sub.6 H.sub.5                                                    149 2-C.sub.6 H.sub.5, 4-Cl                                                    150 2-C.sub.6 H.sub.5, 4-Br                                                    151 2-CH.sub.2 C.sub.6 H.sub.5, 4-Cl                                           152 2-CH.sub.2 C.sub.6 H.sub.5, 4-Br                                           153 2-Cl, 4-CH.sub.2 C.sub.6 H.sub.5                                           154 2-Br, 4-CH.sub.2 C.sub.6 H.sub.5                                           155 2-cyclo-C.sub.6 H.sub.11, 4-Cl                                             156 2-cyclo-C.sub.6 H.sub.11, 4-Br                                             157 2-Cl, 4-cyclo-C.sub.6 H.sub.11                                             158 2-Br, 4-cyclo-C.sub.6 H.sub.11                                             159 2-OCH.sub.3                                                                160 3-OCH.sub.3                                                                161 4-OCH.sub.3                                                                162 2-OC.sub.2 H.sub.5                                                         163 3-O--C.sub.2 H.sub.5                                                       164 4-O--C.sub.2 H.sub.5                                                       165 2-O-n-C.sub.3 H.sub.7                                                      166 3-O-n-C.sub.3 H.sub.7                                                      167 4-O-n-C.sub.3 H.sub.7                                                      168 2-O-i-C.sub.3 H.sub.7                                                      169 3-O-i-C.sub.3 H.sub.7                                                      170 4-O-i-C.sub.3 H.sub.7                                                      171 2-O-n-C.sub.6 H.sub.13                                                     172 3-O-n-C.sub.6 H.sub.13                                                     173 4-O-n-C.sub.6 H.sub.13                                                     174 2-O-n-C.sub.8 H.sub.17                                                     175 3-O-n-C.sub.8 H.sub.17                                                     176 4-O-n-C.sub.8 H.sub.17                                                     177 2-O--CH.sub.2 C.sub.6 H.sub.5                                              178 3-O--CH.sub.2 C.sub.6 H.sub.5                                              179 4-O--CH.sub.2 C.sub.6 H.sub.5                                              180 2-O--(CH.sub.2).sub.3 C.sub.6 H.sub.5                                      181 3-O--(CH.sub.2).sub.3 C.sub.6 H.sub.5                                      182 4-O--(CH.sub.2).sub.3 C.sub.6 H.sub.5                                      183 2,4-(OCH.sub.3).sub.2                                                      184 2-CF.sub.3                                                                 185 3-CF.sub.3                                                                 186 4-CF.sub.3                                                                 187 2-OCF.sub.3                                                                188 3-OCF.sub.3                                                                189 4-OCF.sub.3                                                                190 3-OCH.sub.2 CHF.sub.2                                                      191 2-NO.sub.2                                                                 192 3-NO.sub.2                                                                 193 4-NO.sub.2                                                                 194 2-CN                                                                       195 3-CN                                                                       196 4-CN                                                                       197 2-CH.sub.3, 3-Cl                                                           198 2-CH.sub.3, 4-Cl                                                           199 2-CH.sub.3, 5-Cl                                                           200 2-CH.sub.3, 6-Cl                                                           201 2-CH.sub.3, 3-F                                                            202 2-CH.sub.3, 4-F                                                            203 2-CH.sub.3, 5-F                                                            204 2-CH.sub.3, 6-F                                                            205 2-CH.sub.3, 3-Br                                                           206 2-CH.sub.3, 4-Br                                                           207 2-CH.sub.3, 5-Br                                                           208 2-CH.sub.3, 6-Br                                                           209 2-Cl, 3-CH.sub.3                                                           210 2-Cl, 4-CH.sub.3                                                           211 2-Cl, 5-CH.sub.3                                                           212 2-F, 3-CH.sub.3                                                            213 2-F, 4-CH.sub.3                                                            214 2-F, 5-CH.sub.3                                                            215 2-Br, 3-CH.sub.3                                                           216 2-Br, 4-CH.sub.3                                                           217 2-Br, 5-CH.sub.3                                                           218 3-CH.sub.3, 4-Cl                                                           219 3-CH.sub.3, 5-Cl                                                           220 3-CH.sub.3, 4-F                                                            221 3-CH.sub.3, 5-F                                                            222 3-CH.sub.3, 4-Br                                                           223 3-CH.sub.3, 5-Br                                                           224 3-F, 4-CH.sub.3                                                            225 3-Cl, 4-CH.sub.3                                                           226 3-Br, 4-CH.sub.3                                                           227 2-Cl, 4,5-(CH.sub.3).sub.2                                                 228 2-Br, 4,5-(CH.sub.3).sub.2                                                 229 2-Cl, 3,5-(CH.sub.3).sub.2                                                 230 2-Br, 3,5-(CH.sub.3).sub.2                                                 231 2,6-Cl.sub.2, 4-CH.sub.3                                                   232 2,6-F.sub.2, 4-CH.sub.3                                                    233 2,6-Br.sub.2, 4-CH.sub.3                                                   234 2,4-Br.sub.2, 6-CH.sub.3                                                   235 2,4-F.sub.2, 6-CH.sub.3                                                    236 2,4-Br.sub.2, 6-CH.sub.3                                                   237 2,6-(CH.sub.3).sub.2, 4-F                                                  238 2,6-(CH.sub.3).sub.2, 4-Cl                                                 239 2,6-(CH.sub.3).sub.2, 4-Br                                                 240 3,5-(CH.sub.3).sub.2, 4-F                                                  241 3,5-(CH.sub.3).sub.2, 4-Cl                                                 242 3,5-(CH.sub.3).sub.2, 4-Br                                                 243 2,3,6-(CH.sub.3).sub.3, 4-F                                                244 2,3,6-(CH.sub.3).sub.3, 4-Cl                                               245 2,3,6-(CH.sub.3).sub.3, 4-Br                                               246 2,4-(CH.sub.3).sub.2, 6-F                                                  247 2,4-(CH.sub.3).sub.2, 6-Cl                                                 248 2,4-(CH.sub.3).sub.2, 6-Br                                                 249 2-i-C.sub.3 H.sub.7, 4-Cl, 5-CH.sub.3                                      250 2-Cl, 4-NO.sub.2                                                           251 2-NO.sub.2, 4-Cl                                                           252 2-OCH.sub.3, 5-NO.sub.2                                                    253 2,4-Cl.sub.2, 5-NO.sub.2                                                   254 2,4-Cl.sub.2, 6-NO.sub.2                                                   255 2,6-Cl.sub.2, 4-NO.sub.2                                                   256 2,6-Br.sub.2, 4-NO.sub.2                                                   257 2,6-I.sub.2, 4-NO.sub.2                                                    258 2-CH.sub.3, 5-i-C.sub.3 H.sub.7, 4-Cl                                      259 2-CO.sub.2 CH.sub.3                                                        260 3-CO.sub.2 CH.sub.3                                                        261 4-CO.sub.2 CH.sub.3                                                        262 2-CO.sub.2 (C.sub.2 H.sub.5)                                               263 3-CO.sub.2 (C.sub.2 H.sub.5)                                               264 4-CO.sub.2 (C.sub.2 H.sub.5)                                               265 2-CO.sub.2 (n-C.sub.3 H.sub.7)                                             266 3-CO.sub.2 (n-C.sub.3 H.sub.7)                                             267 4-CO.sub.2 (n-C.sub.3 H.sub.7)                                             268 2-CO.sub.2 (i-C.sub.3 H.sub.7)                                             269 3-CO.sub.2 (i-C.sub.3 H.sub.7)                                             270 4-CO.sub.2 (i-C.sub.3 H.sub.7)                                             271 2-CO.sub.2 (n-C.sub.6 H.sub.13)                                            272 3-CO.sub.2 (n-C.sub.6 H.sub.13)                                            273 4-CO.sub.2 (n-C.sub.6 H.sub.13)                                            274 2-CH.sub.2 --OCH.sub.3                                                     275 3-CH.sub.2 --OCH.sub.3                                                     276 4-CH.sub.2 --OCH.sub.3                                                     277 2-CH.sub.2 O(C.sub.2 H.sub.5)                                              278 3-CH.sub.2 O(C.sub.2 H.sub.5)                                              279 4-CH.sub.2 O(C.sub.2 H.sub.5)                                              280 2-CH.sub.2 O(n-C.sub.3 H.sub.7)                                            281 3-CH.sub.2 O(n-C.sub.3 H.sub.7)                                            282 4-CH.sub.2 O(n-C.sub.3 H.sub.7)                                            283 2-CH.sub.2 O(i-C.sub.3 H.sub.7)                                            284 3-CH.sub.2 O(i-C.sub.3 H.sub.7)                                            285 4-CH.sub.2 O(i-C.sub.3 H.sub.7)                                            286 2-CHO                                                                      287 3-CHO                                                                      288 4-CHO                                                                      289 2-CO--CH.sub.3                                                             290 3-CO--CH.sub.3                                                             291 4-CO--CH.sub.3                                                             292 2-CO--CH.sub.2 --CH.sub.3                                                  293 3-CO--CH.sub.2 --CH.sub.3                                                  294 4-CO--CH.sub.2 --CH.sub.3                                                  295 2-CO--CH.sub.2 --CH.sub.2 --CH.sub.3                                       296 3-CO--CH.sub.2 --CH.sub.2 --CH.sub.3                                       297 4-CO--CH.sub.2 --CH.sub.2 --CH.sub.3                                       298 2-CO--CH(CH.sub.3)--CH.sub.3                                               299 3-CO--CH(CH.sub.3)--CH.sub.3                                               300 4-CO--CH(CH.sub.3)--CH.sub.3                                               301 2-Me-4-CHO                                                                 302 2-Me-4-CH.sub.3 --CO                                                       303 2-Me-4-CH.sub.3 --CH.sub.2 --CO                                            304 2-Me-4-CH.sub.3 --CH.sub.2 --CH.sub.2 --CO                                 305 2-Me-4-CH.sub.3 --CH(CH.sub.3)--CO                                         306 2,5-Me.sub.2 -4-CHO                                                        307 2,5-Me.sub.2 -4-CH.sub.3 --CO                                              308 2,5-Me.sub.2 -4-CH.sub.3 --CH.sub.2 --CO                                   309 2,5-Me.sub.2 -4-CH.sub.3 --CH.sub.2 --CH.sub.2 --CO                        310 2,5-Me.sub.2 -4-CO--CH(CH.sub.3)--CO                                       311 2-Cl-4-CHO                                                                 312 2-Cl-4-CH.sub.3 --CO                                                       313 2-Cl-4-CH.sub.3 --CH.sub.2 --CO                                            314 2-Cl-4-CH.sub.3 --CH(CH.sub.3)--CO                                         315 2,5-Cl.sub.2 -4-CHO                                                        316 2,5-Cl.sub.2 -4-CH.sub.3 --CO                                              317 2,5-Cl.sub.2 -4-CH.sub.3 --CH.sub.2 --CO                                   318 2,5-Cl.sub.2 -4-CH.sub.3 --CH.sub.2 --CH.sub.2 --CO                        319 2,5-Cl.sub.2 -4-CH.sub.3 --CH(CH.sub.3)--CO                                320 2-C(═NOCH.sub.3)--CH.sub.3                                             321 3-C(═NOCH.sub.3)--CH.sub.3                                             322 4-C(═NOCH.sub.3)--CH.sub.3                                             323 2-C(═NOC.sub.2 H.sub.5)--CH.sub.3                                      324 3-C(═NOC.sub.2 H.sub.5)--CH.sub.3                                      325 4-C(═NOC.sub.2 H.sub.5)--CH.sub.3                                      326 2-C(═NO-n-C.sub.3 H.sub.7)--CH.sub.3                                   327 3-C(═NO-n-C.sub.3 H.sub.7)--CH.sub.3                                   328 4-C(═NO-n-C.sub.3 H.sub.7)--CH.sub.3                                   329 2-C(═NO-i-C.sub.3 H.sub.7)--CH.sub.3                                   330 3-C(═NO-i-C.sub.3 H.sub.7)--CH.sub.3                                   331 4-C(═NO-i-C.sub.3 H.sub.7)--CH.sub.3                                   332 2-C(═NO-Allyl)--CH.sub.3                                               333 3-C(═NO-Allyl)--CH.sub.3                                               334 4-C(═NO-Allyl)--CH.sub.3                                               335 2-C(═NO-trans-Chloroallyl)--CH.sub.3                                   336 3-C(═NO-trans-Chloroallyl)--CH.sub.3                                   337 4-C(═NO-trans-Chloroallyl)--CH.sub.3                                   338 2-C(═NO-Propargyl)--CH.sub.3                                           339 3-C(═NO-Propargyl)--CH.sub.3                                           340 4-C(═NO-Propargyl)--CH.sub.3                                           341 2-C(═NO-n-C.sub.4 H.sub.9)--CH.sub.3                                   342 3-C(═NO-n-C.sub.4 H.sub.9)--CH.sub.3                                   343 4-C(═NO-n-C.sub.4 H.sub.9)--CH.sub.3                                   344 2-C(═NO--CH.sub.2 --C.sub.6 H.sub.5)--CH.sub.3                         345 3-C(═NO--CH.sub.2 --C.sub.6 H.sub.5)--CH.sub.3                         346 4-C(═NO--CH.sub.2 --C.sub.6 H.sub.5)--CH.sub.3                         347 2-CH.sub.3 -4-CH═NOCH.sub.3                                            348 2-CH.sub.3 -4-CH═NOC.sub.2 H.sub.5                                     349 2-CH.sub.3 -4-CH═NO-n-C.sub.3 H.sub.7                                  350 2-CH.sub.3 -4-CH═NO-i-C.sub.3 H.sub.7                                  351 2-CH.sub.3 -4-CH═NO-Allyl                                              352 2-CH.sub.3 -4-CH═NO-(trans-Chloroallyl)                                353 2-CH.sub.3 -4-CH═NO-Propargyl                                          354 2-CH.sub.3 -4-CH═NO-n-C.sub.4 H.sub.9                                  355 2-CH.sub.3 -4-CH═NO--CH.sub.2 --C.sub.6 H.sub.5                        356 2-CH.sub.3 -4-(CH.sub.3 --C═NOCH.sub.3)                                357 2-CH.sub.3 -4-(CH.sub.3 --C═NOC.sub.2 H.sub.5)                         358 2-CH.sub.3 -4-(CH.sub.3 --C═NO-n-C.sub.3 H.sub.7)                      359 2-CH.sub.3 -4-(CH.sub.3 --C═NO-i-C.sub.3 H.sub.7)                      360 2-CH.sub.3 -4-(CH.sub.3 --C═NO-Allyl)                                  361 2-CH.sub.3 -4-(CH.sub.3 --C═NO-trans-Chloroallyl)                      362 2-CH.sub.3 -4-(CH.sub.3 --C═NO-Propargyl)                              363 2-CH.sub.3 -4-(CH.sub.3 --C═NO-n-C.sub.4 H.sub.9)                      364 2-CH.sub.3 -4-(CH.sub.3 --C═NO--CH.sub.2 --C.sub.6 H.sub.5)                     365 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C═NO--CH.sub.3)                       366 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C═NO--C.sub.2                        H.sub.5)                                                               367 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C═NO-n-C.sub.3 H.sub.7)                        368 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C═NO-i-C.sub.3                       H.sub.7                                                                369 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C═NO-Allyl)                           370 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C═NO-trans-Chloroallyl)                        371 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C═NO-Propargyl)                       372 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C═NO-n-C.sub.4                       H.sub.9)                                                               373 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C═NO--CH.sub.2 --C.sub.6                      H.sub.5)                                                               374 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C═NOCH.sub.3)                      375 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C═NOC.sub.2 H.sub.5)                        376 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C═NO-n-C.sub.3                    H.sub.7)                                                               377 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C═NO-i-C.sub.3 H.sub.7)                     378 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C═NO-Allyl)                        379 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C═NO-trans-Chloroal               lyl)                                                                   380 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C═NO-Proparyl)                     381 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C═NO-n-C.sub.4 H.sub.9)                     382 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C═NO--CH.sub.2                    --C.sub.6 H.sub.5)                                                     383 2-C.sub.6 H.sub.5                                                          384 3-C.sub.6 H.sub.5                                                          385 4-C.sub.6 H.sub.5                                                          386 2-(2'-F--C.sub.6 H.sub.4)                                                  387 2-(3'-F--C.sub.6 H.sub.4)                                                  388 2-(4'-F--C.sub.6 H.sub.4)                                                  389 3-(2'-F--C.sub.6 H.sub.4)                                                  390 3-(3'-F--C.sub.6 H.sub.4)                                                  391 3-(4'-F--C.sub.6 H.sub.4)                                                  392 4-(2'-F--C.sub.6 H.sub.4)                                                  393 4-(3'-F--C.sub.6 H.sub.4)                                                  394 4-(4'-F--C.sub.6 H.sub.4)                                                  395 2-(2'-Cl--C.sub.6 H.sub.4)                                                 396 2-(3'-Cl--C.sub.6 H.sub.4)                                                 397 2-(4'-Cl--C.sub.6 H.sub.4)                                                 398 3-(2'-Cl--C.sub.6 H.sub.4)                                                 399 3-(3'-Cl--C.sub.6 H.sub.4)                                                 400 3-(4'-Cl--C.sub.6 H.sub.4)                                                 401 4-(2'-Cl--C.sub.6 H.sub.4)                                                 402 4-(3'-Cl--C.sub.6 H.sub.4)                                                 403 4-(4'-Cl--C.sub.6 H.sub.4)                                                 405 2-(2'-CH.sub.3 --C.sub.6 H.sub.4)                                          406 2-(3'-CH.sub.3 --C.sub.6 H.sub.4)                                          407 2-(4'-CH.sub.3 --C.sub.6 H.sub.4)                                          408 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)                                          409 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)                                          410 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)                                          411 4-(2'-CH.sub.3 --C.sub.6 H.sub.4)                                          412 4-(3'-CH.sub.3 --C.sub.6 H.sub.4)                                          413 4-(4'-CH.sub.3 --C.sub.6 H.sub.4)                                          414 2-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                      415 2-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                      416 2-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                      417 3-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                      418 3-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                      419 3-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                      420 4-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                      421 4-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                      422 4-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                      423 2-(2'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                       424 2-(3'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                       425 2-(4'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                       426 3-(2'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                       427 3-(3'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                       428 3-(4'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                       429 4-(2'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                       430 4-(3'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                       431 4-(4'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                       432 2-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                                 433 2-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                                 434 2-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                                 435 3-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                                 436 3-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                                 437 3-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                                 438 4-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                                 439 4-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                                 440 4-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                                 441 2-(2'-CH.sub.3 O--C.sub.6 H.sub.4)                                         442 2-(3'-CH.sub.3 O--C.sub.6 H.sub.4)                                         443 2-(4'-CH.sub.3 O--C.sub.6 H.sub.4)                                         444 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)                                         445 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)                                         446 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)                                         447 4-(2'-CH.sub.3 O--C.sub.6 H.sub.4)                                         448 4-(3'-CH.sub.3 O--C.sub.6 H.sub.4)                                         449 4-(4'-CH.sub.3 O--C.sub.6 H.sub.4)                                         450 2-(2'-O.sub.2 N--C.sub.6 H.sub.4)                                          451 2-(3'-O.sub.2 N--C.sub.6 H.sub.4)                                          452 2-(4'-O.sub.2 N--C.sub.6 H.sub.4)                                          453 3-(2'-O.sub.2 N--C.sub.6 H.sub.4)                                          454 3-(3'-O.sub.2 N--C.sub.6 H.sub.4)                                          455 3-(4'-O.sub.2 N--C.sub.6 H.sub.4)                                          456 4-(2'-O.sub.2 N--C.sub.6 H.sub.4)                                          457 4-(3'-O.sub.2 N--C.sub.6 H.sub.4)                                          458 4-(4'-O.sub.2 N--C.sub.6 H.sub.4)                                          459 2-(2'-NC--C.sub.6 H.sub.4)                                                 460 2-(3'-NC--C.sub.6 H.sub.4)                                                 461 2-(4'-NC--C.sub.6 H.sub.4)                                                 462 3-(2'-NC--C.sub.6 H.sub.4)                                                 463 3-(3'-NC--C.sub.6 H.sub.4)                                                 464 3-(4'-NC--C.sub.6 H.sub.4)                                                 465 4-(2'-NC--C.sub.6 H.sub.4)                                                 466 4-(3'-NC--C.sub.6 H.sub.4)                                                 467 4-(4'-NC--C.sub.6 H.sub.4)                                                 468 2-(2'-CF.sub.3 --C.sub.6 H.sub.4)                                          469 2-(3'-CF.sub.3 --C.sub.6 H.sub.4)                                          470 2-(4'-CF.sub.3 --C.sub.6 H.sub.4)                                          471 3-(2'-CF.sub.3 --C.sub.6 H.sub.4)                                          472 3-(3'-CF.sub.3 --C.sub.6 H.sub.4)                                          473 3-(4'-CF.sub.3 --C.sub.6 H.sub.4)                                          474 4-(2'-CF.sub.3 --C.sub.6 H.sub.4)                                          475 4-(3'-CF.sub.3 --C.sub.6 H.sub.4)                                          476 4-(4'-CF.sub.3 --C.sub.6 H.sub.4)                                          477 2-O--C.sub.6 H.sub.5                                                       475 3-O--C.sub.6 H.sub.5                                                       476 4-O--C.sub.6 H.sub.5                                                       478 2-O-(2'-F--C.sub.6 H.sub.4)                                                479 2-O-(3'-F--C.sub.6 H.sub.4)                                                480 2-O-(4'-F--C.sub.6 H.sub.4)                                                481 3-O-(2'-F--C.sub.6 H.sub.4)                                                482 3-O-(3'-F--C.sub.6 H.sub.4)                                                483 3-O-(4'-F--C.sub.6 H.sub.4)                                                484 4-O-(2'-F--C.sub.6 H.sub.4)                                                485 4-O-(3'-F--C.sub.6 H.sub.4)                                                486 4-O-(4'-F--C.sub.6 H.sub.4)                                                487 2-O-(2'-Cl--C.sub.6 H.sub.4)                                               488 2-O-(3'-Cl--C.sub.6 H.sub.4)                                               489 2-O-(4'-Cl--C.sub.6 H.sub.4)                                               490 3-O-(2'-Cl--C.sub.6 H.sub.4)                                               491 3-O-(3'-Cl--C.sub.6 H.sub.4)                                               492 3-O-(4'-Cl--C.sub.6 H.sub.4)                                               493 3-O-(4'-Cl--C.sub.6 H.sub.4)                                               494 4-O-(2'-Cl--C.sub.6 H.sub.4)                                               495 4-O-(3'-Cl--C.sub.6 H.sub.4)                                               496 4-O-(4'-Cl--C.sub.6 H.sub.4)                                               497 2-O-(2'-CH.sub.3 --C.sub.6 H.sub.4)                                        498 2-O-(3'-CH.sub.3 --C.sub.6 H.sub.4)                                        499 2-O-(4'-CH.sub.3 --C.sub.6 H.sub.4)                                        500 3-O-(2'-CH.sub.3 --C.sub.6 H.sub.4)                                        501 3-O-(3'-CH.sub.3 --C.sub.6 H.sub.4)                                        502 3-O-(4'-CH.sub.3 --C.sub.6 H.sub.4)                                        503 4-O-(2'-CH.sub.3 --C.sub.6 H.sub.4)                                        504 4-O-(3'-CH.sub.3 --C.sub.6 H.sub.4)                                        505 4-O-(4'-CH.sub.3 --C.sub.6 H.sub.4)                                        506 2-O-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                    507 2-O-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                    508 2-O-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                    509 3-O-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                    510 3-O-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                    511 3-O-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                    512 4-O-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                    513 4-O-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                    514 4-O-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                    515 2-O-(2'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                     516 2-O-(3'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                     517 2-O-(4'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                     518 3-O-(2'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                     519 3-O-(3'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                     520 3-O-(4'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                     521 4-O-(2'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                     522 4-O-(3'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                     523 4-O-(4'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                     524 2-O-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                               525 2-O-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                               526 2-O-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                               527 3-O-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                               528 3-O-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                               529 3-O-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                               530 4-O-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                               531 4-O-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                               532 4-O-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                               533 2-O-(2'-CH.sub.3 O--C.sub.6 H.sub.4)                                       534 2-O-(3'-CH.sub.3 O--C.sub.6 H.sub.4)                                       535 2-O-(4'-CH.sub.3 O--C.sub.6 H.sub.4)                                       536 3-O-(2'-CH.sub.3 O--C.sub.6 H.sub.4)                                       537 3-O-(3'-CH.sub.3 O--C.sub.6 H.sub.4)                                       538 3-O-(4'-CH.sub.3 O--C.sub.6 H.sub.4)                                       539 4-O-(2'-CH.sub.3 O--C.sub.6 H.sub.4)                                       540 4-O-(3'-CH.sub.3 O--C.sub.6 H.sub.4)                                       541 4-O-(4'-CH.sub.3 O--C.sub.6 H.sub.4)                                       542 2-O-(2'-O.sub.2 N--C.sub.6 H.sub.4)                                        543 2-O-(3'-O.sub.2 N--C.sub.6 H.sub.4)                                        544 2-O-(4'-O.sub.2 N--C.sub.6 H.sub.4)                                        545 3-O-(2'-O.sub.2 N--C.sub.6 H.sub.4)                                        546 3-O-(3'-O.sub.2 N--C.sub.6 H.sub.4)                                        547 3-O-(4'-O.sub.2 N--C.sub.6 H.sub.4)                                        548 4-O-(2'-O.sub.2 N--C.sub.6 H.sub.4)                                        549 4-O-(3'-O.sub.2 N--C.sub.6 H.sub.4)                                        550 4-O-(4'-O.sub.2 N--C.sub.6 H.sub.4)                                        551 2-O-(2'-NC--C.sub.6 H.sub.4)                                               552 2-O-(3'-NC--C.sub.6 H.sub.4)                                               553 2-O-(4'-NC--C.sub.6 H.sub.4)                                               554 3-O-(2'-NC--C.sub.6 H.sub.4)                                               555 3-O-(3'-NC--C.sub.6 H.sub.4)                                               556 3-O-(4'-NC--C.sub.6 H.sub.4)                                               557 4-O-(2'-NC--C.sub.6 H.sub.4)                                               558 4-O-(3'-NC--C.sub.6 H.sub.4)                                               559 4-O-(4'-NC--C.sub.6 H.sub.4)                                               560 2-O-(2'-CF.sub.3 --C.sub.6 H.sub.4)                                        561 2-O-(3'-CF.sub.3 --C.sub.6 H.sub.4)                                        562 2-O-(4'-CF.sub.3 --C.sub.6 H.sub.4)                                        563 3-O-(2'-CF.sub.3 --C.sub.6 H.sub.4)                                        564 3-O-(3'-CF.sub.3 --C.sub.6 H.sub.4)                                        565 3-O-(4'-CF.sub.3 --C.sub.6 H.sub.4)                                        566 4-O-(2'-CF.sub.3 --C.sub.6 H.sub.4)                                        567 4-O-(3'-CF.sub.3 --C.sub.6 H.sub.4)                                        568 4-O-(4'-CF.sub.3 --C.sub.6 H.sub.4)                                        569 2-Pyridinyl-2'                                                             570 2-Pyridinyl-3'                                                             571 2-Pyridinyl-4'                                                             572 3-Pyridinyl-2'                                                             573 3-Pyridinyl-3'                                                             574 3-Pyridinyl-4'                                                             575 4-Pyridinyl-2'                                                             576 4-Pyridinyl-3'                                                             577 4-Pyridinyl-4'                                                             578 2-Pyrimidinyl-2'                                                           579 2-Pyrimidinyl-3'                                                           580 2-Pyrimidinyl-4'                                                           581 3-Pyrimidinyl-2'                                                           582 3-Pyrimidinyl-3'                                                           583 3-Pyrimidinyl-4'                                                           584 4-Pyrimidinyl-2'                                                           585 4-Pyrimidinyl-3'                                                           586 4-Pyrimidinyl-4'                                                           587 2-Pyrazolyl-1'                                                             588 2-Pyrazolyl-3'                                                             589 2-Pyrazolyl-4'                                                             590 3-Pyrazolyl-1'                                                             591 3-Pyrazolyl-3'                                                             592 3-Pyrazolyl-4'                                                             593 4-Pyrazolyl-1'                                                             594 4-Pyrazolyl-3'                                                             595 4-Pyrazolyl-4'                                                             596 2-Isoxazolyl-3'                                                            597 2-Isoxazolyl-4'                                                            598 2-Isoxazolyl-5'                                                            599 3-Isoxazolyl-3'                                                            600 3-Isoxazolyl-4'                                                            601 3-Isoxazolyl-5'                                                            602 4-Isoxazolyl-3'                                                            603 4-Isoxazolyl-4'                                                            604 4-Isoxazolyl-5'                                                            605 2-Isothiazolyl-3'                                                          606 2-Isothiazolyl-4'                                                          607 2-Isothiazolyl-5'                                                          608 3-Isothiazolyl-3'                                                          609 3-Isothiazolyl-4'                                                          610 3-Isothiazolyl-5'                                                          611 4-Isothiazolyl-3'                                                          612 4-Isothiazolyl-4'                                                          613 4-Isothiazolyl-5'                                                          614 2-Imidazolyl-1'                                                            615 2-Imidazolyl-2'                                                            616 2-Imidazolyl-4'                                                            617 3-Imidazolyl-1'                                                            618 3-Imidazolyl-2'                                                            619 3-Imidazolyl-4'                                                            620 4-Imidazolyl-1'                                                            621 4-Imidazolyl-2'                                                            622 4-Imidazolyl-4'                                                            623 2-Oxazolyl-2'                                                              624 2-Oxazolyl-4'                                                              625 2-Oxazolyl-5'                                                              626 3-Oxazolyl-2'                                                              627 3-Oxazolyl-4'                                                              628 3-Oxazolyl-5'                                                              629 4-Oxazolyl-2'                                                              630 4-Oxazolyl-4'                                                              631 4-Oxazolyl-5'                                                              632 2-Thiazolyl-2'                                                             633 2-Thiazolyl-4'                                                             634 2-Thiazolyl-5'                                                             635 3-Thiazolyl-2'                                                             636 3-Thiazolyl-4'                                                             637 3-Thiazolyl-5'                                                             638 4-Thiazolyl-2'                                                             639 4-Thiazolyl-4'                                                             640 4-Thiazolyl-5'                                                             641 2-CH.sub.3 -4-(CH.sub.3 --C═N--O--CH.sub.2 --CH.sub.2 --OCH.sub.               3)                                                                     642 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C═N--O--CH.sub.2 --CH.sub.2                   --OCH.sub.3)                                                           643 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C═N--O--CH.sub.2 --CH.sub.2                --OCH.sub.3)                                                           644 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C═N--OCH.sub.3)                     645 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C═N--OC.sub.2 H.sub.5)                       646 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C═N--O-n-C.sub.3                   H.sub.7)                                                               647 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C═N--O-i-C.sub.3 H.sub.7)                    648 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C═N--O-Allyl)                       649 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C═N--O-trans-Chloroa               llyl)                                                                  650 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C═N--O-Propargyl)                   651 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C═N--O-n-C.sub.4 H.sub.9)                    652 2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 --C═N--O--CH.sub.2                   --C.sub.6 H.sub.5)                                                     653 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C═N--OCH.sub.3)                     654 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C═N--OC.sub.2 H.sub.5)                       655 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C═N--O-n-C.sub.3                   H.sub.7)                                                               656 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C═N--O-i-C.sub.3 H.sub.7)                    657 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C═N--O-Allyl)                       658 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C═N--O-trans-Chloroa               llyl)                                                                  659 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C═N--O-Propargyl)                   660 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C═N--O-n-C.sub.4 H.sub.9)                    661 2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 --C═N--O--CH.sub.2                   --C.sub.6 H.sub.5)                                                     662 2-O-n-C.sub.4 H.sub.9                                                      663 2-O-i-C.sub.4 H.sub.9                                                      664 2-O-s-C.sub.4 H.sub.9                                                      665 2-O-t-C.sub.4 H.sub.9                                                      666 2-Neopentyloxy                                                             667 3-O-n-C.sub.4 H.sub.9                                                      668 3-O-i-C.sub.4 H.sub.9                                                      669 3-O-s-C.sub.4 H.sub.9                                                      670 3-O-t-C.sub.4 H.sub.9                                                      671 3-Neopentyloxy                                                             672 4-O-n-C.sub.4 H.sub.9                                                      673 4-O-i-C.sub.4 H.sub.9                                                      674 4-O-s-C.sub.4 H.sub.9                                                      675 4-O-t-C.sub.4 H.sub.9                                                      676 4-Neopentyloxy                                                             677 3-CH.sub.3 -4-OCH.sub.3                                                    678 3-CH.sub.3 -4-OC.sub.2 H.sub.5                                             679 3-CH.sub.3 -4-O-n-C.sub.3 H.sub.7                                          680 3-CH.sub.3 -4-O-n-C.sub.4 H.sub.9                                          681 3-CH.sub.3 -4-O-i-C.sub.4 H.sub.9                                          682 3-CH.sub.3 -4-O-s-C.sub.4 H.sub.9                                          683 3-CH.sub.3 -4-O-t-C.sub.4 H.sub.9                                          684 3-CH.sub.3 -4-Neopentyloxy                                                 685 2-CH.sub.3 -3-OCH.sub.3                                                    686 2-CH.sub.3 -4-OCH.sub.3                                                    687 2-CH.sub.3 -5-OCH.sub.3                                                    688 2-CH.sub.3 -6-OCH.sub.3                                                    689 3-CH.sub.3 -4-OCH.sub.3                                                    690 3-CH.sub.3 -5-OCH.sub.3                                                    691 3-CH.sub.3 -6-OCH.sub.3                                                    692 4-CH.sub.3 -5-O--CH.sub.3                                                  693 4-CH.sub.3 -6-O--CH.sub.3                                                  694 4-CH.sub.3 -6-OCH.sub.3                                                    695 2-CH.sub.3 -3-O-i-C.sub.3 H.sub.7                                          696 2-CH.sub.3 -4-O-i-C.sub.3 H.sub.7                                          697 2-CH.sub.3 -5-O-i-C.sub.3 H.sub.7                                          698 2-CH.sub.3 -6-O-i-C.sub.3 H.sub.7                                          699 3-CH.sub.3 -4-O-i-C.sub.3 H.sub.7                                          700 3-CH.sub.3 -5-O-i-C.sub.3 H.sub.7                                          701 3-CH.sub.3 -6-O-i-C.sub.3 H.sub.7                                          702 4-CH.sub.3 -5-O-i-C.sub.3 H.sub.7                                          703 4-CH.sub.3 -6-O-i-C.sub.3 H.sub.7                                          704 5-CH.sub.3 -6-O-i-C.sub.3 H.sub.7                                          705 2-Cl-3-OCH.sub.3                                                           706 2-Cl-4-OCH.sub.3                                                           707 2-Cl-5-OCH.sub.3                                                           708 2-Cl-6-OCH.sub.3                                                           709 3-Cl-4-OCH.sub.3                                                           710 3-Cl-5-OCH.sub.3                                                           711 3-Cl-6-OCH.sub.3                                                           712 4-Cl-5-OCH.sub.3                                                           713 4-Cl-6-OCH.sub.3                                                           714 5-Cl-6-OCH.sub.3                                                         ______________________________________                                    

                  TABLE 44                                                         ______________________________________                                         0  STR277##                                                                       -                                                                             I: R.sup.1 = H, X = CH.sub.3                                                   II: R.sup.1 = CH.sub.3, X = CH.sub.3                                           III: R.sup.1 = C.sub.2 H.sub.5, X = CH.sub.3                                   IV: R.sup.1 = Allyl, X = CH.sub.3                                              V: R.sup.1 = Propargyl, X = CH.sub.3                                           VI: R.sup.1 = CH.sub.2 --OCH.sub.3, X = CH.sub.3                               VII: R.sup.1 = CO.sub.2 CH.sub.3, X = CH.sub.3                                 VIII: R.sup.1 = H, X = Cl                                                      IX: R.sup.1 = CH.sub.3, X = Cl                                                 X: R.sup.1 = C.sub.2 H.sub.5, X = Cl                                           XI: R.sup.1 = Allyl, X = Cl                                                    XII: R.sup.1 = Propargyl, X = Cl                                               XIII: R.sup.1 = CH.sub.2 --OCH.sub.3, X = Cl                                   XIV: R.sup.1 = CO.sub.2 CH.sub.3, X = Cl                                        -                                                                           No.       B                                                                    ______________________________________                                         1         Pyrrolyl-3                                                             2 N--CH.sub.3 -Pyrrolyl-3                                                      3 N--C.sub.6 H.sub.5 -Pyrrolyl-3                                               4 N-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrrolyl-3                                 5 N-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrrolyl-3                                 6 N-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrrolyl-3                                 7 N-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrrolyl-3                                8 N-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrrolyl-3                                9 N-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrrolyl-3                                10 N-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrrolyl-3                                11 N-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrrolyl-3                                12 N-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrrolyl-3                                13 N-(4'-CN--C.sub.6 H.sub.4)-Pyrrolyl-3                                       14 N-(3'-CN--C.sub.6 H.sub.4)-Pyrrolyl-3                                       15 N-(2'-CN--C.sub.6 H.sub.4)-Pyrrolyl-3                                       16 N-(4'-Cl--C.sub.6 H.sub.4)-Pyrrolyl-3                                       17 N-(3'-Cl--C.sub.6 H.sub.4)-Pyrrolyl-3                                       18 N-(2'-Cl--C.sub.6 H.sub.4)-Pyrrolyl-3                                       19 Pyrrolyl-2                                                                  20 N--CH.sub.3 -Pyrrolyl-2                                                     21 N--C.sub.6 H.sub.5 -Pyrrolyl-2                                              22 N-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrrolyl-2                                23 N-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrrolyl-2                                24 N-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrrolyl-2                                25 N-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrrolyl-2                               26 N-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrrolyl-2                               27 N-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrrolyl-2                               28 N-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrrolyl-2                                29 N-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrrolyl-2                                30 N-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrrolyl-2                                31 N-(4'-CN--C.sub.6 H.sub.4)-Pyrrolyl-2                                       32 N-(3'-CN--C.sub.6 H.sub.4)-Pyrrolyl-2                                       33 N-(2'-CN--C.sub.6 H.sub.4)-Pyrrolyl-2                                       34 N-(4'-Cl--C.sub.6 H.sub.4)-Pyrrolyl-2                                       35 N-(3'-Cl--C.sub.6 H.sub.4)-Pyrrolyl-2                                       36 N-(2'-Cl--C.sub.6 H.sub.4)-Pyrrolyl-2                                       37 Furyl-2                                                                     38 5-CH.sub.3 -Furyl-2                                                         39 5-C.sub.6 H.sub.5 -Furyl-2                                                  40 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Furyl-2                                   41 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Furyl-2                                   42 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Furyl-2                                   43 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Furyl-2                                  44 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Furyl-2                                  45 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Furyl-2                                  46 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Furyl-2                                   47 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Furyl-2                                   48 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Furyl-2                                   49 5-(4'-CN--C.sub.6 H.sub.4)-Furyl-2                                          50 5-(3'-CN--C.sub.6 H.sub.4)-Furyl-2                                          51 5-(2'-CN--C.sub.6 H.sub.4)-Furyl-2                                          52 5-(4'-Cl--C.sub.6 H.sub.4)-Furyl-2                                          53 5-(3'-Cl--C.sub.6 H.sub.4)-Furyl-2                                          54 5-(2'-Cl--C.sub.6 H.sub.4)-Furyl-2                                          55 4-CH.sub.3 -Furyl-2                                                         56 4-C.sub.6 H.sub.5 -Furyl-2                                                  57 4-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Furyl-2                                   58 4-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Furyl-2                                   59 4-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Furyl-2                                   60 4-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Furyl-2                                  61 4-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Furyl-2                                  62 4-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Furyl-2                                  63 4-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Furyl-2                                   64 4-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Furyl-2                                   65 4-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Furyl-2                                   66 4-(4'-CN--C.sub.6 H.sub.4)-Furyl-2                                          67 4-(3'-CN--C.sub.6 H.sub.4)-Furyl-2                                          68 4-(2'-CN--C.sub.6 H.sub.4)-Furyl-2                                          69 4-(4'-Cl--C.sub.6 H.sub.4)-Furyl-2                                          70 4-(3'-Cl--C.sub.6 H.sub.4)-Furyl-2                                          71 4-(2'-Cl--C.sub.6 H.sub.4)-Furyl-2                                          72 Thienyl-2                                                                   73 5-CH.sub.3 -Thienyl-2                                                       74 5-C.sub.6 H.sub.5 -Thienyl-2                                                75 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-2                                 76 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-2                                 77 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-2                                 78 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-2                                79 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-2                                80 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-2                                81 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-2                                 82 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-2                                 83 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-2                                 84 5-(4'-CN--C.sub.6 H.sub.4)-Thienyl-2                                        85 5-(3'-CN--C.sub.6 H.sub.4)-Thienyl-2                                        86 5-(2'-CN--C.sub.6 H.sub.4)-Thienyl-2                                        87 5-(4'-Cl--C.sub.6 H.sub.4)-Thienyl-2                                        88 5-(3'-Cl--C.sub.6 H.sub.4)-Thienyl-2                                        89 5-(2'-Cl--C.sub.6 H.sub.4)-Thienyl-2                                        90 4-CH.sub.3 -Thienyl-2                                                       91 4-C.sub.6 H.sub.5 -Thienyl-2                                                92 4-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-2                                 93 4-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-2                                 94 4-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-2                                 95 4-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-2                                96 4-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-2                                97 4-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-2                                98 4-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-2                                 99 4-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-2                                 100 4-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-2                                101 4-(4'-CN--C.sub.6 H.sub.4)-Thienyl-2                                       102 4-(3'-CN--C.sub.6 H.sub.4)-Thienyl-2                                       103 4-(2'-CN--C.sub.6 H.sub.4)-Thienyl-2                                       104 4-(4'-Cl--C.sub.6 H.sub.4)-Thienyl-2                                       105 4-(3'-Cl--C.sub.6 H.sub.4)-Thienyl-2                                       106 4-(2'-Cl--C.sub.6 H.sub.4)-Thienyl-2                                       107 Thienyl-3                                                                  108 5-CH.sub.3 -Thienyl-3                                                      109 5-C.sub.6 H.sub.5 -Thienyl-3                                               110 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-3                                111 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-3                                112 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-3                                113 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-3                               114 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-3                               115 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-3                               116 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-3                                117 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-3                                118 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-3                                119 5-(4'-CN--C.sub.6 H.sub.4)-Thienyl-3                                       120 5-(3'-CN--C.sub.6 H.sub.4)-Thienyl-3                                       121 5-(2'-CN--C.sub.6 H.sub.4)-Thienyl-3                                       122 5-(4'-Cl--C.sub.6 H.sub.4)-Thienyl-3                                       123 5-(3'-Cl--C.sub.6 H.sub.4)-Thienyl-3                                       124 5-(2'-Cl--C.sub.6 H.sub.4)-Thienyl-3                                       125 Pyrazolyl-4                                                                126 N--CH.sub.3 -Pyrazolyl-4                                                   127 N-C.sub.6 H.sub.5 -Pyrazolyl-4                                             128 N-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrazolyl-4                              129 N-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrazolyl-4                              130 N-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrazolyl-4                              131 N-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrazolyl-4                             132 N-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrazolyl-4                             133 N-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrazolyl-4                             134 N-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrazolyl-4                              135 N-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrazolyl-4                              136 N-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrazolyl-4                              137 N-(4'-CN--C.sub.6 H.sub.4)-Pyrazolyl-4                                     138 N-(3'-CN--C.sub.6 H.sub.4)-Pyrazolyl-4                                     139 N-(2'-CN--C.sub.6 H.sub.4)-Pyrazolyl-4                                     140 N-(4'-Cl--C.sub.6 H.sub.4)-Pyrazolyl-4                                     141 N-(3'-Cl--C.sub.6 H.sub.4)-Pyrazolyl-4                                     142 N-(2'-Cl--C.sub.6 H.sub.4)-Pyrazolyl-4                                     143 3-CH.sub.3 --N-Methylpyrazolyl-4                                           144 3-C.sub.6 H.sub.5 --N-Methylpyrazolyl-4                                    145 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)-N-Methylpyrazolyl-4                      146 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)-N-Methylpyrazolyl-4                      147 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)-N-Methylpyrazolyl-4                      148 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-N-Methylpyrazolyl-4                     149 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-N-Methylpyrazolyl-4                     150 3-(2'-CH.sub.3 O-C.sub.6 H.sub.4)-N-Methylpyrazolyl-4                      151 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)-N-Methylpyrazolyl-4                      152 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)-N-Methylpyrazolyl-4                      153 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)-N-Methylpyrazolyl-4                      154 3-(4'-CN--C.sub.6 H.sub.4)-N-Methylpyrazolyl-4                             155 3-(3'-CN--C.sub.6 H.sub.4)-N-Methylpyrazolyl-4                             156 3-(2'-CN--C.sub.6 H.sub.4)-N-Methylpyrazolyl-4                             157 3-(4'-Cl--C.sub.6 H.sub.4)-N-Methylpyrazolyl-4                             158 3-(3'-Cl--C.sub.6 H.sub.4)-N-Methylpyrazolyl-4                             159 3-(2'-Cl--C.sub.6 H.sub.4)-N-Methylpyrazolyl-4                             160 Isoxazolyl-5                                                               161 3-CH.sub.3 -Isoxazolyl-5                                                   162 3-C.sub.6 H.sub.5 -Isoxazolyl-5                                            163 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Isoxazolyl-5                             164 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Isoxazolyl-5                             165 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Isoxazolyl-5                             166 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Isoxazolyl-5                            167 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Isoxazolyl-5                            168 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Isoxazolyl-5                            169 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Isoxazolyl-5                             170 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Isoxazolyl-5                             171 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Isoxazolyl-5                             172 3-(4'-CN--C.sub.6 H.sub.4)-Isoxazolyl-5                                    173 3-(3'-CN--C.sub.6 H.sub.4)-Isoxazolyl-5                                    174 3-(2'-CN--C.sub.6 H.sub.4)-Isoxazolyl-5                                    175 3-(4'-Cl--C.sub.6 H.sub.4)-Isoxazolyl-5                                    176 3-(3'-Cl--C.sub.6 H.sub.4)-Isoxazolyl-5                                    177 3-(2'-Cl--C.sub.6 H.sub.4)-Isoxazolyl-5                                    178 4-Chloroisoxazolyl-5                                                       179 3-CH.sub.3 -4-Chloroisoxazolyl-5                                           180 3-C.sub.6 H.sub.5 -4-Chloroisoxazolyl-5                                    181 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                     182 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                     183 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                     184 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                    185 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                    186 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                    187 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                     188 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                     189 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                     190 3-(4'-CN--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                            191 3-(3'-CN--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                            192 3-(2'-CN--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                            193 3-(4'-Cl--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                            194 3-(3'-Cl--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                            195 3-(2'-Cl--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                            196 Isoxazolyl-3                                                               197 5-CH.sub.3 -Isoxazolyl-3                                                   198 5-C.sub.6 H.sub.5 -Isoxazolyl-3                                            199 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Isoxazolyl-3                             200 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Isoxazolyl-3                             201 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Isoxazolyl-3                             202 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Isoxazolyl-3                            203 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Isoxazolyl-3                            204 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Isoxazolyl-3                            205 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Isoxazolyl-3                             206 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Isoxazolyl-3                             207 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Isoxazolyl-3                             208 5-(4'-CN--C.sub.6 H.sub.4)-Isoxazolyl-3                                    209 5-(3'-CN--C.sub.6 H.sub.4)-Isoxazolyl-3                                    210 5-(2'-CN--C.sub.6 H.sub.4)-Isoxazolyl-3                                    211 5-(4'-Cl--C.sub.6 H.sub.4)-Isoxazolyl-3                                    212 5-(3'-Cl--C.sub.6 H.sub.4)-Isoxazolyl-3                                    213 5-(2'-Cl--C.sub.6 H.sub.4)-Isoxazolyl-3                                    214 Isothiazolyl-5                                                             215 3-CH.sub.3 -Isothiazolyl-5                                                 216 3-C.sub.6 H.sub.5 -Isothiazolyl-5                                          217 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Isothiazolyl-5                           218 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Isothiazolyl-5                           219 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Isothiazolyl-5                           220 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Isothiazolyl-5                          221 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Isothiazolyl-5                          222 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Isothiazolyl-5                          223 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Isothiazolyl-5                           224 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Isothiazolyl-5                           225 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Isothiazolyl-5                           226 3-(4'-CN--C.sub.6 H.sub.4)-Isothiazolyl-5                                  227 3-(3'-CN--C.sub.6 H.sub.4)-Isothiazolyl-5                                  228 3-(2'-CN--C.sub.6 H.sub.4)-Isothiazolyl-5                                  229 3-(4'-Cl--C.sub.6 H.sub.4)-Isothiazolyl-5                                  230 3-(3'-Cl--C.sub.6 H.sub.4)-Isothiazolyl-5                                  231 3-(2'-Cl--C.sub.6 H.sub.4)-Isothiazolyl-5                                  232 Oxazolyl-4                                                                 233 3-CH.sub.3 -Oxazolyl-4                                                     234 3-C.sub.6 H.sub.5 -Oxazolyl-4                                              235 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Oxazolyl-4                               236 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Oxazolyl-4                               237 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Oxazolyl-4                               238 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Oxazolyl-4                              239 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Oxazolyl-4                              240 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Oxazolyl-4                              241 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Oxazolyl-4                               242 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Oxazolyl-4                               243 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Oxazolyl-4                               244 3-(4'-CN--C.sub.6 H.sub.4)-Oxazolyl-4                                      245 3-(3'-CN--C.sub.6 H.sub.4)-Oxazolyl-4                                      246 3-(2'-CN--C.sub.6 H.sub.4)-Oxazolyl-4                                      247 3-(4'-Cl--C.sub.6 H.sub.4)-Oxazolyl-4                                      248 3-(3'-Cl--C.sub.6 H.sub.4)-Oxazolyl-4                                      249 3-(2'-Cl--C.sub.6 H.sub.4)-Oxazolyl-4                                      250 Thiazolyl-4                                                                251 2-CH.sub.3 -Thiazolyl-4                                                    252 2-C.sub.6 H.sub.5 -Thiazolyl-4                                             253 2-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Thiazolyl-4                              254 2-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Thiazolyl-4                              255 2-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Thiazolyl-4                              256 2-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Thiazolyl-4                             267 2-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Thiazolyl-4                             258 2-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Thiazolyl-4                             259 2-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Thiazolyl-4                              260 2-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Thiazolyl-4                              261 2-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Thiazolyl-4                              262 2-(4'-CN--C.sub.6 H.sub.4)-Thiazolyl-4                                     263 2-(3'-CN--C.sub.6 H.sub.4)-Thiazolyl-4                                     264 2-(2'-CN--C.sub.6 H.sub.4)-Thiazolyl-4                                     265 2-(4'-Cl--C.sub.6 H.sub.4)-Thiazolyl-4                                     266 2-(3'-Cl--C.sub.6 H.sub.4)-Thiazolyl-4                                     267 2-(2'-Cl--C.sub.6 H.sub.4)-Thiazolyl-4                                     268 N--CH.sub.3 -1,2,4-Triazolyl-5                                             269 3-CH.sub.3 --N--CH.sub.3 -1,2,4-Triazolyl-5                                270 3-C.sub.6 H.sub.5 --N--CH.sub.3 -1,2,4-Triazolyl-5                         271 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)-N--CH.sub.3 -1,2,4-Triazolyl-5                    272 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)-N--CH.sub.3 -1,2,4-Triazo               lyl-5                                                                  273 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)-N--CH.sub.3 -1,2,4-Triazolyl-5                    274 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-N--CH.sub.3 -1,2,4-Triaz               olyl-5                                                                 275 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-N--CH.sub.3 -1,2,4-Triazolyl-5                   276 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-N--CH.sub.3 -1,2,4-Triaz               olyl-5                                                                 277 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)-N--CH.sub.3 -1,2,4-Triazolyl-5                    278 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)-N--CH.sub.3 -1,2,4-Triazo               lyl-5                                                                  279 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)-N--CH.sub.3 -1,2,4-Triazolyl-5                    280 3-(4'-CN--C.sub.6 H.sub.4)-N--CH.sub.3 -1,2,4-Triazolyl-5                  281 3-(3'-CN--C.sub.6 H.sub.4)-N--CH.sub.3 -1,2,4-Triazolyl-5                  282 3-(2'-CN--C.sub.6 H.sub.4)-N--CH.sub.3 -1,2,4-Triazolyl-5                  283 3-(4'-Cl--C.sub.6 H.sub.4)-N--CH.sub.3 -1,2,4-Triazolyl-5                  284 3-(3'-Cl--C.sub.6 H.sub.4)-N--CH.sub.3 -1,2,4-Triazolyl-5                  285 3-(2'-Cl--C.sub.6 H.sub.4)-N--CH.sub.3 -1,2,4-Triazolyl-5                  286 1,3,4-Oxadiazolyl-2                                               287 5-CH.sub.3 -1,3,4-Oxadiazolyl-2                                            288 5-C.sub.6 H.sub.5 -1,3,4-Oxadiazolyl-2                                     289 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                      290 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                      291 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                      292 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                     293 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                     294 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                     295 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                      296 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                      297 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                      298 5-(4'-CN--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                             299 5-(3'-CN--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                             300 5-(2'-CN--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                             301 5-(4'-Cl--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                             302 5-(3'-Cl--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                             303 5-(2'-Cl--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                             304 1,2,4-Oxadiazolyl-3                                                        305 5-CH.sub.3 -1,2,4-Oxadiazolyl-3                                            306 5-C.sub.6 H.sub.5 -1,2,4-Oxadiazolyl-3                                     307 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                      308 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                      309 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                      310 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                     311 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                     312 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-1,214-Oxadiazolyl-3                     313 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                      314 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                      315 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                      316 5-(4'-CN--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                             317 5-(3'-CN--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                             318 5-(2'-CN--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                             319 5-(4'-Cl--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                             320 5-(3'-Cl--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                             321 5-(2'-Cl--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                             322 1,2,4-Oxadiazolyl-5                                                        323 3-CH.sub.3 -1,2,4-Oxadiazolyl-5                                            324 3-C.sub.6 H.sub.5 -1,2,4-Oxadiazolyl-5                                     325 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                      326 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                      327 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                      328 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                     329 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                     330 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                     331 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                      332 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                      333 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                      334 3-(4'-CN--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                             335 3-(3'-CN--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                             336 3-(2'-CN--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                             337 3-(4'-Cl--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                             338 3-(3'-Cl--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                             339 3-(2'-Cl--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                             340 1,2,4-Thiadiazolyl-3                                                       341 5-CH.sub.3 -1,2,4-Thiadiazolyl-3                                           342 5-C.sub.6 H.sub.5 -1,2,4-Thiadiazolyl-3                                    343 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                     344 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                     345 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                     346 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                    347 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                    348 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                    349 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                     350 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                     351 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                     352 5-(4'-CN--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                            353 5-(3'-CN--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                            354 5-(2'-CN--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                            355 5-(4'-Cl--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                            356 5-(3'-Cl--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                            357 5-(2'-Cl--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                            358 1,3,4-Thiadiazolyl-2                                                       359 5-CH.sub.3 -1,3,4-Thiadiazolyl-2                                           360 5-C.sub.6 H.sub.5 -1,3,4-Thiadiazolyl-2                                    361 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                     362 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                     363 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                     364 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                    365 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                    366 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                    367 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                     368 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                     369 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                     370 5-(4'-CN--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                            371 5-(3'-CN--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                            372 5-(2'-CN--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                            373 5-(4'-Cl--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                            374 5-(3'-Cl--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                            375 5-(2'-Cl--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                            376 Pyridinyl-2                                                                377 Pyridinyl-4                                                                378 Pyridazinyl-3                                                              379 Pyridazinyl-4                                                              380 Pyridazinyl-2                                                              381 Pyrimidinyl-4                                                              382 Pyrimidinyl-5                                                              383 Pyrimidinyl-2                                                              384 1-Naphthyl                                                                 385 2-Naphthyl                                                               ______________________________________                                    

                  TABLE 45                                                         ______________________________________                                         6  STR278##                                                                       - I: R.sup.1 = H, X = CH.sub.3                                                II: R.sup.1 = CH.sub.3, X = CH.sub.3                                           III: R.sup.1 = C.sub.2 H.sub.5, X = CH.sub.3                                   IV: R.sup.1 = Allyl, X = CH.sub.3                                              V: R.sup.1 = Propargyl, X = CH.sub.3                                           VI: R.sup.1 = CH.sub.2 --OCH.sub.3, X = CH.sub.3                               VII: R.sup.1 = CO.sub.2 CH.sub.3, X = CH.sub.3                                 VIII: R.sup.1 = H, X = Cl                                                      IX: R.sup.1 = CH.sub.3, X = Cl                                                 X: R.sup.1 = C.sub.2 H.sub.5, X = Cl                                           XI: R.sup.1 = Allyl, X = Cl                                                    XII: R.sup.1 = Propargyl, X = Cl                                               XIII: R.sup.1 = CH.sub.2 --OCH.sub.3, X = Cl                                   XIV: R.sup.1 = CO.sub.2 CH.sub.3, X = Cl                                       No.        T.sub.m                                                           ______________________________________                                          1       H                                                                        2 2-F                                                                          3 3-F                                                                          4 4-F                                                                          5 2,4-F.sub.2                                                                  6 2,4,6-F.sub.3                                                                7 2,3,4,5,6-F.sub.5                                                            8 2,3-F.sub.2                                                                  9 2-Cl                                                                         10 3-Cl                                                                        11 4-Cl                                                                        12 2,3-Cl.sub.2                                                                13 2,4-Cl.sub.2                                                                14 2,5-Cl.sub.2                                                                15 2,6-Cl.sub.2                                                                16 3,4-Cl.sub.2                                                                17 3,5-Cl.sub.2                                                                18 2,3,4-Cl.sub.3                                                              19 2,3,5-Cl.sub.3                                                              20 2,3,6-Cl.sub.3                                                              21 2,4,5-Cl.sub.3                                                              22 2,4,6-Cl.sub.3                                                              23 3,4,5-Cl.sub.3                                                              24 2,3,4,6-Cl.sub.4                                                            25 2,3,5,6-Cl.sub.4                                                            26 2,3,4,5,6-Cl.sub.5                                                          27 2-Br                                                                        28 3-Br                                                                        29 4-Br                                                                        30 2,4-Br.sub.2                                                                31 2,5-Br.sub.2                                                                32 2,6-Br.sub.2                                                                33 2,4,6-Br.sub.3                                                              34 2,3,4,5,6-Br.sub.5                                                          35 2-I                                                                         36 3-I                                                                         37 4-I                                                                         38 2,4-I.sub.2                                                                 39 2-Cl, 3-F                                                                   40 2-Cl, 4-F                                                                   41 2-Cl, 5-F                                                                   42 2-Cl, 6-F                                                                   43 2-Cl, 3-Br                                                                  44 2-Cl, 4-Br                                                                  45 2-Cl, 5-Br                                                                  46 2-Cl, 6-Br                                                                  47 2-Br, 3-Cl                                                                  48 2-Br, 4-Cl                                                                  49 2-Br, 5-Cl                                                                  50 2-Br, 3-F                                                                   51 2-Br, 4-F                                                                   52 2-Br, 5-F                                                                   53 2-Br, 6-F                                                                   54 2-F, 3-Cl                                                                   55 2-F, 4-Cl                                                                   56 2-F, 5-Cl                                                                   57 3-Cl, 4-F                                                                   58 3-Cl, 5-F                                                                   59 3-Cl, 4-Br                                                                  60 3-Cl, 5-Br                                                                  61 3-F, 4-Cl                                                                   62 3-F, 4-Br                                                                   63 3-Br, 4-Cl                                                                  64 3-Br, 4-F                                                                   65 2,6-Cl.sub.2, 4-Br                                                          66 2-CH.sub.3                                                                  67 3-CH.sub.3                                                                  68 4-CH.sub.3                                                                  69 2,3-(CH.sub.3).sub.2                                                        70 2,4-(CH.sub.3).sub.2                                                        71 2,5-(CH.sub.3).sub.2                                                        72 2,6-(CH.sub.3).sub.2                                                        73 3,4-(CH.sub.3).sub.2                                                        74 3,5-(CH.sub.3).sub.2                                                        75 2,3,5-(CH.sub.3).sub.3                                                      76 2,3,4-(CH.sub.3).sub.3                                                      77 2,3,6-(CH.sub.3).sub.3                                                      78 2,4,5-(CH.sub.3).sub.3                                                      79 2,4,6-(CH.sub.3).sub.3                                                      80 3,4,5-(CH.sub.3).sub.3                                                      81 2,3,4,6-(CH.sub.3).sub.4                                                    82 2,3,5,6-(CH.sub.3).sub.4                                                    83 2,3,4,5,6-(CH.sub.3).sub.5                                                  84 2-C.sub.2 H.sub.5                                                           85 3-C.sub.2 H.sub.5                                                           86 4-C.sub.2 H.sub.5                                                           87 2,4-(C.sub.2 H.sub.5).sub.2                                                 88 2,6-(C.sub.2 H.sub.5).sub.2                                                 89 3,5-(C.sub.2 H.sub.5).sub.2                                                 90 2,4,6-(C.sub.2 H.sub.5).sub.3                                               91 2-n-C.sub.3 H.sub.7                                                         92 3-n-C.sub.3 H.sub.7                                                         93 4-n-C.sub.3 H.sub.7                                                         94 2-i-C.sub.3 H.sub.7                                                         95 3-i-C.sub.3 H.sub.7                                                         96 4-i-C.sub.3 H.sub.7                                                         97 2,4-(i-C.sub.3 H.sub.7).sub.2                                               98 2,6-(i-C.sub.3 H.sub.7).sub.2                                               99 3,5-(i-C.sub.3 H.sub.7).sub.2                                              100 2,4,6-(i-C.sub.3 H.sub.7).sub.3                                            101 2-s-C.sub.4 H.sub.9                                                        102 3-s-C.sub.4 H.sub.9                                                        103 4-s-C.sub.4 H.sub.9                                                        104 2-t-C.sub.4 H.sub.9                                                        105 3-t-C.sub.4 H.sub.9                                                        106 4-t-C.sub.4 H.sub.9                                                        107 2,3-(t-C.sub.4 H.sub.9).sub.2                                              108 2,4-(t-C.sub.4 H.sub.9).sub.2                                              109 2,5-(t-C.sub.4 H.sub.9).sub.2                                              110 2,6-(t-C.sub.4 H.sub.9).sub.2                                              111 3,4-(t-C.sub.4 H.sub.9).sub.2                                              112 2,4,6-(t-C.sub.4 H.sub.9).sub.3                                            113 4-n-C.sub.9 H.sub.19                                                       114 4-n-C.sub.12 H.sub.25                                                      115 4-n-C.sub.15 H.sub.31                                                      116 4-(1,1,3,3-Tetramethylbutyl)                                               117 4-(2,4,4-Trimethylpropyl)                                                  118 2-t-C.sub.4 H.sub.9, 4-CH.sub.3                                            119 2-t-C.sub.4 H.sub.9, 5-CH.sub.3                                            120 2,6-(t-C.sub.4 H.sub.9).sub.2, 4-CH.sub.3                                  121 2-CH.sub.3, 4-t-C.sub.4 H.sub.9                                            122 2-CH.sub.3, 6-t-C.sub.4 H.sub.9                                            123 2-CH.sub.3, 4-i-C.sub.3 H.sub.7                                            124 2-CH.sub.3, 5-i-C.sub.3 H.sub.7                                            125 3-CH.sub.3, 4-i-C.sub.3 H.sub.7                                            126 2-i-C.sub.3 H.sub.7, 5-CH.sub.3                                            127 2,4-(t-C.sub.4 H.sub.9).sub.2, 6-i-C.sub.3 H.sub.7                         128 2-Allyl                                                                    129 3-Allyl                                                                    130 4-Allyl                                                                    131 2-Allyl, 6-CH.sub.3                                                        132 2-cyclo-C.sub.6 H.sub.11                                                   133 3-cyclo-C.sub.6 H.sub.11                                                   134 4-cyclo-C.sub.6 H.sub.11                                                   135 2,4-(cyclo-C.sub.6 H.sub.11).sub.2, 6-CH.sub.3                             136 2-CH.sub.3, 4-cyclo-C.sub.6 H.sub.11                                       137 2-CH.sub.2 --C.sub.6 H.sub.5                                               138 3-CH.sub.2 --C.sub.6 H.sub.5                                               139 4-CH.sub.2 --C.sub.6 H.sub.5                                               140 2-CH.sub.2 --C.sub.6 H.sub.5, 4-CH.sub.3                                   141 2-CH.sub.3, 4-CH.sub.2 --C.sub.6 H.sub.5                                   142 2-C.sub.6 H.sub.5                                                          143 3-C.sub.6 H.sub.5                                                          144 4-C.sub.6 H.sub.5                                                          145 4-(2-i-C.sub.3 H.sub.7 --C.sub.6 H.sub.4)                                  146 4-C.sub.6 H.sub.5, 2,6-(CH.sub.3).sub.2                                    147 2-Cl, 4-C.sub.6 H.sub.5                                                    148 2-Br, 4-C.sub.6 H.sub.5                                                    149 2-C.sub.6 H.sub.5, 4-Cl                                                    150 2-C.sub.6 H.sub.5, 4-Br                                                    151 2-CH.sub.2 C.sub.6 H.sub.5, 4-Cl                                           152 2-CH.sub.2 C.sub.6 H.sub.5, 4-Br                                           153 2-Cl, 4-CH.sub.2 C.sub.6 H.sub.5                                           154 2-Br, 4-CH.sub.2 C.sub.6 H.sub.5                                           155 2-cyclo-C.sub.6 H.sub.11, 4-Cl                                             156 2-cyclo-C.sub.6 H.sub.11, 4-Br                                             157 2-Cl, 4-cyclo-C.sub.6 H.sub.11                                             158 2-Br, 4-cyclo-C.sub.6 H.sub.11                                             159 2-OCH.sub.3                                                                160 3-OCH.sub.3                                                                161 4-OCH.sub.3                                                                162 2-OC.sub.2 H.sub.5                                                         163 3-O--C.sub.2 H.sub.5                                                       164 4-O--C.sub.2 H.sub.5                                                       165 2-O-n-C.sub.3 H.sub.7                                                      166 3-O-n-C.sub.3 H.sub.7                                                      167 4-O-n-C.sub.3 H.sub.7                                                      168 2-O-i-C.sub.3 H.sub.7                                                      169 3-O-i-C.sub.3 H.sub.7                                                      170 4-O-i-C.sub.3 H.sub.7                                                      171 2-O-n-C.sub.6 H.sub.13                                                     172 3-O-n-C.sub.6 H.sub.13                                                     173 4-O-n-C.sub.6 H.sub.13                                                     174 2-O-n-C.sub.8 H.sub.17                                                     175 3-O-n-C.sub.8 H.sub.17                                                     176 4-O-n-C.sub.8 H.sub.17                                                     177 2-O-CH.sub.2 C.sub.6 H.sub.5                                               178 3-O-CH.sub.2 C.sub.6 H.sub.5                                               179 4-O-CH.sub.2 C.sub.6 H.sub.5                                               180 2-O-(CH.sub.2).sub.3 C.sub.6 H.sub.5                                       181 3-O-(CH.sub.2).sub.3 C.sub.6 H.sub.5                                       182 4-O-(CH.sub.2).sub.3 C.sub.6 H.sub.5                                       183 2,4-(OCH.sub.3).sub.2                                                      184 2-CF.sub.3                                                                 185 3-CF.sub.3                                                                 186 4-CF.sub.3                                                                 187 2-OCF.sub.3                                                                188 3-OCF.sub.3                                                                189 4-OCF.sub.3                                                                190 3-OCH.sub.2 CHF.sub.2                                                      191 2-NO.sub.2                                                                 192 3-NO.sub.2                                                                 193 4-NO.sub.2                                                                 194 2-CN                                                                       195 3-CN                                                                       196 4-CN                                                                       197 2-CH.sub.3, 3-Cl                                                           198 2-CH.sub.3, 4-Cl                                                           199 2-CH.sub.3, 5-Cl                                                           200 2-CH.sub.3, 6-Cl                                                           201 2-CH.sub.3, 3-F                                                            202 2-CH.sub.3, 4-F                                                            203 2-CH.sub.3, 5-F                                                            204 2-CH.sub.3, 6-F                                                            205 2-CH.sub.3, 3-Br                                                           206 2-CH.sub.3, 4-Br                                                           207 2-CH.sub.3, 5-Br                                                           208 2-CH.sub.3, 6-Br                                                           209 2-Cl, 3-CH.sub.3                                                           210 2-Cl, 4-CH.sub.3                                                           211 2-Cl, 5-CH.sub.3                                                           212 2-F, 3-CH.sub.3                                                            213 2-F, 4-CH.sub.3                                                            214 2-F, 5-CH.sub.3                                                            215 2-Br, 3-CH.sub.3                                                           216 2-Br, 4-CH.sub.3                                                           217 2-Br, 5-CH.sub.3                                                           218 3-CH.sub.3, 4-Cl                                                           219 3-CH.sub.3, 5-Cl                                                           220 3-CH.sub.3, 4-F                                                            221 3-CH.sub.3, 5-F                                                            222 3-CH.sub.3, 4-Br                                                           223 3-CH.sub.3, 5-Br                                                           224 3-F, 4-CH.sub.3                                                            225 3-Cl, 4-CH.sub.3                                                           226 3-Br, 4-CH.sub.3                                                           227 2-Cl, 4,5-(CH.sub.3).sub.2                                                 228 2-Br, 4,5-(CH.sub.3).sub.2                                                 229 2-Cl, 3,5-(CH.sub.3).sub.2                                                 230 2-Br, 3,5-(CH.sub.3).sub.2                                                 231 2,6-Cl.sub.2, 4-CH.sub.3                                                   232 2,6-F.sub.2, 4-CH.sub.3                                                    233 2,6-Br.sub.2, 4-CH.sub.3                                                   234 2,4-Br.sub.2, 6-CH.sub.3                                                   235 2,4-F.sub.2, 6-CH.sub.3                                                    236 2,4-Br.sub.2, 6-CH.sub.3                                                   237 2,6-(CH.sub.3).sub.2, 4-F                                                  238 2,6-(CH.sub.3).sub.2, 4-Cl                                                 239 2,6-(CH.sub.3).sub.2, 4-Br                                                 240 3,5-(CH.sub.3).sub.2, 4-F                                                  241 3,5-(CH.sub.3).sub.2, 4-Cl                                                 242 3,5-(CH.sub.3).sub.2, 4-Br                                                 243 2,3,6-(CH.sub.3).sub.3, 4-F                                                244 2,3,6-(CH.sub.3).sub.3, 4-Cl                                               245 2,3,6-(CH.sub.3).sub.3, 4-Br                                               246 2,4-(CH.sub.3).sub.2, 6-F                                                  247 2,4-(CH.sub.3).sub.2, 6-Cl                                                 248 2,4-(CH.sub.3).sub.2, 6-Br                                                 249 2-i-C.sub.3 H.sub.7, 4-Cl, 5-CH.sub.3                                      250 2-Cl, 4-NO.sub.2                                                           251 2-NO.sub.2, 4-Cl                                                           252 2-OCH.sub.3, 5-NO.sub.2                                                    253 2,4-Cl.sub.2, 5-NO.sub.2                                                   254 2,4-Cl.sub.2, 6-NO.sub.2                                                   255 2,6-Cl.sub.2, 4-NO.sub.2                                                   256 2,6-Br.sub.2, 4-NO.sub.2                                                   257 2,6-I.sub.2, 4-NO.sub.2                                                    258 2-CH.sub.3, 5-i-C.sub.3 H.sub.7, 4-Cl                                      259 2-CO.sub.2 CH.sub.3                                                        260 3-CO.sub.2 CH.sub.3                                                        261 4-CO.sub.2 CH.sub.3                                                        262 2-CO.sub.2 (C.sub.2 H.sub.5)                                               263 3-CO.sub.2 (C.sub.2 H.sub.5)                                               264 4-CO.sub.2 (C.sub.2 H.sub.5)                                               265 2-CO.sub.2 (n-C.sub.3 H.sub.7)                                             266 3-CO.sub.2 (n-C.sub.3 H.sub.7)                                             267 4-CO.sub.2 (n-C.sub.3 H.sub.7)                                             268 2-CO.sub.2 (i-C.sub.3 H.sub.7)                                             269 3-CO.sub.2 (i-C.sub.3 H.sub.7)                                             270 4-CO.sub.2 (i-C.sub.3 H.sub.7)                                             271 2-CO.sub.2 (n-C.sub.6 H.sub.13)                                            272 3-CO.sub.2 (n-C.sub.6 H.sub.13)                                            273 4-CO.sub.2 (n-C.sub.6 H.sub.13)                                            274 2-CH.sub.2 --OCH.sub.3                                                     275 3-CH.sub.2 --OCH.sub.3                                                     276 4-CH.sub.2 --OCH.sub.3                                                     277 2-CH.sub.2 O(C.sub.2 H.sub.5)                                              278 3-CH.sub.2 O(C.sub.2 H.sub.5)                                              279 4-CH.sub.2 O(C.sub.2 H.sub.5)                                              280 2-CH.sub.2 O(n-C.sub.3 H.sub.7)                                            281 3-CH.sub.2 O(n-C.sub.3 H.sub.7)                                            282 4-CH.sub.2 O(n-C.sub.3 H.sub.7)                                            283 2-CH.sub.2 O(i-C.sub.3 H.sub.7)                                            284 3-CH.sub.2 O(i-C.sub.3 H.sub.7)                                            285 4-CH.sub.2 O(i-C.sub.3 H.sub.7)                                            286 2-CHO                                                                      287 3-CHO                                                                      288 4-CHO                                                                      289 2-CO--CH.sub.3                                                             290 3-CO--CH.sub.3                                                             291 4-CO--CH.sub.3                                                             292 2-CO--CH.sub.2 --CH.sub.3                                                  293 3-CO--CH.sub.2 --CH.sub.3                                                  294 4-CO--CH.sub.2 --CH.sub.3                                                  295 2-CO--CH.sub.2 --CH.sub.2 --CH.sub.3                                       296 3-CO--CH.sub.2 --CH.sub.2 --CH.sub.3                                       297 4-CO--CH.sub.2 --CH.sub.2 --CH.sub.3                                       298 2-CO--CH(CH.sub.3)--CH.sub.3                                               299 3-CO--CH(CH.sub.3)--CH.sub.3                                               300 4-CO--CH(CH.sub.3)--CH.sub.3                                               301 2-Me-4-CHO                                                                 302 2-Me-4-CH.sub.3 --CO                                                       303 2-Me-4-CH.sub.3 --CH.sub.2 --CO                                            304 2-Me-4-CH.sub.3 --CH.sub.2 --CH.sub.2 --CO                                 305 2-Me-4-CH.sub.3 --CH(CH.sub.3)--CO                                         306 2,5-Me.sub.2 -4-CHO                                                        307 2,5-Me.sub.2 -4-CH.sub.3 --CO                                              308 2,5-Me.sub.2 -4-CH.sub.3 --CH.sub.2 --CO                                   309 2,5-Me.sub.2 -4-CH.sub.3 --CH.sub.2 --CH.sub.2 --CO                        310 2,5-Me.sub.2 -4-CH.sub.3 --CH(CH.sub.3)--CO                                311 2-Cl-4-CHO                                                                 312 2-Cl-4-CH.sub.3 --CO                                                       313 2-Cl-4-CH.sub.3 --CH.sub.2 --CO                                            314 2-Cl-4-CH.sub.3 --CH(CH.sub.3)--CO                                         315 2,5-Cl.sub.2 -4-CHO                                                        316 2,5-Cl.sub.2 -4-CH.sub.3 --CO                                              317 2,5-Cl.sub.2 -4-CH.sub.3 --CH.sub.2 --CO                                   318 2,5-Cl.sub.2 -4-CH.sub.3 --CH.sub.2 --CH.sub.2 --CO                        319 2,5-Cl.sub.2 -4-CH.sub.3 --CH(CH.sub.3)--CO                                320 2-C(═NOCH.sub.3)--CH.sub.3                                             321 3-C(═NOCH.sub.3)--CH.sub.3                                             322 4-C(═NOCH.sub.3)--CH.sub.3                                             323 2-C(═NOC.sub.2 H.sub.5)--CH.sub.3                                      324 3-C(═NOC.sub.2 H.sub.5)--CH.sub.3                                      325 4-C(═NOC.sub.2 H.sub.5)--CH.sub.3                                      326 2-C(═NO-n-C.sub.3 H.sub.7)--CH.sub.3                                   327 3-C(═NO-n-C.sub.3 H.sub.7)--CH.sub.3                                   328 4-C(═NO-n-C.sub.3 H.sub.7)--CH.sub.3                                   329 2-C(═NO-i-C.sub.3 H.sub.7)--CH.sub.3                                   330 3-C(═NO-i-C.sub.3 H.sub.7)--CH.sub.3                                   331 4-C(═NO-i-C.sub.3 H.sub.7)--CH.sub.3                                   332 2-C(═NO-Allyl)--CH.sub.3                                               333 3-C(═NO-Allyl)--CH.sub.3                                               334 4-C(═NO-Allyl)--CH.sub.3                                               335 2-C(═NO-trans-Chloroallyl)--CH.sub.3                                   336 3-C(═NO-trans-Chloroallyl)--CH.sub.3                                   337 4-C(═NO-trans-Chloroallyl)--CH.sub.3                                   338 2-C(═NO-Propargyl)--CH.sub.3                                           339 3-C(═NO-Propargyl)--CH.sub.3                                           340 4-C(═NO-Propargyl)--CH.sub.3                                           341 2-C(═NO-n-C.sub.4 H.sub.9)--CH.sub.3                                   342 3-C(═NO-n-C.sub.4 H.sub.9)--CH.sub.3                                   343 4-C(═NO-n-C.sub.4 H.sub.9)--CH.sub.3                                   344 2-C(═NO--CH.sub.2 --C.sub.6 H.sub.5)--CH.sub.3                         345 3-C(═NO--CH.sub.2 --C.sub.6 H.sub.5)--CH.sub.3                         346 4-C(═NO--CH.sub.2 --C.sub.6 H.sub.5)--CH.sub.3                         347 2-CH.sub.3 -4-CH═NOCH.sub.3                                            348 2-CH.sub.3 -4-CH═NOC.sub.2 H.sub.5                                     349 2-CH.sub.3 -4-CH═NO-n-C.sub.3 H.sub.7                                  350 2-CH.sub.3 -4-CH═NO-i-C.sub.3 H.sub.7                                  351 2-CH.sub.3 -4-CH═NO-Allyl                                              352 2-CH.sub.3 -4-CH═NO-(trans-Chloroallyl)                                353 2-CH.sub.3 -4-CH═NO-Propargyl                                          354 2-CH.sub.3 -4-CH═NO-n-C.sub.4 H.sub.9                                  355 2-CH.sub.3 -4-CH═NO--CH.sub.2 --C.sub.6 H.sub.5                        356 2-CH.sub.3 -4-(CH.sub.3 --C═NOCH.sub.3)                                357 2-CH.sub.3 -4-(CH.sub.3 --C═NOC.sub.2 H.sub.5)                         358 2-CH.sub.3 -4-(CH.sub.3 --C═NO-n-C.sub.3 H.sub.7)                      359 2-CH.sub.3 -4-(CH.sub.3 --C═NO-i-C.sub.3 H.sub.7)                      360 2-CH.sub.3 -4-(CH.sub.3 --C═NO-Allyl)                                  361 2-CH.sub.3 -4-(CH.sub.3 --C═NO-trans-Chloroallyl)                      362 2-CH.sub.3 -4-(CH.sub.3 --C═NO-Propargyl)                              363 2-CH.sub.3 -4-(CH.sub.3 --C═NO-n-C.sub.4 H.sub.9)                      364 2-CH.sub.3 -4-(CH.sub.3 --C═NO--CH.sub.2 --C.sub.6 H.sub.5)                    365 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C═NO--CH.sub.3)                       366 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C═NO--C.sub.2 H.sub.5)        367 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C═NO-n-C.sub.3 H.sub.7)                       368 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C═NO-i-C.sub.3 H.sub.7        369 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C═NO-Allyl)                           370 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C═NO-trans-Chloroallyl)                       371 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C═NO-Propargyl)                       372 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C═NO-n-C.sub.4                       H.sub.9)                                                                373 2-CH.sub.3 -4-(C.sub.2 H.sub.5 --C═NO--CH.sub.2 --C.sub.6                     H.sub.5)                                                                374 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C═NOCH.sub.3)                      375 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C═NOC.sub.2 H.sub.5)                       376 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C═NO-n-C.sub.3                    H.sub.7)                                                                377 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C═NO-i-C.sub.3 H.sub.7)                    378 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C═NO-Allyl)                        379 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C═NO-trans-Chloroall              yl)                                                                     380 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C═NO-Proparyl)                     381 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C═NO-n-C.sub.4 H.sub.9)                    382 2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 --C═NO--CH.sub.2                    --C.sub.6 H.sub.5)                                                      383 2-C.sub.6 H.sub.5                                                          384 3-C.sub.6 H.sub.5                                                          385 4-C.sub.6 H.sub.5                                                          386 2-(2'-F--C.sub.6 H.sub.4)                                                  387 2-(3'-F--C.sub.6 H.sub.4)                                                  388 2-(4'-F--C.sub.6 H.sub.4)                                                  389 3-(2'-F--C.sub.6 H.sub.4)                                                  390 3-(3'-F--C.sub.6 H.sub.4)                                                  391 3-(4'-F--C.sub.6 H.sub.4)                                                  392 4-(2'-F--C.sub.6 H.sub.4)                                                  393 4-(3'-F--C.sub.6 H.sub.4)                                                  394 4-(4'-F--C.sub.6 H.sub.4)                                                  395 2-(2'-Cl--C.sub.6 H.sub.4)                                                 396 2-(3'-Cl--C.sub.6 H.sub.4)                                                 397 2-(4'-Cl--C.sub.6 H.sub.4)                                                 398 3-(2'-Cl--C.sub.6 H.sub.4)                                                 399 3-(3'-Cl--C.sub.6 H.sub.4)                                                 400 3-(4'-Cl--C.sub.6 H.sub.4)                                                 401 4-(2'-Cl--C.sub.6 H.sub.4)                                                 402 4-(3'-Cl--C.sub.6 H.sub.4)                                                 403 4-(4'-Cl--C.sub.6 H.sub.4)                                                 405 2-(2'-CH.sub.3 --C.sub.6 H.sub.4)                                          406 2-(3'-CH.sub.3 --C.sub.6 H.sub.4)                                          407 2-(4'-CH.sub.3 --C.sub.6 H.sub.4)                                          408 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)                                          409 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)                                          410 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)                                          411 4-(2'-CH.sub.3 --C.sub.6 H.sub.4)                                          412 4-(3'-CH.sub.3 --C.sub.6 H.sub.4)                                          413 4-(4'-CH.sub.3 --C.sub.6 H.sub.4)                                          414 2-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                      415 2-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                      416 2-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                      417 3-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                      418 3-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                      419 3-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                      420 4-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                      421 4-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                      422 4-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                      423 2-(2'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                       424 2-(3'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                       425 2-(4'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                       426 3-(2'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                       427 3-(3'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                       428 3-(4'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                       429 4-(2'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                       430 4-(3'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                       431 4-(4'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                       432 2-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                                 433 2-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                                 434 2-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                                 435 3-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                                 436 3-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                                 437 3-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                                 438 4-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                                 439 4-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                                 440 4-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                                 441 2-(2'-CH.sub.3 O--C.sub.6 H.sub.4)                                         442 2-(3'-CH.sub.3 O--C.sub.6 H.sub.4)                                         443 2-(4'-CH.sub.3 O--C.sub.6 H.sub.4)                                         444 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)                                         445 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)                                         446 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)                                         447 4-(2'-CH.sub.3 O--C.sub.6 H.sub.4)                                         448 4-(3'-CH.sub.3 O--C.sub.6 H.sub.4)                                         449 4-(4'-CH.sub.3 O--C.sub.6 H.sub.4)                                         450 2-(2'-O.sub.2 N--C.sub.6 H.sub.4)                                          451 2-(3'-O.sub.2 N--C.sub.6 H.sub.4)                                          452 2-(4'-O.sub.2 N--C.sub.6 H.sub.4)                                          453 3-(2'-O.sub.2 N--C.sub.6 H.sub.4)                                          454 3-(3'-O.sub.2 N--C.sub.6 H.sub.4)                                          455 3-(4'-O.sub.2 N--C.sub.6 H.sub.4)                                          456 4-(2'-O.sub.2 N--C.sub.6 H.sub.4)                                          457 4-(3'-O.sub.2 N--C.sub.6 H.sub.4)                                          458 4-(4'-O.sub.2 N--C.sub.6 H.sub.4)                                          459 2-(2'-NC--C.sub.6 H.sub.4)                                                 460 2-(3'-NC--C.sub.6 H.sub.4)                                                 461 2-(4'-NC--C.sub.6 H.sub.4)                                                 462 3-(2'-NC--C.sub.6 H.sub.4)                                                 463 3-(3'-NC--C.sub.6 H.sub.4)                                                 464 3-(4'-NC--C.sub.6 H.sub.4)                                                 465 4-(2'-NC--C.sub.6 H.sub.4)                                                 466 4-(3'-NC--C.sub.6 H.sub.4)                                                 467 4-(4'-NC--C.sub.6 H.sub.4)                                                 468 2-(2'-CF.sub.3 --C.sub.6 H.sub.4)                                          469 2-(3'-CF.sub.3 --C.sub.6 H.sub.4)                                          470 2-(4'-CF.sub.3 --C.sub.6 H.sub.4)                                          471 3-(2'-CF.sub.3 --C.sub.6 H.sub.4)                                          472 3-(3'-CF.sub.3 --C.sub.6 H.sub.4)                                          473 3-(4'-CF.sub.3 --C.sub.6 H.sub.4)                                          474 4-(2'-CF.sub.3 --C.sub.6 H.sub.4)                                          475 4-(3'-CF.sub.3 --C.sub.6 H.sub.4)                                          476 4-(4'-CF.sub.3 --C.sub.6 H.sub.4)                                          477 2-O-C.sub.6 H.sub.5                                                        475 3-O-C.sub.6 H.sub.5                                                        476 4-O-C.sub.6 H.sub.5                                                        478 2-O-(2'-F--C.sub.6 H.sub.4)                                                479 2-O-(3'-F--C.sub.6 H.sub.4)                                                480 2-O-(4'-F--C.sub.6 H.sub.4)                                                481 3-O-(2'-F--C.sub.6 H.sub.4)                                                482 3-O-(3'-F--C.sub.6 H.sub.4)                                                483 3-O-(4'-F--C.sub.6 H.sub.4)                                                484 4-O-(2'-F--C.sub.6 H.sub.4)                                                485 4-O-(3'-F--C.sub.6 H.sub.4)                                                486 4-O-(4'-F--C.sub.6 H.sub.4)                                                487 2-O-(2'-Cl--C.sub.6 H.sub.4)                                               488 2-O-(3'-Cl--C.sub.6 H.sub.4)                                               489 2-O-(4'-Cl--C.sub.6 H.sub.4)                                               490 3-O-(2'-Cl--C.sub.6 H.sub.4)                                               491 3-O-(3'-Cl--C.sub.6 H.sub.4)                                               492 3-O-(4'-Cl--C.sub.6 H.sub.4)                                               493 3-O-(4'-Cl--C.sub.6 H.sub.4)                                               494 4-O-(2'-Cl--C.sub.6 H.sub.4)                                               495 4-O-(3'-Cl--C.sub.6 H.sub.4)                                               496 4-O-(4'-Cl--C.sub.6 H.sub.4)                                               497 2-O-(2'-CH.sub.3 --C.sub.6 H.sub.4)                                        498 2-O-(3'-CH.sub.3 --C.sub.6 H.sub.4)                                        499 2-O-(4'-CH.sub.3 --C.sub.6 H.sub.4)                                        500 3-O-(2'-CH.sub.3 --C.sub.6 H.sub.4)                                        501 3-O-(3'-CH.sub.3 --C.sub.6 H.sub.4)                                        502 3-O-(4'-CH.sub.3 --C.sub.6 H.sub.4)                                        503 4-O-(2'-CH.sub.3 --C.sub.6 H.sub.4)                                        504 4-O-(3'-CH.sub.3 --C.sub.6 H.sub.4)                                        505 4-O-(4'-CH.sub.3 --C.sub.6 H.sub.4)                                        506 2-O-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                    507 2-O-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                    508 2-O-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                    509 3-O-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                    510 3-O-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                    511 3-O-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                    512 4-O-(2'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                    513 4-O-(3'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                    514 4-O-(4'-CH.sub.3 --CO--C.sub.6 H.sub.4)                                    515 2-O-(2'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                     516 2-O-(3'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                     517 2-O-(4'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                     518 3-O-(2'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                     519 3-O-(3'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                     520 3-O-(4'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                     521 4-O-(2'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                     522 4-O-(3'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                     523 4-O-(4'-(CH.sub.3 --C(═NOAllyl))--C.sub.6 H.sub.4)                     524 2-O-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                               525 2-O-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                               526 2-O-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                               527 3-O-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                               528 3-O-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                               529 3-O-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                               530 4-O-(2'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                               531 4-O-(3'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                               532 4-O-(4'-CH.sub.3 O.sub.2 C--C.sub.6 H.sub.4)                               533 2-O-(2'-CH.sub.3 O--C.sub.6 H.sub.4)                                       534 2-O-(3'-CH.sub.3 O--C.sub.6 H.sub.4)                                       535 2-O-(4'-CH.sub.3 O--C.sub.6 H.sub.4)                                       536 3-O-(2'-CH.sub.3 O--C.sub.6 H.sub.4)                                       537 3-O-(3'-CH.sub.3 O--C.sub.6 H.sub.4)                                       538 3-O-(4'-CH.sub.3 O--C.sub.6 H.sub.4)                                       539 4-O-(2'-CH.sub.3 O--C.sub.6 H.sub.4)                                       540 4-O-(3'-CH.sub.3 O--C.sub.6 H.sub.4)                                       541 4-O-(4'-CH.sub.3 O--C.sub.6 H.sub.4)                                       542 2-O-(2'-O.sub.2 N--C.sub.6 H.sub.4)                                        543 2-O-(3'-O.sub.2 N--C.sub.6 H.sub.4)                                        544 2-O-(4'-O.sub.2 N--C.sub.6 H.sub.4)                                        545 3-O-(2'-O.sub.2 N--C.sub.6 H.sub.4)                                        546 3-O-(3'-O.sub.2 N--C.sub.6 H.sub.4)                                        547 3-O-(4'-O.sub.2 N--C.sub.6 H.sub.4)                                        548 4-O-(2'-O.sub.2 N--C.sub.6 H.sub.4)                                        549 4-O-(3'-O.sub.2 N--C.sub.6 H.sub.4)                                        550 4-O-(4'-O.sub.2 N--C.sub.6 H.sub.4)                                        551 2-O-(2'-NC--C.sub.6 H.sub.4)                                               552 2-O-(3'-NC--C.sub.6 H.sub.4)                                               553 2-O-(4'-NC--C.sub.6 H.sub.4)                                               554 3-O-(2'-NC--C.sub.6 H.sub.4)                                               555 3-O-(3'-NC--C.sub.6 H.sub.4)                                               556 3-O-(4'-NC--C.sub.6 H.sub.4)                                               557 4-O-(2'-NC--C.sub.6 H.sub.4)                                               558 4-O-(3'-NC--C.sub.6 H.sub.4)                                               559 4-O-(4'-NC--C.sub.6 H.sub.4)                                               560 2-O-(2'-CF.sub.3 --C.sub.6 H.sub.5)                                        561 2-O-(3'-CF.sub.3 --C.sub.6 H.sub.5)                                        562 2-O-(4'-CF.sub.3 --C.sub.6 H.sub.5)                                        563 3-O-(2'-CF.sub.3 --C.sub.6 H.sub.5)                                        564 3-O-(3'-CF.sub.3 --C.sub.6 H.sub.5)                                        565 3-O-(4'-CF.sub.3 --C.sub.6 H.sub.5)                                        566 4-O-(2'-CF.sub.3 --C.sub.6 H.sub.5)                                        567 4-O-(3'-CF.sub.3 --C.sub.6 H.sub.5)                                        568 4-O-(4'-CF.sub.3 --C.sub.6 H.sub.5)                                        569 2-Pyridinyl-2'                                                             570 2-Pyridinyl-3'                                                             571 2-Pyridinyl-4'                                                             572 3-Pyridinyl-2'                                                             573 3-Pyridinyl-3'                                                             574 3-Pyridinyl-4'                                                             575 4-Pyridinyl-2'                                                             576 4-Pyridinyl-3'                                                             577 4-Pyridinyl-4'                                                             578 2-Pyrimidinyl-2'                                                           579 2-Pyrimidinyl-3'                                                           580 2-Pyrimidinyl-4'                                                           581 3-Pyrimidinyl-2'                                                           582 3-Pyrimidinyl-3'                                                           583 3-Pyrimidinyl-4'                                                           584 4-Pyrimidinyl-2'                                                           585 4-Pyrimidinyl-3'                                                           586 4-Pyrimidinyl-4'                                                           587 2-Pyrazolyl-1'                                                             588 2-Pyrazolyl-3'                                                             589 2-Pyrazolyl-4'                                                             590 3-Pyrazolyl-1'                                                             591 3-Pyrazolyl-3'                                                             592 3-Pyrazolyl-4'                                                             593 4-Pyrazolyl-1'                                                             594 4-Pyrazolyl-3'                                                             595 4-Pyrazolyl-4'                                                             596 2-Isoxazolyl-3'                                                            597 2-Isoxazolyl-4'                                                            598 2-Isoxazolyl-5'                                                            599 3-Isoxazolyl-3'                                                            600 3-Isoxazolyl-4'                                                            601 3-Isoxazolyl-5'                                                            602 4-Isoxazolyl-3'                                                            603 4-Isoxazolyl-4'                                                            604 4-Isoxazolyl-5'                                                            605 2-Isothiazolyl-3'                                                          606 2-Isothiazolyl-4'                                                          607 2-Isothiazolyl-5'                                                          608 3-Isothiazolyl-3'                                                          609 3-Isothiazolyl-4'                                                          610 3-Isothiazolyl-5'                                                          611 4-Isothiazolyl-3'                                                          612 4-Isothiazolyl-4'                                                          613 4-Isothiazolyl-5'                                                          614 2-Imidazolyl-1'                                                            615 2-Imidazolyl-2'                                                            616 2-Imidazolyl-4'                                                            617 3-Imidazolyl-1'                                                            618 3-Imidazolyl-2'                                                            619 3-Imidazolyl-4'                                                            620 4-Imidazolyl-1'                                                            621 4-Imidazolyl-2'                                                            622 4-Imidazolyl-4'                                                            623 2-Oxazolyl-2'                                                              624 2-Oxazolyl-4'                                                              625 2-Oxazolyl-5'                                                              626 3-Oxazolyl-2'                                                              627 3-Oxazolyl-4'                                                              628 3-Oxazolyl-5'                                                              629 4-Oxazolyl-2'                                                              630 4-Oxazolyl-4'                                                              631 4-Oxazolyl-5'                                                              632 2-Thiazolyl-2'                                                             633 2-Thiazolyl-4'                                                             634 2-Thiazolyl-5'                                                             635 3-Thiazolyl-2'                                                             636 3-Thiazolyl-4'                                                             637 3-Thiazolyl-5'                                                             638 4-Thiazolyl-2'                                                             639 4-Thiazolyl-4'                                                             640 4-Thiazolyl-5'                                                           ______________________________________                                    

                  TABLE 46                                                         ______________________________________                                         3  STR279##                                                                       - I: R.sup.1 = H, X = CH.sub.3                                                II: R.sup.1 = CH.sub.3, X = CH.sub.3                                           III: R.sup.1 = C.sub.2 H.sub.5, X = CH.sub.3                                   IV: R.sup.1 = Allyl, X = CH.sub.3                                              V: R.sup.1 = Propargyl, X = CH.sub.3                                           VI: R.sup.1 = CH.sub.2 --OCH.sub.3, X = CH.sub.3                               VII: R.sup.1 = CO.sub.2 CH.sub.3, X = CH.sub.3                                 VIII: R.sup.1 = H, X = Cl                                                      IX: R.sup.1 = CH.sub.3, X = Cl                                                 X: R.sup.1 = C.sub.2 H.sub.5, X = Cl                                           XI: R.sup.1 = Allyl, X = Cl                                                    XII: R.sup.1 = Propargyl, X = Cl                                               XIII: R.sup.1 = CH.sub.2 --OCH.sub.3, X = Cl                                   XIV: R.sup.1 = CO.sub.2 CH.sub.3, X = Cl                                       No.         B                                                                ______________________________________                                         1         Pyrrolyl-3                                                             2 N--CH.sub.3 -Pyrrolyl-3                                                      3 N--C.sub.6 H.sub.5 -Pyrrolyl-3                                               4 N-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrrolyl-3                                 5 N-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrrolyl-3                                 6 N-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrrolyl-3                                 7 N-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrrolyl-3                                8 N-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrrolyl-3                                9 N-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrrolyl-3                                10 N-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrrolyl-3                                11 N-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrrolyl-3                                12 N-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrrolyl-3                                13 N-(4'-CN--C.sub.6 H.sub.4)-Pyrrolyl-3                                       14 N-(3'-CN--C.sub.6 H.sub.4)-Pyrrolyl-3                                       15 N-(2'-CN--C.sub.6 H.sub.4)-Pyrrolyl-3                                       16 N-(4'-Cl--C.sub.6 H.sub.4)-Pyrrolyl-3                                       17 N-(3'-Cl--C.sub.6 H.sub.4)-Pyrrolyl-3                                       18 N-(2'-Cl--C.sub.6 H.sub.4)-Pyrrolyl-3                                       19 Pyrrolyl-2                                                                  20 N--CH.sub.3 -Pyrrolyl-2                                                     21 N--C.sub.6 H.sub.5 -Pyrrolyl-2                                              22 N-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrrolyl-2                                23 N-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrrolyl-2                                24 N-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrrolyl-2                                25 N-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrrolyl-2                               26 N-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrrolyl-2                               27 N-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrrolyl-2                               28 N-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrrolyl-2                                29 N-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrrolyl-2                                30 N-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrrolyl-2                                31 N-(4'-CN--C.sub.6 H.sub.4)-Pyrrolyl-2                                       32 N-(3'-CN--C.sub.6 H.sub.4)-Pyrrolyl-2                                       33 N-(2'-CN--C.sub.6 H.sub.4)-Pyrrolyl-2                                       34 N-(4'-Cl--C.sub.6 H.sub.4)-Pyrrolyl-2                                       35 N-(3'-Cl--C.sub.6 H.sub.4)-Pyrrolyl-2                                       36 N-(2'-Cl--C.sub.6 H.sub.4)-Pyrrolyl-2                                       37 Furyl-2                                                                     38 5-CH.sub.3 -Furyl-2                                                         39 5-C.sub.6 H.sub.5 -Furyl-2                                                  40 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Furyl-2                                   41 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Furyl-2                                   42 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Furyl-2                                   43 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Furyl-2                                  44 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Furyl-2                                  45 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Furyl-2                                  46 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Furyl-2                                   47 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Furyl-2                                   48 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Furyl-2                                   49 5-(4'-CN--C.sub.6 H.sub.4)-Furyl-2                                          50 5-(3'-CN--C.sub.6 H.sub.4)-Furyl-2                                          51 5-(2'-CN--C.sub.6 H.sub.4)-Furyl-2                                          52 5-(4'-Cl--C.sub.6 H.sub.4)-Furyl-2                                          53 5-(3'-Cl--C.sub.6 H.sub.4)-Furyl-2                                          54 5-(2'-Cl--C.sub.6 H.sub.4)-Furyl-2                                          55 4-CH.sub.3 -Furyl-2                                                         56 4-C.sub.6 H.sub.5 -Furyl-2                                                  57 4-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Furyl-2                                   58 4-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Furyl-2                                   59 4-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Furyl-2                                   60 4-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Furyl-2                                  61 4-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Furyl-2                                  62 4-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Furyl-2                                  63 4-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Furyl-2                                   64 4-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Furyl-2                                   65 4-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Furyl-2                                   66 4-(4'-CN--C.sub.6 H.sub.4)-Furyl-2                                          67 4-(3'-CN--C.sub.6 H.sub.4)-Furyl-2                                          68 4-(2'-CN--C.sub.6 H.sub.4)-Furyl-2                                          69 4-(4'-Cl--C.sub.6 H.sub.4)-Furyl-2                                          70 4-(3'-Cl--C.sub.6 H.sub.4)-Furyl-2                                          71 4-(2'-Cl--C.sub.6 H.sub.4)-Furyl-2                                          72 Thienyl-2                                                                   73 5-CH.sub.3 -Thienyl-2                                                       74 5-C.sub.6 H.sub.5 -Thienyl-2                                                75 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-2                                 76 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-2                                 77 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-2                                 78 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-2                                79 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-2                                80 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-2                                81 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-2                                 82 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-2                                 83 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-2                                 84 5-(4'-CN--C.sub.6 H.sub.4)-Thienyl-2                                        85 5-(3'-CN--C.sub.6 H.sub.4)-Thienyl-2                                        86 5-(2'-CN--C.sub.6 H.sub.4)-Thienyl-2                                        87 5-(4'-Cl--C.sub.6 H.sub.4)-Thienyl-2                                        88 5-(3'-Cl--C.sub.6 H.sub.4)-Thienyl-2                                        89 5-(2'-Cl--C.sub.6 H.sub.4)-Thienyl-2                                        90 4-CH.sub.3 -Thienyl-2                                                       91 4-C.sub.6 H.sub.5 -Thienyl-2                                                92 4-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-2                                 93 4-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-2                                 94 4-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-2                                 95 4-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-2                                96 4-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-2                                97 4-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-2                                98 4-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-2                                 99 4-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-2                                 100 4-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-2                                101 4-(4'-CN--C.sub.6 H.sub.4)-Thienyl-2                                       102 4-(3'-CN--C.sub.6 H.sub.4)-Thienyl-2                                       103 4-(2'-CN--C.sub.6 H.sub.4)-Thienyl-2                                       104 4-(4'-Cl--C.sub.6 H.sub.4)-Thienyl-2                                       105 4-(3'-Cl--C.sub.6 H.sub.4)-Thienyl-2                                       106 4-(2'-Cl--C.sub.6 H.sub.4)-Thienyl-2                                       107 Thienyl-3                                                                  108 5-CH.sub.3 -Thienyl-3                                                      109 5-C.sub.6 H.sub.5 -Thienyl-3                                               110 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-3                                111 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-3                                112 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Thienyl-3                                113 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-3                               114 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-3                               115 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Thienyl-3                               116 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-3                                117 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-3                                118 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Thienyl-3                                119 5-(4'-CN--C.sub.6 H.sub.4)-Thienyl-3                                       120 5-(3'-CN--C.sub.6 H.sub.4)-Thienyl-3                                       121 5-(2'-CN--C.sub.6 H.sub.4)-Thienyl-3                                       122 5-(4'-Cl--C.sub.6 H.sub.4)-Thienyl-3                                       123 5-(3'-Cl--C.sub.6 H.sub.4)-Thienyl-3                                       124 5-(2'-Cl--C.sub.6 H.sub.4)-Thienyl-3                                       125 Pyrazolyl-4                                                                126 N--CH.sub.3 -Pyrazolyl-4                                                   127 N--C.sub.6 H.sub.5 -Pyrazolyl-4                                            128 N-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrazolyl-4                              129 N-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrazolyl-4                              130 N-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Pyrazolyl-4                              131 N-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrazolyl-4                             132 N-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrazolyl-4                             133 N-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Pyrazolyl-4                             134 N-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrazolyl-4                              135 N-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrazolyl-4                              136 N-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Pyrazolyl-4                              137 N-(4'-CN--C.sub.6 H.sub.4)-Pyrazolyl-4                                     138 N-(3'-CN--C.sub.6 H.sub.4)-Pyrazolyl-4                                     139 N-(2'-CN--C.sub.6 H.sub.4)-Pyrazolyl-4                                     140 N-(4'-Cl--C.sub.6 H.sub.4)-Pyrazolyl-4                                     141 N-(3'-Cl--C.sub.6 H.sub.4)-Pyrazolyl-4                                     142 N-(2'-Cl--C.sub.6 H.sub.4)-Pyrazolyl-4                                     143 3-CH.sub.3 --N-Methylpyrazolyl-4                                           144 3-C.sub.6 H.sub.5 --N-Methylpyrazolyl-4                                    145 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)-N-Methylpyrazolyl-4                      146 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)-N-Methylpyrazolyl-4                      147 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)-N-Methylpyrazolyl-4                      148 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-N-Methylpyrazolyl-4                     149 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-N-Methylpyrazolyl-4                     150 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-N-Methylpyrazolyl-4                     151 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)-N-Methylpyrazolyl-4                      152 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)-N-Methylpyrazolyl-4                      153 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)-N-Methylpyrazolyl-4                      154 3-(4'-CN--C.sub.6 H.sub.4)-N-Methylpyrazolyl-4                             155 3-(3'-CN--C.sub.6 H.sub.4)-N-Methylpyrazolyl-4                             156 3-(2'-CN--C.sub.6 H.sub.4)-N-Methylpyrazolyl-4                             157 3-(4'-Cl--C.sub.6 H.sub.4)-N-Methylpyrazolyl-4                             158 3-(3'-Cl--C.sub.6 H.sub.4)-N-Methylpyrazolyl-4                             159 3-(2'-Cl--C.sub.6 H.sub.4)-N-Methylpyrazolyl-4                             160 Isoxazolyl-5                                                               161 3-CH.sub.3 -Isoxazolyl-5                                                   162 3-C.sub.6 H.sub.5 -Isoxazolyl-5                                            163 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Isoxazolyl-5                             164 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Isoxazolyl-5                             165 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Isoxazolyl-5                             166 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Isoxazolyl-5                            167 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Isoxazolyl-5                            168 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Isoxazolyl-5                            169 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Isoxazolyl-5                             170 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Isoxazolyl-5                             171 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Isoxazolyl-5                             172 3-(4'-CN--C.sub.6 H.sub.4)-Isoxazolyl-5                                    173 3-(3'-CN--C.sub.6 H.sub.4)-Isoxazolyl-5                                    174 3-(2'-CN--C.sub.6 H.sub.4)-Isoxazolyl-5                                    175 3-(4'-Cl--C.sub.6 H.sub.4)-Isoxazolyl-5                                    176 3-(3'-Cl--C.sub.6 H.sub.4)-Isoxazolyl-5                                    177 3-(2'-Cl--C.sub.6 H.sub.4)-Isoxazolyl-5                                    178 4-Chloroisoxazolyl-5                                                       179 3-CH.sub.3 -4-Chloroisoxazolyl-5                                           180 3-C.sub.6 H.sub.5 -4-Chloroisoxazolyl-5                                    181 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                     182 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                     183 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                     184 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                    185 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                    186 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                    187 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                     188 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                     189 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                     190 3-(4'-CN--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                            191 3-(3'-CN--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                            192 3-(2'-CN--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                            193 3-(4'-Cl--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                            194 3-(3'-Cl--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                            195 3-(2'-Cl--C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                            196 Isoxazolyl-3                                                               197 5-CH.sub.3 -Isoxazolyl-3                                                   198 5-C.sub.6 H.sub.5 -Isoxazolyl-3                                            199 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Isoxazolyl-3                             200 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Isoxazolyl-3                             201 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Isoxazolyl-3                             202 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Isoxazolyl-3                            203 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Isoxazolyl-3                            204 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Isoxazolyl-3                            205 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Isoxazolyl-3                             206 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Isoxazolyl-3                             207 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Isoxazolyl-3                             208 5-(4'-CN--C.sub.6 H.sub.4)-Isoxazolyl-3                                    209 5-(3'-CN--C.sub.6 H.sub.4)-Isoxazolyl-3                                    210 5-(2'-CN--C.sub.6 H.sub.4)-Isoxazolyl-3                                    211 5-(4'-Cl--C.sub.6 H.sub.4)-Isoxazolyl-3                                    212 5-(3'-Cl--C.sub.6 H.sub.4)-Isoxazolyl-3                                    213 5-(2'-Cl--C.sub.6 H.sub.4)-Isoxazolyl-3                                    214 Isothiazolyl-5                                                             215 3-CH.sub.3 -Isothiazolyl-5                                                 216 3-C.sub.6 H.sub.5 -Isothiazolyl-5                                          217 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Isothiazolyl-5                           218 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Isothiazolyl-5                           219 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Isothiazolyl-5                           220 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Isothiazolyl-5                          221 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Isothiazolyl-5                          222 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Isothiazolyl-5                          223 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Isothiazolyl-5                           224 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Isothiazolyl-5                           225 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Isothiazolyl-5                           226 3-(4'-CN--C.sub.6 H.sub.4)-Isothiazolyl-5                                  227 3-(3'-CN--C.sub.6 H.sub.4)-Isothiazolyl-5                                  228 3-(2'-CN--C.sub.6 H.sub.4)-Isothiazolyl-5                                  229 3-(4'-Cl--C.sub.6 H.sub.4)-Isothiazolyl-5                                  230 3-(3'-Cl--C.sub.6 H.sub.4)-Isothiazolyl-5                                  231 3-(2'-Cl--C.sub.6 H.sub.4)-Isothiazolyl-5                                  232 Oxazolyl-4                                                                 233 3-CH.sub.3 -Oxazolyl-4                                                     234 3-C.sub.6 H.sub.5 -Oxazolyl-4                                              235 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Oxazolyl-4                               236 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Oxazolyl-4                               237 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Oxazolyl-4                               238 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Oxazolyl-4                              239 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Oxazolyl-4                              240 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Oxazolyl-4                              241 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Oxazolyl-4                               242 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Oxazolyl-4                               243 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Oxazolyl-4                               244 3-(4'-CN--C.sub.6 H.sub.4)-Oxazolyl-4                                      245 3-(3'-CN--C.sub.6 H.sub.4)-Oxazolyl-4                                      246 3-(2'-CN--C.sub.6 H.sub.4)-Oxazolyl-4                                      247 3-(4'-Cl--C.sub.6 H.sub.4)-Oxazolyl-4                                      248 3-(3'-Cl--C.sub.6 H.sub.4)-Oxazolyl-4                                      249 3-(2'-Cl--C.sub.6 H.sub.4)-Oxazolyl-4                                      250 Thiazolyl-4                                                                251 2-CH.sub.3 -Thiazolyl-4                                                    252 2-C.sub.6 H.sub.5 -Thiazolyl-4                                             253 2-(4'-CH.sub.3 --C.sub.6 H.sub.4)-Thiazolyl-4                              254 2-(3'-CH.sub.3 --C.sub.6 H.sub.4)-Thiazolyl-4                              255 2-(2'-CH.sub.3 --C.sub.6 H.sub.4)-Thiazolyl-4                              256 2-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-Thiazolyl-4                             267 2-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-Thiazolyl-4                             258 2-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-Thiazolyl-4                             259 2-(4'-NO.sub.2 --C.sub.6 H.sub.4)-Thiazoly1-4                              260 2-(3'-NO.sub.2 --C.sub.6 H.sub.4)-Thiazolyl-4                              261 2-(2'-NO.sub.2 --C.sub.6 H.sub.4)-Thiazolyl-4                              262 2-(4'-CN--C.sub.6 H.sub.4)-Thiazolyl-4                                     263 2-(3'-CN--C.sub.6 H.sub.4)-Thiazolyl-4                                     264 2-(2'-CN--C.sub.6 H.sub.4)-Thiazolyl-4                                     265 2-(4'-Cl--C.sub.6 H.sub.4)-Thiazolyl-4                                     266 2-(3'-Cl--C.sub.6 H.sub.4)-Thiazolyl-4                                     267 2-(2'-Cl--C.sub.6 H.sub.4)-Thiazolyl-4                                     268 N--CH.sub.3 -1,2,4-Triazolyl-5                                             269 3-CH.sub.3 --N--CH.sub.3 -1,2,4-Triazolyl-5                                270 3-C.sub.6 H.sub.5 --N--CH.sub.3 -1,2,4-Triazolyl-5                         271 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)-N--CH.sub.3 -1,2,4-Triazolyl-5                    272 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)-N--CH.sub.3 -1,2,4-Triazo               lyl-5                                                                  273 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)-N--CH.sub.3 -1,2,4-Triazolyl-5                    274 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-N--CH.sub.3 -1,2,4-Triaz               olyl-5                                                                 275 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-N--CH.sub.3 -1,2,4-Triazolyl-5                   276 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-N--CH.sub.3 -1,2,4-Triaz               olyl-5                                                                 277 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)-N--CH.sub.3 -1,2,4-Triazolyl-5                    278 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)-N--CH.sub.3 -1 2,4-Triazo               lyl-5                                                                  279 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)-N--CH.sub.3 -1,2,4-Triazolyl-5                    280 3-(4'-CN--C.sub.6 H.sub.4)-N--CH.sub.3 -1,2,4-Triazolyl-5                  281 3-(3'-CN--C.sub.6 H.sub.4)-N--CH.sub.3 -1,2,4-Triazolyl-5                  282 3-(2'-CN--C.sub.6 H.sub.4)-N--CH.sub.3 -1,2,4-Triazolyl-5                  283 3-(4'-Cl--C.sub.6 H.sub.4)-N--CH.sub.3 -1,2,4-Triazolyl-5                  284 3-(3'-Cl--C.sub.6 H.sub.4)-N--CH.sub.3 -1,2,4-Triazolyl-5                  285 3-(2'-Cl--C.sub.6 H.sub.4)-N--CH.sub.3 -1,2,4-Triazolyl-5                  286 1,3,4-Oxadiazolyl-2                                               287 5-CH.sub.3 -1,3,4-Oxadiazolyl-2                                            288 5-C.sub.6 H.sub.5 -1,3,4-Oxadiazolyl-2                                     289 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                      290 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                      291 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                      292 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                     293 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                     294 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                     295 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                      296 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                      297 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                      298 5-(4'-CN--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                             299 5-(3'-CN--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                             300 5-(2'-CN--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                             301 S-(4'-Cl--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                             302 S-(3'-Cl--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                             303 S-(2'-Cl--C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                             304 1,2,4-Oxadiazolyl-3                                                        305 5-CH.sub.3 -1,2,4-Oxadiazolyl-3                                            306 5-C.sub.6 H.sub.5 -1,2,4-Oxadiazolyl-3                                     307 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                      308 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                      309 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                      310 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                     311 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                     312 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                     313 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                      314 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                      315 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                      316 5-(4'-CN--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                             317 5-(3'-CN--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                             318 5-(2'-CN--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                             319 5-(4'-Cl--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                             320 5-(3'-Cl--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                             321 5-(2'-Cl--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                             322 1,2,4-Oxadiazolyl-5                                                        323 3-CH.sub.3 -1,2,4-Oxadiazolyl-5                                            324 3-C.sub.6 H.sub.5 -1,2,4-Oxadiazolyl-5                                     325 3-(4'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                      326 3-(3'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                      327 3-(2'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                      328 3-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                     329 3-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                     330 3-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                     331 3-(4'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                      332 3-(3'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                      333 3-(2'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                      334 3-(4'-CN--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                             335 3-(3'-CN--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                             336 3-(2'-CN--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                             337 3-(4'-Cl--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                             338 3-(3'-Cl--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                             339 3-(2'-Cl--C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                             340 1,2,4-Thiadiazolyl-3                                                       341 5-CH.sub.3 -1,2,4-Thiadiazolyl-3                                           342 5-C.sub.6 H.sub.5 -1,2,4-Thiadiazolyl-3                                    343 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                     344 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                     345 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                     346 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                    347 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                    348 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                    349 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                     350 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                     351 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                     352 5-(4'-CN--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                            353 5-(3'-CN--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                            354 5-(2'-CN--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                            355 5-(4'-Cl--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                            356 5-(3'-Cl--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                            357 5-(2'-Cl--C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                            358 1,3,4-Thiadiazolyl-2                                                       359 5-CH.sub.3 -1,3,4-Thiadiazolyl-2                                           360 5-C.sub.6 H.sub.5 -1,3,4-Thiadiazolyl-2                                    361 5-(4'-CH.sub.3 --C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                     362 5-(3'-CH.sub.3 --C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                     363 5-(2'-CH.sub.3 --C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                     364 5-(4'-CH.sub.3 O--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                    365 5-(3'-CH.sub.3 O--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                    366 5-(2'-CH.sub.3 O--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                    367 5-(4'-NO.sub.2 --C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                     368 5-(3'-NO.sub.2 --C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                     369 5-(2'-NO.sub.2 --C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                     370 5-(4'-CN--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                            371 5-(3'-CN--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                            372 5-(2'-CN--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                            373 5-(4'-Cl--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                            374 5-(3'-Cl--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                            375 5-(2'-Cl--C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                            376 Pyridinyl-2                                                                377 Pyridinyl-4                                                                378 Pyridazinyl-3                                                              379 Pyridazinyl-4                                                              380 Pyridazinyl-2                                                              381 Pyrimidinyl-4                                                              382 Pyrimidinyl-5                                                              383 Pyrimidinyl-2                                                            ______________________________________                                    

                  TABLE 47                                                         ______________________________________                                         Selected physical data of some compounds                                       2  STR280##                                                                       -                        IR (cm.sup.-1) or                                    No. Xm R.sup.1 .sup.1 H--NMR (ppm) mp                                        ______________________________________                                         1    4-Cl      H                        133                                      2 3,4-Cl.sub.2 H  109                                                          3 4-t-C.sub.4 H.sub.9 H  86                                                    4 4-CH.sub.3 H  117                                                            5 4-CF.sub.3 H  103                                                            6 3-Br H  99                                                                   7 3-Cl H  93                                                                   8 3-CF.sub.3 H  88                                                             9 3,5-Cl.sub.2 H  100                                                          10 3,4-(CH.sub.3).sub.2 H  127                                                 11 3,4-Cl.sub.2 CH.sub.3  74                                                   12 3,4-Cl.sub.2 Allyl 3.65(S, 3H); 2.2(S, 6H)                                  13 3,4-Cl.sub.2 Propargyl 3.65(S, 3H); 2.3(S, 3H);                                2.2(S, 3H)                                                                  14 3,4-Cl.sub.2 CH.sub.2 --OCH.sub.3 3.65(S, 3H); 2.3(S, 3H);                     2.2(S, 3H)                                                                  15 3,4-Cl.sub.2 CO--OCH.sub.3  137                                             16 4-t-C.sub.4 H.sub.9 CH.sub.3 3.65(S, 3H); 2.25(S, 3H);                         2.2(S, 3H)                                                                  17 4-t-C.sub.4 H.sub.9 Allyl  69                                               18 4-t-C.sub.4 H.sub.9 Propargyl  117                                          19 4-t-C.sub.4 H.sub.9 CH.sub.2 --OCH.sub.3 3.65(S, 3H); 2.25(S, 3H);                                                117                                         2.2(S, 3H)                                                                  20 4-t-C.sub.4 H.sub.9 CO--OCH.sub.3 3.65; 2.1 119                             21 4-CH.sub.3 CH.sub.3  69                                                     22 4-CH.sub.3 Allyl 3.65(S, 3H); 2.25(S, 3H);                                     2.2(S, 3H)                                                                  23 4-CH.sub.3 Propargyl 3.65(S, 3H); 2.3(S, 3H);                                  2.2(S, 3H)                                                                  24 4-CH.sub.3 CH.sub.2 --OCH.sub.3 3.65(S, 3H); 2.3(S, 3H);                       2.2(S, 3H)                                                                  25 4-CH.sub.3 CO--OCH.sub.3  97                                                26 4-CF.sub.3 CH.sub.3  76                                                     27 4-CF.sub.3 Allyl 3.65(S, 3H); 2.3(S, 3H);                                      2.25(S, 3H)                                                                 28 4-CF.sub.3 Propargyl 3.65(S, 3H); 2.3(S, 3H);                                  2.25(S, 3H)                                                                 29 4-CF.sub.3 CH.sub.2 --OCH.sub.3 3.65(S, 3H); 2.25(S, 6H)                    30 4-CF.sub.3 CO--OCH.sub.3  103                                               31 4-Cl CH.sub.3  106                                                          32 4-Cl Allyl 3.65(S, 3H); 2.2(2S,                                                each 3H)                                                                    33 4-Cl Propargyl 3.65(S, 3H); 2.3(S, 3H;                                         2.2(S, 3H)                                                                  34 4-Cl CH.sub.2 --OCH.sub.3 3.65(S, 3H); 2.25(S, 3H;                             2.2(S, 3H)                                                                  35 4-Cl CO--OCH.sub.3  109                                                     36 3-Br CH.sub.3  75                                                           37 3-Br Allyl 3.65(S, 3H); 2.2(2S,                                                each 3H                                                                     38 3-Br Propargyl 3.65(S, 3H); 2.3(S, 3H);                                        2.2(S, 3H)                                                                  39 3-Br CH.sub.2 --OCH.sub.3  72                                               40 3-Br CO--OCH.sub.3  131                                                     41 3-Cl CH.sub.3  84                                                           42 3-Cl Allyl 3.65(S, 3H); 2.25(S, 3H);                                           2.2(S, 3H)                                                                  43 3-Cl Propargyl 3.65(S, 3H); 2.3(S, 3H);                                        2.2(S, 3H)                                                                  44 3-Cl CH.sub.2 --OCH.sub.3  66                                               45 3-Cl CO--OCH.sub.3  123                                                     46 3-CF.sub.3 CH.sub.3  63                                                     47 3-CF.sub.3 Allyl  64                                                        48 3-CF.sub.3 Propargyl 3.65(S, 3H); 2.3(S, 3H);                                  2.25(S, 3H)                                                                 49 3-CF.sub.3 CH.sub.2 --OCH.sub.3  89                                         50 3-CF.sub.3 CO--OCH.sub.3  136                                               51 4-Br CO--OCH.sub.3  103                                                     52 4-Br H  108                                                                 53 4-Br Propargyl 1710, 1486, 1469, 1447,                                         1376, 1299, 1252, 1026,                                                        1008, 774                                                                   54 4-Br CH.sub.2 --OCH.sub.3 1715, 1468, 1445, 1370,                              1301, 1274, 1090, 1059,                                                        1008, 775                                                                   55 3,4-(CH.sub.3).sub.2 CH.sub.3  oil                                          56 3,4-(CH.sub.3).sub.2 Allyl  oil                                             57 3,4-(CH.sub.3).sub.2 Propargyl  oil                                         58 3,4-(CH.sub.3).sub.2 CH.sub.2 --OCH.sub.3  oil                              59 3,4-(CH.sub.3).sub.2 CO--COH.sub.3  135                                     60 3,5-Cl.sub.2 CH.sub.3  95                                                   61 3,5-Cl.sub.2 Allyl  97                                                      62 3,5-Cl.sub.2 Propargyl  100                                                 63 3,5-Cl.sub.2 CH.sub.2 --OCH.sub.3  112                                      64 3,5-Cl.sub.2 CO--OCH.sub.3  160                                           ______________________________________                                    

                  TABLE 48                                                         ______________________________________                                         Selected physical data of some compounds                                          -                                                                           2  STR281##                                                                       -                             IR (cm.sup.-1) or                                  .sup.1 H-NMR                                                                No. X.sub.m R.sup.1 (ppm) mp                                                 ______________________________________                                          1   2-CH.sub.3 -4-C(CH.sub.3)═                                                                 H                   82                                       N--OCH.sub.3                                                                   2 2,4-(CH.sub.3).sub.2 H  131                                                  3 2,5-(CH.sub.3).sub.2 H  124                                                  4 2-CH.sub.3 -4-C(CH.sub.3)═ H  102                                        N--OC.sub.2 H.sub.5                                                            5 2,5-(CH.sub.3).sub.2 -4-C(CH.sub.3)═ H  116                              N--OC.sub.2 H.sub.5                                                            6 2,5-(CH.sub.3).sub.2 -4-C(CH.sub.3)═ H  122                              N--OCH.sub.3                                                                   7 2-CH.sub.3 -4-C(CH.sub.3)═ CH.sub.3 4.0(S, 3H);                          N--OCH.sub.3  3.65(S, 3H)                                                      8 2-CH.sub.3 -4-C(CH.sub.3)═ Allyl  101                                    N--OCH.sub.3                                                                   9 2-CH.sub.3 -4-C(CH.sub.3)═ Propargyl 4.0(S, 3H);                         N--OCH.sub.3  3.65(S, 3H)                                                     10 2-CH.sub.3 -4-C(CH.sub.3)═ CH.sub.2 --OCH.sub.3 4.0(S, 3H);                                                     N--OCH.sub.3  3.65(S, 3H)                                                     11 2-CH.sub.3 -4-C(CH.sub.3)═                                              CO--OCH.sub.3  122                       N--OCH.sub.3                                                                  12 2,4-(CH.sub.3).sub.2 CH.sub.3 3.65(S, 3H);                                     2.25(2s,                                                                       each 3H)                                                                    13 2,4-(CH.sub.3).sub.2 Allyl   59                                             14 2,4-(CH.sub.3).sub.2 Propargyl 3.65(S, 3H);                                    2.25(3s,                                                                       each 3H)                                                                    15 2,4-(CH.sub.3).sub.2 CH.sub.2 --OCH.sub.3   76                              16 2,4-(CH.sub.3).sub.2 CO--OCH.sub.3  133                                     17 2,5-(CH.sub.3).sub.2 CH.sub.3 3.65(S, 3H);                                     2.3(S, 3H)                                                                  18 2,5-(CH.sub.3).sub.2 Allyl   56                                             19 2,5-(CH.sub.3).sub.2 Propargyl   80                                         20 2,5-(CH.sub.3).sub.2 CH.sub.2 --OCH.sub.3 3.65(S, 3H);  80                     2.3(S, 3H)                                                                  21 2,5-(CH.sub.3).sub.2 CH.sub.2 --OCH.sub.3  140                              22 2-CH.sub.3 H  107                                                           23 2-CH.sub.3 Propargyl  oil                                                   24 2-CH.sub.3 CO--OCH.sub.3  135                                               25 2-CH.sub.3 CH.sub.2 --OCH.sub.3  oil                                        26 2-CH.sub.3 -4-C(CH.sub.3)═N--O- H   97                                   Allyl                                                                         27 2-CH.sub.3 -4-C(CH.sub.3)═N--O- Propargyl  oil                           Allyl                                                                         28 2-CH.sub.3 -4-C(CH.sub.3)═N--O- CO--OCH.sub.3  130                       Allyl                                                                         29 2-CH.sub.3 -4-C(CH.sub.3)═N--O- CH.sub.2 --OCH.sub.3  oil                                                       Allyl                                  30 2-CH.sub.3 -4-C(CH.sub.3)═N-- CH.sub.3  oil                              O--C.sub.2 H.sub.5                                                            31 2-CH.sub.3 -4-C(CH.sub.3)═N-- Allyl   75                                 O--C.sub.2 H.sub.5                                                            32 2-CH.sub.3 -4-C(CH.sub.3)═N-- Propargyl   77                             O--C.sub.2 H.sub.5                                                            33 2-CH.sub.3 -4-C(CH.sub.3)═N-- CH.sub.2 --OCH.sub.3  oil                  O--C.sub.2 H.sub.5                                                            34 2-CH.sub.3 -4-C(CH.sub.3)═N-- CO--OCH.sub.3  oil                         O--C.sub.2 H.sub.5                                                            35 2,5-(CH.sub.3).sub.2 -4-C(CH.sub.3)═ CH.sub.3  oil                       N--OCH.sub.3                                                                  36 2,5-(CH.sub.3).sub.2 -4-C(CH.sub.3)═ Allyl  104                          N--OCH.sub.3                                                                  37 2,5-(CH.sub.3).sub.2 -4-C(CH.sub.3)═ Propargyl  oil                      N--OCH.sub.3                                                                  38 2,5-(CH.sub.3).sub.2 -4-C(CH.sub.3)═ CH.sub.2 --OCH.sub.3  oil                                                  N--OCH.sub.3                           39 2,5-(CH.sub.3).sub.2 -4-C(CH.sub.3)═ CO--OCH.sub.3  158                  N--OCH.sub.3                                                                  40 2,5-(CH.sub.3).sub.2 -4-C(CH.sub.3)═ CH.sub.3  oil                       N--OC.sub.2 H.sub.5                                                           41 2,5-(CH.sub.3).sub.2 -4-C(CH.sub.3)═ Allyl   71                          N--OC.sub.2 H.sub.5                                                           42 2,5-(CH.sub.3).sub.2 -4-C(CH.sub.3)═ Propargyl  oil                      N--OC.sub.2 H.sub.5                                                           43 2,5-(CH.sub.3).sub.2 -4-C(CH.sub.3)═ CH.sub.2 --OCH.sub.3  oil                                                  N--OC.sub.2 H.sub.5                    44 2,5-(CH.sub.3).sub.2 -4-C(CH.sub.3)═ CO--OCH.sub.3  128                  N--OC.sub.2 H.sub.5                                                         ______________________________________                                    

                  TABLE 49                                                         ______________________________________                                         2  STR282##                                                                       -                                                                               I: R.sup.1 = H, X = CH.sub.3                                                                     VIII: R.sup.1 = H, X = Cl                                  II: R.sup.1 = CH.sub.3, X = CH.sub.3 IX: R.sup.1 = CH.sub.3, X = Cl                                 III: R.sup.1 = C.sub.2 H.sub.5, X = CH.sub.3 X:                               R.sup.1 = C.sub.2 H.sub.5, X = Cl                          IV: R.sup.1 = Allyl, X = CH.sub.3 XI: R.sup.1 = Allyl, X = Cl                  V: R.sup.1 = Propargyl, X = CH.sub.3 XII: R.sup.1 = Propargyl, X = Cl                               VI: R.sup.1 = CH.sub.2 --OCH.sub.3, X = CH.sub.3                              XIII: R.sup.1 = CH.sub.2 --OCH.sub.3, X = Cl                                    VII: R.sup.1 = CO.sub.2 CH.sub.3, X = CH.sub.3                                XIV: R.sup.1 = CO.sub.2 CH.sub.3, X = Cl                 No.     B                                                                      ______________________________________                                         1       2-Pyridyl                                                                2 3-Trifluoromethyl-2-pyridyl                                                  3 5-Trifluoromethyl-2-pyridyl                                                  4 3,5-Bis-(trifluoromethyl)-2-pyridyl                                          5 3,5-Dichloro-2-pyridyl                                                       6 3-Chloro-5-trifluoromethyl-2-pyridyl                                         7 3,5-Dichloro-2-pyridyl                                                       8 2-Chloro-4-trifluoromethylphenyl                                             9 2-Benzothiazolyl                                                             10  5-Chloro-1-methyl-2-benzimidazolyl                                         11  2-Benzoxazolyl                                                             12  1-Methyl-5-trifluoromethylimide-azo[5,4-a]-pyridin-2-yl                    13  5-Chloro-2-pyrimidinyl                                                     14  4-Methyl-5-phenyl-2-thiazolin-2-yl                                         15  4-Methyl-5-phenyl-2-oxazolin-2-yl                                          16  7-Trifluoromethyl-4-quinolinyl                                           ______________________________________                                    

                  TABLE 50                                                         ______________________________________                                         Selected physical data of some compounds                                       3  STR283##                                                                      No.      X.sub.m     IR(cm.sup.-1) or .sup.1 H-NMR (ppm)                                                          mp                                        ______________________________________                                          1     4-NO.sub.2                  112                                            2 3,4-Cl.sub.2 3.8(s, 3H); 3.75(s, 3H)                                         3 2,4-(CH.sub.3).sub.2 3.75(s, 3H); 3.7(s, 3H)                                 4 H 3.75(2s, each 3H)                                                          5 4-i-C.sub.3 H.sub.7 3.8(s, 3H); 3.75(s, 3H)                                  6 3,4-(CH.sub.3).sub.2 3.8(s, 3H); 3.75(s, 3H)                                 7 3-CH.sub.3 -4-OCH.sub.3 3.85(s, 3H); 3.8(s, 3H);                              3.75(s, 3H)                                                                   8 3-CH.sub.3 -4-O- 3.8(2s, each 3H)                                            i-C.sub.3 H.sub.7                                                              9 4-CF.sub.3 3.8(s, 3H); 3.75(s, 3H)                                          10 3-CH.sub.3 3.8(2s, each 3H)                                                 11 3-CF.sub.3 3.8(s, 3H); 3.75(s, 3H)                                          12 4-F 3.8(s, 3H); 3.75(s, 3H)                                                 13 4-Br 3.8(s, 3H); 3.75(s, 3H)                                                14 3-Br 3.8(s, 3H); 3.75(s, 3H)                                                15 4-t-Bu 3.8(s, 3H); 3.75(s, 3H)                                              16 4-OCH.sub.3 3.85(s, 3H); 3.8(s, 3H);                                          3.75(s, 3H)                                                                  17 2-CH.sub.3 3.8(s, 3H); 3.75(s, 3H)                                          18 3-Cl 3.8(s, 3H); 3.75(s, 3H)                                                19 4-CN 3.8(s, 3H); 3.75(s, 3H)                                                20 4-C.sub.2 H.sub.5 3.8(s, 3H); 3.75(s, 3H)                                 ______________________________________                                    

                  TABLE 51                                                         ______________________________________                                         Selected physical data of some compounds                                          -                                                                           2  STR284##                                                                      No.     X.sub.m         IR (cm.sup.-1) or .sup.1 H-NMR (ppm)                                                          mp                                    ______________________________________                                         1     4-Cl            3.8(s, 3H); 3.75(s, 3H)                                    2 2-Cl 3.8(s, 3H); 3.75(s, 3H)                                                 3 2,5-(CH.sub.3).sub.2 -4-C(C.sub.2 H.sub.5)═ 3.8(s, 3H); 3.75(s,                              3H)                                                         N--O-Allyl                                                                    4 2,5-(CH.sub.3).sub.2 -4-C(C.sub.2 H.sub.5)═ 3.9(s, 3H); 3,8(s,                               3H);                                                        N--O--CH.sub.3 3.75(s, 3H)                                                    5 2-CH.sub.3 -4-C(C.sub.2 H.sub.5)═N--O- 3.8(s, 3H); 3.75(s, 3H)                                 trans-Cl-Allyl                                           6 2-CH.sub.3 -4-C(C.sub.2 H.sub.5)═N--O- 3.8(s, 3H); 3.75(s, 3H)                                 Allyl                                                    7 2-CH.sub.3 -4-Cl 3.8(s, 3H); 3.75(s, 3H)                                     8 2-Cl-4-CH.sub.3 3.8(s, 3H); 3.75(s, 3H)                                      9 2-Cl-5-CH.sub.3 3.8(s, 3H); 3.75(s, 3H)                                      10  2-CH.sub.3 -4-C(C.sub.2 H.sub.5)═N-- 4.2(q, 2H); 3.8(s, 3H);                                 O--C.sub.2 H.sub.5 3.75(s, 3H)                           11  2-CH.sub.3 -4-C(C.sub.2 H.sub.5)═N-- 3.95(s, 3H); 3.8(s, 3H);                                O--CH.sub.3 3.75(s, 3H)                                  12  2,5-(CH.sub.3).sub.2 -4-C(CH.sub.3)═ 3.8(s, 3H); 3.75(s, 3H)                                 N--O-trans-Cl-Allyl                                      13  2,5-(CH.sub.3).sub.2 -4-C(CH.sub.3)═ 4.2(t, 2H); 3.8(s, 3H);                                 --N--O--C.sub.2 H.sub.5 3.75(s, 3H)                      14  2,5-(CH.sub.3).sub.2 -4-C(CH.sub.3)═ 3.95(s, 3H); 3.8(s, 3H);                                N--O--CH.sub.3 3.75(s, 3H)                               15  2-CH.sub.3 -4-C(CH.sub.3)═N--O- 3.8(s, 3H); 3.75(s, 3H)                                      trans-Cl-Allyl                                           16  2-CH.sub.3 -4-C(CH.sub.3)═N-- 4.2(t, 2H); 3.8(s, 3H);                   O--C.sub.2 H.sub.5 3.75(s, 3H)                                                17  2,5-(CH.sub.3).sub.2 -4-C(C.sub.2 H.sub.5)═ 4.2(t, 2H); 3.8(s,                             3H);                                                        N--O--C.sub.2 H.sub.5 3.75(s, 3H)                                           ______________________________________                                    

                  TABLE 60                                                         ______________________________________                                         3  STR285##                                                                      No.           B                                                              ______________________________________                                         1           Phenyl                                                               2 3-Phenoxyphenyl                                                              3 3-(2-Cyanophenoxy)-phenyl                                                    4 4-Chlorophenyl                                                               5 3-Trifluoromethylphenyl                                                      6 3-tert.-Butoxyphenyl                                                         7 3,5-Dichlorophenyl                                                           8 3,5-Diethylphenyl                                                            9 2-Pyridyl                                                                    10  4-Pyrimidinyl                                                              11  6-Phenoxy-pyrimidin-4-yl                                                   12  6-Chloropyrimidin-4-yl                                                     13  6-(2-Fluorophenoxy)-pyrimidin-4-yl                                         14  6-(2-Methylphenoxy)-pyrimidin-4-yl                                         15  6-(2-Cyanophenoxy)-pyrimidin-4-yl                                          16  6-(2,6-Difluorophenoxy)-pyrimidin-4-yl                                   ______________________________________                                    

The novel compounds are suitable as fungicides.

The fungicidal compounds according to the invention, or agents containing them, may be applied for instance in the form of directly sprayable solutions, powders, suspensions (including high-percentage aqueous, oily or other suspensions), dispersions, emulsions, oil dispersions, pastes, dusts, broadcasting agents, or granules by spraying, atomizing, dusting, broadcasting or watering. The forms of application depend entirely on the purpose for which the agents are being used, but they must ensure as fine a distribution of the active ingredients according to the invention as possible.

Normally, the plants are sprayed or dusted with the active ingredients, or the seeds of the plants are treated with the active ingredients.

The formulations are produced in known manner, for example by extending the active ingredient with solvents and/or carriers, with or without the use of emulsifiers and dispersants; water is used as solvent, it is also possible to employ other organic solvents as auxiliary solvents. Suitable auxiliaries for this purpose are solvents such as aromatics (e.g., xylene), chlorinated aromatics (e.g., chlorobenzenes), paraffins (e.g., crude oil fractions), alcohols (e.g., methanol, butanol), ketones (e.g., cyclohexanone), amines (e.g., ethanolamine, dimethylformamide), and water; carriers such as ground natural minerals (e.g., kaolins, aluminas, talc and chalk) and ground synthetic minerals (e.g., highly disperse silica and silicates); emulsifiers such as nonionic and anionic emulsifiers (e.g., polyoxyethylene fatty alcohol ethers, alkyl sulfonates and aryl sulfonates); and dispersants such as lignin-sulfite waste liquors and methylcellulose.

Examples of surfactants are: alkali metal, alkaline earth metal and ammonium salts of aromatic sulfonic acids, e.g., ligninsulfonic acid, phenolsulfonic acid, naphthalenesulfonic acid and dibutylnaphthalenesulfonic acid, and of fatty acids, alkyl and alkylaryl sulfonates, and alkyl, lauryl ether and fatty alcohol sulfates, and salts of sulfated hexadecanols, heptadecanols, and octadecanols, salts of fatty alcohol glycol ethers, condensation products of sulfonated naphthalene and naphthalene derivatives with formaldehyde, condensation products of naphthalene or naphthalenesulfonic acids with phenol and formaldehyde, polyoxyethylene octylphenol ethers, ethoxylated isooctylphenol, ethoxylated octylphenol and ethoxylated nonylphenol, alkylphenol polyglycol ethers, tributylphenyl polyglycol ethers, alkylaryl polyether alcohols, isotridecyl alcohol, fatty alcohol ethylene oxide condensates, ethoxylated castor oil, polyoxyethylene alkyl ethers, ethoxylated polyoxypropylene, lauryl alcohol polyglycol ether acetal, sorbitol esters, lignin-sulfite waste liquors and methyl cellulose.

Powders, dusts and broadcasting agents may be prepared by mixing or grinding the active ingredients with a solid carrier.

Granules, e.g., coated, impregnated or homogeneous granules, may be prepared by bonding the active ingredients to solid carriers. Examples of solid carriers are mineral earths such as silicic acids, silica gels, silicates, talc, kaolin, attapulgus clay, limestone, lime, chalk, bole, loess, clay, dolomite, diatomaceous earth, calcium sulfate, magnesium sulfate, magnesium oxide, ground plastics, fertilizers such as ammonium sulfate, ammonium phosphate, ammonium nitrate, and ureas, and vegetable products such as grain meals, bark meal, wood meal, and nutshell meal, cellulosic powders, etc.

Examples of formulations are given below.

I. A solution of 90 parts by weight of the compound from Table 7, No. 1 (7/1) and 10 parts by weight of N-methyl-α-pyrrolidone, which is suitable for application in the form of very fine drops.

II. A mixture of 20 parts by weight of compound 7/2, 80 parts by weight of xylene, 10 parts by weight of the adduct of 8 to 10 moles of ethylene oxide and 1 mole of oleic acid-N-monoethanolamide, 5 parts by weight of the calcium salt of dodecylbenzenesulfonic acid, and 5 parts by weight of the adduct of 40 moles of ethylene oxide and 1 mole of castor oil. By finely dispersing the mixture in water, a dispersion is obtained.

III. An aqueous dispersion of 20 parts by weight of compound 7/3, 40 parts by weight of cyclohexanone, 30 parts by weight of isobutanol, 20 parts by weight of the adduct of 40 moles of ethylene oxide and 1 mole of castor oil.

IV. An aqueous dispersion of 20 parts by weight of compound 7/4, 25 parts by weight of cyclohexanol, 65 parts by weight of a mineral oil fraction having a boiling point between 210 and 280° C., and 10 parts by weight of the adduct of 40 moles of ethylene oxide and 1 mole of castor oil.

V. A hammer-milled mixture of 80 parts by weight of compound 7/5, 3 parts by weight of the sodium salt of diisobutylnaphthalene-α-sulfonic acid, 10 parts by weight of the sodium salt of a lignin-sulfonic acid obtained from a sulfite waste liquor, and 7 parts by weight of powdered silica gel. By finely dispersing the mixture in water, a spray liquor is obtained.

VI. An intimate mixture of 3 parts by weight of compound 7/6 and 97 parts by weight of particulate kaolin. The dust contains 3wt % of the active ingredient.

VII. An intimate mixture of 30 parts by weight of compound 7/7, 92 parts by weight of powdered silica gel and 8 parts by weight of paraffin oil sprayed onto the surface of this silica gel. This formulation of the active ingredient exhibits good adherence.

VIII. A stable aqueous dispersion of 40 parts by weight of compound 7/8, 10 parts of the sodium salt of a phenolsulfonic acid-urea-formaldehyde condensate, 2 parts of silica gel and 48 parts of water, which dispersion can be further diluted.

IX. A stable oily dispersion of 20 parts by weight of compound 7/9, 2 parts by weight of the calcium salt of dodecylbenzenesulfonic acid, 8 parts by weight of a fatty alcohol polyglycol ether, 2 parts by weight of the sodium salt of a phenolsulfonic acid-urea-formaldehyde condensate and 68 parts by weight of a paraffinic mineral oil.

The novel compounds are extremely effective on a broad spectrum of phytopathogenic fungi, in particular those from the class consisting of the Ascomycetes and Basidiomycetes. Some of them have a systemic action and can be used as foliar and soil fungicides.

The fungicidal compounds are of particular interest for controlling a large number of fungi in various crops or their seeds, especially wheat, rye, barley, oats, rice, Indian corn, lawns, cotton, soybeans, coffee, sugar cane, fruit and ornamentals in horticulture and viticulture, and in vegetables such as cucumbers, beans and cucurbits.

The compounds are applied by treating the fungi, or the seeds, plants, materials or soil to be protected against fungus attack with a fungicidally effective amount of the active ingredients.

The agents may be applied before or after infection of the materials, plants or seed by the fungi.

The compounds I are particularly useful for controlling the following plant diseases:

Erysiphe graminis in cereals,

Erysiphe cichoracearum and Sphaerotheca fuliginea in cucurbits,

Podosphaera leucotricha in apples,

Uncinula necator in vines,

Puccinia species in cereals,

Rhizoctonia solani in cotton,

Ustilago species in cereals and sugar cane,

Venturia inaequalis (scab) in apples,

Helminthosporium species in cereals,

Septoria nodorum in wheat,

Botrytis cinerea (gray mold) in strawberries and grapes,

Cercospora arachidicola in groundnuts,

Pseudocercosporella herpotrichoides in wheat and barley,

Pyricularia oryzae in rice,

Phytophthora infestans in potatoes and tomatoes,

Fusarium and Verticillium species in various plants,

Plasmopara viticola in grapes,

Alternaria species in fruit and vegetables.

The novel compounds may also be used for protecting materials (timber), for instance against Paecilomyces variotii.

The fungicidal agents generally contain from 0.1 to 95, an preferably from 0.5 to 90, wt % of active ingredient.

The application rates depend on the effect desired, and are from 0.02 to 3 kg of active ingredient per hectare.

When the active ingredients are used for treating seed, amounts of from 0.001 to 50, and preferably from 0.01 to 10, g per kg of seed are generally needed.

When the agents according to the invention are used as fungicides, they may be present together with other active ingredients, e.g., herbicides, insecticides, growth regulators, other fungicides, and fertilizers.

When they are mixed with other fungicides, the spectrum of fungicidal action is in many cases increased.

USE EXAMPLES

The active ingredients used for comparison purposes were isopropyl N-phenylcarbamate (A)--known from GB 574 995--, isopropyl N-3-chlorophenylcarbamate (B)--known from GB 574 995--and methyl N-3,4-dichlorophenylcarbamate (C)--known from BE 612 550.

Example 1

Action on Wheat Mildew

Leaves of pot-grown wheat seedlings of the "Fruhgold" variety were sprayed with aqueous liquors containing (dry basis) 80% of active ingredient and 20% of emulsifier, and dusted, 24 hours after the sprayed-on layer had dried, with spores of wheat mildew (Erysiphe graminis var. tritici). The plants were then set up in the greenhouse at from 20 to 22° C. and a relative humidity of from 75 to 80%. The extent of mildew spread was assessed after 7 days.

The results show that active ingredients nos. 1, 2, 3, 4, 8, 9, 20, 23, 31, 33, 34, 35, 36, 42, 43, 44, 47, 48, 52, 53, 54, 55, 56, 57, 60, 61, 62, 63, 64, 67, 69, 70, 71, 72, 74, 78, 79, 85, 87, 89, 90, 91, 92, 93, 94, 95, 104, 105, 106 and 107 from Table 7 have, when applied as spray liquors containing 250 ppm of active ingredient, a better fungicidal action (95%) than prior art comparative agents A (45%), B (45%) and C (45%).

Example 2

Action on Pyricularia oryzae (Protective)

Leaves of pot-grown rice seedlings of the "Bahia" variety were sprayed to runoff with aqueous emulsions containing (dry basis) 80% of active ingredient and 20% of emulsifier, and inoculated 24 hours later with an aqueous spore suspension of Pyricularia oryzae. The plants were then set up in climatic cabinets at 22 to 24° C. and 95 to 99% relative humidity. The extent of fungus attack was assessed after 6 days.

The results show that active ingredients nos. 1, 2, 12, 18, 19, 22, 29, 39, 40, 42, 47, 49, 50, 52, 53, 54, 60, 61, 62, 63, 69, 70, 71, 72, 73, 74, 81, 83, 85, 87, 89, 90, 91, 92, 94, 95, 104, 105, 106 and 107 from Table 7 have, when applied as spray liquors containing 250 ppm of active ingredient, a better fungicidal action (95%) than prior art comparative agents A (30%), B (30%) and C (30%).

Example 3

Action on Wheat Mildew

Leaves of pot-grown wheat seedlings of the "Fruhgold" variety were sprayed with aqueous liquors containing (dry basis) 80% of active ingredient and 20% of emulsifier, and dusted, 24 hours after the sprayed-on layer had dried, with spores of wheat mildew (Erysiphe graminis var. tritici). The plants were then set up in the greenhouse at from 20 to 22° C. and a relative humidity of from 75 to 80%. The extent of mildew spread was assessed after 7 days.

The results show that active ingredient no. 3 from Table 14, nos. 3 and 4 from Table 21, nos. 1, 3, 4, 5, 6, 7, 8, 9, 10, 11, 15, 17, 18, 19, 20, 21, 22, 23, 24, 25, 26, 27, 28, 29, 30, 31, 32, 33, 34, 35, 36, 37, 38, 39, 40 41, 42, 43 and 44 from Table 48, nos. 7, 8, 9, 10, 11, 13, 14, 15, 16, 17, 18, 20 and 23 from Table 14, nos. 1, 2, 3, 4, 5, 6, 7, 8, 9, 10, 11, 12, 13, 14, 15, 16, 17, 18 and 19 from Table 52, and nos. 1, 2, 3, 4, 5, 6, 7, 8, 9, 10, 11, 12, 13, 14, 15, 16 and 17 from Table 53 have, when applied as spray liquors containing 250 ppm of active ingredient, a better fungicidal action (100%) than prior art comparative agents A, B and C

Example 4

Action on Pyricularia oryzae (Protective)

Leaves of pot-grown rice seedlings of the "Bahia" variety were sprayed to runoff with aqueous emulsions containing (dry basis) 80% of active ingredient and 20% of emulsifier, and inoculated 24 hours later with an aqueous spore suspension of Pyricularia oryzae. The plants were then set up in climatic cabinets at 22 to 24° C. and 95 to 99% relative humidity. The extent of fungus attack was assessed after 6 days.

The results show that active ingredient nos. 3, 7, 8, 9, 10, 11, 13, 14, 15, 16, 17, 18, 20, 21, 22 and 24 from Table 14, nos. 1, 2, 3, 4, 5, 6, 7, 8, 9, 10, 11, 12, 13, 14, 15, 16, 17, 18, 19 and 20 from Table 52, nos. 1, 2, 3, 4, 5, 6, 7, 8, 9, 10, 11, 12, 13, 14, 15, 16 and 17 from Table 53, nos. 3 and 4 from Table 21, nos. 4 and 5 from Table 38, nos. 4, 7, 10, 16, 20, 21, 22, 23, 24, 25, 41, 42, 55, 56, 57, 58 and 59 from Table 47, and nos. 1, 4, 5, 6, 7, 8, 11, 20, 21, 22, 23, 24, 25, 26, 27, 28, 29, 30, 31, 32, 33, 34, 35, 36, 37, 38, 39, 40, 41, 42, 43 and 44 from Table 48 have, when applied as spray liquors containing 250 ppm of active ingredient, a better fungicidal action (100%) than prior art comparative agents A, B and C (0%).

Use Example 5

Action on Botrytis cinerea

Paprika seedlings of the "Neusiedler Ideal Elite" variety were sprayed, after 4 to 5 leaves were well developed, to runoff with aqueous suspensions containing (dry basis) 80% of active ingredient and 20% of emulsifier. After the sprayed-on layer had dried, the plants were sprinkled with a conidial suspension of the fungus Botrytis cinerea, and placed at 22 to 24° C. in a chamber of high humidity. After 5 days, the disease had spread to such a great extent on the untreated plants that the necroses covered the major portion of the leaves.

    ______________________________________                                                         Percentage leaf attack after                                      spraying with aqueous for-                                                     mulations containing 500 ppm                                                  Active ingredient of active ingredient                                       ______________________________________                                         Table 30, active ingr. no. 2                                                                    5                                                               Comparative substance A 100                                                    Comparative substance B 100                                                    Comparative substance C 100                                                    Untreated 100                                                                ______________________________________                                    

Use Example 6

Action on Plasmopara viticola

Leaves of potted vines of the Muller-Thurgau variety were sprayed with aqueous suspensions containing (dry basis) 80% of active ingredient and 20% of emulsifier. To assess the duration of action, the plants were set up, after the sprayed-on layer had dried, for 8 days in the greenhouse. Then the leaves were infected with a zoospore suspension of Plasmopara viticola. The plants were first placed for 48 hours in a water vapor-saturated chamber at 24° C. and then in a greenhouse for 5 days at from 20 to 30° C. To accelerate and intensify the sporangiophore discharge, the plants were then again placed in the moist chamber for 16 hours. The extent of fungus attack was then assessed on the undersides of the leaves.

    ______________________________________                                                         Percentage leaf attack after                                      applying aqueous formula-                                                      tions containing 500 ppm of                                                   Active ingredient active ingredient                                          ______________________________________                                         Table 21, active ingr. no. 3                                                                   5                                                                Table 21, active ingr. no. 4 0                                                 Table 30, active ingr. no. 1 15                                                Comparative substance A 65                                                     Comparative substance B 40                                                     Comparative substance C 25                                                     Untreated 65                                                                 ______________________________________                                     

We claim:
 1. A carbamate of the formula VII ##STR286## where the substituents have the following meanings: X and Y are identical or different and each is hydrogen, F, Cl, Br, CF₃, CN, NO₂, alkoxy, alkenyloxy, alkynyloxy, alkyl, alkenyl or alkynyl or may together be condensed to form a substituted or unsubstituted aromatic or heteroaromatic, alicyclic or heterocyclic, partially or completely hydrogenated ring,R¹ is substituted or unsubstituted and is alkyl, alkenyl, alkynyl, cycloalkyl, cycloalkenyl or --CO₂ -alkyl, A is --O--, S--S, --CR² ═CR³ --, CHR² --O--, --CHR² --S--, --CHR² --O--N═C(R⁴)--, --CR² ═N--O--, --O--N═C(R⁴)--, --C═C--, --CHR² --CHR³ --, --CHR² --O--CO--, --O--CHR² -- or a single bond, B is a substituted or unsubstituted, saturated or unsaturated heterocyclic group, R² and R³ are identical or different and each is hydrogen, alkyl, alkenyl, alkynyl or cycloalkyl and R⁴ is hydrogen, cyano, alkyl, alkenyl, alkynyl, cycloalkyl or alkoxy, or plant-tolerated acid and base adducts.
 2. A carbamate of the formula VIII ##STR287## where A, B, and R¹ have the meanings given in claim
 1. 3. A carbamate of the formula IX ##STR288## where R¹ and B have the meanings given in claim
 1. 4. A carbamate of the formula X ##STR289## where R¹ and B have the meanings given in claim
 1. 5. Hydroxylamine derivatives of the formula XIV ##STR290## where the substituents have the following meanings: Z is NH₂, NHCH₃, N(CH₃)₂, CH₃, C₂ H₅, CF₃ or CCl₃,X and Y are identical or different and each is hydrogen, F, Cl, Br, CF₃, CN, NO₂, alkoxy, alkenyloxy, alkynyloxy, alkyl, alkenyl or alkynyl or together may be condensed to form a substituted or unsubstituted aromatic or heteroaromatic, alicyclic or heterocyclic, partially or completely hydrogenated ring, R¹ is substituted or unsubstituted and is alkyl, alkenyl, alkynyl, cycloalkyl, cycloalkenyl or --CO₂ -alkyl, A is --O--, --S--, --CR² ═CR³ --, CHR² --O--, --CHR² --S--, --CHR² --O--N═C(R⁴)--, --CR² ═N--O--, --O--N═C(R⁴)--, --C═C--, --CHR² --CHR³ --, --CHR² --O--CO--, --O--CHR² -- or a single bond, B is a substituted or unsubstituted, saturated or unsaturated heterocyclic group, R² and R³ are identical or different and each is hydrogen, alkyl, alkenyl, alkynyl or cycloalkyl and R⁴ is hydrogen, cyano, alkyl, alkenyl, alkynyl, cycloalkyl or alkoxy, or its plant-tolerated acid and base adducts.
 6. A compound of the formula XV ##STR291## where A is --O--, --S--, --CR² ═CR³ --, CHR² --O----CHR² --S--, --CHR² --O--N═C(R⁴)--, --CR² ═N--O--, --O--N═C(R⁴)--, --C═C--, --CHR² --CHR³ --, --CHR² --O--CO--, --O--CHR² -- or a single bond, B is a substituted or unsubstituted saturated or unsaturated heterocyclic group, Z is methoxy, NH₂, NHCH₃, N(CH₃)₂, CH₃, C₂ H₅, CF₃ or CCl₃, R¹ is substituted or unsubstituted and is alkyl, alkenyl, alkynyl, cycloalkyl, cycloalkenyl or --CO₂ -alkyl and X and Y are identical or different and each is hydrogen, F, Cl, Br, C₁ -C₄ -alkyl, C₁ -C₄ -alkoxy or cyano.
 7. A compound of the formula XV as set forth in claim 6, where Y is hydrogen.
 8. A compound of the formula XV as set forth in claim 6, where X and Y are hydrogen.
 9. A compound of the formula XVI ##STR292## where R¹, X, Y, Z and B have the meanings given in claim
 6. 10. A compound of the formula XVII ##STR293## where R¹, X, Y, Z and B have the meanings given in claim
 6. 11. A compound of the formula XIX ##STR294## where R¹, X, Y, z and B have the meanings given in claim
 6. 12. A compound of the formula XIX ##STR295## where R¹ is hydrogen, alkyl, alkenyl, alkynyl, cyclopropyl, cyclopropylmethyl, cyclobutyl, --CH₂ --CN, --CH₂ --O--CH₃, or --CO₂ CH₃, X and Y are identical or different and each is hydrogen, F, Cl, Br, CF₃, CN, NO₂, alkoxy, alkenyloxy, alkynyloxy, alkyl, alkenyl or alkynyl, or may be condensed together to form a phenyl ring, Z is methoxy, B is a substituted or unsubstituted saturated or unsaturated heterocyclic group.
 13. A compound of the formula XVI as set forth in claim 9, Y denoting hydrogen.
 14. A compound of the formula XVI as set forth in claim 9, X and Y denoting hydrogen.
 15. A compound of the formula XXV ##STR296## where the substituents have the following meanings: X and Y are identical or different and each is F, Cl, Br, CF₃, CN, NO₂, alkoxy, alkenyloxy, alkynyloxy, alkyl, alkenyl or alkynyl or may together be condensed to form a substituted or unsubstituted aromatic or heteroaromatic, alicyclic or heterocyclic, partially or completely hydrogenated ring, or Y is hydrogen,R¹ is substituted or unsubstituted and is alkyl, alkenyl, alkynyl, cycloalkyl, cycloalkenyl or --CO₂ -alkyl, A is --O----S--, --CR² ═CR³ --, CHR² --O--, --CHR² --S--, --CHR² --O--N═C(R⁴)--, --CR² ═N--O--, --O--N═C(R⁴)--, --C═C--, --CHR² --CHR³ --, --CHR² --O--CO--, --O--CHR² -- or a single bond, B is a substituted or unsubstituted, saturated or unsaturated heterocyclic group. R² and R³ are identical or different and each is hydrogen, alkyl, alkenyl, alkynyl or cycloalkyl and R⁴ is hydrogen, cyano, alkyl, alkenyl, alkynyl, cycloalkyl or alkoxy, or its plant-tolerated acid and base adducts.
 16. A compound of the formula XXVI ##STR297## where A, B and R¹ have the meanings given in claim 15 and X and Y are identical or different and each is F, Cl, Br, C₁ -C₄ -alkyl, C₁ -C₄ -alkoxy or cyano.
 17. A compound of the formula XXVI as set forth in claim 16, Y denoting hydrogen.
 18. A compound of the formula XXVII ##STR298## where R¹, X, Y and B have the meanings given in claim
 15. 19. A compound of the formula XXVIII ##STR299## where R¹, X, Y and B have the meanings given in claim
 15. 20. A compound of the formula XXIX ##STR300## where R¹, X, Y and B have the meanings given in claim
 15. 21. A compound of the formula XXX ##STR301## where R¹, X, Y and B have the meanings given in claim
 15. 22. A compound of the formula XXVII as set forth in claim 18, Y denoting hydrogen.
 23. An aniline derivative of the formula XXXVI ##STR302## where the substituents have the following meanings: Z is NH₂, NHCH₃, N(CH₃)₂, CH₃, C₂ H₅, CF₃, or CCl₃, X and Y are H,R¹ is H, A is --O--, B is pyrimidin-6-yl-4-O-2-methylphenyl, or its plant-tolerated acid and base adducts.
 24. A carbamate of the formula I ##STR303## where the substitutents have the following meanings: Z is methoxy,X and Y are H, R¹ is H, A is --O--, B is pyrimidin-6-yl-4-O-2-methylphenyl, or its plant-tolerated acid and base adducts. 